Details of the Target

General Information of Target

Target ID LDTP04689
Target Name Adenosine kinase (ADK)
Gene Name ADK
Gene ID 132
Synonyms
Adenosine kinase; AK; EC 2.7.1.20; Adenosine 5'-phosphotransferase
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MAAAEEEPKPKKLKVEAPQALRENILFGMGNPLLDISAVVDKDFLDKYSLKPNDQILAED
KHKELFDELVKKFKVEYHAGGSTQNSIKVAQWMIQQPHKAATFFGCIGIDKFGEILKRKA
AEAHVDAHYYEQNEQPTGTCAACITGDNRSLIANLAAANCYKKEKHLDLEKNWMLVEKAR
VCYIAGFFLTVSPESVLKVAHHASENNRIFTLNLSAPFISQFYKESLMKVMPYVDILFGN
ETEAATFAREQGFETKDIKEIAKKTQALPKMNSKRQRIVIFTQGRDDTIMATESEVTAFA
VLDQDQKEIIDTNGAGDAFVGGFLSQLVSDKPLTECIRAGHYAASIIIRRTGCTFPEKPD
FH
Target Type
Clinical trial
Target Bioclass
Enzyme
Family
Carbohydrate kinase PfkB family
Subcellular location
Cytoplasm; Nucleus
Function
Catalyzes the phosphorylation of the purine nucleoside adenosine at the 5' position in an ATP-dependent manner. Serves as a potential regulator of concentrations of extracellular adenosine and intracellular adenine nucleotides.
TTD ID
T91661
Uniprot ID
P55263
DrugMap ID
TTL732K
Ensemble ID
ENST00000372734.5
HGNC ID
HGNC:257
ChEMBL ID
CHEMBL3589

Target Site Mutations in Different Cell Lines

Cell line Mutation details Probe for labeling this protein in this cell
HT115 SNV: p.E131K DBIA    Probe Info 
LS180 Deletion: p.I310del DBIA    Probe Info 
MELHO SNV: p.E260D DBIA    Probe Info 

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 28 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
m-APA
 Probe Info  		14.35  LDD0402  [1]
TH211
 Probe Info  		Y77(7.14)  LDD0260  [2]
IBr-1b
 Probe Info  		20.00  LDD0306  [3]
STPyne
 Probe Info  		K162(1.16); K256(9.72); K264(10.00); K72(5.56)  LDD0277  [4]
Probe 1
 Probe Info  		Y48(9.93)  LDD3495  [5]
Dasatinib-CA-4PAP
 Probe Info  		9.79  LDD0270  [6]
JZ128-DTB
 Probe Info  		N.A.  LDD0462  [7]
BTD
 Probe Info  		C353(1.74)  LDD1700  [8]
HHS-475
 Probe Info  		Y223(1.10)  LDD0264  [9]
DBIA
 Probe Info  		C353(1.28)  LDD0078  [10]
5E-2FA
 Probe Info  		H201(0.00); H202(0.00); H78(0.00)  LDD2235  [11]
ATP probe
 Probe Info  		K162(0.00); K163(0.00); K74(0.00)  LDD0199  [12]
4-Iodoacetamidophenylacetylene
 Probe Info  		C106(0.00); C336(0.00); C160(0.00); C353(0.00)  LDD0038  [13]
IA-alkyne
 Probe Info  		C106(0.00); C336(0.00); C353(0.00); C160(0.00)  LDD0036  [13]
IPIAA_H
 Probe Info  		N.A.  LDD0030  [14]
IPIAA_L
 Probe Info  		N.A.  LDD0031  [14]
Lodoacetamide azide
 Probe Info  		C106(0.00); C336(0.00); C160(0.00); C353(0.00)  LDD0037  [13]
JW-RF-010
 Probe Info  		N.A.  LDD0026  [15]
NAIA_4
 Probe Info  		C160(0.00); C336(0.00); 0.00  LDD2226  [16]
TFBX
 Probe Info  		C160(0.00); C143(0.00); C140(0.00); C353(0.00)  LDD0027  [15]
WYneN
 Probe Info  		N.A.  LDD0021  [17]
IPM
 Probe Info  		N.A.  LDD0005  [17]
NHS
 Probe Info  		N.A.  LDD0010  [17]
Phosphinate-6
 Probe Info  		N.A.  LDD0018  [18]
Acrolein
 Probe Info  		C160(0.00); C353(0.00); H201(0.00)  LDD0217  [19]
Methacrolein
 Probe Info  		C160(0.00); C353(0.00)  LDD0218  [19]
AOyne
 Probe Info  		15.00  LDD0443  [20]
NAIA_5
 Probe Info  		C106(0.00); C336(0.00); C353(0.00); C160(0.00)  LDD2223  [16]
PAL-AfBPP Probe
Click To Hide/Show 51 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
PARPYnD
 Probe Info  		2.44  LDD0374  [21]
C003
 Probe Info  		20.39  LDD1713  [22]
C006
 Probe Info  		6.23  LDD1715  [22]
C017
 Probe Info  		23.75  LDD1725  [22]
C027
 Probe Info  		7.67  LDD1733  [22]
C040
 Probe Info  		41.36  LDD1740  [22]
C055
 Probe Info  		45.57  LDD1752  [22]
C056
 Probe Info  		21.56  LDD1753  [22]
C063
 Probe Info  		20.97  LDD1760  [22]
C087
 Probe Info  		8.17  LDD1779  [22]
C091
 Probe Info  		10.63  LDD1782  [22]
C095
 Probe Info  		5.28  LDD1786  [22]
C131
 Probe Info  		16.68  LDD1813  [22]
C158
 Probe Info  		12.30  LDD1838  [22]
C166
 Probe Info  		11.63  LDD1846  [22]
C174
 Probe Info  		25.63  LDD1854  [22]
C187
 Probe Info  		20.11  LDD1865  [22]
C191
 Probe Info  		11.47  LDD1868  [22]
C199
 Probe Info  		15.14  LDD1875  [22]
C229
 Probe Info  		28.84  LDD1902  [22]
C232
 Probe Info  		42.81  LDD1905  [22]
C233
 Probe Info  		13.83  LDD1906  [22]
C235
 Probe Info  		53.82  LDD1908  [22]
C252
 Probe Info  		10.27  LDD1925  [22]
C266
 Probe Info  		10.20  LDD1937  [22]
C269
 Probe Info  		11.16  LDD1939  [22]
C270
 Probe Info  		16.11  LDD1940  [22]
C289
 Probe Info  		28.44  LDD1959  [22]
C292
 Probe Info  		7.73  LDD1962  [22]
C299
 Probe Info  		9.25  LDD1968  [22]
C303
 Probe Info  		8.63  LDD1972  [22]
C348
 Probe Info  		99.73  LDD2009  [22]
C353
 Probe Info  		7.41  LDD2014  [22]
C361
 Probe Info  		34.30  LDD2022  [22]
C364
 Probe Info  		14.83  LDD2025  [22]
C391
 Probe Info  		13.00  LDD2050  [22]
C399
 Probe Info  		7.62  LDD2058  [22]
C407
 Probe Info  		26.54  LDD2064  [22]
C413
 Probe Info  		17.15  LDD2069  [22]
C417
 Probe Info  		27.86  LDD2072  [22]
C420
 Probe Info  		21.71  LDD2075  [22]
C426
 Probe Info  		54.95  LDD2081  [22]
C433
 Probe Info  		5.66  LDD2088  [22]
FFF probe2
 Probe Info  		20.00  LDD0463  [23]
FFF probe3
 Probe Info  		20.00  LDD0465  [23]
FFF probe6
 Probe Info  		20.00  LDD0468  [23]
Dasatinib-CA-3PAP
 Probe Info  		4.39  LDD0365  [6]
Dasatinib-CA-8PAP
 Probe Info  		4.78  LDD0364  [6]
EN
 Probe Info  		1.82  LDD0418  [24]
DA-2
 Probe Info  		N.A.  LDD0070  [25]
STS-1
 Probe Info  		N.A.  LDD0069  [26]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0524  2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide MDA-MB-231 C353(1.16); C160(0.77)  LDD2117  [8]
 LDCM0558  2-Cyano-N-phenylacetamide MDA-MB-231 C353(1.00)  LDD2152  [8]
 LDCM0539  3-(4-Isopropylpiperazin-1-yl)-3-oxopropanenitrile MDA-MB-231 C353(0.39)  LDD2132  [8]
 LDCM0538  4-(Cyanoacetyl)morpholine MDA-MB-231 C353(0.62)  LDD2131  [8]
 LDCM0214  AC1 HCT 116 C160(0.84); C353(1.09)  LDD0531  [10]
 LDCM0215  AC10 HCT 116 C160(0.98); C353(1.12)  LDD0532  [10]
 LDCM0216  AC100 HCT 116 C353(1.11)  LDD0533  [10]
 LDCM0217  AC101 HCT 116 C353(1.08)  LDD0534  [10]
 LDCM0218  AC102 HCT 116 C353(0.97)  LDD0535  [10]
 LDCM0219  AC103 HCT 116 C353(1.18)  LDD0536  [10]
 LDCM0220  AC104 HCT 116 C353(0.99)  LDD0537  [10]
 LDCM0221  AC105 HCT 116 C353(1.13)  LDD0538  [10]
 LDCM0222  AC106 HCT 116 C353(1.17)  LDD0539  [10]
 LDCM0223  AC107 HCT 116 C353(1.02)  LDD0540  [10]
 LDCM0224  AC108 HCT 116 C353(0.98)  LDD0541  [10]
 LDCM0225  AC109 HCT 116 C353(0.85)  LDD0542  [10]
 LDCM0226  AC11 HCT 116 C160(1.16); C353(1.14)  LDD0543  [10]
 LDCM0227  AC110 HCT 116 C353(0.98)  LDD0544  [10]
 LDCM0228  AC111 HCT 116 C353(0.96)  LDD0545  [10]
 LDCM0229  AC112 HCT 116 C353(1.01)  LDD0546  [10]
 LDCM0230  AC113 HCT 116 C353(1.01)  LDD0547  [10]
 LDCM0231  AC114 HCT 116 C353(0.95)  LDD0548  [10]
 LDCM0232  AC115 HCT 116 C353(0.97)  LDD0549  [10]
 LDCM0233  AC116 HCT 116 C353(0.96)  LDD0550  [10]
 LDCM0234  AC117 HCT 116 C353(0.98)  LDD0551  [10]
 LDCM0235  AC118 HCT 116 C353(0.94)  LDD0552  [10]
 LDCM0236  AC119 HCT 116 C353(0.97)  LDD0553  [10]
 LDCM0237  AC12 HCT 116 C160(1.05); C353(0.97)  LDD0554  [10]
 LDCM0238  AC120 HCT 116 C353(0.87)  LDD0555  [10]
 LDCM0239  AC121 HCT 116 C353(0.88)  LDD0556  [10]
 LDCM0240  AC122 HCT 116 C353(0.98)  LDD0557  [10]
 LDCM0241  AC123 HCT 116 C353(0.90)  LDD0558  [10]
 LDCM0242  AC124 HCT 116 C353(0.85)  LDD0559  [10]
 LDCM0243  AC125 HCT 116 C353(0.88)  LDD0560  [10]
 LDCM0244  AC126 HCT 116 C353(0.92)  LDD0561  [10]
 LDCM0245  AC127 HCT 116 C353(0.90)  LDD0562  [10]
 LDCM0246  AC128 HCT 116 C160(0.68); C353(0.90)  LDD0563  [10]
 LDCM0247  AC129 HCT 116 C160(1.20); C353(1.17)  LDD0564  [10]
 LDCM0249  AC130 HCT 116 C160(0.96); C353(1.24)  LDD0566  [10]
 LDCM0250  AC131 HCT 116 C160(1.17); C353(1.01)  LDD0567  [10]
 LDCM0251  AC132 HCT 116 C160(1.20); C353(1.22)  LDD0568  [10]
 LDCM0252  AC133 HCT 116 C160(1.02); C353(1.17)  LDD0569  [10]
 LDCM0253  AC134 HCT 116 C160(1.05); C353(1.34)  LDD0570  [10]
 LDCM0254  AC135 HCT 116 C160(0.95); C353(1.02)  LDD0571  [10]
 LDCM0255  AC136 HCT 116 C160(1.00); C353(1.20)  LDD0572  [10]
 LDCM0256  AC137 HCT 116 C160(1.12); C353(1.35)  LDD0573  [10]
 LDCM0257  AC138 HCT 116 C160(1.04); C353(1.67)  LDD0574  [10]
 LDCM0258  AC139 HCT 116 C160(1.13); C353(1.34)  LDD0575  [10]
 LDCM0259  AC14 HCT 116 C160(1.03); C353(1.03)  LDD0576  [10]
 LDCM0260  AC140 HCT 116 C160(0.98); C353(1.63)  LDD0577  [10]
 LDCM0261  AC141 HCT 116 C160(1.12); C353(1.59)  LDD0578  [10]
 LDCM0262  AC142 HCT 116 C160(1.12); C353(1.36)  LDD0579  [10]
 LDCM0263  AC143 HCT 116 C160(0.92); C353(1.21)  LDD0580  [10]
 LDCM0264  AC144 HCT 116 C160(0.82); C353(1.49)  LDD0581  [10]
 LDCM0265  AC145 HCT 116 C160(0.86); C353(1.20)  LDD0582  [10]
 LDCM0266  AC146 HCT 116 C160(0.96); C353(1.29)  LDD0583  [10]
 LDCM0267  AC147 HCT 116 C160(0.75); C353(1.39)  LDD0584  [10]
 LDCM0268  AC148 HCT 116 C160(0.31); C353(1.71)  LDD0585  [10]
 LDCM0269  AC149 HCT 116 C160(0.75); C353(1.52)  LDD0586  [10]
 LDCM0270  AC15 HCT 116 C160(1.01); C353(1.03)  LDD0587  [10]
 LDCM0271  AC150 HCT 116 C160(1.06); C353(1.18)  LDD0588  [10]
 LDCM0272  AC151 HCT 116 C160(1.05); C353(1.17)  LDD0589  [10]
 LDCM0273  AC152 HCT 116 C160(0.68); C353(1.23)  LDD0590  [10]
 LDCM0274  AC153 HCT 116 C160(0.22); C353(2.08)  LDD0591  [10]
 LDCM0621  AC154 HCT 116 C160(0.83); C353(1.29)  LDD2158  [10]
 LDCM0622  AC155 HCT 116 C160(0.87); C353(1.15)  LDD2159  [10]
 LDCM0623  AC156 HCT 116 C160(0.92); C353(1.00)  LDD2160  [10]
 LDCM0624  AC157 HCT 116 C160(0.97); C353(0.93)  LDD2161  [10]
 LDCM0276  AC17 HCT 116 C353(1.10); C160(1.11)  LDD0593  [10]
 LDCM0277  AC18 HCT 116 C160(0.97); C353(1.20)  LDD0594  [10]
 LDCM0278  AC19 HCT 116 C353(1.09); C160(1.26)  LDD0595  [10]
 LDCM0279  AC2 HCT 116 C160(0.92); C353(1.11)  LDD0596  [10]
 LDCM0280  AC20 HCT 116 C160(1.15); C353(1.16)  LDD0597  [10]
 LDCM0281  AC21 HCT 116 C160(0.98); C353(1.10)  LDD0598  [10]
 LDCM0282  AC22 HCT 116 C160(1.11); C353(1.12)  LDD0599  [10]
 LDCM0283  AC23 HCT 116 C160(1.01); C353(1.08)  LDD0600  [10]
 LDCM0284  AC24 HCT 116 C353(1.00); C160(1.08)  LDD0601  [10]
 LDCM0285  AC25 HCT 116 C353(1.05)  LDD0602  [10]
 LDCM0286  AC26 HCT 116 C353(1.18)  LDD0603  [10]
 LDCM0287  AC27 HCT 116 C353(1.05)  LDD0604  [10]
 LDCM0288  AC28 HCT 116 C353(1.03)  LDD0605  [10]
 LDCM0289  AC29 HCT 116 C353(1.14)  LDD0606  [10]
 LDCM0290  AC3 HCT 116 C160(0.93); C353(1.16)  LDD0607  [10]
 LDCM0291  AC30 HCT 116 C353(1.18)  LDD0608  [10]
 LDCM0292  AC31 HCT 116 C353(1.16)  LDD0609  [10]
 LDCM0293  AC32 HCT 116 C353(1.43)  LDD0610  [10]
 LDCM0294  AC33 HCT 116 C353(1.18)  LDD0611  [10]
 LDCM0295  AC34 HCT 116 C353(1.17)  LDD0612  [10]
 LDCM0296  AC35 HCT 116 C160(0.88); C353(0.88); C106(1.42)  LDD0613  [10]
 LDCM0297  AC36 HCT 116 C353(0.92); C160(0.96); C106(1.16)  LDD0614  [10]
 LDCM0298  AC37 HCT 116 C353(0.89); C160(0.92); C106(1.30)  LDD0615  [10]
 LDCM0299  AC38 HCT 116 C353(0.93); C160(0.94); C106(1.16)  LDD0616  [10]
 LDCM0300  AC39 HCT 116 C160(0.85); C353(0.97); C106(0.98)  LDD0617  [10]
 LDCM0301  AC4 HCT 116 C160(0.93); C353(1.21)  LDD0618  [10]
 LDCM0302  AC40 HCT 116 C106(0.88); C353(0.97); C160(1.21)  LDD0619  [10]
 LDCM0303  AC41 HCT 116 C353(0.96); C160(0.99); C106(1.14)  LDD0620  [10]
 LDCM0304  AC42 HCT 116 C353(0.95); C106(1.02); C160(1.08)  LDD0621  [10]
 LDCM0305  AC43 HCT 116 C160(1.02); C353(1.02); C106(1.15)  LDD0622  [10]
 LDCM0306  AC44 HCT 116 C353(0.91); C106(0.95); C160(1.12)  LDD0623  [10]
 LDCM0307  AC45 HCT 116 C106(0.73); C353(0.99); C160(1.01)  LDD0624  [10]
 LDCM0308  AC46 HCT 116 C106(0.98); C160(1.02); C353(1.15)  LDD0625  [10]
 LDCM0309  AC47 HCT 116 C106(0.86); C160(0.98); C353(1.20)  LDD0626  [10]
 LDCM0310  AC48 HCT 116 C160(0.92); C106(0.98); C353(1.32)  LDD0627  [10]
 LDCM0311  AC49 HCT 116 C106(0.33); C160(0.69); C353(1.38)  LDD0628  [10]
 LDCM0312  AC5 HCT 116 C160(0.91); C353(1.33)  LDD0629  [10]
 LDCM0313  AC50 HCT 116 C106(0.44); C160(0.78); C353(1.41)  LDD0630  [10]
 LDCM0314  AC51 HCT 116 C160(0.98); C353(1.01); C106(1.28)  LDD0631  [10]
 LDCM0315  AC52 HCT 116 C106(0.94); C160(1.05); C353(1.25)  LDD0632  [10]
 LDCM0316  AC53 HCT 116 C106(0.60); C160(0.96); C353(1.14)  LDD0633  [10]
 LDCM0317  AC54 HCT 116 C106(0.61); C160(0.83); C353(1.14)  LDD0634  [10]
 LDCM0318  AC55 HCT 116 C106(0.33); C160(0.81); C353(1.51)  LDD0635  [10]
 LDCM0319  AC56 HCT 116 C106(0.14); C160(0.59); C353(2.26)  LDD0636  [10]
 LDCM0320  AC57 HCT 116 C106(0.78); C160(0.98); C353(1.37)  LDD0637  [10]
 LDCM0321  AC58 HCT 116 C106(0.80); C160(1.04); C353(1.55)  LDD0638  [10]
 LDCM0322  AC59 HCT 116 C106(0.62); C160(0.99); C353(1.59)  LDD0639  [10]
 LDCM0323  AC6 HCT 116 C160(0.85); C353(1.26)  LDD0640  [10]
 LDCM0324  AC60 HCT 116 C160(0.92); C106(0.92); C353(1.44)  LDD0641  [10]
 LDCM0325  AC61 HCT 116 C106(0.88); C160(0.93); C353(1.51)  LDD0642  [10]
 LDCM0326  AC62 HCT 116 C106(0.56); C160(0.83); C353(1.97)  LDD0643  [10]
 LDCM0327  AC63 HCT 116 C106(0.81); C160(0.84); C353(1.32)  LDD0644  [10]
 LDCM0328  AC64 HCT 116 C106(0.59); C160(0.92); C353(1.79)  LDD0645  [10]
 LDCM0329  AC65 HCT 116 C106(0.90); C160(0.97); C353(1.73)  LDD0646  [10]
 LDCM0330  AC66 HCT 116 C106(0.99); C160(1.00); C353(1.65)  LDD0647  [10]
 LDCM0331  AC67 HCT 116 C106(0.24); C160(1.07); C353(2.12)  LDD0648  [10]
 LDCM0332  AC68 HCT 116 C106(0.86); C160(0.93); C353(1.16)  LDD0649  [10]
 LDCM0333  AC69 HCT 116 C106(0.69); C160(0.90); C353(1.14)  LDD0650  [10]
 LDCM0334  AC7 HCT 116 C160(0.94); C353(0.99)  LDD0651  [10]
 LDCM0335  AC70 HCT 116 C106(0.39); C160(0.43); C353(1.37)  LDD0652  [10]
 LDCM0336  AC71 HCT 116 C106(1.09); C353(1.12); C160(1.25)  LDD0653  [10]
 LDCM0337  AC72 HCT 116 C106(0.71); C160(0.83); C353(1.28)  LDD0654  [10]
 LDCM0338  AC73 HCT 116 C160(0.22); C106(0.22); C353(1.81)  LDD0655  [10]
 LDCM0339  AC74 HCT 116 C160(0.27); C106(0.28); C353(1.64)  LDD0656  [10]
 LDCM0340  AC75 HCT 116 C106(0.13); C160(0.13); C353(2.34)  LDD0657  [10]
 LDCM0341  AC76 HCT 116 C106(0.55); C160(0.56); C353(1.33)  LDD0658  [10]
 LDCM0342  AC77 HCT 116 C106(0.54); C160(0.59); C353(1.41)  LDD0659  [10]
 LDCM0343  AC78 HCT 116 C106(0.91); C160(1.13); C353(1.16)  LDD0660  [10]
 LDCM0344  AC79 HCT 116 C106(0.94); C160(0.98); C353(1.19)  LDD0661  [10]
 LDCM0345  AC8 HCT 116 C160(0.88); C353(1.02)  LDD0662  [10]
 LDCM0346  AC80 HCT 116 C106(0.72); C160(0.75); C353(1.18)  LDD0663  [10]
 LDCM0347  AC81 HCT 116 C106(0.79); C353(1.07); C160(1.10)  LDD0664  [10]
 LDCM0348  AC82 HCT 116 C106(0.10); C160(0.10); C353(2.45)  LDD0665  [10]
 LDCM0349  AC83 HCT 116 C160(0.85); C353(1.27)  LDD0666  [10]
 LDCM0350  AC84 HCT 116 C160(0.86); C353(1.21)  LDD0667  [10]
 LDCM0351  AC85 HCT 116 C160(1.08); C353(1.28)  LDD0668  [10]
 LDCM0352  AC86 HCT 116 C160(1.05); C353(1.22)  LDD0669  [10]
 LDCM0353  AC87 HCT 116 C160(0.93); C353(1.14)  LDD0670  [10]
 LDCM0354  AC88 HCT 116 C160(1.01); C353(1.22)  LDD0671  [10]
 LDCM0355  AC89 HCT 116 C160(0.95); C353(1.20)  LDD0672  [10]
 LDCM0357  AC90 HCT 116 C160(1.23); C353(1.34)  LDD0674  [10]
 LDCM0358  AC91 HCT 116 C160(0.85); C353(1.18)  LDD0675  [10]
 LDCM0359  AC92 HCT 116 C160(0.88); C353(1.26)  LDD0676  [10]
 LDCM0360  AC93 HCT 116 C160(0.77); C353(1.17)  LDD0677  [10]
 LDCM0361  AC94 HCT 116 C160(0.74); C353(1.09)  LDD0678  [10]
 LDCM0362  AC95 HCT 116 C160(0.83); C353(1.19)  LDD0679  [10]
 LDCM0363  AC96 HCT 116 C160(0.94); C353(1.04)  LDD0680  [10]
 LDCM0364  AC97 HCT 116 C160(0.81); C353(1.33)  LDD0681  [10]
 LDCM0365  AC98 HCT 116 C353(1.89)  LDD0682  [10]
 LDCM0366  AC99 HCT 116 C353(1.09)  LDD0683  [10]
 LDCM0545  Acetamide MDA-MB-231 C353(0.59)  LDD2138  [8]
 LDCM0248  AKOS034007472 HCT 116 C160(1.12); C353(0.94)  LDD0565  [10]
 LDCM0356  AKOS034007680 HCT 116 C160(1.08); C353(1.12)  LDD0673  [10]
 LDCM0275  AKOS034007705 HCT 116 C160(0.89); C353(1.57)  LDD0592  [10]
 LDCM0156  Aniline NCI-H1299 13.77  LDD0403  [1]
 LDCM0020  ARS-1620 HCC44 C353(1.28)  LDD0078  [10]
 LDCM0103  BDHI 10 Jurkat C353(4.78)  LDD0205  [27]
 LDCM0498  BS-3668 MDA-MB-231 C353(0.60)  LDD2091  [8]
 LDCM0630  CCW28-3 231MFP C353(1.11)  LDD2214  [28]
 LDCM0108  Chloroacetamide HeLa C353(0.00); H201(0.00); C106(0.00); C160(0.00)  LDD0222  [19]
 LDCM0632  CL-Sc Hep-G2 C160(0.85); C353(0.80); C353(0.71)  LDD2227  [16]
 LDCM0367  CL1 HCT 116 C353(0.83); C160(1.00)  LDD0684  [10]
 LDCM0368  CL10 HCT 116 C160(0.83); C353(1.20)  LDD0685  [10]
 LDCM0369  CL100 HCT 116 C160(0.86); C353(1.23)  LDD0686  [10]
 LDCM0370  CL101 HCT 116 C160(0.97); C353(1.11)  LDD0687  [10]
 LDCM0371  CL102 HCT 116 C353(0.87); C160(0.89)  LDD0688  [10]
 LDCM0372  CL103 HCT 116 C353(0.89); C160(1.03)  LDD0689  [10]
 LDCM0373  CL104 HCT 116 C160(0.90); C353(0.98)  LDD0690  [10]
 LDCM0374  CL105 HCT 116 C160(1.11); C353(1.22)  LDD0691  [10]
 LDCM0375  CL106 HCT 116 C160(1.26); C353(1.62)  LDD0692  [10]
 LDCM0376  CL107 HCT 116 C160(1.12); C353(1.52)  LDD0693  [10]
 LDCM0377  CL108 HCT 116 C160(1.15); C353(1.43)  LDD0694  [10]
 LDCM0378  CL109 HCT 116 C160(1.03); C353(1.19)  LDD0695  [10]
 LDCM0379  CL11 HCT 116 C160(0.93); C353(1.14)  LDD0696  [10]
 LDCM0380  CL110 HCT 116 C160(0.95); C353(1.19)  LDD0697  [10]
 LDCM0381  CL111 HCT 116 C160(0.99); C353(1.13)  LDD0698  [10]
 LDCM0382  CL112 HCT 116 C353(0.85)  LDD0699  [10]
 LDCM0383  CL113 HCT 116 C353(1.22)  LDD0700  [10]
 LDCM0384  CL114 HCT 116 C353(1.06)  LDD0701  [10]
 LDCM0385  CL115 HCT 116 C353(1.03)  LDD0702  [10]
 LDCM0386  CL116 HCT 116 C353(1.10)  LDD0703  [10]
 LDCM0387  CL117 HCT 116 C106(0.31); C353(1.20); C160(1.31)  LDD0704  [10]
 LDCM0388  CL118 HCT 116 C106(0.88); C160(0.93); C353(1.01)  LDD0705  [10]
 LDCM0389  CL119 HCT 116 C106(0.88); C160(0.94); C353(0.98)  LDD0706  [10]
 LDCM0390  CL12 HCT 116 C160(0.96); C353(1.45)  LDD0707  [10]
 LDCM0391  CL120 HCT 116 C160(0.94); C353(1.02); C106(1.11)  LDD0708  [10]
 LDCM0392  CL121 HCT 116 C106(0.78); C353(0.79); C160(0.83)  LDD0709  [10]
 LDCM0393  CL122 HCT 116 C106(0.82); C160(0.97); C353(1.16)  LDD0710  [10]
 LDCM0394  CL123 HCT 116 C106(0.60); C160(0.69); C353(1.47)  LDD0711  [10]
 LDCM0395  CL124 HCT 116 C106(0.46); C160(0.77); C353(1.36)  LDD0712  [10]
 LDCM0396  CL125 HCT 116 C160(1.00); C106(1.03); C353(1.14)  LDD0713  [10]
 LDCM0397  CL126 HCT 116 C160(0.93); C106(1.06); C353(1.14)  LDD0714  [10]
 LDCM0398  CL127 HCT 116 C160(0.96); C106(1.01); C353(1.23)  LDD0715  [10]
 LDCM0399  CL128 HCT 116 C106(0.72); C160(0.97); C353(1.50)  LDD0716  [10]
 LDCM0400  CL13 HCT 116 C160(0.96); C353(0.97)  LDD0717  [10]
 LDCM0401  CL14 HCT 116 C353(0.90); C160(1.09)  LDD0718  [10]
 LDCM0402  CL15 HCT 116 C353(1.02); C160(1.06)  LDD0719  [10]
 LDCM0403  CL16 HCT 116 C353(1.01); C160(1.24)  LDD0720  [10]
 LDCM0404  CL17 HCT 116 C353(1.00)  LDD0721  [10]
 LDCM0405  CL18 HCT 116 C353(1.08)  LDD0722  [10]
 LDCM0406  CL19 HCT 116 C353(0.99)  LDD0723  [10]
 LDCM0407  CL2 HCT 116 C353(0.94); C160(1.01)  LDD0724  [10]
 LDCM0408  CL20 HCT 116 C353(1.15)  LDD0725  [10]
 LDCM0409  CL21 HCT 116 C353(1.12)  LDD0726  [10]
 LDCM0410  CL22 HCT 116 C353(1.52)  LDD0727  [10]
 LDCM0411  CL23 HCT 116 C353(0.99)  LDD0728  [10]
 LDCM0412  CL24 HCT 116 C353(1.27)  LDD0729  [10]
 LDCM0413  CL25 HCT 116 C353(1.19)  LDD0730  [10]
 LDCM0414  CL26 HCT 116 C353(1.10)  LDD0731  [10]
 LDCM0415  CL27 HCT 116 C353(1.12)  LDD0732  [10]
 LDCM0416  CL28 HCT 116 C353(1.15)  LDD0733  [10]
 LDCM0417  CL29 HCT 116 C353(1.15)  LDD0734  [10]
 LDCM0418  CL3 HCT 116 C160(1.00); C353(0.94)  LDD0735  [10]
 LDCM0419  CL30 HCT 116 C353(1.00)  LDD0736  [10]
 LDCM0420  CL31 HCT 116 C160(0.91); C353(1.01)  LDD0737  [10]
 LDCM0421  CL32 HCT 116 C160(0.75); C353(1.23)  LDD0738  [10]
 LDCM0422  CL33 HCT 116 C160(0.75); C353(1.10)  LDD0739  [10]
 LDCM0423  CL34 HCT 116 C160(0.66); C353(1.40)  LDD0740  [10]
 LDCM0424  CL35 HCT 116 C160(0.74); C353(1.41)  LDD0741  [10]
 LDCM0425  CL36 HCT 116 C160(0.80); C353(1.24)  LDD0742  [10]
 LDCM0426  CL37 HCT 116 C160(0.72); C353(1.36)  LDD0743  [10]
 LDCM0428  CL39 HCT 116 C160(0.80); C353(1.37)  LDD0745  [10]
 LDCM0429  CL4 HCT 116 C160(0.91); C353(0.82)  LDD0746  [10]
 LDCM0430  CL40 HCT 116 C160(0.74); C353(1.20)  LDD0747  [10]
 LDCM0431  CL41 HCT 116 C160(0.81); C353(1.24)  LDD0748  [10]
 LDCM0432  CL42 HCT 116 C160(0.51); C353(1.88)  LDD0749  [10]
 LDCM0433  CL43 HCT 116 C160(0.72); C353(1.53)  LDD0750  [10]
 LDCM0434  CL44 HCT 116 C160(0.77); C353(1.30)  LDD0751  [10]
 LDCM0435  CL45 HCT 116 C160(0.70); C353(1.39)  LDD0752  [10]
 LDCM0436  CL46 HCT 116 C160(1.19); C353(0.99)  LDD0753  [10]
 LDCM0437  CL47 HCT 116 C160(0.93); C353(0.90)  LDD0754  [10]
 LDCM0438  CL48 HCT 116 C160(1.26); C353(0.94)  LDD0755  [10]
 LDCM0439  CL49 HCT 116 C160(1.30); C353(0.90)  LDD0756  [10]
 LDCM0440  CL5 HCT 116 C160(1.03); C353(1.05)  LDD0757  [10]
 LDCM0441  CL50 HCT 116 C160(1.25); C353(0.87)  LDD0758  [10]
 LDCM0442  CL51 HCT 116 C160(1.14); C353(0.95)  LDD0759  [10]
 LDCM0443  CL52 HCT 116 C160(1.18); C353(0.95)  LDD0760  [10]
 LDCM0444  CL53 HCT 116 C160(0.73); C353(0.79)  LDD0761  [10]
 LDCM0445  CL54 HCT 116 C160(1.03); C353(0.89)  LDD0762  [10]
 LDCM0446  CL55 HCT 116 C160(1.02); C353(0.85)  LDD0763  [10]
 LDCM0447  CL56 HCT 116 C160(1.05); C353(0.97)  LDD0764  [10]
 LDCM0448  CL57 HCT 116 C160(0.97); C353(0.83)  LDD0765  [10]
 LDCM0449  CL58 HCT 116 C160(1.16); C353(0.85)  LDD0766  [10]
 LDCM0450  CL59 HCT 116 C160(1.08); C353(0.87)  LDD0767  [10]
 LDCM0451  CL6 HCT 116 C160(0.92); C353(0.93)  LDD0768  [10]
 LDCM0452  CL60 HCT 116 C160(1.15); C353(0.94)  LDD0769  [10]
 LDCM0453  CL61 HCT 116 C353(1.10)  LDD0770  [10]
 LDCM0454  CL62 HCT 116 C353(1.12)  LDD0771  [10]
 LDCM0455  CL63 HCT 116 C353(1.19)  LDD0772  [10]
 LDCM0456  CL64 HCT 116 C353(1.41)  LDD0773  [10]
 LDCM0457  CL65 HCT 116 C353(1.07)  LDD0774  [10]
 LDCM0458  CL66 HCT 116 C353(1.47)  LDD0775  [10]
 LDCM0459  CL67 HCT 116 C353(1.22)  LDD0776  [10]
 LDCM0460  CL68 HCT 116 C353(1.13)  LDD0777  [10]
 LDCM0461  CL69 HCT 116 C353(1.01)  LDD0778  [10]
 LDCM0462  CL7 HCT 116 C160(1.02); C353(1.10)  LDD0779  [10]
 LDCM0463  CL70 HCT 116 C353(1.17)  LDD0780  [10]
 LDCM0464  CL71 HCT 116 C353(1.16)  LDD0781  [10]
 LDCM0465  CL72 HCT 116 C353(1.07)  LDD0782  [10]
 LDCM0466  CL73 HCT 116 C353(1.18)  LDD0783  [10]
 LDCM0467  CL74 HCT 116 C353(1.19)  LDD0784  [10]
 LDCM0469  CL76 HCT 116 C160(0.86); C353(1.17)  LDD0786  [10]
 LDCM0470  CL77 HCT 116 C160(0.77); C353(0.95)  LDD0787  [10]
 LDCM0471  CL78 HCT 116 C160(1.03); C353(1.33)  LDD0788  [10]
 LDCM0472  CL79 HCT 116 C160(0.86); C353(1.33)  LDD0789  [10]
 LDCM0473  CL8 HCT 116 C160(0.85); C353(1.05)  LDD0790  [10]
 LDCM0474  CL80 HCT 116 C160(1.04); C353(1.05)  LDD0791  [10]
 LDCM0475  CL81 HCT 116 C160(1.02); C353(1.17)  LDD0792  [10]
 LDCM0476  CL82 HCT 116 C160(0.69); C353(1.56)  LDD0793  [10]
 LDCM0477  CL83 HCT 116 C160(0.70); C353(1.63)  LDD0794  [10]
 LDCM0478  CL84 HCT 116 C160(0.55); C353(2.16)  LDD0795  [10]
 LDCM0479  CL85 HCT 116 C160(0.78); C353(1.22)  LDD0796  [10]
 LDCM0480  CL86 HCT 116 C160(0.97); C353(1.13)  LDD0797  [10]
 LDCM0481  CL87 HCT 116 C160(0.87); C353(1.23)  LDD0798  [10]
 LDCM0482  CL88 HCT 116 C160(0.68); C353(1.41)  LDD0799  [10]
 LDCM0483  CL89 HCT 116 C160(0.67); C353(2.58)  LDD0800  [10]
 LDCM0484  CL9 HCT 116 C160(1.00); C353(1.05)  LDD0801  [10]
 LDCM0485  CL90 HCT 116 C160(0.82); C353(0.90)  LDD0802  [10]
 LDCM0486  CL91 HCT 116 C160(0.85); C353(1.08)  LDD0803  [10]
 LDCM0487  CL92 HCT 116 C160(0.88); C353(0.91)  LDD0804  [10]
 LDCM0488  CL93 HCT 116 C160(0.99); C353(1.04)  LDD0805  [10]
 LDCM0489  CL94 HCT 116 C160(0.92); C353(1.09)  LDD0806  [10]
 LDCM0490  CL95 HCT 116 C160(0.91); C353(1.12)  LDD0807  [10]
 LDCM0491  CL96 HCT 116 C160(0.94); C353(1.01)  LDD0808  [10]
 LDCM0492  CL97 HCT 116 C160(0.85); C353(1.11)  LDD0809  [10]
 LDCM0493  CL98 HCT 116 C160(0.86); C353(1.21)  LDD0810  [10]
 LDCM0494  CL99 HCT 116 C160(0.87); C353(1.13)  LDD0811  [10]
 LDCM0182  Compound 18 HEK-293T 9.22  LDD0501  [23]
 LDCM0191  Compound 21 HEK-293T 6.13  LDD0493  [23]
 LDCM0190  Compound 34 HEK-293T 14.93  LDD0497  [23]
 LDCM0193  Compound 36 HEK-293T 5.99  LDD0494  [23]
 LDCM0196  Compound 39 HEK-293T 10.64  LDD0496  [23]
 LDCM0197  Compound 40 HEK-293T 10.47  LDD0495  [23]
 LDCM0181  Compound 41 HEK-293T 6.67  LDD0502  [23]
 LDCM0634  CY-0357 Hep-G2 C353(1.03)  LDD2228  [16]
 LDCM0097  Dasatinib K562 9.79  LDD0270  [6]
 LDCM0495  E2913 HEK-293T C353(0.97); C336(1.10); C160(1.07); C140(1.02)  LDD1698  [29]
 LDCM0213  Electrophilic fragment 2 MDA-MB-231 C160(1.54); C353(1.18)  LDD1702  [8]
 LDCM0163  Entinostat Hep-G2 1.82  LDD0418  [24]
 LDCM0625  F8 Ramos C353(1.54); C160(0.92)  LDD2187  [30]
 LDCM0572  Fragment10 MDA-MB-231 C353(1.45)  LDD1389  [31]
 LDCM0573  Fragment11 MDA-MB-231 C353(1.02)  LDD1391  [31]
 LDCM0574  Fragment12 MDA-MB-231 C353(1.13)  LDD1393  [31]
 LDCM0575  Fragment13 MDA-MB-231 C353(0.97)  LDD1395  [31]
 LDCM0576  Fragment14 MDA-MB-231 C353(1.33)  LDD1397  [31]
 LDCM0577  Fragment15 MDA-MB-231 C353(3.65)  LDD1399  [31]
 LDCM0579  Fragment20 MDA-MB-231 C353(1.51)  LDD1402  [31]
 LDCM0580  Fragment21 MDA-MB-231 C353(0.90)  LDD1404  [31]
 LDCM0581  Fragment22 MDA-MB-231 C353(0.99)  LDD1406  [31]
 LDCM0582  Fragment23 Ramos C353(2.15)  LDD2196  [30]
 LDCM0583  Fragment24 Ramos C353(1.04)  LDD1410  [31]
 LDCM0584  Fragment25 MDA-MB-231 C353(1.04)  LDD1411  [31]
 LDCM0585  Fragment26 Ramos C353(0.91)  LDD1412  [31]
 LDCM0578  Fragment27 MDA-MB-231 C353(0.93)  LDD1401  [31]
 LDCM0586  Fragment28 MDA-MB-231 C353(0.94)  LDD1415  [31]
 LDCM0587  Fragment29 MDA-MB-231 C353(1.01)  LDD1417  [31]
 LDCM0588  Fragment30 MDA-MB-231 C353(0.76)  LDD1419  [31]
 LDCM0589  Fragment31 MDA-MB-231 C353(2.48)  LDD1421  [31]
 LDCM0590  Fragment32 MDA-MB-231 C353(1.73)  LDD1423  [31]
 LDCM0468  Fragment33 HCT 116 C353(1.12)  LDD0785  [10]
 LDCM0592  Fragment34 MDA-MB-231 C353(0.75)  LDD1427  [31]
 LDCM0593  Fragment35 MDA-MB-231 C353(0.79)  LDD1429  [31]
 LDCM0595  Fragment37 Ramos C353(1.12)  LDD1432  [31]
 LDCM0596  Fragment38 MDA-MB-231 C353(1.21)  LDD1433  [31]
 LDCM0597  Fragment39 MDA-MB-231 C353(1.17)  LDD1435  [31]
 LDCM0566  Fragment4 MDA-MB-231 C353(1.19)  LDD1378  [31]
 LDCM0598  Fragment40 MDA-MB-231 C353(0.81)  LDD1436  [31]
 LDCM0599  Fragment41 MDA-MB-231 C353(1.28)  LDD1438  [31]
 LDCM0600  Fragment42 Ramos C353(1.10)  LDD1440  [31]
 LDCM0601  Fragment43 MDA-MB-231 C353(0.96)  LDD1441  [31]
 LDCM0602  Fragment44 MDA-MB-231 C353(0.79)  LDD1443  [31]
 LDCM0603  Fragment45 MDA-MB-231 C353(2.05)  LDD1444  [31]
 LDCM0604  Fragment46 MDA-MB-231 C353(0.82)  LDD1445  [31]
 LDCM0605  Fragment47 MDA-MB-231 C353(1.39)  LDD1446  [31]
 LDCM0607  Fragment49 MDA-MB-231 C353(1.61)  LDD1448  [31]
 LDCM0608  Fragment50 MDA-MB-231 C353(14.39)  LDD1449  [31]
 LDCM0427  Fragment51 HCT 116 C160(0.57); C353(1.73)  LDD0744  [10]
 LDCM0610  Fragment52 MDA-MB-231 C353(1.16)  LDD1452  [31]
 LDCM0611  Fragment53 MDA-MB-231 C353(0.92)  LDD1454  [31]
 LDCM0612  Fragment54 MDA-MB-231 C353(1.03)  LDD1456  [31]
 LDCM0613  Fragment55 MDA-MB-231 C353(0.88)  LDD1457  [31]
 LDCM0614  Fragment56 MDA-MB-231 C353(0.87)  LDD1458  [31]
 LDCM0569  Fragment7 Ramos C353(4.56)  LDD1384  [31]
 LDCM0570  Fragment8 MDA-MB-231 C353(0.97)  LDD1385  [31]
 LDCM0571  Fragment9 MDA-MB-231 C353(0.99)  LDD1387  [31]
 LDCM0116  HHS-0101 DM93 Y223(1.10)  LDD0264  [9]
 LDCM0117  HHS-0201 DM93 Y223(0.41)  LDD0265  [9]
 LDCM0118  HHS-0301 DM93 Y223(0.30)  LDD0266  [9]
 LDCM0119  HHS-0401 DM93 Y223(0.49)  LDD0267  [9]
 LDCM0120  HHS-0701 DM93 Y223(1.02)  LDD0268  [9]
 LDCM0107  IAA HeLa C160(0.00); H78(0.00); H201(0.00); H202(0.00)  LDD0221  [19]
 LDCM0179  JZ128 PC-3 N.A.  LDD0462  [7]
 LDCM0022  KB02 MDA-MB-231 C353(2.61)  LDD1374  [31]
 LDCM0023  KB03 Jurkat C353(5.21)  LDD0315  [32]
 LDCM0024  KB05 G361 C89(1.58); C160(1.22)  LDD3311  [33]
 LDCM0109  NEM HeLa H78(0.00); H201(0.00); H341(0.00)  LDD0223  [19]
 LDCM0496  Nucleophilic fragment 11a MDA-MB-231 C353(0.67)  LDD2089  [8]
 LDCM0500  Nucleophilic fragment 13a MDA-MB-231 C353(1.02)  LDD2093  [8]
 LDCM0505  Nucleophilic fragment 15b MDA-MB-231 C353(0.97)  LDD2098  [8]
 LDCM0506  Nucleophilic fragment 16a MDA-MB-231 C353(1.01)  LDD2099  [8]
 LDCM0507  Nucleophilic fragment 16b MDA-MB-231 C353(0.92)  LDD2100  [8]
 LDCM0511  Nucleophilic fragment 18b MDA-MB-231 C353(1.09)  LDD2104  [8]
 LDCM0514  Nucleophilic fragment 20a MDA-MB-231 C353(0.82); C160(0.71)  LDD2107  [8]
 LDCM0518  Nucleophilic fragment 22a MDA-MB-231 C353(1.00)  LDD2111  [8]
 LDCM0525  Nucleophilic fragment 25b MDA-MB-231 C353(0.49)  LDD2118  [8]
 LDCM0526  Nucleophilic fragment 26a MDA-MB-231 C353(2.35)  LDD2119  [8]
 LDCM0532  Nucleophilic fragment 29a MDA-MB-231 C353(0.83)  LDD2125  [8]
 LDCM0533  Nucleophilic fragment 29b MDA-MB-231 C353(0.44)  LDD2126  [8]
 LDCM0536  Nucleophilic fragment 31 MDA-MB-231 C353(1.03)  LDD2129  [8]
 LDCM0541  Nucleophilic fragment 36 MDA-MB-231 C353(0.45)  LDD2134  [8]
 LDCM0542  Nucleophilic fragment 37 MDA-MB-231 C353(1.26)  LDD2135  [8]
 LDCM0543  Nucleophilic fragment 38 MDA-MB-231 C353(1.29)  LDD2136  [8]
 LDCM0544  Nucleophilic fragment 39 MDA-MB-231 C353(1.17)  LDD2137  [8]
 LDCM0211  Nucleophilic fragment 3b MDA-MB-231 C353(1.74)  LDD1700  [8]
 LDCM0546  Nucleophilic fragment 40 MDA-MB-231 C353(0.80)  LDD2140  [8]
 LDCM0547  Nucleophilic fragment 41 MDA-MB-231 C353(0.78)  LDD2141  [8]
 LDCM0549  Nucleophilic fragment 43 MDA-MB-231 C353(1.11)  LDD2143  [8]
 LDCM0550  Nucleophilic fragment 5a MDA-MB-231 C353(1.89)  LDD2144  [8]
 LDCM0551  Nucleophilic fragment 5b MDA-MB-231 C106(0.40)  LDD2145  [8]
 LDCM0552  Nucleophilic fragment 6a MDA-MB-231 C353(1.29)  LDD2146  [8]
 LDCM0554  Nucleophilic fragment 7a MDA-MB-231 C353(0.64)  LDD2148  [8]
 LDCM0627  NUDT7-COV-1 HEK-293T C353(1.01); C353(0.31)  LDD2206  [34]
 LDCM0628  OTUB2-COV-1 HEK-293T C353(1.43); C353(0.82)  LDD2207  [34]
 LDCM0131  RA190 MM1.R C353(1.12)  LDD0304  [35]
 LDCM0021  THZ1 HCT 116 C353(1.15)  LDD2173  [10]

The Interaction Atlas With This Target

The Drug(s) Related To This Target

Approved
Click To Hide/Show 4 Drug(s) Interacting with This Target
Drug Name Drug Type External ID
Abacavir Small molecular drug DB01048
Adenosine Small molecular drug DB00640
Adenosine Phosphate Small molecular drug DB00131
Ribavirin Small molecular drug DB00811
Phase 1
Click To Hide/Show 1 Drug(s) Interacting with This Target
Drug Name Drug Type External ID
Gp-3269 . D01GVC
Investigative
Click To Hide/Show 9 Drug(s) Interacting with This Target
Drug Name Drug Type External ID
5'-iodotubercidin Small molecular drug D00RDY
5-iodo,5'-deoxytubercidin Small molecular drug D03SHX
6-benzylthioinosine Small molecular drug D0K1YY
7-(5-deoxy-beta-d-ribofuranosyl)-5-iodo-7h-pyrrolo[23-d]Pyrimidin-4-amine Small molecular drug DB07173
Atp Small molecular drug DB00171
Gp515 Small molecular drug D07OAC
Iodotubercidin Small molecular drug D0S2FW
5-[4-(Dimethylamino)Phenyl]-6-[(6-morpholin-4-ylpyridin-3-yl)Ethynyl]Pyrimidin-4-amine . DB07280
Mb-03966 . D00WHC
Discontinued
Click To Hide/Show 3 Drug(s) Interacting with This Target
Drug Name Drug Type External ID
A-134974 Small molecular drug D0S9XV
Abt-702 Small molecular drug D08LUT
Gp-683 Small molecular drug D0JI1J

References

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Mass spectrometry data entry: PXD044402
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