Details of the Target

General Information of Target

Target ID LDTP05511
Target Name Cytoskeleton-associated protein 4 (CKAP4)
Gene Name CKAP4
Gene ID 10970
Synonyms
Cytoskeleton-associated protein 4; 63-kDa cytoskeleton-linking membrane protein; Climp-63; p63
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MPSAKQRGSKGGHGAASPSEKGAHPSGGADDVAKKPPPAPQQPPPPPAPHPQQHPQQHPQ
NQAHGKGGHRGGGGGGGKSSSSSSASAAAAAAAASSSASCSRRLGRALNFLFYLALVAAA
AFSGWCVHHVLEEVQQVRRSHQDFSRQREELGQGLQGVEQKVQSLQATFGTFESILRSSQ
HKQDLTEKAVKQGESEVSRISEVLQKLQNEILKDLSDGIHVVKDARERDFTSLENTVEER
LTELTKSINDNIAIFTEVQKRSQKEINDMKAKVASLEESEGNKQDLKALKEAVKEIQTSA
KSREWDMEALRSTLQTMESDIYTEVRELVSLKQEQQAFKEAADTERLALQALTEKLLRSE
ESVSRLPEEIRRLEEELRQLKSDSHGPKEDGGFRHSEAFEALQQKSQGLDSRLQHVEDGV
LSMQVASARQTESLESLLSKSQEHEQRLAALQGRLEGLGSSEADQDGLASTVRSLGETQL
VLYGDVEELKRSVGELPSTVESLQKVQEQVHTLLSQDQAQAARLPPQDFLDRLSSLDNLK
ASVSQVEADLKMLRTAVDSLVAYSVKIETNENNLESAKGLLDDLRNDLDRLFVKVEKIHE
KV
Target Bioclass
Transporter and channel
Subcellular location
Endoplasmic reticulum membrane
Function
Mediates the anchoring of the endoplasmic reticulum to microtubules.; High-affinity epithelial cell surface receptor for the FZD8-related low molecular weight sialoglycopeptide APF/antiproliferative factor. Mediates the APF antiproliferative signaling within cells.
Uniprot ID
Q07065
Ensemble ID
ENST00000378026.5
HGNC ID
HGNC:16991
ChEMBL ID
CHEMBL4296025

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 46 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
HDSF-alk
 Probe Info  		2.11  LDD0197  [2]
CHEMBL5175495
 Probe Info  		13.13  LDD0196  [3]
CY-1
 Probe Info  		100.00  LDD0243  [4]
CY4
 Probe Info  		100.00  LDD0244  [4]
N1
 Probe Info  		100.00  LDD0242  [4]
TG42
 Probe Info  		8.35  LDD0326  [5]
W1
 Probe Info  		35.50  LDD0235  [6]
FBP2
 Probe Info  		2.74  LDD0317  [7]
YN-1
 Probe Info  		12.26  LDD0444  [8]
YN-4
 Probe Info  		100.00  LDD0445  [8]
ONAyne
 Probe Info  		K182(0.82); K191(0.97); K223(2.86); K290(1.20)  LDD0274  [9]
OPA-S-S-alkyne
 Probe Info  		K339(1.14); K405(1.20); K223(2.50); K388(2.60)  LDD3494  [10]
IA-alkyne
 Probe Info  		C100(3.94)  LDD0304  [11]
m-APA
 Probe Info  		11.81  LDD0403  [12]
Alkylaryl probe 2
 Probe Info  		4.00  LDD0392  [13]
P26
 Probe Info  		1.48  LDD0409  [14]
JZ128-DTB
 Probe Info  		N.A.  LDD0462  [15]
BTD
 Probe Info  		C100(0.40)  LDD2089  [16]
Sulforaphane-probe2
 Probe Info  		2.54  LDD0042  [17]
Curcusone 37
 Probe Info  		2.15  LDD0188  [18]
Johansson_61
 Probe Info  		_(20.00)  LDD1485  [19]
YY4-yne
 Probe Info  		2.37  LDD0400  [20]
AHL-Pu-1
 Probe Info  		C100(2.12)  LDD0171  [21]
HPAP
 Probe Info  		3.14  LDD0062  [22]
DBIA
 Probe Info  		C100(1.65)  LDD0078  [23]
5E-2FA
 Probe Info  		H13(0.00); H181(0.00); H511(0.00)  LDD2235  [24]
ATP probe
 Probe Info  		K223(0.00); K388(0.00); K206(0.00); K21(0.00)  LDD0199  [25]
ATP probe
 Probe Info  		K223(0.00); K78(0.00)  LDD0035  [26]
JW-RF-010
 Probe Info  		N.A.  LDD0026  [27]
NAIA_4
 Probe Info  		N.A.  LDD2226  [28]
TFBX
 Probe Info  		N.A.  LDD0027  [27]
WYneN
 Probe Info  		N.A.  LDD0021  [29]
WYneO
 Probe Info  		N.A.  LDD0022  [29]
ENE
 Probe Info  		N.A.  LDD0006  [29]
IPM
 Probe Info  		N.A.  LDD0005  [29]
NHS
 Probe Info  		K294(0.00); K21(0.00); K260(0.00); K223(0.00)  LDD0010  [29]
STPyne
 Probe Info  		K223(0.00); K213(0.00)  LDD0009  [29]
VSF
 Probe Info  		N.A.  LDD0007  [29]
Phosphinate-6
 Probe Info  		N.A.  LDD0018  [30]
1c-yne
 Probe Info  		K206(0.00); K540(0.00)  LDD0228  [31]
Acrolein
 Probe Info  		H511(0.00); H13(0.00); H24(0.00); C100(0.00)  LDD0217  [32]
Cinnamaldehyde
 Probe Info  		N.A.  LDD0220  [32]
Crotonaldehyde
 Probe Info  		C100(0.00); H13(0.00); H395(0.00); H24(0.00)  LDD0219  [32]
Methacrolein
 Probe Info  		N.A.  LDD0218  [32]
AOyne
 Probe Info  		4.60  LDD0443  [33]
NAIA_5
 Probe Info  		N.A.  LDD2223  [28]
PAL-AfBPP Probe
Click To Hide/Show 106 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
DR-1
 Probe Info  		3.97  LDD0398  [34]
C003
 Probe Info  		12.47  LDD1713  [35]
C004
 Probe Info  		5.78  LDD1714  [35]
C017
 Probe Info  		7.62  LDD1725  [35]
C022
 Probe Info  		17.88  LDD1728  [35]
C027
 Probe Info  		5.54  LDD1733  [35]
C040
 Probe Info  		24.42  LDD1740  [35]
C041
 Probe Info  		9.19  LDD1741  [35]
C052
 Probe Info  		5.86  LDD1750  [35]
C053
 Probe Info  		6.19  LDD1751  [35]
C055
 Probe Info  		13.36  LDD1752  [35]
C056
 Probe Info  		26.72  LDD1753  [35]
C063
 Probe Info  		13.55  LDD1760  [35]
C070
 Probe Info  		12.30  LDD1766  [35]
C087
 Probe Info  		7.57  LDD1779  [35]
C091
 Probe Info  		14.72  LDD1782  [35]
C092
 Probe Info  		21.41  LDD1783  [35]
C094
 Probe Info  		25.28  LDD1785  [35]
C095
 Probe Info  		6.68  LDD1786  [35]
C100
 Probe Info  		10.06  LDD1789  [35]
C106
 Probe Info  		39.95  LDD1793  [35]
C107
 Probe Info  		6.92  LDD1794  [35]
C112
 Probe Info  		47.84  LDD1799  [35]
C129
 Probe Info  		5.13  LDD1811  [35]
C134
 Probe Info  		33.82  LDD1816  [35]
C135
 Probe Info  		9.58  LDD1817  [35]
C138
 Probe Info  		6.36  LDD1820  [35]
C140
 Probe Info  		7.89  LDD1822  [35]
C143
 Probe Info  		13.09  LDD1825  [35]
C153
 Probe Info  		16.56  LDD1834  [35]
C158
 Probe Info  		8.94  LDD1838  [35]
C161
 Probe Info  		11.71  LDD1841  [35]
C163
 Probe Info  		6.54  LDD1843  [35]
C166
 Probe Info  		6.54  LDD1846  [35]
C169
 Probe Info  		30.27  LDD1849  [35]
C177
 Probe Info  		9.25  LDD1856  [35]
C178
 Probe Info  		16.80  LDD1857  [35]
C187
 Probe Info  		38.05  LDD1865  [35]
C194
 Probe Info  		8.88  LDD1870  [35]
C201
 Probe Info  		99.73  LDD1877  [35]
C206
 Probe Info  		28.25  LDD1881  [35]
C207
 Probe Info  		19.56  LDD1882  [35]
C210
 Probe Info  		56.49  LDD1884  [35]
C218
 Probe Info  		19.84  LDD1892  [35]
C219
 Probe Info  		5.24  LDD1893  [35]
C220
 Probe Info  		19.84  LDD1894  [35]
C228
 Probe Info  		24.42  LDD1901  [35]
C231
 Probe Info  		20.82  LDD1904  [35]
C232
 Probe Info  		42.52  LDD1905  [35]
C234
 Probe Info  		6.15  LDD1907  [35]
C235
 Probe Info  		33.13  LDD1908  [35]
C238
 Probe Info  		12.04  LDD1911  [35]
C244
 Probe Info  		22.16  LDD1917  [35]
C246
 Probe Info  		19.43  LDD1919  [35]
C265
 Probe Info  		18.64  LDD1936  [35]
C277
 Probe Info  		8.82  LDD1947  [35]
C285
 Probe Info  		25.11  LDD1955  [35]
C289
 Probe Info  		43.41  LDD1959  [35]
C293
 Probe Info  		22.94  LDD1963  [35]
C296
 Probe Info  		19.97  LDD1966  [35]
C299
 Probe Info  		6.82  LDD1968  [35]
C310
 Probe Info  		9.19  LDD1977  [35]
C313
 Probe Info  		12.55  LDD1980  [35]
C314
 Probe Info  		13.27  LDD1981  [35]
C317
 Probe Info  		10.70  LDD1983  [35]
C326
 Probe Info  		7.16  LDD1990  [35]
C338
 Probe Info  		13.83  LDD2001  [35]
C339
 Probe Info  		11.31  LDD2002  [35]
C343
 Probe Info  		16.91  LDD2005  [35]
C348
 Probe Info  		17.51  LDD2009  [35]
C349
 Probe Info  		20.11  LDD2010  [35]
C350
 Probe Info  		74.03  LDD2011  [35]
C354
 Probe Info  		7.57  LDD2015  [35]
C355
 Probe Info  		32.90  LDD2016  [35]
C356
 Probe Info  		8.75  LDD2017  [35]
C362
 Probe Info  		99.73  LDD2023  [35]
C363
 Probe Info  		31.34  LDD2024  [35]
C364
 Probe Info  		30.06  LDD2025  [35]
C366
 Probe Info  		8.88  LDD2027  [35]
C367
 Probe Info  		7.89  LDD2028  [35]
C382
 Probe Info  		10.13  LDD2041  [35]
C383
 Probe Info  		34.30  LDD2042  [35]
C388
 Probe Info  		76.64  LDD2047  [35]
C390
 Probe Info  		99.73  LDD2049  [35]
C391
 Probe Info  		22.01  LDD2050  [35]
C393
 Probe Info  		5.78  LDD2052  [35]
C403
 Probe Info  		28.44  LDD2061  [35]
C407
 Probe Info  		20.25  LDD2064  [35]
C413
 Probe Info  		15.45  LDD2069  [35]
C420
 Probe Info  		12.04  LDD2075  [35]
C431
 Probe Info  		15.89  LDD2086  [35]
FFF probe11
 Probe Info  		20.00  LDD0471  [36]
FFF probe12
 Probe Info  		20.00  LDD0473  [36]
FFF probe13
 Probe Info  		20.00  LDD0475  [36]
FFF probe14
 Probe Info  		20.00  LDD0477  [36]
FFF probe15
 Probe Info  		11.18  LDD0478  [36]
FFF probe2
 Probe Info  		20.00  LDD0463  [36]
FFF probe3
 Probe Info  		20.00  LDD0464  [36]
FFF probe6
 Probe Info  		20.00  LDD0482  [36]
FFF probe9
 Probe Info  		20.00  LDD0470  [36]
JN0003
 Probe Info  		20.00  LDD0469  [36]
STS-1
 Probe Info  		4.70  LDD0136  [37]
STS-2
 Probe Info  		9.90  LDD0138  [37]
Diazir
 Probe Info  		N.A.  LDD0011  [29]
BD-F
 Probe Info  		A92(0.00); A90(0.00); A94(0.00)  LDD0024  [38]
OEA-DA
 Probe Info  		3.40  LDD0046  [39]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0548  1-(4-(Benzo[d][1,3]dioxol-5-ylmethyl)piperazin-1-yl)-2-nitroethan-1-one MDA-MB-231 C100(1.08)  LDD2142  [16]
 LDCM0519  1-(6-methoxy-3,4-dihydroquinolin-1(2H)-yl)-2-nitroethan-1-one MDA-MB-231 C100(1.50)  LDD2112  [16]
 LDCM0524  2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide MDA-MB-231 C100(0.82)  LDD2117  [16]
 LDCM0558  2-Cyano-N-phenylacetamide MDA-MB-231 C100(1.19)  LDD2152  [16]
 LDCM0026  4SU-RNA+native RNA DM93 C100(2.12)  LDD0171  [21]
 LDCM0214  AC1 HCT 116 C100(0.90)  LDD0531  [23]
 LDCM0215  AC10 HCT 116 C100(0.69)  LDD0532  [23]
 LDCM0216  AC100 HCT 116 C100(0.83)  LDD0533  [23]
 LDCM0217  AC101 HCT 116 C100(1.16)  LDD0534  [23]
 LDCM0218  AC102 HCT 116 C100(1.01)  LDD0535  [23]
 LDCM0219  AC103 HCT 116 C100(1.10)  LDD0536  [23]
 LDCM0220  AC104 HCT 116 C100(1.04)  LDD0537  [23]
 LDCM0221  AC105 HCT 116 C100(1.10)  LDD0538  [23]
 LDCM0222  AC106 HCT 116 C100(0.96)  LDD0539  [23]
 LDCM0223  AC107 HCT 116 C100(1.14)  LDD0540  [23]
 LDCM0224  AC108 HCT 116 C100(1.22)  LDD0541  [23]
 LDCM0225  AC109 HCT 116 C100(0.86)  LDD0542  [23]
 LDCM0226  AC11 HCT 116 C100(0.85)  LDD0543  [23]
 LDCM0227  AC110 HCT 116 C100(1.00)  LDD0544  [23]
 LDCM0228  AC111 HCT 116 C100(1.06)  LDD0545  [23]
 LDCM0229  AC112 HCT 116 C100(1.18)  LDD0546  [23]
 LDCM0230  AC113 HCT 116 C100(0.99)  LDD0547  [23]
 LDCM0231  AC114 HCT 116 C100(1.18)  LDD0548  [23]
 LDCM0232  AC115 HCT 116 C100(1.11)  LDD0549  [23]
 LDCM0233  AC116 HCT 116 C100(0.95)  LDD0550  [23]
 LDCM0234  AC117 HCT 116 C100(1.00)  LDD0551  [23]
 LDCM0235  AC118 HCT 116 C100(0.85)  LDD0552  [23]
 LDCM0236  AC119 HCT 116 C100(0.88)  LDD0553  [23]
 LDCM0237  AC12 HCT 116 C100(0.84)  LDD0554  [23]
 LDCM0238  AC120 HCT 116 C100(1.07)  LDD0555  [23]
 LDCM0239  AC121 HCT 116 C100(0.82)  LDD0556  [23]
 LDCM0240  AC122 HCT 116 C100(0.83)  LDD0557  [23]
 LDCM0241  AC123 HCT 116 C100(1.05)  LDD0558  [23]
 LDCM0242  AC124 HCT 116 C100(0.87)  LDD0559  [23]
 LDCM0243  AC125 HCT 116 C100(0.94)  LDD0560  [23]
 LDCM0244  AC126 HCT 116 C100(1.17)  LDD0561  [23]
 LDCM0245  AC127 HCT 116 C100(0.99)  LDD0562  [23]
 LDCM0246  AC128 HCT 116 C100(1.35)  LDD0563  [23]
 LDCM0247  AC129 HCT 116 C100(1.19)  LDD0564  [23]
 LDCM0249  AC130 HCT 116 C100(1.20)  LDD0566  [23]
 LDCM0250  AC131 HCT 116 C100(1.38)  LDD0567  [23]
 LDCM0251  AC132 HCT 116 C100(1.09)  LDD0568  [23]
 LDCM0252  AC133 HCT 116 C100(1.25)  LDD0569  [23]
 LDCM0253  AC134 HCT 116 C100(1.56)  LDD0570  [23]
 LDCM0254  AC135 HCT 116 C100(1.15)  LDD0571  [23]
 LDCM0255  AC136 HCT 116 C100(1.33)  LDD0572  [23]
 LDCM0256  AC137 HCT 116 C100(1.21)  LDD0573  [23]
 LDCM0257  AC138 HCT 116 C100(1.59)  LDD0574  [23]
 LDCM0258  AC139 HCT 116 C100(1.19)  LDD0575  [23]
 LDCM0259  AC14 HCT 116 C100(0.73)  LDD0576  [23]
 LDCM0260  AC140 HCT 116 C100(1.57)  LDD0577  [23]
 LDCM0261  AC141 HCT 116 C100(1.66)  LDD0578  [23]
 LDCM0262  AC142 HCT 116 C100(1.20)  LDD0579  [23]
 LDCM0263  AC143 HCT 116 C100(1.06)  LDD0580  [23]
 LDCM0264  AC144 HCT 116 C100(1.07)  LDD0581  [23]
 LDCM0265  AC145 HCT 116 C100(1.06)  LDD0582  [23]
 LDCM0266  AC146 HCT 116 C100(1.08)  LDD0583  [23]
 LDCM0267  AC147 HCT 116 C100(1.02)  LDD0584  [23]
 LDCM0268  AC148 HCT 116 C100(1.10)  LDD0585  [23]
 LDCM0269  AC149 HCT 116 C100(1.12)  LDD0586  [23]
 LDCM0270  AC15 HCT 116 C100(0.73)  LDD0587  [23]
 LDCM0271  AC150 HCT 116 C100(1.25)  LDD0588  [23]
 LDCM0272  AC151 HCT 116 C100(0.86)  LDD0589  [23]
 LDCM0273  AC152 HCT 116 C100(1.03)  LDD0590  [23]
 LDCM0274  AC153 HCT 116 C100(1.10)  LDD0591  [23]
 LDCM0621  AC154 HCT 116 C100(1.01)  LDD2158  [23]
 LDCM0622  AC155 HCT 116 C100(1.01)  LDD2159  [23]
 LDCM0623  AC156 HCT 116 C100(0.90)  LDD2160  [23]
 LDCM0624  AC157 HCT 116 C100(0.83)  LDD2161  [23]
 LDCM0276  AC17 HCT 116 C100(1.52)  LDD0593  [23]
 LDCM0277  AC18 HCT 116 C100(1.15)  LDD0594  [23]
 LDCM0278  AC19 HCT 116 C100(1.50)  LDD0595  [23]
 LDCM0279  AC2 HCT 116 C100(0.77)  LDD0596  [23]
 LDCM0280  AC20 HCT 116 C100(1.29)  LDD0597  [23]
 LDCM0281  AC21 HCT 116 C100(1.42)  LDD0598  [23]
 LDCM0282  AC22 HCT 116 C100(1.10)  LDD0599  [23]
 LDCM0283  AC23 HCT 116 C100(2.22)  LDD0600  [23]
 LDCM0284  AC24 HCT 116 C100(1.39)  LDD0601  [23]
 LDCM0285  AC25 HCT 116 C100(0.95)  LDD0602  [23]
 LDCM0286  AC26 HCT 116 C100(0.94)  LDD0603  [23]
 LDCM0287  AC27 HCT 116 C100(0.94)  LDD0604  [23]
 LDCM0288  AC28 HCT 116 C100(1.35)  LDD0605  [23]
 LDCM0289  AC29 HCT 116 C100(1.04)  LDD0606  [23]
 LDCM0290  AC3 HCT 116 C100(0.71)  LDD0607  [23]
 LDCM0291  AC30 HCT 116 C100(0.96)  LDD0608  [23]
 LDCM0292  AC31 HCT 116 C100(0.92)  LDD0609  [23]
 LDCM0293  AC32 HCT 116 C100(1.06)  LDD0610  [23]
 LDCM0294  AC33 HCT 116 C100(1.09)  LDD0611  [23]
 LDCM0295  AC34 HCT 116 C100(1.38)  LDD0612  [23]
 LDCM0296  AC35 HCT 116 C100(0.91)  LDD0613  [23]
 LDCM0297  AC36 HCT 116 C100(0.96)  LDD0614  [23]
 LDCM0298  AC37 HCT 116 C100(0.91)  LDD0615  [23]
 LDCM0299  AC38 HCT 116 C100(0.94)  LDD0616  [23]
 LDCM0300  AC39 HCT 116 C100(0.78)  LDD0617  [23]
 LDCM0301  AC4 HCT 116 C100(0.73)  LDD0618  [23]
 LDCM0302  AC40 HCT 116 C100(1.09)  LDD0619  [23]
 LDCM0303  AC41 HCT 116 C100(0.97)  LDD0620  [23]
 LDCM0304  AC42 HCT 116 C100(1.01)  LDD0621  [23]
 LDCM0305  AC43 HCT 116 C100(0.92)  LDD0622  [23]
 LDCM0306  AC44 HCT 116 C100(0.82)  LDD0623  [23]
 LDCM0307  AC45 HCT 116 C100(0.87)  LDD0624  [23]
 LDCM0308  AC46 HCT 116 C100(1.22)  LDD0625  [23]
 LDCM0309  AC47 HCT 116 C100(1.07)  LDD0626  [23]
 LDCM0310  AC48 HCT 116 C100(0.90)  LDD0627  [23]
 LDCM0311  AC49 HCT 116 C100(1.37)  LDD0628  [23]
 LDCM0312  AC5 HCT 116 C100(0.68)  LDD0629  [23]
 LDCM0313  AC50 HCT 116 C100(1.62)  LDD0630  [23]
 LDCM0314  AC51 HCT 116 C100(1.07)  LDD0631  [23]
 LDCM0315  AC52 HCT 116 C100(1.16)  LDD0632  [23]
 LDCM0316  AC53 HCT 116 C100(1.51)  LDD0633  [23]
 LDCM0317  AC54 HCT 116 C100(0.95)  LDD0634  [23]
 LDCM0318  AC55 HCT 116 C100(1.48)  LDD0635  [23]
 LDCM0319  AC56 HCT 116 C100(1.66)  LDD0636  [23]
 LDCM0320  AC57 HCT 116 C100(0.84)  LDD0637  [23]
 LDCM0321  AC58 HCT 116 C100(1.02)  LDD0638  [23]
 LDCM0322  AC59 HCT 116 C100(0.90)  LDD0639  [23]
 LDCM0323  AC6 HCT 116 C100(0.92)  LDD0640  [23]
 LDCM0324  AC60 HCT 116 C100(0.86)  LDD0641  [23]
 LDCM0325  AC61 HCT 116 C100(0.62)  LDD0642  [23]
 LDCM0326  AC62 HCT 116 C100(0.89)  LDD0643  [23]
 LDCM0327  AC63 HCT 116 C100(0.97)  LDD0644  [23]
 LDCM0328  AC64 HCT 116 C100(0.77)  LDD0645  [23]
 LDCM0329  AC65 HCT 116 C100(0.76)  LDD0646  [23]
 LDCM0330  AC66 HCT 116 C100(0.86)  LDD0647  [23]
 LDCM0331  AC67 HCT 116 C100(0.77)  LDD0648  [23]
 LDCM0332  AC68 HCT 116 C100(0.88)  LDD0649  [23]
 LDCM0333  AC69 HCT 116 C100(0.96)  LDD0650  [23]
 LDCM0334  AC7 HCT 116 C100(0.82)  LDD0651  [23]
 LDCM0335  AC70 HCT 116 C100(1.09)  LDD0652  [23]
 LDCM0336  AC71 HCT 116 C100(0.77)  LDD0653  [23]
 LDCM0337  AC72 HCT 116 C100(1.09)  LDD0654  [23]
 LDCM0338  AC73 HCT 116 C100(1.18)  LDD0655  [23]
 LDCM0339  AC74 HCT 116 C100(1.23)  LDD0656  [23]
 LDCM0340  AC75 HCT 116 C100(1.24)  LDD0657  [23]
 LDCM0341  AC76 HCT 116 C100(0.98)  LDD0658  [23]
 LDCM0342  AC77 HCT 116 C100(1.31)  LDD0659  [23]
 LDCM0343  AC78 HCT 116 C100(0.87)  LDD0660  [23]
 LDCM0344  AC79 HCT 116 C100(0.96)  LDD0661  [23]
 LDCM0345  AC8 HCT 116 C100(0.79)  LDD0662  [23]
 LDCM0346  AC80 HCT 116 C100(0.87)  LDD0663  [23]
 LDCM0347  AC81 HCT 116 C100(0.92)  LDD0664  [23]
 LDCM0348  AC82 HCT 116 C100(1.17)  LDD0665  [23]
 LDCM0349  AC83 HCT 116 C100(1.32)  LDD0666  [23]
 LDCM0350  AC84 HCT 116 C100(1.32)  LDD0667  [23]
 LDCM0351  AC85 HCT 116 C100(1.29)  LDD0668  [23]
 LDCM0352  AC86 HCT 116 C100(1.48)  LDD0669  [23]
 LDCM0353  AC87 HCT 116 C100(1.24)  LDD0670  [23]
 LDCM0354  AC88 HCT 116 C100(1.34)  LDD0671  [23]
 LDCM0355  AC89 HCT 116 C100(1.40)  LDD0672  [23]
 LDCM0357  AC90 HCT 116 C100(1.18)  LDD0674  [23]
 LDCM0358  AC91 HCT 116 C100(1.42)  LDD0675  [23]
 LDCM0359  AC92 HCT 116 C100(1.41)  LDD0676  [23]
 LDCM0360  AC93 HCT 116 C100(1.23)  LDD0677  [23]
 LDCM0361  AC94 HCT 116 C100(1.39)  LDD0678  [23]
 LDCM0362  AC95 HCT 116 C100(2.18)  LDD0679  [23]
 LDCM0363  AC96 HCT 116 C100(1.44)  LDD0680  [23]
 LDCM0364  AC97 HCT 116 C100(1.32)  LDD0681  [23]
 LDCM0365  AC98 HCT 116 C100(1.26)  LDD0682  [23]
 LDCM0366  AC99 HCT 116 C100(1.11)  LDD0683  [23]
 LDCM0520  AKOS000195272 MDA-MB-231 C100(0.77)  LDD2113  [16]
 LDCM0248  AKOS034007472 HCT 116 C100(0.66)  LDD0565  [23]
 LDCM0356  AKOS034007680 HCT 116 C100(0.75)  LDD0673  [23]
 LDCM0275  AKOS034007705 HCT 116 C100(0.87)  LDD0592  [23]
 LDCM0156  Aniline NCI-H1299 11.81  LDD0403  [12]
 LDCM0020  ARS-1620 HCC44 C100(1.65)  LDD0078  [23]
 LDCM0498  BS-3668 MDA-MB-231 C100(0.58)  LDD2091  [16]
 LDCM0630  CCW28-3 231MFP C100(1.53)  LDD2214  [40]
 LDCM0108  Chloroacetamide HeLa C100(0.00); H24(0.00); H13(0.00); H395(0.00)  LDD0222  [32]
 LDCM0632  CL-Sc Hep-G2 C100(0.37)  LDD2227  [28]
 LDCM0367  CL1 HCT 116 C100(1.84)  LDD0684  [23]
 LDCM0368  CL10 HCT 116 C100(3.26)  LDD0685  [23]
 LDCM0369  CL100 HCT 116 C100(1.21)  LDD0686  [23]
 LDCM0370  CL101 HCT 116 C100(1.20)  LDD0687  [23]
 LDCM0371  CL102 HCT 116 C100(0.67)  LDD0688  [23]
 LDCM0372  CL103 HCT 116 C100(1.33)  LDD0689  [23]
 LDCM0373  CL104 HCT 116 C100(1.58)  LDD0690  [23]
 LDCM0374  CL105 HCT 116 C100(1.41)  LDD0691  [23]
 LDCM0375  CL106 HCT 116 C100(2.03)  LDD0692  [23]
 LDCM0376  CL107 HCT 116 C100(1.14)  LDD0693  [23]
 LDCM0377  CL108 HCT 116 C100(1.30)  LDD0694  [23]
 LDCM0378  CL109 HCT 116 C100(2.60)  LDD0695  [23]
 LDCM0379  CL11 HCT 116 C100(2.94)  LDD0696  [23]
 LDCM0380  CL110 HCT 116 C100(3.79)  LDD0697  [23]
 LDCM0381  CL111 HCT 116 C100(2.55)  LDD0698  [23]
 LDCM0382  CL112 HCT 116 C100(1.05)  LDD0699  [23]
 LDCM0383  CL113 HCT 116 C100(1.15)  LDD0700  [23]
 LDCM0384  CL114 HCT 116 C100(6.85)  LDD0701  [23]
 LDCM0385  CL115 HCT 116 C100(1.06)  LDD0702  [23]
 LDCM0386  CL116 HCT 116 C100(0.89)  LDD0703  [23]
 LDCM0387  CL117 HCT 116 C100(1.30)  LDD0704  [23]
 LDCM0388  CL118 HCT 116 C100(0.93)  LDD0705  [23]
 LDCM0389  CL119 HCT 116 C100(1.21)  LDD0706  [23]
 LDCM0390  CL12 HCT 116 C100(1.43)  LDD0707  [23]
 LDCM0391  CL120 HCT 116 C100(0.84)  LDD0708  [23]
 LDCM0392  CL121 HCT 116 C100(0.89)  LDD0709  [23]
 LDCM0393  CL122 HCT 116 C100(2.17)  LDD0710  [23]
 LDCM0394  CL123 HCT 116 C100(9.16)  LDD0711  [23]
 LDCM0395  CL124 HCT 116 C100(2.21)  LDD0712  [23]
 LDCM0396  CL125 HCT 116 C100(0.84)  LDD0713  [23]
 LDCM0397  CL126 HCT 116 C100(1.48)  LDD0714  [23]
 LDCM0398  CL127 HCT 116 C100(0.82)  LDD0715  [23]
 LDCM0399  CL128 HCT 116 C100(0.80)  LDD0716  [23]
 LDCM0400  CL13 HCT 116 C100(1.09)  LDD0717  [23]
 LDCM0401  CL14 HCT 116 C100(1.61)  LDD0718  [23]
 LDCM0402  CL15 HCT 116 C100(2.21)  LDD0719  [23]
 LDCM0403  CL16 HCT 116 C100(1.03)  LDD0720  [23]
 LDCM0404  CL17 HCT 116 C100(5.44)  LDD0721  [23]
 LDCM0405  CL18 HCT 116 C100(1.29)  LDD0722  [23]
 LDCM0406  CL19 HCT 116 C100(1.09)  LDD0723  [23]
 LDCM0407  CL2 HCT 116 C100(0.95)  LDD0724  [23]
 LDCM0408  CL20 HCT 116 C100(1.46)  LDD0725  [23]
 LDCM0409  CL21 HCT 116 C100(6.97)  LDD0726  [23]
 LDCM0410  CL22 HCT 116 C100(1.77)  LDD0727  [23]
 LDCM0411  CL23 HCT 116 C100(1.49)  LDD0728  [23]
 LDCM0412  CL24 HCT 116 C100(1.50)  LDD0729  [23]
 LDCM0413  CL25 HCT 116 C100(4.27)  LDD0730  [23]
 LDCM0414  CL26 HCT 116 C100(1.18)  LDD0731  [23]
 LDCM0415  CL27 HCT 116 C100(1.12)  LDD0732  [23]
 LDCM0416  CL28 HCT 116 C100(1.65)  LDD0733  [23]
 LDCM0417  CL29 HCT 116 C100(1.37)  LDD0734  [23]
 LDCM0418  CL3 HCT 116 C100(2.20)  LDD0735  [23]
 LDCM0419  CL30 HCT 116 C100(1.07)  LDD0736  [23]
 LDCM0420  CL31 HCT 116 C100(1.60)  LDD0737  [23]
 LDCM0421  CL32 HCT 116 C100(1.52)  LDD0738  [23]
 LDCM0422  CL33 HCT 116 C100(11.23)  LDD0739  [23]
 LDCM0423  CL34 HCT 116 C100(2.65)  LDD0740  [23]
 LDCM0424  CL35 HCT 116 C100(2.21)  LDD0741  [23]
 LDCM0425  CL36 HCT 116 C100(3.18)  LDD0742  [23]
 LDCM0426  CL37 HCT 116 C100(2.95)  LDD0743  [23]
 LDCM0428  CL39 HCT 116 C100(2.16)  LDD0745  [23]
 LDCM0429  CL4 HCT 116 C100(4.34)  LDD0746  [23]
 LDCM0430  CL40 HCT 116 C100(4.46)  LDD0747  [23]
 LDCM0431  CL41 HCT 116 C100(2.37)  LDD0748  [23]
 LDCM0432  CL42 HCT 116 C100(6.63)  LDD0749  [23]
 LDCM0433  CL43 HCT 116 C100(2.52)  LDD0750  [23]
 LDCM0434  CL44 HCT 116 C100(2.26)  LDD0751  [23]
 LDCM0435  CL45 HCT 116 C100(3.61)  LDD0752  [23]
 LDCM0436  CL46 HCT 116 C100(1.46)  LDD0753  [23]
 LDCM0437  CL47 HCT 116 C100(1.25)  LDD0754  [23]
 LDCM0438  CL48 HCT 116 C100(1.69)  LDD0755  [23]
 LDCM0439  CL49 HCT 116 C100(2.43)  LDD0756  [23]
 LDCM0440  CL5 HCT 116 C100(0.94)  LDD0757  [23]
 LDCM0441  CL50 HCT 116 C100(2.06)  LDD0758  [23]
 LDCM0442  CL51 HCT 116 C100(1.90)  LDD0759  [23]
 LDCM0443  CL52 HCT 116 C100(1.67)  LDD0760  [23]
 LDCM0444  CL53 HCT 116 C100(6.39)  LDD0761  [23]
 LDCM0445  CL54 HCT 116 C100(4.81)  LDD0762  [23]
 LDCM0446  CL55 HCT 116 C100(1.78)  LDD0763  [23]
 LDCM0447  CL56 HCT 116 C100(1.11)  LDD0764  [23]
 LDCM0448  CL57 HCT 116 C100(1.55)  LDD0765  [23]
 LDCM0449  CL58 HCT 116 C100(1.40)  LDD0766  [23]
 LDCM0450  CL59 HCT 116 C100(1.17)  LDD0767  [23]
 LDCM0451  CL6 HCT 116 C100(3.57)  LDD0768  [23]
 LDCM0452  CL60 HCT 116 C100(1.57)  LDD0769  [23]
 LDCM0453  CL61 HCT 116 C100(1.08)  LDD0770  [23]
 LDCM0454  CL62 HCT 116 C100(1.06)  LDD0771  [23]
 LDCM0455  CL63 HCT 116 C100(2.43)  LDD0772  [23]
 LDCM0456  CL64 HCT 116 C100(3.04)  LDD0773  [23]
 LDCM0457  CL65 HCT 116 C100(1.20)  LDD0774  [23]
 LDCM0458  CL66 HCT 116 C100(1.16)  LDD0775  [23]
 LDCM0459  CL67 HCT 116 C100(1.07)  LDD0776  [23]
 LDCM0460  CL68 HCT 116 C100(1.20)  LDD0777  [23]
 LDCM0461  CL69 HCT 116 C100(2.13)  LDD0778  [23]
 LDCM0462  CL7 HCT 116 C100(1.14)  LDD0779  [23]
 LDCM0463  CL70 HCT 116 C100(1.28)  LDD0780  [23]
 LDCM0464  CL71 HCT 116 C100(1.23)  LDD0781  [23]
 LDCM0465  CL72 HCT 116 C100(0.92)  LDD0782  [23]
 LDCM0466  CL73 HCT 116 C100(1.93)  LDD0783  [23]
 LDCM0467  CL74 HCT 116 C100(1.21)  LDD0784  [23]
 LDCM0469  CL76 HCT 116 C100(1.07)  LDD0786  [23]
 LDCM0470  CL77 HCT 116 C100(2.48)  LDD0787  [23]
 LDCM0471  CL78 HCT 116 C100(1.63)  LDD0788  [23]
 LDCM0472  CL79 HCT 116 C100(1.72)  LDD0789  [23]
 LDCM0473  CL8 HCT 116 C100(7.53)  LDD0790  [23]
 LDCM0474  CL80 HCT 116 C100(1.15)  LDD0791  [23]
 LDCM0475  CL81 HCT 116 C100(1.33)  LDD0792  [23]
 LDCM0476  CL82 HCT 116 C100(1.69)  LDD0793  [23]
 LDCM0477  CL83 HCT 116 C100(3.99)  LDD0794  [23]
 LDCM0478  CL84 HCT 116 C100(4.29)  LDD0795  [23]
 LDCM0479  CL85 HCT 116 C100(1.55)  LDD0796  [23]
 LDCM0480  CL86 HCT 116 C100(1.47)  LDD0797  [23]
 LDCM0481  CL87 HCT 116 C100(1.23)  LDD0798  [23]
 LDCM0482  CL88 HCT 116 C100(1.29)  LDD0799  [23]
 LDCM0483  CL89 HCT 116 C100(1.78)  LDD0800  [23]
 LDCM0484  CL9 HCT 116 C100(1.47)  LDD0801  [23]
 LDCM0485  CL90 HCT 116 C100(5.99)  LDD0802  [23]
 LDCM0486  CL91 HCT 116 C100(1.04)  LDD0803  [23]
 LDCM0487  CL92 HCT 116 C100(2.18)  LDD0804  [23]
 LDCM0488  CL93 HCT 116 C100(1.64)  LDD0805  [23]
 LDCM0489  CL94 HCT 116 C100(1.63)  LDD0806  [23]
 LDCM0490  CL95 HCT 116 C100(4.35)  LDD0807  [23]
 LDCM0491  CL96 HCT 116 C100(1.68)  LDD0808  [23]
 LDCM0492  CL97 HCT 116 C100(2.07)  LDD0809  [23]
 LDCM0493  CL98 HCT 116 C100(1.19)  LDD0810  [23]
 LDCM0494  CL99 HCT 116 C100(0.87)  LDD0811  [23]
 LDCM0185  Compound 17 HEK-293T 12.12  LDD0512  [36]
 LDCM0191  Compound 21 HEK-293T 8.13  LDD0508  [36]
 LDCM0190  Compound 34 HEK-293T 12.12  LDD0510  [36]
 LDCM0192  Compound 35 HEK-293T 9.52  LDD0509  [36]
 LDCM0193  Compound 36 HEK-293T 6.60  LDD0511  [36]
 LDCM0033  Curcusone1d MCF-7 2.15  LDD0188  [18]
 LDCM0495  E2913 HEK-293T C100(1.28)  LDD1698  [41]
 LDCM0213  Electrophilic fragment 2 MDA-MB-231 C100(35.85)  LDD1702  [16]
 LDCM0204  EV-97 T cell C100(7.48)  LDD0524  [42]
 LDCM0625  F8 Ramos C100(1.83)  LDD2187  [43]
 LDCM0572  Fragment10 Ramos C100(5.14)  LDD2189  [43]
 LDCM0573  Fragment11 MDA-MB-231 C100(0.97)  LDD1467  [19]
 LDCM0574  Fragment12 MDA-MB-231 C100(20.00)  LDD1468  [19]
 LDCM0575  Fragment13 MDA-MB-231 C100(1.62)  LDD1469  [19]
 LDCM0576  Fragment14 MDA-MB-231 C100(11.16)  LDD1471  [19]
 LDCM0579  Fragment20 Ramos C100(4.62)  LDD2194  [43]
 LDCM0580  Fragment21 MDA-MB-231 C100(2.23)  LDD1473  [19]
 LDCM0582  Fragment23 Ramos C100(0.87)  LDD2196  [43]
 LDCM0578  Fragment27 Ramos C100(1.13)  LDD2197  [43]
 LDCM0586  Fragment28 Ramos C100(2.04)  LDD2198  [43]
 LDCM0588  Fragment30 Ramos C100(2.58)  LDD2199  [43]
 LDCM0589  Fragment31 Ramos C100(1.81)  LDD2200  [43]
 LDCM0590  Fragment32 Ramos C100(3.35)  LDD2201  [43]
 LDCM0468  Fragment33 HCT 116 C100(0.91)  LDD0785  [23]
 LDCM0596  Fragment38 Ramos C100(3.85)  LDD2203  [43]
 LDCM0566  Fragment4 Ramos C100(6.84)  LDD2184  [43]
 LDCM0599  Fragment41 MDA-MB-231 C100(1.01)  LDD1481  [19]
 LDCM0603  Fragment45 MDA-MB-231 C100(20.00)  LDD1482  [19]
 LDCM0427  Fragment51 HCT 116 C100(2.41)  LDD0744  [23]
 LDCM0610  Fragment52 Ramos C100(2.52)  LDD2204  [43]
 LDCM0614  Fragment56 Ramos C100(1.63)  LDD2205  [43]
 LDCM0615  Fragment63-R Jurkat _(20.00)  LDD1487  [19]
 LDCM0617  Fragment63-S Jurkat _(20.00)  LDD1490  [19]
 LDCM0569  Fragment7 Jurkat _(20.00)  LDD1485  [19]
 LDCM0571  Fragment9 MDA-MB-231 C100(15.44)  LDD1463  [19]
 LDCM0149  GA MCF-7 C100(3.08)  LDD0379  [44]
 LDCM0107  IAA HeLa H511(0.00); H24(0.00); H13(0.00); H395(0.00)  LDD0221  [32]
 LDCM0179  JZ128 PC-3 N.A.  LDD0462  [15]
 LDCM0022  KB02 HCT 116 C100(20.00)  LDD0080  [23]
 LDCM0023  KB03 HCT 116 C100(20.00)  LDD0081  [23]
 LDCM0024  KB05 HCT 116 C100(20.00)  LDD0082  [23]
 LDCM0169  KB63 Ramos 7.42  LDD0432  [45]
 LDCM0528  N-(4-bromophenyl)-2-cyano-N-phenylacetamide MDA-MB-231 C100(0.31)  LDD2121  [16]
 LDCM0109  NEM HeLa H511(0.00); C100(0.00); H415(0.00); H395(0.00)  LDD0223  [32]
 LDCM0496  Nucleophilic fragment 11a MDA-MB-231 C100(0.40)  LDD2089  [16]
 LDCM0497  Nucleophilic fragment 11b MDA-MB-231 C100(1.84)  LDD2090  [16]
 LDCM0499  Nucleophilic fragment 12b MDA-MB-231 C100(1.08)  LDD2092  [16]
 LDCM0500  Nucleophilic fragment 13a MDA-MB-231 C100(0.80)  LDD2093  [16]
 LDCM0501  Nucleophilic fragment 13b MDA-MB-231 C100(1.20)  LDD2094  [16]
 LDCM0504  Nucleophilic fragment 15a MDA-MB-231 C100(1.26)  LDD2097  [16]
 LDCM0505  Nucleophilic fragment 15b MDA-MB-231 C100(1.54)  LDD2098  [16]
 LDCM0506  Nucleophilic fragment 16a MDA-MB-231 C100(0.89)  LDD2099  [16]
 LDCM0507  Nucleophilic fragment 16b MDA-MB-231 C100(2.27)  LDD2100  [16]
 LDCM0511  Nucleophilic fragment 18b MDA-MB-231 C100(1.68)  LDD2104  [16]
 LDCM0512  Nucleophilic fragment 19a MDA-MB-231 C100(0.94)  LDD2105  [16]
 LDCM0513  Nucleophilic fragment 19b MDA-MB-231 C100(1.33)  LDD2106  [16]
 LDCM0514  Nucleophilic fragment 20a MDA-MB-231 C100(0.73)  LDD2107  [16]
 LDCM0515  Nucleophilic fragment 20b MDA-MB-231 C100(0.98)  LDD2108  [16]
 LDCM0516  Nucleophilic fragment 21a MDA-MB-231 C100(0.88)  LDD2109  [16]
 LDCM0517  Nucleophilic fragment 21b MDA-MB-231 C100(2.47)  LDD2110  [16]
 LDCM0521  Nucleophilic fragment 23b MDA-MB-231 C100(1.63)  LDD2114  [16]
 LDCM0522  Nucleophilic fragment 24a MDA-MB-231 C100(0.77)  LDD2115  [16]
 LDCM0527  Nucleophilic fragment 26b MDA-MB-231 C100(1.11)  LDD2120  [16]
 LDCM0530  Nucleophilic fragment 28a MDA-MB-231 C100(0.48)  LDD2123  [16]
 LDCM0531  Nucleophilic fragment 28b MDA-MB-231 C100(1.24)  LDD2124  [16]
 LDCM0534  Nucleophilic fragment 30a MDA-MB-231 C100(1.15)  LDD2127  [16]
 LDCM0540  Nucleophilic fragment 35 MDA-MB-231 C100(0.64)  LDD2133  [16]
 LDCM0541  Nucleophilic fragment 36 MDA-MB-231 C100(0.78)  LDD2134  [16]
 LDCM0542  Nucleophilic fragment 37 MDA-MB-231 C100(0.69)  LDD2135  [16]
 LDCM0543  Nucleophilic fragment 38 MDA-MB-231 C100(1.54)  LDD2136  [16]
 LDCM0546  Nucleophilic fragment 40 MDA-MB-231 C100(0.61)  LDD2140  [16]
 LDCM0547  Nucleophilic fragment 41 MDA-MB-231 C100(0.76)  LDD2141  [16]
 LDCM0549  Nucleophilic fragment 43 MDA-MB-231 C100(1.18)  LDD2143  [16]
 LDCM0552  Nucleophilic fragment 6a MDA-MB-231 C100(0.66)  LDD2146  [16]
 LDCM0554  Nucleophilic fragment 7a MDA-MB-231 C100(0.60)  LDD2148  [16]
 LDCM0556  Nucleophilic fragment 8a MDA-MB-231 C100(0.56)  LDD2150  [16]
 LDCM0559  Nucleophilic fragment 9b MDA-MB-231 C100(2.31)  LDD2153  [16]
 LDCM0627  NUDT7-COV-1 HEK-293T C100(0.07)  LDD2206  [46]
 LDCM0159  P28 BxPC-3 1.48  LDD0409  [14]
 LDCM0014  Panhematin HEK-293T 3.14  LDD0062  [22]
 LDCM0099  Phenelzine MDA-MB-231 4.00  LDD0392  [13]
 LDCM0131  RA190 MM1.R C100(3.94)  LDD0304  [11]
 LDCM0003  Sulforaphane MCF-7 2.54  LDD0042  [17]
 LDCM0021  THZ1 HCT 116 C100(1.17)  LDD2173  [23]
 LDCM0154  YY4 T cell 2.37  LDD0400  [20]

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