Details of the Target

General Information of Target

Target ID	LDTP18448
Target Name	Transmembrane 9 superfamily member 3 (TM9SF3)
Gene Name	TM9SF3
Gene ID	56889
Synonyms	SMBP; Transmembrane 9 superfamily member 3; EP70-P-iso; SM-11044-binding protein
3D Structure	Download 2D Sequence (FASTA) Download 3D Structure (PDB) Download
Sequence	MKMKKFQIPVSFQDLTVNFTQEEWQQLDPAQRLLYRDVMLENYSNLVSVGYHVSKPDVIF KLEQGEEPWIVEEFSNQNYPDIDDALEKNKEIQDKHLTQTVFFSNKTLITERENVFGKTL NLGMNSVPSRKMPYKCNPGGNSLKTNSEVIVAKKSKENRKIPDGYSGFGKHEKSHLGMKK YRYNPMRKASNQNENLILHQNIQILKQPFDYNKCGKTFFKRAILITQKGRQTERKPNECN ECRKTFSKRSTLIVHQRIHTGEKPYVCSDCRKTFRVKTSLTRHRRIHTGERPYECSECRK TFIDKSALIVHQKIHGGEKSYECNECGKTFFRKSALAEHFRSHTGEKPYECKECGNAFSK KSYLVVHQRTHRGEKPNECKECGKTFFCQSALTAHQRIHTGEKPYECSECEKTFFCQSAL NVHRRSHTGEKPYECSQCGKFLCTKSALIAHQITHRGKKSYECNECGKFFCHKSTLTIHQ RTHTGEKHGVFNKCGRISIVKSNCSQCKRMNTKENLYECSEHGHAVSKNSHLIVHQRTIW ERPYECNECGRTYCRKSALTHHQRTHTGQRPYECNECGKTFCQKFSFVEHQRTHTGEKPY ECNECGKSFCHKSAFRVHRRIHTGEKPYECNQCGKTYRRLWTLTEHQKIHTGEKPYECNK CEKTFRHKSNFLLHQKSHKE
Target Bioclass	Transporter and channel
Family	Nonaspanin (TM9SF) (TC 9.A.2) family
Subcellular location	Membrane
Uniprot ID	Q9HD45
Ensemble ID	ENST00000371142.9
HGNC ID	HGNC:21529

Probe(s) Labeling This Target

ABPP Probe

Click To Hide/Show 32 Probe Related to This Target

Probe name	Binding Site(Ratio)	Interaction ID	Ref
m-APA Probe Info	5.79	LDD0402	[1]
FBPP2 Probe Info	2.06	LDD0318	[2]
CY4 Probe Info	100.00	LDD0244	[3]
TH211 Probe Info	Y122(20.00); Y583(20.00); Y76(20.00); Y272(8.28)	LDD0260	[4]
YN-4 Probe Info	100.00	LDD0445	[5]
STPyne Probe Info	K440(6.92); K581(3.56)	LDD0277	[6]
ONAyne Probe Info	K581(8.71)	LDD0275	[6]
AHL-Pu-1 Probe Info	C66(2.10)	LDD0168	[7]
HPAP Probe Info	3.02	LDD0063	[8]
EA-probe Probe Info	N.A.	LDD0440	[9]
DBIA Probe Info	C428(1.05)	LDD0078	[10]
4-Iodoacetamidophenylacetylene Probe Info	C428(0.00); C66(0.00)	LDD0038	[11]
IA-alkyne Probe Info	C66(0.00); C428(0.00)	LDD0032	[12]
Lodoacetamide azide Probe Info	C428(0.00); C66(0.00)	LDD0037	[11]
BTD Probe Info	N.A.	LDD0004	[13]
JW-RF-010 Probe Info	N.A.	LDD0026	[14]
WYneN Probe Info	N.A.	LDD0021	[13]
WYneO Probe Info	N.A.	LDD0022	[13]
Compound 10 Probe Info	C428(0.00); C66(0.00)	LDD2216	[15]
Compound 11 Probe Info	N.A.	LDD2213	[15]
ENE Probe Info	N.A.	LDD0006	[13]
IPM Probe Info	N.A.	LDD0005	[13]
SF Probe Info	N.A.	LDD0028	[16]
TFBX Probe Info	N.A.	LDD0148	[14]
VSF Probe Info	N.A.	LDD0007	[13]
Acrolein Probe Info	C428(0.00); C66(0.00)	LDD0217	[17]
Cinnamaldehyde Probe Info	N.A.	LDD0220	[17]
Crotonaldehyde Probe Info	C428(0.00); H52(0.00); C66(0.00)	LDD0219	[17]
Methacrolein Probe Info	N.A.	LDD0218	[17]
W1 Probe Info	C428(0.00); D213(0.00); Q218(0.00); S215(0.00)	LDD0236	[18]
AOyne Probe Info	13.70	LDD0443	[19]
NAIA_5 Probe Info	N.A.	LDD2223	[20]

PAL-AfBPP Probe

Click To Hide/Show 156 Probe Related to This Target

Probe name	Binding Site(Ratio)	Interaction ID	Ref
DR-1 Probe Info	3.94	LDD0398	[21]
C004 Probe Info	9.32	LDD1714	[22]
C011 Probe Info	5.06	LDD1720	[22]
C017 Probe Info	7.11	LDD1725	[22]
C022 Probe Info	14.93	LDD1728	[22]
C026 Probe Info	6.36	LDD1732	[22]
C039 Probe Info	5.54	LDD1739	[22]
C040 Probe Info	12.38	LDD1740	[22]
C041 Probe Info	7.62	LDD1741	[22]
C053 Probe Info	5.39	LDD1751	[22]
C055 Probe Info	24.08	LDD1752	[22]
C056 Probe Info	25.46	LDD1753	[22]
C059 Probe Info	4.96	LDD1756	[22]
C063 Probe Info	19.97	LDD1760	[22]
C064 Probe Info	9.06	LDD1761	[22]
C067 Probe Info	5.28	LDD1763	[22]
C070 Probe Info	13.93	LDD1766	[22]
C072 Probe Info	12.04	LDD1768	[22]
C087 Probe Info	8.63	LDD1779	[22]
C091 Probe Info	19.03	LDD1782	[22]
C092 Probe Info	27.67	LDD1783	[22]
C094 Probe Info	32.45	LDD1785	[22]
C095 Probe Info	6.73	LDD1786	[22]
C106 Probe Info	23.59	LDD1793	[22]
C107 Probe Info	10.13	LDD1794	[22]
C108 Probe Info	16.91	LDD1795	[22]
C112 Probe Info	28.25	LDD1799	[22]
C129 Probe Info	6.02	LDD1811	[22]
C130 Probe Info	8.34	LDD1812	[22]
C134 Probe Info	26.17	LDD1816	[22]
C135 Probe Info	17.51	LDD1817	[22]
C139 Probe Info	23.43	LDD1821	[22]
C140 Probe Info	7.73	LDD1822	[22]
C141 Probe Info	14.22	LDD1823	[22]
C143 Probe Info	25.99	LDD1825	[22]
C147 Probe Info	7.57	LDD1829	[22]
C153 Probe Info	22.94	LDD1834	[22]
C159 Probe Info	10.93	LDD1839	[22]
C160 Probe Info	15.14	LDD1840	[22]
C161 Probe Info	15.67	LDD1841	[22]
C163 Probe Info	10.70	LDD1843	[22]
C165 Probe Info	15.56	LDD1845	[22]
C166 Probe Info	10.93	LDD1846	[22]
C169 Probe Info	39.67	LDD1849	[22]
C170 Probe Info	11.47	LDD1850	[22]
C173 Probe Info	5.28	LDD1853	[22]
C178 Probe Info	19.29	LDD1857	[22]
C186 Probe Info	10.48	LDD1864	[22]
C187 Probe Info	61.82	LDD1865	[22]
C191 Probe Info	46.85	LDD1868	[22]
C193 Probe Info	17.39	LDD1869	[22]
C194 Probe Info	11.88	LDD1870	[22]
C196 Probe Info	17.15	LDD1872	[22]
C197 Probe Info	6.28	LDD1873	[22]
C198 Probe Info	16.45	LDD1874	[22]
C201 Probe Info	63.56	LDD1877	[22]
C204 Probe Info	5.31	LDD1879	[22]
C206 Probe Info	44.02	LDD1881	[22]
C207 Probe Info	18.38	LDD1882	[22]
C210 Probe Info	73.01	LDD1884	[22]
C211 Probe Info	9.25	LDD1885	[22]
C213 Probe Info	18.00	LDD1887	[22]
C216 Probe Info	5.90	LDD1890	[22]
C217 Probe Info	6.02	LDD1891	[22]
C218 Probe Info	32.90	LDD1892	[22]
C219 Probe Info	14.32	LDD1893	[22]
C220 Probe Info	38.59	LDD1894	[22]
C225 Probe Info	6.92	LDD1898	[22]
C226 Probe Info	8.22	LDD1899	[22]
C228 Probe Info	21.41	LDD1901	[22]
C229 Probe Info	12.13	LDD1902	[22]
C231 Probe Info	35.75	LDD1904	[22]
C232 Probe Info	59.71	LDD1905	[22]
C233 Probe Info	18.00	LDD1906	[22]
C234 Probe Info	10.63	LDD1907	[22]
C235 Probe Info	40.79	LDD1908	[22]
C238 Probe Info	21.26	LDD1911	[22]
C239 Probe Info	5.35	LDD1912	[22]
C240 Probe Info	11.88	LDD1913	[22]
C243 Probe Info	14.93	LDD1916	[22]
C244 Probe Info	16.00	LDD1917	[22]
C246 Probe Info	18.13	LDD1919	[22]
C249 Probe Info	13.00	LDD1922	[22]
C252 Probe Info	11.79	LDD1925	[22]
C264 Probe Info	22.01	LDD1935	[22]
C265 Probe Info	20.82	LDD1936	[22]
C270 Probe Info	9.25	LDD1940	[22]
C273 Probe Info	6.63	LDD1943	[22]
C277 Probe Info	11.71	LDD1947	[22]
C280 Probe Info	11.71	LDD1950	[22]
C282 Probe Info	24.42	LDD1952	[22]
C285 Probe Info	28.64	LDD1955	[22]
C286 Probe Info	6.87	LDD1956	[22]
C287 Probe Info	16.00	LDD1957	[22]
C288 Probe Info	13.18	LDD1958	[22]
C289 Probe Info	40.50	LDD1959	[22]
C290 Probe Info	9.19	LDD1960	[22]
C293 Probe Info	25.11	LDD1963	[22]
C296 Probe Info	19.84	LDD1966	[22]
C299 Probe Info	8.34	LDD1968	[22]
C305 Probe Info	10.27	LDD1974	[22]
C307 Probe Info	5.74	LDD1975	[22]
C310 Probe Info	14.52	LDD1977	[22]
C314 Probe Info	15.67	LDD1981	[22]
C322 Probe Info	9.19	LDD1988	[22]
C326 Probe Info	11.00	LDD1990	[22]
C338 Probe Info	12.73	LDD2001	[22]
C339 Probe Info	9.71	LDD2002	[22]
C343 Probe Info	15.56	LDD2005	[22]
C348 Probe Info	14.83	LDD2009	[22]
C349 Probe Info	19.43	LDD2010	[22]
C350 Probe Info	38.59	LDD2011	[22]
C353 Probe Info	8.69	LDD2014	[22]
C354 Probe Info	6.96	LDD2015	[22]
C355 Probe Info	25.46	LDD2016	[22]
C356 Probe Info	9.58	LDD2017	[22]
C357 Probe Info	6.45	LDD2018	[22]
C362 Probe Info	37.27	LDD2023	[22]
C363 Probe Info	19.70	LDD2024	[22]
C364 Probe Info	21.26	LDD2025	[22]
C366 Probe Info	12.64	LDD2027	[22]
C367 Probe Info	7.21	LDD2028	[22]
C373 Probe Info	5.31	LDD2033	[22]
C376 Probe Info	11.24	LDD2036	[22]
C378 Probe Info	6.59	LDD2037	[22]
C380 Probe Info	6.45	LDD2039	[22]
C382 Probe Info	15.35	LDD2041	[22]
C390 Probe Info	37.27	LDD2049	[22]
C399 Probe Info	9.65	LDD2058	[22]
C403 Probe Info	25.28	LDD2061	[22]
C405 Probe Info	5.35	LDD2063	[22]
C407 Probe Info	38.05	LDD2064	[22]
C408 Probe Info	6.73	LDD2065	[22]
C409 Probe Info	8.57	LDD2066	[22]
C413 Probe Info	15.03	LDD2069	[22]
C419 Probe Info	10.34	LDD2074	[22]
C423 Probe Info	10.27	LDD2078	[22]
C424 Probe Info	9.38	LDD2079	[22]
C426 Probe Info	22.16	LDD2081	[22]
C429 Probe Info	16.34	LDD2084	[22]
C431 Probe Info	20.82	LDD2086	[22]
FFF probe11 Probe Info	20.00	LDD0471	[23]
FFF probe12 Probe Info	6.83	LDD0473	[23]
FFF probe13 Probe Info	20.00	LDD0475	[23]
FFF probe14 Probe Info	20.00	LDD0477	[23]
FFF probe15 Probe Info	17.36	LDD0478	[23]
FFF probe2 Probe Info	20.00	LDD0463	[23]
FFF probe3 Probe Info	20.00	LDD0464	[23]
FFF probe4 Probe Info	20.00	LDD0466	[23]
FFF probe7 Probe Info	10.58	LDD0483	[23]
FFF probe9 Probe Info	13.71	LDD0470	[23]
JN0003 Probe Info	20.00	LDD0469	[23]
STS-2 Probe Info	N.A.	LDD0138	[24]
VE-P Probe Info	N.A.	LDD0396	[25]
AX-1 Probe Info	3.10	LDD0441	[26]
OEA-DA Probe Info	20.00	LDD0046	[27]

Competitor(s) Related to This Target

Competitor ID	Name	Cell line	Binding Site(Ratio)	Interaction ID	Ref
LDCM0548	1-(4-(Benzo[d][1,3]dioxol-5-ylmethyl)piperazin-1-yl)-2-nitroethan-1-one	MDA-MB-231	C428(0.97); C108(0.86)	LDD2142	[28]
LDCM0519	1-(6-methoxy-3,4-dihydroquinolin-1(2H)-yl)-2-nitroethan-1-one	MDA-MB-231	C428(1.17)	LDD2112	[28]
LDCM0537	2-Cyano-N,N-dimethylacetamide	MDA-MB-231	C428(1.00)	LDD2130	[28]
LDCM0524	2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide	MDA-MB-231	C428(0.87)	LDD2117	[28]
LDCM0558	2-Cyano-N-phenylacetamide	MDA-MB-231	C428(1.11)	LDD2152	[28]
LDCM0510	3-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-3-oxopropanenitrile	MDA-MB-231	C428(1.12)	LDD2103	[28]
LDCM0539	3-(4-Isopropylpiperazin-1-yl)-3-oxopropanenitrile	MDA-MB-231	C428(0.59)	LDD2132	[28]
LDCM0538	4-(Cyanoacetyl)morpholine	MDA-MB-231	C428(1.08)	LDD2131	[28]
LDCM0025	4SU-RNA	HEK-293T	C66(2.10)	LDD0168	[7]
LDCM0026	4SU-RNA+native RNA	HEK-293T	C428(2.02)	LDD0169	[7]
LDCM0176	9im	MDA-MB-231	3.10	LDD0441	[26]
LDCM0214	AC1	HCT 116	C428(1.17)	LDD0531	[10]
LDCM0215	AC10	HCT 116	C428(1.15)	LDD0532	[10]
LDCM0216	AC100	HCT 116	C428(0.93)	LDD0533	[10]
LDCM0217	AC101	HCT 116	C428(0.85)	LDD0534	[10]
LDCM0218	AC102	HCT 116	C428(0.87)	LDD0535	[10]
LDCM0219	AC103	HCT 116	C428(0.89)	LDD0536	[10]
LDCM0220	AC104	HCT 116	C428(0.85)	LDD0537	[10]
LDCM0221	AC105	HCT 116	C428(0.88)	LDD0538	[10]
LDCM0222	AC106	HCT 116	C428(0.81)	LDD0539	[10]
LDCM0223	AC107	HCT 116	C428(0.81)	LDD0540	[10]
LDCM0224	AC108	HCT 116	C428(0.84)	LDD0541	[10]
LDCM0225	AC109	HCT 116	C428(0.89)	LDD0542	[10]
LDCM0226	AC11	HCT 116	C428(0.93)	LDD0543	[10]
LDCM0227	AC110	HCT 116	C428(0.94)	LDD0544	[10]
LDCM0228	AC111	HCT 116	C428(0.85)	LDD0545	[10]
LDCM0229	AC112	HCT 116	C428(0.90)	LDD0546	[10]
LDCM0230	AC113	HCT 116	C428(1.06)	LDD0547	[10]
LDCM0231	AC114	HCT 116	C428(1.17)	LDD0548	[10]
LDCM0232	AC115	HCT 116	C428(1.18)	LDD0549	[10]
LDCM0233	AC116	HCT 116	C428(1.39)	LDD0550	[10]
LDCM0234	AC117	HCT 116	C428(0.97)	LDD0551	[10]
LDCM0235	AC118	HCT 116	C428(1.07)	LDD0552	[10]
LDCM0236	AC119	HCT 116	C428(1.11)	LDD0553	[10]
LDCM0237	AC12	HCT 116	C428(0.94)	LDD0554	[10]
LDCM0238	AC120	HCT 116	C428(1.07)	LDD0555	[10]
LDCM0239	AC121	HCT 116	C428(1.05)	LDD0556	[10]
LDCM0240	AC122	HCT 116	C428(1.10)	LDD0557	[10]
LDCM0241	AC123	HCT 116	C428(1.34)	LDD0558	[10]
LDCM0242	AC124	HCT 116	C428(1.14)	LDD0559	[10]
LDCM0243	AC125	HCT 116	C428(1.12)	LDD0560	[10]
LDCM0244	AC126	HCT 116	C428(1.32)	LDD0561	[10]
LDCM0245	AC127	HCT 116	C428(1.12)	LDD0562	[10]
LDCM0246	AC128	HCT 116	C428(1.40)	LDD0563	[10]
LDCM0247	AC129	HCT 116	C428(1.45)	LDD0564	[10]
LDCM0249	AC130	HCT 116	C428(1.37)	LDD0566	[10]
LDCM0250	AC131	HCT 116	C428(1.30)	LDD0567	[10]
LDCM0251	AC132	HCT 116	C428(1.19)	LDD0568	[10]
LDCM0252	AC133	HCT 116	C428(1.24)	LDD0569	[10]
LDCM0253	AC134	HCT 116	C428(1.16)	LDD0570	[10]
LDCM0254	AC135	HCT 116	C428(1.28)	LDD0571	[10]
LDCM0255	AC136	HCT 116	C428(1.15)	LDD0572	[10]
LDCM0256	AC137	HCT 116	C428(1.10)	LDD0573	[10]
LDCM0257	AC138	HCT 116	C428(1.00)	LDD0574	[10]
LDCM0258	AC139	HCT 116	C428(1.10)	LDD0575	[10]
LDCM0259	AC14	HCT 116	C428(0.94)	LDD0576	[10]
LDCM0260	AC140	HCT 116	C428(1.00)	LDD0577	[10]
LDCM0261	AC141	HCT 116	C428(1.03)	LDD0578	[10]
LDCM0262	AC142	HCT 116	C428(1.15)	LDD0579	[10]
LDCM0263	AC143	HCT 116	C428(0.97)	LDD0580	[10]
LDCM0264	AC144	HCT 116	C428(1.10)	LDD0581	[10]
LDCM0265	AC145	HCT 116	C428(1.12)	LDD0582	[10]
LDCM0266	AC146	HCT 116	C428(1.14)	LDD0583	[10]
LDCM0267	AC147	HCT 116	C428(1.07)	LDD0584	[10]
LDCM0268	AC148	HCT 116	C428(1.16)	LDD0585	[10]
LDCM0269	AC149	HCT 116	C428(1.29)	LDD0586	[10]
LDCM0270	AC15	HCT 116	C428(1.13)	LDD0587	[10]
LDCM0271	AC150	HCT 116	C428(1.04)	LDD0588	[10]
LDCM0272	AC151	HCT 116	C428(1.32)	LDD0589	[10]
LDCM0273	AC152	HCT 116	C428(1.10)	LDD0590	[10]
LDCM0274	AC153	HCT 116	C428(1.38)	LDD0591	[10]
LDCM0621	AC154	HCT 116	C428(1.22)	LDD2158	[10]
LDCM0622	AC155	HCT 116	C428(1.25)	LDD2159	[10]
LDCM0623	AC156	HCT 116	C428(1.34)	LDD2160	[10]
LDCM0624	AC157	HCT 116	C428(1.26)	LDD2161	[10]
LDCM0276	AC17	HCT 116	C428(1.04)	LDD0593	[10]
LDCM0277	AC18	HCT 116	C428(0.92)	LDD0594	[10]
LDCM0278	AC19	HCT 116	C428(1.05)	LDD0595	[10]
LDCM0279	AC2	HCT 116	C428(1.06)	LDD0596	[10]
LDCM0280	AC20	HCT 116	C428(0.89)	LDD0597	[10]
LDCM0281	AC21	HCT 116	C428(1.16)	LDD0598	[10]
LDCM0282	AC22	HCT 116	C428(1.09)	LDD0599	[10]
LDCM0283	AC23	HCT 116	C428(0.86)	LDD0600	[10]
LDCM0284	AC24	HCT 116	C428(0.97)	LDD0601	[10]
LDCM0285	AC25	HCT 116	C428(0.92)	LDD0602	[10]
LDCM0286	AC26	HCT 116	C428(1.12)	LDD0603	[10]
LDCM0287	AC27	HCT 116	C428(0.99)	LDD0604	[10]
LDCM0288	AC28	HCT 116	C428(1.41)	LDD0605	[10]
LDCM0289	AC29	HCT 116	C428(1.04)	LDD0606	[10]
LDCM0290	AC3	HCT 116	C428(1.11)	LDD0607	[10]
LDCM0291	AC30	HCT 116	C428(1.07)	LDD0608	[10]
LDCM0292	AC31	HCT 116	C428(1.28)	LDD0609	[10]
LDCM0293	AC32	HCT 116	C428(1.11)	LDD0610	[10]
LDCM0294	AC33	HCT 116	C428(0.95)	LDD0611	[10]
LDCM0295	AC34	HCT 116	C428(1.00)	LDD0612	[10]
LDCM0296	AC35	HCT 116	C428(1.14)	LDD0613	[10]
LDCM0297	AC36	HCT 116	C428(0.95)	LDD0614	[10]
LDCM0298	AC37	HCT 116	C428(1.06)	LDD0615	[10]
LDCM0299	AC38	HCT 116	C428(0.99)	LDD0616	[10]
LDCM0300	AC39	HCT 116	C428(0.79)	LDD0617	[10]
LDCM0301	AC4	HCT 116	C428(1.32)	LDD0618	[10]
LDCM0302	AC40	HCT 116	C428(0.97)	LDD0619	[10]
LDCM0303	AC41	HCT 116	C428(0.91)	LDD0620	[10]
LDCM0304	AC42	HCT 116	C428(0.85)	LDD0621	[10]
LDCM0305	AC43	HCT 116	C428(0.86)	LDD0622	[10]
LDCM0306	AC44	HCT 116	C428(0.95)	LDD0623	[10]
LDCM0307	AC45	HCT 116	C428(1.08)	LDD0624	[10]
LDCM0308	AC46	HCT 116	C428(1.01)	LDD0625	[10]
LDCM0309	AC47	HCT 116	C428(1.16)	LDD0626	[10]
LDCM0310	AC48	HCT 116	C428(1.09)	LDD0627	[10]
LDCM0311	AC49	HCT 116	C428(0.98)	LDD0628	[10]
LDCM0312	AC5	HCT 116	C428(1.38)	LDD0629	[10]
LDCM0313	AC50	HCT 116	C428(1.05)	LDD0630	[10]
LDCM0314	AC51	HCT 116	C428(1.01)	LDD0631	[10]
LDCM0315	AC52	HCT 116	C428(1.03)	LDD0632	[10]
LDCM0316	AC53	HCT 116	C428(1.03)	LDD0633	[10]
LDCM0317	AC54	HCT 116	C428(1.01)	LDD0634	[10]
LDCM0318	AC55	HCT 116	C428(1.03)	LDD0635	[10]
LDCM0319	AC56	HCT 116	C428(1.00)	LDD0636	[10]
LDCM0320	AC57	HCT 116	C428(1.00)	LDD0637	[10]
LDCM0321	AC58	HCT 116	C428(1.03)	LDD0638	[10]
LDCM0322	AC59	HCT 116	C428(1.01)	LDD0639	[10]
LDCM0323	AC6	HCT 116	C428(0.96)	LDD0640	[10]
LDCM0324	AC60	HCT 116	C428(0.98)	LDD0641	[10]
LDCM0325	AC61	HCT 116	C428(1.06)	LDD0642	[10]
LDCM0326	AC62	HCT 116	C428(1.02)	LDD0643	[10]
LDCM0327	AC63	HCT 116	C428(1.02)	LDD0644	[10]
LDCM0328	AC64	HCT 116	C428(1.11)	LDD0645	[10]
LDCM0329	AC65	HCT 116	C428(1.03)	LDD0646	[10]
LDCM0330	AC66	HCT 116	C428(1.05)	LDD0647	[10]
LDCM0331	AC67	HCT 116	C428(1.18)	LDD0648	[10]
LDCM0332	AC68	HCT 116	C428(0.96)	LDD0649	[10]
LDCM0333	AC69	HCT 116	C428(1.01)	LDD0650	[10]
LDCM0334	AC7	HCT 116	C428(0.90)	LDD0651	[10]
LDCM0335	AC70	HCT 116	C428(0.92)	LDD0652	[10]
LDCM0336	AC71	HCT 116	C428(0.92)	LDD0653	[10]
LDCM0337	AC72	HCT 116	C428(0.99)	LDD0654	[10]
LDCM0338	AC73	HCT 116	C428(0.82)	LDD0655	[10]
LDCM0339	AC74	HCT 116	C428(0.85)	LDD0656	[10]
LDCM0340	AC75	HCT 116	C428(1.10)	LDD0657	[10]
LDCM0341	AC76	HCT 116	C428(1.03)	LDD0658	[10]
LDCM0342	AC77	HCT 116	C428(0.96)	LDD0659	[10]
LDCM0343	AC78	HCT 116	C428(0.89)	LDD0660	[10]
LDCM0344	AC79	HCT 116	C428(1.00)	LDD0661	[10]
LDCM0345	AC8	HCT 116	C428(0.96)	LDD0662	[10]
LDCM0346	AC80	HCT 116	C428(0.96)	LDD0663	[10]
LDCM0347	AC81	HCT 116	C428(1.00)	LDD0664	[10]
LDCM0348	AC82	HCT 116	C428(0.98)	LDD0665	[10]
LDCM0349	AC83	HCT 116	C428(0.97)	LDD0666	[10]
LDCM0350	AC84	HCT 116	C428(0.96)	LDD0667	[10]
LDCM0351	AC85	HCT 116	C428(1.05)	LDD0668	[10]
LDCM0352	AC86	HCT 116	C428(1.06)	LDD0669	[10]
LDCM0353	AC87	HCT 116	C428(1.11)	LDD0670	[10]
LDCM0354	AC88	HCT 116	C428(0.98)	LDD0671	[10]
LDCM0355	AC89	HCT 116	C428(1.06)	LDD0672	[10]
LDCM0357	AC90	HCT 116	C428(1.03)	LDD0674	[10]
LDCM0358	AC91	HCT 116	C428(1.18)	LDD0675	[10]
LDCM0359	AC92	HCT 116	C428(1.04)	LDD0676	[10]
LDCM0360	AC93	HCT 116	C428(0.98)	LDD0677	[10]
LDCM0361	AC94	HCT 116	C428(1.08)	LDD0678	[10]
LDCM0362	AC95	HCT 116	C428(0.96)	LDD0679	[10]
LDCM0363	AC96	HCT 116	C428(1.00)	LDD0680	[10]
LDCM0364	AC97	HCT 116	C428(0.97)	LDD0681	[10]
LDCM0365	AC98	HCT 116	C428(0.84)	LDD0682	[10]
LDCM0366	AC99	HCT 116	C428(0.86)	LDD0683	[10]
LDCM0545	Acetamide	MDA-MB-231	C428(0.56)	LDD2138	[28]
LDCM0520	AKOS000195272	MDA-MB-231	C428(0.95)	LDD2113	[28]
LDCM0248	AKOS034007472	HCT 116	C428(1.17)	LDD0565	[10]
LDCM0356	AKOS034007680	HCT 116	C428(0.98)	LDD0673	[10]
LDCM0275	AKOS034007705	HCT 116	C428(1.09)	LDD0592	[10]
LDCM0020	ARS-1620	HCC44	C428(1.05)	LDD0078	[10]
LDCM0498	BS-3668	MDA-MB-231	C428(0.67)	LDD2091	[28]
LDCM0108	Chloroacetamide	HeLa	C108(0.00); C428(0.00); C66(0.00)	LDD0222	[17]
LDCM0367	CL1	HCT 116	C428(1.13)	LDD0684	[10]
LDCM0368	CL10	HCT 116	C428(1.11)	LDD0685	[10]
LDCM0369	CL100	HCT 116	C428(1.16)	LDD0686	[10]
LDCM0370	CL101	HCT 116	C428(0.89)	LDD0687	[10]
LDCM0371	CL102	HCT 116	C428(0.93)	LDD0688	[10]
LDCM0372	CL103	HCT 116	C428(1.03)	LDD0689	[10]
LDCM0373	CL104	HCT 116	C428(0.95)	LDD0690	[10]
LDCM0374	CL105	HCT 116	C428(0.96)	LDD0691	[10]
LDCM0375	CL106	HCT 116	C428(1.08)	LDD0692	[10]
LDCM0376	CL107	HCT 116	C428(1.03)	LDD0693	[10]
LDCM0377	CL108	HCT 116	C428(1.13)	LDD0694	[10]
LDCM0378	CL109	HCT 116	C428(0.94)	LDD0695	[10]
LDCM0379	CL11	HCT 116	C428(1.16)	LDD0696	[10]
LDCM0380	CL110	HCT 116	C428(1.02)	LDD0697	[10]
LDCM0381	CL111	HCT 116	C428(1.01)	LDD0698	[10]
LDCM0382	CL112	HCT 116	C428(1.03)	LDD0699	[10]
LDCM0383	CL113	HCT 116	C428(1.19)	LDD0700	[10]
LDCM0384	CL114	HCT 116	C428(0.91)	LDD0701	[10]
LDCM0385	CL115	HCT 116	C428(0.96)	LDD0702	[10]
LDCM0386	CL116	HCT 116	C428(0.96)	LDD0703	[10]
LDCM0387	CL117	HCT 116	C428(0.87)	LDD0704	[10]
LDCM0388	CL118	HCT 116	C428(1.17)	LDD0705	[10]
LDCM0389	CL119	HCT 116	C428(1.12)	LDD0706	[10]
LDCM0390	CL12	HCT 116	C428(1.19)	LDD0707	[10]
LDCM0391	CL120	HCT 116	C428(1.00)	LDD0708	[10]
LDCM0392	CL121	HCT 116	C428(0.79)	LDD0709	[10]
LDCM0393	CL122	HCT 116	C428(1.00)	LDD0710	[10]
LDCM0394	CL123	HCT 116	C428(0.89)	LDD0711	[10]
LDCM0395	CL124	HCT 116	C428(0.99)	LDD0712	[10]
LDCM0396	CL125	HCT 116	C428(0.93)	LDD0713	[10]
LDCM0397	CL126	HCT 116	C428(1.00)	LDD0714	[10]
LDCM0398	CL127	HCT 116	C428(1.11)	LDD0715	[10]
LDCM0399	CL128	HCT 116	C428(1.05)	LDD0716	[10]
LDCM0400	CL13	HCT 116	C428(1.09)	LDD0717	[10]
LDCM0401	CL14	HCT 116	C428(1.19)	LDD0718	[10]
LDCM0402	CL15	HCT 116	C428(1.04)	LDD0719	[10]
LDCM0403	CL16	HCT 116	C428(0.98)	LDD0720	[10]
LDCM0404	CL17	HCT 116	C428(0.95)	LDD0721	[10]
LDCM0405	CL18	HCT 116	C428(1.08)	LDD0722	[10]
LDCM0406	CL19	HCT 116	C428(1.02)	LDD0723	[10]
LDCM0407	CL2	HCT 116	C428(1.19)	LDD0724	[10]
LDCM0408	CL20	HCT 116	C428(1.15)	LDD0725	[10]
LDCM0409	CL21	HCT 116	C428(1.15)	LDD0726	[10]
LDCM0410	CL22	HCT 116	C428(1.13)	LDD0727	[10]
LDCM0411	CL23	HCT 116	C428(1.10)	LDD0728	[10]
LDCM0412	CL24	HCT 116	C428(1.42)	LDD0729	[10]
LDCM0413	CL25	HCT 116	C428(0.98)	LDD0730	[10]
LDCM0414	CL26	HCT 116	C428(0.99)	LDD0731	[10]
LDCM0415	CL27	HCT 116	C428(1.26)	LDD0732	[10]
LDCM0416	CL28	HCT 116	C428(1.10)	LDD0733	[10]
LDCM0417	CL29	HCT 116	C428(1.42)	LDD0734	[10]
LDCM0418	CL3	HCT 116	C428(1.02)	LDD0735	[10]
LDCM0419	CL30	HCT 116	C428(1.11)	LDD0736	[10]
LDCM0420	CL31	HCT 116	C428(1.18)	LDD0737	[10]
LDCM0421	CL32	HCT 116	C428(0.94)	LDD0738	[10]
LDCM0422	CL33	HCT 116	C428(0.82)	LDD0739	[10]
LDCM0423	CL34	HCT 116	C428(0.92)	LDD0740	[10]
LDCM0424	CL35	HCT 116	C428(1.06)	LDD0741	[10]
LDCM0425	CL36	HCT 116	C428(0.85)	LDD0742	[10]
LDCM0426	CL37	HCT 116	C428(1.05)	LDD0743	[10]
LDCM0428	CL39	HCT 116	C428(0.95)	LDD0745	[10]
LDCM0429	CL4	HCT 116	C428(1.08)	LDD0746	[10]
LDCM0430	CL40	HCT 116	C428(0.89)	LDD0747	[10]
LDCM0431	CL41	HCT 116	C428(0.99)	LDD0748	[10]
LDCM0432	CL42	HCT 116	C428(0.95)	LDD0749	[10]
LDCM0433	CL43	HCT 116	C428(1.20)	LDD0750	[10]
LDCM0434	CL44	HCT 116	C428(1.14)	LDD0751	[10]
LDCM0435	CL45	HCT 116	C428(0.97)	LDD0752	[10]
LDCM0436	CL46	HCT 116	C428(1.13)	LDD0753	[10]
LDCM0437	CL47	HCT 116	C428(0.97)	LDD0754	[10]
LDCM0438	CL48	HCT 116	C428(1.23)	LDD0755	[10]
LDCM0439	CL49	HCT 116	C428(1.32)	LDD0756	[10]
LDCM0440	CL5	HCT 116	C428(1.19)	LDD0757	[10]
LDCM0441	CL50	HCT 116	C428(1.09)	LDD0758	[10]
LDCM0442	CL51	HCT 116	C428(1.16)	LDD0759	[10]
LDCM0443	CL52	HCT 116	C428(0.98)	LDD0760	[10]
LDCM0444	CL53	HCT 116	C428(1.04)	LDD0761	[10]
LDCM0445	CL54	HCT 116	C428(1.11)	LDD0762	[10]
LDCM0446	CL55	HCT 116	C428(1.05)	LDD0763	[10]
LDCM0447	CL56	HCT 116	C428(0.99)	LDD0764	[10]
LDCM0448	CL57	HCT 116	C428(1.04)	LDD0765	[10]
LDCM0449	CL58	HCT 116	C428(1.28)	LDD0766	[10]
LDCM0450	CL59	HCT 116	C428(1.17)	LDD0767	[10]
LDCM0451	CL6	HCT 116	C428(1.02)	LDD0768	[10]
LDCM0452	CL60	HCT 116	C428(1.08)	LDD0769	[10]
LDCM0453	CL61	HCT 116	C428(1.08)	LDD0770	[10]
LDCM0454	CL62	HCT 116	C428(1.06)	LDD0771	[10]
LDCM0455	CL63	HCT 116	C428(1.04)	LDD0772	[10]
LDCM0456	CL64	HCT 116	C428(0.92)	LDD0773	[10]
LDCM0457	CL65	HCT 116	C428(1.20)	LDD0774	[10]
LDCM0458	CL66	HCT 116	C428(0.99)	LDD0775	[10]
LDCM0459	CL67	HCT 116	C428(0.86)	LDD0776	[10]
LDCM0460	CL68	HCT 116	C428(1.08)	LDD0777	[10]
LDCM0461	CL69	HCT 116	C428(0.95)	LDD0778	[10]
LDCM0462	CL7	HCT 116	C428(1.19)	LDD0779	[10]
LDCM0463	CL70	HCT 116	C428(0.99)	LDD0780	[10]
LDCM0464	CL71	HCT 116	C428(1.21)	LDD0781	[10]
LDCM0465	CL72	HCT 116	C428(1.07)	LDD0782	[10]
LDCM0466	CL73	HCT 116	C428(1.10)	LDD0783	[10]
LDCM0467	CL74	HCT 116	C428(0.92)	LDD0784	[10]
LDCM0469	CL76	HCT 116	C428(1.00)	LDD0786	[10]
LDCM0470	CL77	HCT 116	C428(0.89)	LDD0787	[10]
LDCM0471	CL78	HCT 116	C428(1.07)	LDD0788	[10]
LDCM0472	CL79	HCT 116	C428(1.15)	LDD0789	[10]
LDCM0473	CL8	HCT 116	C428(1.01)	LDD0790	[10]
LDCM0474	CL80	HCT 116	C428(0.95)	LDD0791	[10]
LDCM0475	CL81	HCT 116	C428(1.16)	LDD0792	[10]
LDCM0476	CL82	HCT 116	C428(1.02)	LDD0793	[10]
LDCM0477	CL83	HCT 116	C428(1.01)	LDD0794	[10]
LDCM0478	CL84	HCT 116	C428(1.05)	LDD0795	[10]
LDCM0479	CL85	HCT 116	C428(0.96)	LDD0796	[10]
LDCM0480	CL86	HCT 116	C428(1.00)	LDD0797	[10]
LDCM0481	CL87	HCT 116	C428(1.13)	LDD0798	[10]
LDCM0482	CL88	HCT 116	C428(1.08)	LDD0799	[10]
LDCM0483	CL89	HCT 116	C428(1.05)	LDD0800	[10]
LDCM0484	CL9	HCT 116	C428(1.25)	LDD0801	[10]
LDCM0485	CL90	HCT 116	C428(1.25)	LDD0802	[10]
LDCM0486	CL91	HCT 116	C428(0.88)	LDD0803	[10]
LDCM0487	CL92	HCT 116	C428(0.84)	LDD0804	[10]
LDCM0488	CL93	HCT 116	C428(0.96)	LDD0805	[10]
LDCM0489	CL94	HCT 116	C428(1.15)	LDD0806	[10]
LDCM0490	CL95	HCT 116	C428(1.01)	LDD0807	[10]
LDCM0491	CL96	HCT 116	C428(1.14)	LDD0808	[10]
LDCM0492	CL97	HCT 116	C428(0.97)	LDD0809	[10]
LDCM0493	CL98	HCT 116	C428(1.19)	LDD0810	[10]
LDCM0494	CL99	HCT 116	C428(1.07)	LDD0811	[10]
LDCM0185	Compound 17	HEK-293T	6.56	LDD0512	[23]
LDCM0191	Compound 21	HEK-293T	8.62	LDD0508	[23]
LDCM0190	Compound 34	HEK-293T	11.30	LDD0510	[23]
LDCM0192	Compound 35	HEK-293T	8.26	LDD0509	[23]
LDCM0193	Compound 36	HEK-293T	11.76	LDD0511	[23]
LDCM0495	E2913	HEK-293T	C108(1.03); C66(0.69)	LDD1698	[29]
LDCM0213	Electrophilic fragment 2	MDA-MB-231	C428(40.31); C66(2.21); C108(1.92)	LDD1702	[28]
LDCM0175	Ethacrynic acid	HeLa	N.A.	LDD0440	[9]
LDCM0625	F8	Ramos	C428(2.21)	LDD2187	[30]
LDCM0572	Fragment10	Ramos	C428(4.84)	LDD2189	[30]
LDCM0573	Fragment11	Ramos	C428(1.59)	LDD2190	[30]
LDCM0574	Fragment12	Ramos	C428(3.54)	LDD2191	[30]
LDCM0575	Fragment13	Ramos	C428(1.45)	LDD2192	[30]
LDCM0576	Fragment14	Ramos	C428(20.00)	LDD2193	[30]
LDCM0580	Fragment21	Ramos	C428(2.22)	LDD2195	[30]
LDCM0582	Fragment23	Ramos	C428(0.20)	LDD2196	[30]
LDCM0578	Fragment27	Ramos	C428(0.70)	LDD2197	[30]
LDCM0586	Fragment28	Ramos	C428(0.40)	LDD2198	[30]
LDCM0588	Fragment30	Ramos	C428(1.28)	LDD2199	[30]
LDCM0589	Fragment31	Ramos	C428(0.83)	LDD2200	[30]
LDCM0590	Fragment32	Ramos	C428(3.87)	LDD2201	[30]
LDCM0468	Fragment33	HCT 116	C428(1.01)	LDD0785	[10]
LDCM0596	Fragment38	Ramos	C428(3.02)	LDD2203	[30]
LDCM0566	Fragment4	Ramos	C428(10.71)	LDD2184	[30]
LDCM0427	Fragment51	HCT 116	C428(0.86)	LDD0744	[10]
LDCM0610	Fragment52	Ramos	C428(0.91)	LDD2204	[30]
LDCM0614	Fragment56	Ramos	C428(0.88)	LDD2205	[30]
LDCM0569	Fragment7	Ramos	C428(20.00)	LDD2186	[30]
LDCM0107	IAA	HeLa	C428(0.00); C66(0.00)	LDD0221	[17]
LDCM0022	KB02	HCT 116	C428(1.17)	LDD0080	[10]
LDCM0023	KB03	HCT 116	C428(1.16)	LDD0081	[10]
LDCM0024	KB05	HCT 116	C428(1.01)	LDD0082	[10]
LDCM0509	N-(4-bromo-3,5-dimethylphenyl)-2-nitroacetamide	MDA-MB-231	C428(1.88)	LDD2102	[28]
LDCM0528	N-(4-bromophenyl)-2-cyano-N-phenylacetamide	MDA-MB-231	C428(0.83)	LDD2121	[28]
LDCM0109	NEM	HeLa	N.A.	LDD0223	[17]
LDCM0496	Nucleophilic fragment 11a	MDA-MB-231	C428(0.91)	LDD2089	[28]
LDCM0497	Nucleophilic fragment 11b	MDA-MB-231	C428(1.57)	LDD2090	[28]
LDCM0499	Nucleophilic fragment 12b	MDA-MB-231	C428(1.19)	LDD2092	[28]
LDCM0500	Nucleophilic fragment 13a	MDA-MB-231	C428(1.08)	LDD2093	[28]
LDCM0501	Nucleophilic fragment 13b	MDA-MB-231	C428(1.52)	LDD2094	[28]
LDCM0504	Nucleophilic fragment 15a	MDA-MB-231	C428(1.05)	LDD2097	[28]
LDCM0505	Nucleophilic fragment 15b	MDA-MB-231	C428(1.49)	LDD2098	[28]
LDCM0506	Nucleophilic fragment 16a	MDA-MB-231	C428(0.88)	LDD2099	[28]
LDCM0507	Nucleophilic fragment 16b	MDA-MB-231	C428(1.76)	LDD2100	[28]
LDCM0508	Nucleophilic fragment 17a	MDA-MB-231	C428(1.25)	LDD2101	[28]
LDCM0511	Nucleophilic fragment 18b	MDA-MB-231	C428(1.27); C108(0.65)	LDD2104	[28]
LDCM0512	Nucleophilic fragment 19a	MDA-MB-231	C428(1.48)	LDD2105	[28]
LDCM0513	Nucleophilic fragment 19b	MDA-MB-231	C428(1.18)	LDD2106	[28]
LDCM0514	Nucleophilic fragment 20a	MDA-MB-231	C428(0.85)	LDD2107	[28]
LDCM0515	Nucleophilic fragment 20b	MDA-MB-231	C428(0.72)	LDD2108	[28]
LDCM0516	Nucleophilic fragment 21a	MDA-MB-231	C428(0.99)	LDD2109	[28]
LDCM0518	Nucleophilic fragment 22a	MDA-MB-231	C428(0.99)	LDD2111	[28]
LDCM0521	Nucleophilic fragment 23b	MDA-MB-231	C428(1.54)	LDD2114	[28]
LDCM0522	Nucleophilic fragment 24a	MDA-MB-231	C428(0.83)	LDD2115	[28]
LDCM0526	Nucleophilic fragment 26a	MDA-MB-231	C428(1.75)	LDD2119	[28]
LDCM0527	Nucleophilic fragment 26b	MDA-MB-231	C428(1.10)	LDD2120	[28]
LDCM0530	Nucleophilic fragment 28a	MDA-MB-231	C428(1.01)	LDD2123	[28]
LDCM0532	Nucleophilic fragment 29a	MDA-MB-231	C428(0.86)	LDD2125	[28]
LDCM0534	Nucleophilic fragment 30a	MDA-MB-231	C428(1.03)	LDD2127	[28]
LDCM0535	Nucleophilic fragment 30b	MDA-MB-231	C428(1.51)	LDD2128	[28]
LDCM0536	Nucleophilic fragment 31	MDA-MB-231	C428(1.07)	LDD2129	[28]
LDCM0540	Nucleophilic fragment 35	MDA-MB-231	C428(0.77)	LDD2133	[28]
LDCM0541	Nucleophilic fragment 36	MDA-MB-231	C428(0.66)	LDD2134	[28]
LDCM0542	Nucleophilic fragment 37	MDA-MB-231	C428(1.10)	LDD2135	[28]
LDCM0543	Nucleophilic fragment 38	MDA-MB-231	C428(1.65)	LDD2136	[28]
LDCM0544	Nucleophilic fragment 39	MDA-MB-231	C428(0.87); C108(0.99)	LDD2137	[28]
LDCM0211	Nucleophilic fragment 3b	MDA-MB-231	C428(1.57)	LDD1700	[28]
LDCM0546	Nucleophilic fragment 40	MDA-MB-231	C428(0.83)	LDD2140	[28]
LDCM0547	Nucleophilic fragment 41	MDA-MB-231	C428(0.69); C108(1.05)	LDD2141	[28]
LDCM0549	Nucleophilic fragment 43	MDA-MB-231	C428(1.12)	LDD2143	[28]
LDCM0550	Nucleophilic fragment 5a	MDA-MB-231	C428(2.85)	LDD2144	[28]
LDCM0551	Nucleophilic fragment 5b	MDA-MB-231	C428(7.98)	LDD2145	[28]
LDCM0552	Nucleophilic fragment 6a	MDA-MB-231	C428(0.90)	LDD2146	[28]
LDCM0553	Nucleophilic fragment 6b	MDA-MB-231	C428(2.76)	LDD2147	[28]
LDCM0554	Nucleophilic fragment 7a	MDA-MB-231	C428(1.06)	LDD2148	[28]
LDCM0559	Nucleophilic fragment 9b	MDA-MB-231	C428(2.24)	LDD2153	[28]
LDCM0628	OTUB2-COV-1	HEK-293T	C428(0.64)	LDD2207	[31]
LDCM0014	Panhematin	K562	3.02	LDD0063	[8]
LDCM0021	THZ1	HCT 116	C428(1.12)	LDD2173	[10]
LDCM0110	W12	Hep-G2	C428(6.20)	LDD0237	[18]
LDCM0111	W14	Hep-G2	C428(1.32)	LDD0238	[18]
LDCM0113	W17	Hep-G2	C428(0.77)	LDD0240	[18]

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Prof. Feng Zhu

Prof. Feng Ni