Probe Name	DA-2					Probe Info
Probe concentration	10 uM
Criteria	Other data
In Vivo Experiment Model	Model Type			Cell lysate
	Derived Tissue			Peripheral blood
	Disease Model		Chronic myeloid leukemia [ICD-11:2A20]
	Model Name		Human chronic myeloid leukemia cell lysate (K562)

Target ID	Target Name
LDTP10869	26S proteasome non-ATPase regulatory subunit 1 (PSMD1)
LDTP00224	26S proteasome non-ATPase regulatory subunit 12 (PSMD12)
LDTP13667	26S proteasome non-ATPase regulatory subunit 13 (PSMD13)
LDTP00294	26S proteasome non-ATPase regulatory subunit 14 (PSMD14)
LDTP05782	26S proteasome non-ATPase regulatory subunit 2 (PSMD2)
LDTP00714	26S proteasome non-ATPase regulatory subunit 3 (PSMD3)
LDTP06532	26S proteasome non-ATPase regulatory subunit 5 (PSMD5)
LDTP10954	3-hydroxyacyl-CoA dehydrogenase type-2 (HSD17B10)
LDTP03291	Acetyl-CoA acetyltransferase, mitochondrial (ACAT1)
LDTP10982	Aconitate hydratase, mitochondrial (ACO2)
LDTP05069	Actin, alpha cardiac muscle 1 (ACTC1)
LDTP06905	Acylglycerol kinase, mitochondrial (AGK)
LDTP02220	Adenine phosphoribosyltransferase (APRT)
LDTP04689	Adenosine kinase (ADK)
LDTP04636	Adenylate kinase 2, mitochondrial (AK2)
LDTP03551	Adenylosuccinate lyase (ADSL)
LDTP03541	Adenylosuccinate synthetase isozyme 2 (ADSS2)
LDTP11127	ADP-dependent glucokinase (ADPGK)
LDTP00776	Aflatoxin B1 aldehyde reductase member 2 (AKR7A2)
LDTP04262	Alanine--tRNA ligase, cytoplasmic (AARS1)
LDTP15371	Aldehyde dehydrogenase family 16 member A1 (ALDH16A1)
LDTP02514	Alkaline phosphatase, germ cell type (ALPG)
LDTP02100	Alkaline phosphatase, placental type (ALPP)
LDTP15993	Aminopeptidase B (RNPEP)
LDTP04601	Arginine--tRNA ligase, cytoplasmic (RARS1)
LDTP02264	Asparagine synthetase [glutamine-hydrolyzing] (ASNS)
LDTP00866	Asparagine--tRNA ligase, cytoplasmic (NARS1)
LDTP01783	Aspartate aminotransferase, mitochondrial (GOT2)
LDTP02752	Aspartate--tRNA ligase, cytoplasmic (DARS1)
LDTP04561	ATP-citrate synthase (ACLY)
LDTP02925	ATP-dependent 6-phosphofructokinase, liver type (PFKL)
LDTP05314	ATP-dependent 6-phosphofructokinase, platelet type (PFKP)
LDTP09766	ATP-dependent RNA helicase DDX1 (DDX1)
LDTP00314	ATP-dependent RNA helicase DDX3X (DDX3X)
LDTP00684	ATP-dependent RNA helicase DHX15 (DHX15)
LDTP00491	Aurora kinase A (AURKA)
LDTP03159	Bifunctional phosphoribosylaminoimidazole carboxylase/phosphoribosylaminoimidazole succinocarboxamide synthetase (PAICS)
LDTP04552	Biliverdin reductase A (BLVRA)
LDTP05992	Bleomycin hydrolase (BLMH)
LDTP12163	Calcyclin-binding protein (CACYBP)
LDTP10215	Carboxymethylenebutenolidase homolog (CMBL)
LDTP01205	Citrate synthase, mitochondrial (CS)
LDTP02616	Creatine kinase B-type (CKB)
LDTP02622	Creatine kinase U-type, mitochondrial (CKMT1A; CKMT1B)
LDTP08296	Cullin-associated NEDD8-dissociated protein 1 (CAND1)
LDTP02149	Cyclin-dependent kinase 1 (CDK1)
LDTP05507	Cyclin-dependent kinase 18 (CDK18)
LDTP03299	Cyclin-dependent kinase 2 (CDK2)
LDTP04263	Cysteine--tRNA ligase, cytoplasmic (CARS1)
LDTP03455	Cytosol aminopeptidase (LAP3)
LDTP03669	Deoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial (DUT)
LDTP02362	Dihydrolipoyl dehydrogenase, mitochondrial (DLD)
LDTP02497	Dihydrolipoyllysine-residue acetyltransferase component of pyruvate dehydrogenase complex, mitochondrial (DLAT)
LDTP03829	Dihydrolipoyllysine-residue succinyltransferase component of 2-oxoglutarate dehydrogenase complex, mitochondrial (DLST)
LDTP03680	DNA replication licensing factor MCM4 (MCM4)
LDTP03681	DNA replication licensing factor MCM5 (MCM5)
LDTP06150	DNA replication licensing factor MCM6 (MCM6)
LDTP03682	DNA replication licensing factor MCM7 (MCM7)
LDTP05136	DNA-dependent protein kinase catalytic subunit (PRKDC)
LDTP02694	Electron transfer flavoprotein subunit alpha, mitochondrial (ETFA)
LDTP03849	Electron transfer flavoprotein subunit beta (ETFB)
LDTP04251	Elongation factor Tu, mitochondrial (TUFM)
LDTP03965	Enoyl-CoA delta isomerase 1, mitochondrial (ECI1)
LDTP03518	Enoyl-CoA hydratase, mitochondrial (ECHS1)
LDTP01785	Epidermal growth factor receptor (EGFR)
LDTP03915	Eukaryotic translation initiation factor 2 subunit 3 (EIF2S3)
LDTP00246	Eukaryotic translation initiation factor 3 subunit F (EIF3F)
LDTP03511	Flavin reductase (NADPH) (BLVRB)
LDTP02386	Fructose-bisphosphate aldolase C (ALDOC)
LDTP02235	Fumarate hydratase, mitochondrial (FH)
LDTP02569	Glucose-6-phosphate 1-dehydrogenase (G6PD)
LDTP01771	Glutathione reductase, mitochondrial (GSR)
LDTP05128	Glutathione S-transferase omega-1 (GSTO1)
LDTP03628	Glycerol kinase (GK)
LDTP04333	GMP synthase [glutamine-hydrolyzing] (GMPS)
LDTP02991	Hexokinase-1 (HK1)
LDTP00479	Histone acetyltransferase type B catalytic subunit (HAT1)
LDTP06645	Hydroxyacyl-coenzyme A dehydrogenase, mitochondrial (HADH)
LDTP01782	Hypoxanthine-guanine phosphoribosyltransferase (HPRT1)
LDTP14854	Inorganic pyrophosphatase (PPA1)
LDTP02611	Inosine-5'-monophosphate dehydrogenase 2 (IMPDH2)
LDTP03003	Interferon-induced, double-stranded RNA-activated protein kinase (EIF2AK2)
LDTP01333	Isocitrate dehydrogenase [NADP] cytoplasmic (IDH1)
LDTP04345	Isocitrate dehydrogenase [NAD] subunit alpha, mitochondrial (IDH3A)
LDTP16025	Ketosamine-3-kinase (FN3KRP)
LDTP05434	Lactoylglutathione lyase (GLO1)
LDTP13056	Leucine--tRNA ligase, cytoplasmic (LARS1)
LDTP03817	Lon protease homolog, mitochondrial (LONP1)
LDTP06294	Lysine--tRNA ligase (KARS1)
LDTP02565	Medium-chain specific acyl-CoA dehydrogenase, mitochondrial (ACADM)
LDTP04730	Methionine--tRNA ligase, cytoplasmic (MARS1)
LDTP05632	Mitochondrial-processing peptidase subunit alpha (PMPCA)
LDTP06547	Mitogen-activated protein kinase 14 (MAPK14)
LDTP06192	Neutral alpha-glucosidase AB (GANAB)
LDTP04051	Nicotinamide phosphoribosyltransferase (NAMPT)
LDTP02796	Nucleoside diphosphate kinase A (NME1)
LDTP12610	Obg-like ATPase 1 (OLA1)
LDTP02021	Ornithine aminotransferase, mitochondrial (OAT)
LDTP03813	Oxygen-dependent coproporphyrinogen-III oxidase, mitochondrial (CPOX)
LDTP10878	Parkinson disease protein 7 (PARK7)
LDTP05372	Peptidyl-prolyl cis-trans isomerase FKBP4 (FKBP4)
LDTP01787	Phosphoglycerate kinase 1 (PGK1)
LDTP02186	Phosphoglycerate kinase 2 (PGK2)
LDTP14198	Phosphoserine aminotransferase (PSAT1)
LDTP13750	Proliferation-associated protein 2G4 (PA2G4)
LDTP03330	Proteasome subunit alpha type-1 (PSMA1)
LDTP03331	Proteasome subunit alpha type-2 (PSMA2)
LDTP03413	Proteasome subunit alpha type-5 (PSMA5)
LDTP00449	Proteasome subunit alpha type-7 (PSMA7)
LDTP03060	Proteasome subunit beta type-1 (PSMB1)
LDTP04285	Proteasome subunit beta type-2 (PSMB2)
LDTP03417	Proteasome subunit beta type-4 (PSMB4)
LDTP10997	Protein arginine N-methyltransferase 1 (PRMT1)
LDTP03521	Protein disulfide-isomerase A3 (PDIA3)
LDTP06314	Protein disulfide-isomerase A6 (PDIA6)
LDTP02123	Protein kinase C beta type (PRKCB)
LDTP04266	Protein phosphatase 1F (PPM1F)
LDTP03146	Protein-glutamine gamma-glutamyltransferase 2 (TGM2)
LDTP02318	Proto-oncogene tyrosine-protein kinase ROS (ROS1)
LDTP02638	Proto-oncogene tyrosine-protein kinase Src (SRC)
LDTP01781	Purine nucleoside phosphorylase (PNP)
LDTP04712	Puromycin-sensitive aminopeptidase (NPEPPS)
LDTP18413	Putative tubulin-like protein alpha-4B (TUBA4B)
LDTP00343	Pyridoxal kinase (PDXK)
LDTP02733	Pyruvate kinase PKM (PKM)
LDTP04895	Ras-related protein Rab-10 (RAB10)
LDTP04910	Ras-related protein Rap-1b (RAP1B)
LDTP03592	Ribonucleoside-diphosphate reductase subunit M2 (RRM2)
LDTP04882	Ribose-phosphate pyrophosphokinase 1 (PRPS1)
LDTP02592	Ribose-phosphate pyrophosphokinase 2 (PRPS2)
LDTP05588	RNA cytosine C(5)-methyltransferase NSUN2 (NSUN2)
LDTP13816	RuvB-like 1 (RUVBL1)
LDTP03577	S-adenosylmethionine synthase isoform type-2 (MAT2A)
LDTP06279	Septin-2 (SEPTIN2)
LDTP04265	Serine--tRNA ligase, cytoplasmic (SARS1)
LDTP00299	Serine/threonine-protein kinase 25 (STK25)
LDTP06536	Serine/threonine-protein kinase N2 (PKN2)
LDTP05232	Serine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B beta isoform (PPP2R2B)
LDTP03522	Serine/threonine-protein phosphatase 2A 65 kDa regulatory subunit A alpha isoform (PPP2R1A)
LDTP03819	Serine/threonine-protein phosphatase PP1-gamma catalytic subunit (PPP1CC)
LDTP05991	Spliceosome RNA helicase DDX39B (DDX39B)
LDTP03572	Succinate dehydrogenase flavoprotein subunit, mitochondrial (SDHA)
LDTP02019	Superoxide dismutase [Mn], mitochondrial (SOD2)
LDTP10887	Synaptic vesicle membrane protein VAT-1 homolog (VAT1)
LDTP04542	Thimet oligopeptidase (THOP1)
LDTP03365	Threonine--tRNA ligase 1, cytoplasmic (TARS1)
LDTP03258	Thymidylate kinase (DTYMK)
LDTP05808	Transcription intermediary factor 1-beta (TRIM28)
LDTP03156	Trifunctional purine biosynthetic protein adenosine-3 (GART)
LDTP03222	Tryptophan--tRNA ligase, cytoplasmic (WARS1)
LDTP07907	Tubulin alpha-1A chain (TUBA1A)
LDTP05478	Tyrosine-protein kinase BTK (BTK)
LDTP03944	Tyrosine-protein kinase CSK (CSK)
LDTP02231	Tyrosine-protein kinase Yes (YES1)
LDTP05449	Tyrosine-protein phosphatase non-receptor type 12 (PTPN12)
LDTP06639	Tyrosine-protein phosphatase non-receptor type 21 (PTPN21)
LDTP04074	Ubiquitin carboxyl-terminal hydrolase 5 (USP5)
LDTP12851	UDP-glucose:glycoprotein glucosyltransferase 1 (UGGT1)
LDTP11571	Uridine-cytidine kinase 2 (UCK2)
LDTP02135	Uroporphyrinogen decarboxylase (UROD)
LDTP03366	Valine--tRNA ligase (VARS1)
LDTP12954	Very-long-chain (3R)-3-hydroxyacyl-CoA dehydratase 3 (HACD3)

Target ID	Target Name
LDTP04969	14-3-3 protein epsilon (YWHAE)
LDTP01601	Activator of 90 kDa heat shock protein ATPase homolog 1 (AHSA1)
LDTP02608	ADP/ATP translocase 1 (SLC25A4)
LDTP16103	ATP-binding cassette sub-family F member 3 (ABCF3)
LDTP05165	Brain acid soluble protein 1 (BASP1)
LDTP03402	Calreticulin (CALR)
LDTP00244	Chloride intracellular channel protein 1 (CLIC1)
LDTP12882	Chloride intracellular channel protein 5 (CLIC5)
LDTP05510	Complement component 1 Q subcomponent-binding protein, mitochondrial (C1QBP)
LDTP13393	Electrogenic aspartate/glutamate antiporter SLC25A13, mitochondrial (SLC25A13)
LDTP00501	Exportin-1 (XPO1)
LDTP04662	Exportin-2 (CSE1L)
LDTP12142	Exportin-5 (XPO5)
LDTP06103	Filamin-C (FLNC)
LDTP06549	Hsp90 co-chaperone Cdc37 (CDC37)
LDTP01574	Importin-7 (IPO7)
LDTP05238	Solute carrier family 25 member 3 (SLC25A3)
LDTP01969	Transferrin receptor protein 1 (TFRC)
LDTP03104	V-type proton ATPase subunit B, brain isoform (ATP6V1B2)
LDTP10741	Vacuolar protein sorting-associated protein 35 (VPS35)
LDTP04071	Voltage-dependent anion-selective channel protein 2 (VDAC2)
LDTP13824	Voltage-dependent anion-selective channel protein 3 (VDAC3)

Target ID	Target Name
LDTP03903	Signal transducer and activator of transcription 3 (STAT3)
LDTP09932	SWI/SNF complex subunit SMARCC1 (SMARCC1)
LDTP05065	Y-box-binding protein 1 (YBX1)

Target ID	Target Name
LDTP05442	14-3-3 protein eta (YWHAH)
LDTP03618	14-3-3 protein sigma (SFN)
LDTP00223	26S proteasome non-ATPase regulatory subunit 11 (PSMD11)
LDTP06273	26S proteasome non-ATPase regulatory subunit 6 (PSMD6)
LDTP03871	Acidic leucine-rich nuclear phosphoprotein 32 family member A (ANP32A)
LDTP09843	Acidic leucine-rich nuclear phosphoprotein 32 family member B (ANP32B)
LDTP04902	Actin-related protein 3 (ACTR3)
LDTP05294	Adenylyl cyclase-associated protein 1 (CAP1)
LDTP03612	Bifunctional purine biosynthesis protein ATIC (ATIC)
LDTP09444	CDK5 and ABL1 enzyme substrate 1 (CABLES1)
LDTP04092	Crk-like protein (CRKL)
LDTP12642	CYFIP-related Rac1 interactor B (CYRIB)
LDTP06543	DNA damage-binding protein 1 (DDB1)
LDTP06450	ELAV-like protein 1 (ELAVL1)
LDTP03283	Elongation factor 1-beta (EEF1B2)
LDTP03499	Elongation factor 1-delta (EEF1D)
LDTP11021	Endophilin-A3 (SH3GL3)
LDTP02101	Eukaryotic translation initiation factor 2 subunit 1 (EIF2S1)
LDTP13813	Eukaryotic translation initiation factor 3 subunit L (EIF3L)
LDTP04544	F-actin-capping protein subunit alpha-1 (CAPZA1)
LDTP04127	F-actin-capping protein subunit beta (CAPZB)
LDTP08263	Fermitin family homolog 3 (FERMT3)
LDTP01922	Hemoglobin subunit epsilon (HBE1)
LDTP05083	Hemoglobin subunit gamma-2 (HBG2)
LDTP00500	Heterogeneous nuclear ribonucleoprotein D-like (HNRNPDL)
LDTP03615	Heterogeneous nuclear ribonucleoprotein H (HNRNPH1)
LDTP02750	Heterogeneous nuclear ribonucleoprotein L (HNRNPL)
LDTP04500	Heterogeneous nuclear ribonucleoprotein M (HNRNPM)
LDTP00991	Heterogeneous nuclear ribonucleoprotein Q (SYNCRIP)
LDTP00756	Heterogeneous nuclear ribonucleoprotein R (HNRNPR)
LDTP02227	Heterogeneous nuclear ribonucleoproteins C1/C2 (HNRNPC)
LDTP05590	Histone-binding protein RBBP4 (RBBP4)
LDTP04367	Hsc70-interacting protein (ST13)
LDTP05688	Interleukin enhancer-binding factor 2 (ILF2)
LDTP04094	Large proline-rich protein BAG6 (BAG6)
LDTP02109	Large ribosomal subunit protein uL10 (RPLP0)
LDTP06220	LIM and SH3 domain protein 1 (LASP1)
LDTP02116	Lupus La protein (SSB)
LDTP04027	Matrin-3 (MATR3)
LDTP13817	Nuclear migration protein nudC (NUDC)
LDTP04684	Nucleosome assembly protein 1-like 1 (NAP1L1)
LDTP01021	Perilipin-3 (PLIN3)
LDTP03520	Phosphatidylethanolamine-binding protein 1 (PEBP1)
LDTP02595	Polyadenylate-binding protein 1 (PABPC1)
LDTP03364	Polypyrimidine tract-binding protein 1 (PTBP1)
LDTP09580	Programmed cell death 6-interacting protein (PDCD6IP)
LDTP02596	Proliferating cell nuclear antigen (PCNA)
LDTP13519	Proteasome activator complex subunit 2 (PSME2)
LDTP04917	Proteasome activator complex subunit 3 (PSME3)
LDTP04355	Rab GDP dissociation inhibitor beta (GDI2)
LDTP02964	Regulator of chromosome condensation (RCC1)
LDTP04510	Rho GDP-dissociation inhibitor 1 (ARHGDIA)
LDTP02480	RNA-binding protein RO60 (RO60)
LDTP13991	Serine-threonine kinase receptor-associated protein (STRAP)
LDTP03719	Serpin B6 (SERPINB6)
LDTP04362	Serpin B9 (SERPINB9)
LDTP04363	Serpin H1 (SERPINH1)
LDTP05002	Small ribosomal subunit protein eS6 (RPS6)
LDTP04964	Small ribosomal subunit protein eS8 (RPS8)
LDTP06280	Squamous cell carcinoma antigen recognized by T-cells 3 (SART3)
LDTP06094	Src substrate cortactin (CTTN)
LDTP03619	Stress-induced-phosphoprotein 1 (STIP1)
LDTP02934	T-complex protein 1 subunit alpha (TCP1)
LDTP05113	T-complex protein 1 subunit beta (CCT2)
LDTP04201	T-complex protein 1 subunit epsilon (CCT5)
LDTP03888	T-complex protein 1 subunit zeta (CCT6A)
LDTP09777	T-complex protein 1 subunit zeta-2 (CCT6B)
LDTP02037	Tubulin beta-4A chain (TUBB4A)
LDTP06809	Tubulin beta-8 chain (TUBB8)
LDTP00759	Tumor protein D54 (TPD52L2)
LDTP05418	UBX domain-containing protein 1 (UBXN1)
LDTP02297	Vimentin (VIM)

1	Cell-based proteome profiling of potential dasatinib targets by use of affinity-based probes. J Am Chem Soc. 2012 Feb 15;134(6):3001-14. doi: 10.1021/ja208518u. Epub 2012 Feb 1.