Details of the Target

General Information of Target

Target ID LDTP07531
Target Name Sideroflexin-4 (SFXN4)
Gene Name SFXN4
Gene ID 119559
Synonyms
BCRM1; Sideroflexin-4; Breast cancer resistance marker 1
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MSLEQEEETQPGRLLGRRDAVPAFIEPNVRFWITERQSFIRRFLQWTELLDPTNVFISVE
SIENSRQLLCTNEDVSSPASADQRIQEAWKRSLATVHPDSSNLIPKLFRPAAFLPFMAPT
VFLSMTPLKGIKSVILPQVFLCAYMAAFNSINGNRSYTCKPLERSLLMAGAVASSTFLGV
IPQFVQMKYGLTGPWIKRLLPVIFLVQASGMNVYMSRSLESIKGIAVMDKEGNVLGHSRI
AGTKAVRETLASRIVLFGTSALIPEVFTYFFKRTQYFRKNPGSLWILKLSCTVLAMGLMV
PFSFSIFPQIGQIQYCSLEEKIQSPTEETEIFYHRGV
Target Bioclass
Transporter and channel
Family
Sideroflexin family
Subcellular location
Mitochondrion inner membrane
Function Mitochondrial amino-acid transporter. Does not act as a serine transporter: not able to mediate transport of serine into mitochondria.
Uniprot ID
Q6P4A7
Ensemble ID
ENST00000355697.7
HGNC ID
HGNC:16088

Target Site Mutations in Different Cell Lines

Cell line Mutation details Probe for labeling this protein in this cell
AGS SNV: p.F332L DBIA    Probe Info 
HELA SNV: p.E330K .
JURKAT SNV: p.A111V .
MCAS SNV: p.F108S DBIA    Probe Info 
MEWO SNV: p.L93F DBIA    Probe Info 
NCIH1975 SNV: p.R18K .

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 16 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
YN-1
 Probe Info  		100.00  LDD0444  [1]
STPyne
 Probe Info  		K90(6.25)  LDD0277  [2]
m-APA
 Probe Info  		13.20  LDD0403  [3]
BTD
 Probe Info  		C159(1.16)  LDD2090  [4]
AHL-Pu-1
 Probe Info  		C70(3.20)  LDD0169  [5]
DBIA
 Probe Info  		C70(1.44)  LDD0531  [6]
4-Iodoacetamidophenylacetylene
 Probe Info  		N.A.  LDD0038  [7]
IA-alkyne
 Probe Info  		N.A.  LDD0036  [7]
Lodoacetamide azide
 Probe Info  		N.A.  LDD0037  [7]
TFBX
 Probe Info  		N.A.  LDD0027  [8]
IPM
 Probe Info  		N.A.  LDD0005  [9]
VSF
 Probe Info  		N.A.  LDD0007  [9]
1d-yne
 Probe Info  		N.A.  LDD0357  [10]
Crotonaldehyde
 Probe Info  		N.A.  LDD0219  [11]
AOyne
 Probe Info  		15.00  LDD0443  [12]
NAIA_5
 Probe Info  		N.A.  LDD2223  [13]
PAL-AfBPP Probe
Click To Hide/Show 75 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
C002
 Probe Info  		5.10  LDD1712  [14]
C004
 Probe Info  		6.06  LDD1714  [14]
C022
 Probe Info  		11.39  LDD1728  [14]
C027
 Probe Info  		8.63  LDD1733  [14]
C040
 Probe Info  		20.53  LDD1740  [14]
C041
 Probe Info  		5.98  LDD1741  [14]
C056
 Probe Info  		21.41  LDD1753  [14]
C063
 Probe Info  		10.13  LDD1760  [14]
C070
 Probe Info  		23.26  LDD1766  [14]
C091
 Probe Info  		21.26  LDD1782  [14]
C092
 Probe Info  		27.86  LDD1783  [14]
C094
 Probe Info  		47.18  LDD1785  [14]
C107
 Probe Info  		5.54  LDD1794  [14]
C112
 Probe Info  		21.86  LDD1799  [14]
C134
 Probe Info  		23.59  LDD1816  [14]
C135
 Probe Info  		11.31  LDD1817  [14]
C141
 Probe Info  		32.67  LDD1823  [14]
C143
 Probe Info  		27.47  LDD1825  [14]
C153
 Probe Info  		15.24  LDD1834  [14]
C159
 Probe Info  		15.89  LDD1839  [14]
C160
 Probe Info  		17.88  LDD1840  [14]
C169
 Probe Info  		29.86  LDD1849  [14]
C177
 Probe Info  		9.25  LDD1856  [14]
C186
 Probe Info  		7.73  LDD1864  [14]
C194
 Probe Info  		8.88  LDD1870  [14]
C198
 Probe Info  		9.65  LDD1874  [14]
C219
 Probe Info  		12.04  LDD1893  [14]
C225
 Probe Info  		6.73  LDD1898  [14]
C228
 Probe Info  		18.38  LDD1901  [14]
C231
 Probe Info  		26.91  LDD1904  [14]
C232
 Probe Info  		39.12  LDD1905  [14]
C233
 Probe Info  		9.25  LDD1906  [14]
C235
 Probe Info  		29.86  LDD1908  [14]
C238
 Probe Info  		11.31  LDD1911  [14]
C239
 Probe Info  		14.32  LDD1912  [14]
C246
 Probe Info  		13.55  LDD1919  [14]
C264
 Probe Info  		26.72  LDD1935  [14]
C277
 Probe Info  		8.88  LDD1947  [14]
C278
 Probe Info  		77.17  LDD1948  [14]
C282
 Probe Info  		40.50  LDD1952  [14]
C284
 Probe Info  		23.75  LDD1954  [14]
C287
 Probe Info  		18.25  LDD1957  [14]
C289
 Probe Info  		29.86  LDD1959  [14]
C296
 Probe Info  		12.30  LDD1966  [14]
C310
 Probe Info  		9.00  LDD1977  [14]
C314
 Probe Info  		22.47  LDD1981  [14]
C317
 Probe Info  		5.82  LDD1983  [14]
C322
 Probe Info  		6.28  LDD1988  [14]
C343
 Probe Info  		11.63  LDD2005  [14]
C349
 Probe Info  		24.42  LDD2010  [14]
C350
 Probe Info  		83.29  LDD2011  [14]
C355
 Probe Info  		24.42  LDD2016  [14]
C356
 Probe Info  		17.51  LDD2017  [14]
C362
 Probe Info  		42.52  LDD2023  [14]
C363
 Probe Info  		18.90  LDD2024  [14]
C364
 Probe Info  		20.82  LDD2025  [14]
C366
 Probe Info  		5.62  LDD2027  [14]
C380
 Probe Info  		6.11  LDD2039  [14]
C388
 Probe Info  		42.22  LDD2047  [14]
C390
 Probe Info  		22.32  LDD2049  [14]
C403
 Probe Info  		21.41  LDD2061  [14]
C407
 Probe Info  		15.78  LDD2064  [14]
C413
 Probe Info  		29.24  LDD2069  [14]
C420
 Probe Info  		17.27  LDD2075  [14]
C424
 Probe Info  		7.73  LDD2079  [14]
C426
 Probe Info  		28.44  LDD2081  [14]
FFF probe11
 Probe Info  		20.00  LDD0471  [15]
FFF probe13
 Probe Info  		20.00  LDD0475  [15]
FFF probe14
 Probe Info  		20.00  LDD0477  [15]
FFF probe2
 Probe Info  		20.00  LDD0463  [15]
FFF probe3
 Probe Info  		14.63  LDD0464  [15]
JN0003
 Probe Info  		20.00  LDD0469  [15]
BD-F
 Probe Info  		E48(0.00); T47(0.00); D51(0.00)  LDD0024  [16]
LD-F
 Probe Info  		D51(0.00); E48(0.00); L50(0.00); T47(0.00)  LDD0015  [16]
OEA-DA
 Probe Info  		13.60  LDD0046  [17]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0539  3-(4-Isopropylpiperazin-1-yl)-3-oxopropanenitrile MDA-MB-231 C159(0.73)  LDD2132  [4]
 LDCM0026  4SU-RNA+native RNA HEK-293T C70(3.20)  LDD0169  [5]
 LDCM0214  AC1 HCT 116 C70(1.44)  LDD0531  [6]
 LDCM0215  AC10 HEK-293T C70(1.05)  LDD1508  [18]
 LDCM0216  AC100 HCT 116 C70(0.88)  LDD0533  [6]
 LDCM0217  AC101 HCT 116 C70(0.96)  LDD0534  [6]
 LDCM0218  AC102 HCT 116 C70(1.02)  LDD0535  [6]
 LDCM0219  AC103 HCT 116 C70(1.05)  LDD0536  [6]
 LDCM0220  AC104 HCT 116 C70(1.05)  LDD0537  [6]
 LDCM0221  AC105 HCT 116 C70(0.99)  LDD0538  [6]
 LDCM0222  AC106 HCT 116 C70(0.94)  LDD0539  [6]
 LDCM0223  AC107 HCT 116 C70(0.85)  LDD0540  [6]
 LDCM0224  AC108 HCT 116 C70(0.99)  LDD0541  [6]
 LDCM0225  AC109 HCT 116 C70(1.05)  LDD0542  [6]
 LDCM0226  AC11 HEK-293T C159(1.06); C70(1.16)  LDD1509  [18]
 LDCM0227  AC110 HCT 116 C70(0.89)  LDD0544  [6]
 LDCM0228  AC111 HCT 116 C70(0.95)  LDD0545  [6]
 LDCM0229  AC112 HCT 116 C70(0.90)  LDD0546  [6]
 LDCM0237  AC12 HEK-293T C159(0.97); C70(1.16)  LDD1510  [18]
 LDCM0259  AC14 HEK-293T C159(1.17); C70(0.89)  LDD1512  [18]
 LDCM0270  AC15 HEK-293T C159(1.15)  LDD1513  [18]
 LDCM0276  AC17 HEK-293T C70(0.85)  LDD1515  [18]
 LDCM0277  AC18 HEK-293T C70(1.10)  LDD1516  [18]
 LDCM0278  AC19 HEK-293T C159(1.08); C70(1.16)  LDD1517  [18]
 LDCM0279  AC2 HCT 116 C70(1.16)  LDD0596  [6]
 LDCM0280  AC20 HEK-293T C159(1.05); C70(1.11)  LDD1519  [18]
 LDCM0281  AC21 HEK-293T C159(1.28); C70(1.13)  LDD1520  [18]
 LDCM0282  AC22 HEK-293T C159(1.16); C70(0.93)  LDD1521  [18]
 LDCM0283  AC23 HEK-293T C159(1.01)  LDD1522  [18]
 LDCM0284  AC24 HEK-293T C159(1.04); C70(0.94)  LDD1523  [18]
 LDCM0285  AC25 HEK-293T C70(0.90)  LDD1524  [18]
 LDCM0286  AC26 HEK-293T C70(1.15)  LDD1525  [18]
 LDCM0287  AC27 HEK-293T C159(1.05); C70(0.93)  LDD1526  [18]
 LDCM0288  AC28 HEK-293T C159(1.07); C70(1.09)  LDD1527  [18]
 LDCM0289  AC29 HEK-293T C159(1.01); C70(1.08)  LDD1528  [18]
 LDCM0290  AC3 HCT 116 C70(1.48)  LDD0607  [6]
 LDCM0291  AC30 HEK-293T C159(1.11); C70(1.08)  LDD1530  [18]
 LDCM0292  AC31 HEK-293T C159(1.06)  LDD1531  [18]
 LDCM0293  AC32 HEK-293T C159(1.14); C70(0.99)  LDD1532  [18]
 LDCM0294  AC33 HEK-293T C70(0.88)  LDD1533  [18]
 LDCM0295  AC34 HEK-293T C70(1.12)  LDD1534  [18]
 LDCM0296  AC35 HEK-293T C70(1.56)  LDD0894  [6]
 LDCM0297  AC36 HEK-293T C70(2.05)  LDD0895  [6]
 LDCM0298  AC37 HEK-293T C70(2.46)  LDD0896  [6]
 LDCM0299  AC38 HEK-293T C70(1.56)  LDD0897  [6]
 LDCM0300  AC39 HEK-293T C70(0.77)  LDD0898  [6]
 LDCM0301  AC4 HCT 116 C70(1.66)  LDD0618  [6]
 LDCM0302  AC40 HEK-293T C70(0.82)  LDD0900  [6]
 LDCM0303  AC41 HEK-293T C70(0.64)  LDD0901  [6]
 LDCM0304  AC42 HEK-293T C70(0.68)  LDD0902  [6]
 LDCM0305  AC43 HEK-293T C70(0.57)  LDD0903  [6]
 LDCM0306  AC44 HEK-293T C70(1.08)  LDD0904  [6]
 LDCM0307  AC45 HEK-293T C70(2.19)  LDD0905  [6]
 LDCM0308  AC46 HEK-293T C70(1.49)  LDD0906  [6]
 LDCM0309  AC47 HEK-293T C70(1.28)  LDD0907  [6]
 LDCM0310  AC48 HEK-293T C70(1.80)  LDD0908  [6]
 LDCM0311  AC49 HEK-293T C70(1.17)  LDD0909  [6]
 LDCM0312  AC5 HCT 116 C70(1.48)  LDD0629  [6]
 LDCM0313  AC50 HEK-293T C70(1.37)  LDD0911  [6]
 LDCM0314  AC51 HEK-293T C70(1.86)  LDD0912  [6]
 LDCM0315  AC52 HEK-293T C70(2.09)  LDD0913  [6]
 LDCM0316  AC53 HEK-293T C70(1.36)  LDD0914  [6]
 LDCM0317  AC54 HEK-293T C70(1.38)  LDD0915  [6]
 LDCM0318  AC55 HEK-293T C70(1.33)  LDD0916  [6]
 LDCM0319  AC56 HEK-293T C70(1.13)  LDD0917  [6]
 LDCM0320  AC57 HEK-293T C70(1.27)  LDD0918  [6]
 LDCM0321  AC58 HEK-293T C70(2.68)  LDD0919  [6]
 LDCM0322  AC59 HEK-293T C70(2.53)  LDD0920  [6]
 LDCM0323  AC6 HEK-293T C159(1.01); C70(1.12)  LDD1562  [18]
 LDCM0324  AC60 HEK-293T C70(2.32)  LDD0922  [6]
 LDCM0325  AC61 HEK-293T C70(2.30)  LDD0923  [6]
 LDCM0326  AC62 HEK-293T C70(3.07)  LDD0924  [6]
 LDCM0327  AC63 HEK-293T C70(2.31)  LDD0925  [6]
 LDCM0328  AC64 HEK-293T C70(3.19)  LDD0926  [6]
 LDCM0329  AC65 HEK-293T C70(3.41)  LDD0927  [6]
 LDCM0330  AC66 HEK-293T C70(2.25)  LDD0928  [6]
 LDCM0331  AC67 HEK-293T C70(2.82)  LDD0929  [6]
 LDCM0332  AC68 HEK-293T C70(0.58)  LDD0930  [6]
 LDCM0333  AC69 HEK-293T C70(0.54)  LDD0931  [6]
 LDCM0334  AC7 HEK-293T C159(1.03)  LDD1568  [18]
 LDCM0335  AC70 HEK-293T C70(0.61)  LDD0933  [6]
 LDCM0336  AC71 HEK-293T C70(0.50)  LDD0934  [6]
 LDCM0337  AC72 HEK-293T C70(0.71)  LDD0935  [6]
 LDCM0338  AC73 HEK-293T C70(0.70)  LDD0936  [6]
 LDCM0339  AC74 HEK-293T C70(0.40)  LDD0937  [6]
 LDCM0340  AC75 HEK-293T C70(0.63)  LDD0938  [6]
 LDCM0341  AC76 HEK-293T C70(0.45)  LDD0939  [6]
 LDCM0342  AC77 HEK-293T C70(0.56)  LDD0940  [6]
 LDCM0343  AC78 HEK-293T C70(1.15)  LDD0941  [6]
 LDCM0344  AC79 HEK-293T C70(1.29)  LDD0942  [6]
 LDCM0345  AC8 HEK-293T C159(1.08); C70(1.00)  LDD1569  [18]
 LDCM0346  AC80 HEK-293T C70(0.67)  LDD0944  [6]
 LDCM0347  AC81 HEK-293T C70(0.53)  LDD0945  [6]
 LDCM0348  AC82 HEK-293T C70(0.64)  LDD0946  [6]
 LDCM0349  AC83 HCT 116 C70(1.17)  LDD0666  [6]
 LDCM0350  AC84 HCT 116 C70(1.17)  LDD0667  [6]
 LDCM0351  AC85 HCT 116 C70(1.12)  LDD0668  [6]
 LDCM0352  AC86 HCT 116 C70(1.16)  LDD0669  [6]
 LDCM0353  AC87 HCT 116 C70(0.91)  LDD0670  [6]
 LDCM0354  AC88 HCT 116 C70(0.99)  LDD0671  [6]
 LDCM0355  AC89 HCT 116 C70(1.24)  LDD0672  [6]
 LDCM0357  AC90 HCT 116 C70(1.16)  LDD0674  [6]
 LDCM0358  AC91 HCT 116 C70(1.44)  LDD0675  [6]
 LDCM0359  AC92 HCT 116 C70(1.40)  LDD0676  [6]
 LDCM0360  AC93 HCT 116 C70(1.16)  LDD0677  [6]
 LDCM0361  AC94 HCT 116 C70(1.11)  LDD0678  [6]
 LDCM0362  AC95 HCT 116 C70(1.19)  LDD0679  [6]
 LDCM0363  AC96 HCT 116 C70(1.22)  LDD0680  [6]
 LDCM0364  AC97 HCT 116 C70(1.42)  LDD0681  [6]
 LDCM0365  AC98 HCT 116 C70(1.13)  LDD0682  [6]
 LDCM0366  AC99 HCT 116 C70(1.01)  LDD0683  [6]
 LDCM0248  AKOS034007472 HEK-293T C159(1.00); C70(1.02)  LDD1511  [18]
 LDCM0356  AKOS034007680 HEK-293T C70(0.96)  LDD1570  [18]
 LDCM0275  AKOS034007705 HEK-293T C159(1.14); C70(1.05)  LDD1514  [18]
 LDCM0156  Aniline NCI-H1299 13.20  LDD0403  [3]
 LDCM0367  CL1 HCT 116 C70(1.03)  LDD0684  [6]
 LDCM0368  CL10 HCT 116 C70(1.78)  LDD0685  [6]
 LDCM0369  CL100 HCT 116 C70(1.65)  LDD0686  [6]
 LDCM0370  CL101 HEK-293T C159(1.08); C70(1.03)  LDD1574  [18]
 LDCM0371  CL102 HEK-293T C70(0.95)  LDD1575  [18]
 LDCM0372  CL103 HEK-293T C70(0.99)  LDD1576  [18]
 LDCM0373  CL104 HEK-293T C70(0.95)  LDD1577  [18]
 LDCM0374  CL105 HEK-293T C159(1.11); C70(0.99)  LDD1578  [18]
 LDCM0375  CL106 HEK-293T C70(0.88)  LDD1579  [18]
 LDCM0376  CL107 HEK-293T C70(1.04)  LDD1580  [18]
 LDCM0377  CL108 HEK-293T C70(1.03)  LDD1581  [18]
 LDCM0378  CL109 HEK-293T C159(1.18); C70(0.97)  LDD1582  [18]
 LDCM0379  CL11 HCT 116 C70(1.53)  LDD0696  [6]
 LDCM0380  CL110 HEK-293T C70(0.91)  LDD1584  [18]
 LDCM0381  CL111 HEK-293T C70(0.98)  LDD1585  [18]
 LDCM0382  CL112 HEK-293T C70(1.06)  LDD1586  [18]
 LDCM0383  CL113 HEK-293T C159(1.07); C70(0.99)  LDD1587  [18]
 LDCM0384  CL114 HEK-293T C70(0.87)  LDD1588  [18]
 LDCM0385  CL115 HEK-293T C70(1.01)  LDD1589  [18]
 LDCM0386  CL116 HEK-293T C70(0.97)  LDD1590  [18]
 LDCM0387  CL117 HEK-293T C70(2.37)  LDD0985  [6]
 LDCM0388  CL118 HEK-293T C70(1.67)  LDD0986  [6]
 LDCM0389  CL119 HEK-293T C70(0.74)  LDD0987  [6]
 LDCM0390  CL12 HCT 116 C70(2.03)  LDD0707  [6]
 LDCM0391  CL120 HEK-293T C70(0.54)  LDD0989  [6]
 LDCM0392  CL121 HEK-293T C70(1.45)  LDD0990  [6]
 LDCM0393  CL122 HEK-293T C70(1.48)  LDD0991  [6]
 LDCM0394  CL123 HEK-293T C70(1.17)  LDD0992  [6]
 LDCM0395  CL124 HEK-293T C70(1.18)  LDD0993  [6]
 LDCM0396  CL125 HEK-293T C70(1.38)  LDD0994  [6]
 LDCM0397  CL126 HEK-293T C70(1.13)  LDD0995  [6]
 LDCM0398  CL127 HEK-293T C70(1.09)  LDD0996  [6]
 LDCM0399  CL128 HEK-293T C70(1.19)  LDD0997  [6]
 LDCM0400  CL13 HCT 116 C70(2.03)  LDD0717  [6]
 LDCM0401  CL14 HCT 116 C70(1.12)  LDD0718  [6]
 LDCM0402  CL15 HCT 116 C70(2.14)  LDD0719  [6]
 LDCM0403  CL16 HEK-293T C70(1.03)  LDD1607  [18]
 LDCM0404  CL17 HEK-293T C70(0.90)  LDD1608  [18]
 LDCM0405  CL18 HEK-293T C70(1.13)  LDD1609  [18]
 LDCM0406  CL19 HEK-293T C159(0.88); C70(1.04)  LDD1610  [18]
 LDCM0407  CL2 HCT 116 C70(1.04)  LDD0724  [6]
 LDCM0408  CL20 HEK-293T C159(0.71); C70(1.09)  LDD1612  [18]
 LDCM0409  CL21 HEK-293T C159(0.76); C70(1.05)  LDD1613  [18]
 LDCM0410  CL22 HEK-293T C159(0.58); C70(0.98)  LDD1614  [18]
 LDCM0411  CL23 HEK-293T C159(0.47)  LDD1615  [18]
 LDCM0412  CL24 HEK-293T C159(0.49); C70(0.98)  LDD1616  [18]
 LDCM0413  CL25 HEK-293T C159(1.14); C70(1.02)  LDD1617  [18]
 LDCM0414  CL26 HEK-293T C70(0.89)  LDD1618  [18]
 LDCM0415  CL27 HEK-293T C70(1.00)  LDD1619  [18]
 LDCM0416  CL28 HEK-293T C70(1.00)  LDD1620  [18]
 LDCM0417  CL29 HEK-293T C70(0.82)  LDD1621  [18]
 LDCM0418  CL3 HCT 116 C70(1.14)  LDD0735  [6]
 LDCM0419  CL30 HEK-293T C70(1.11)  LDD1623  [18]
 LDCM0420  CL31 HCT 116 C70(0.83)  LDD0737  [6]
 LDCM0421  CL32 HCT 116 C70(0.83)  LDD0738  [6]
 LDCM0422  CL33 HCT 116 C70(0.88)  LDD0739  [6]
 LDCM0423  CL34 HCT 116 C70(1.09)  LDD0740  [6]
 LDCM0424  CL35 HCT 116 C70(0.95)  LDD0741  [6]
 LDCM0425  CL36 HCT 116 C70(0.96)  LDD0742  [6]
 LDCM0426  CL37 HCT 116 C70(0.90)  LDD0743  [6]
 LDCM0428  CL39 HCT 116 C70(0.99)  LDD0745  [6]
 LDCM0429  CL4 HCT 116 C70(1.25)  LDD0746  [6]
 LDCM0430  CL40 HCT 116 C70(0.93)  LDD0747  [6]
 LDCM0431  CL41 HCT 116 C70(1.16)  LDD0748  [6]
 LDCM0432  CL42 HCT 116 C70(1.07)  LDD0749  [6]
 LDCM0433  CL43 HCT 116 C70(1.02)  LDD0750  [6]
 LDCM0434  CL44 HCT 116 C70(0.91)  LDD0751  [6]
 LDCM0435  CL45 HCT 116 C70(1.10)  LDD0752  [6]
 LDCM0436  CL46 HEK-293T C159(0.52); C70(1.04)  LDD1640  [18]
 LDCM0437  CL47 HEK-293T C159(0.44)  LDD1641  [18]
 LDCM0438  CL48 HEK-293T C159(0.36); C70(1.00)  LDD1642  [18]
 LDCM0439  CL49 HEK-293T C159(1.04); C70(1.14)  LDD1643  [18]
 LDCM0440  CL5 HCT 116 C70(1.89)  LDD0757  [6]
 LDCM0441  CL50 HEK-293T C70(0.86)  LDD1645  [18]
 LDCM0443  CL52 HEK-293T C70(0.96)  LDD1646  [18]
 LDCM0444  CL53 HEK-293T C70(0.90)  LDD1647  [18]
 LDCM0445  CL54 HEK-293T C70(1.09)  LDD1648  [18]
 LDCM0446  CL55 HEK-293T C159(0.90); C70(1.04)  LDD1649  [18]
 LDCM0447  CL56 HEK-293T C159(0.68); C70(1.15)  LDD1650  [18]
 LDCM0448  CL57 HEK-293T C159(0.75); C70(1.25)  LDD1651  [18]
 LDCM0449  CL58 HEK-293T C159(0.54); C70(1.04)  LDD1652  [18]
 LDCM0450  CL59 HEK-293T C159(0.49)  LDD1653  [18]
 LDCM0451  CL6 HCT 116 C70(1.38)  LDD0768  [6]
 LDCM0452  CL60 HEK-293T C159(0.52); C70(1.00)  LDD1655  [18]
 LDCM0453  CL61 HCT 116 C70(1.81)  LDD0770  [6]
 LDCM0454  CL62 HCT 116 C70(0.88)  LDD0771  [6]
 LDCM0455  CL63 HCT 116 C70(1.16)  LDD0772  [6]
 LDCM0456  CL64 HCT 116 C70(1.05)  LDD0773  [6]
 LDCM0457  CL65 HCT 116 C70(0.98)  LDD0774  [6]
 LDCM0458  CL66 HCT 116 C70(1.64)  LDD0775  [6]
 LDCM0459  CL67 HCT 116 C70(1.41)  LDD0776  [6]
 LDCM0460  CL68 HCT 116 C70(1.24)  LDD0777  [6]
 LDCM0461  CL69 HCT 116 C70(1.08)  LDD0778  [6]
 LDCM0462  CL7 HCT 116 C70(1.26)  LDD0779  [6]
 LDCM0463  CL70 HCT 116 C70(1.39)  LDD0780  [6]
 LDCM0464  CL71 HCT 116 C70(0.97)  LDD0781  [6]
 LDCM0465  CL72 HCT 116 C70(1.10)  LDD0782  [6]
 LDCM0466  CL73 HCT 116 C70(1.09)  LDD0783  [6]
 LDCM0467  CL74 HCT 116 C70(1.06)  LDD0784  [6]
 LDCM0469  CL76 PaTu 8988t C70(0.63)  LDD1348  [6]
 LDCM0470  CL77 PaTu 8988t C70(0.66)  LDD1349  [6]
 LDCM0471  CL78 PaTu 8988t C70(0.72)  LDD1350  [6]
 LDCM0472  CL79 PaTu 8988t C70(0.92)  LDD1351  [6]
 LDCM0473  CL8 HCT 116 C70(1.50)  LDD0790  [6]
 LDCM0474  CL80 PaTu 8988t C70(0.85)  LDD1353  [6]
 LDCM0475  CL81 PaTu 8988t C70(0.79)  LDD1354  [6]
 LDCM0476  CL82 PaTu 8988t C70(0.91)  LDD1355  [6]
 LDCM0477  CL83 PaTu 8988t C70(1.02)  LDD1356  [6]
 LDCM0478  CL84 PaTu 8988t C70(0.96)  LDD1357  [6]
 LDCM0479  CL85 PaTu 8988t C70(0.86)  LDD1358  [6]
 LDCM0480  CL86 PaTu 8988t C70(0.83)  LDD1359  [6]
 LDCM0481  CL87 PaTu 8988t C70(1.16)  LDD1360  [6]
 LDCM0482  CL88 PaTu 8988t C70(0.99)  LDD1361  [6]
 LDCM0483  CL89 PaTu 8988t C70(0.98)  LDD1362  [6]
 LDCM0484  CL9 HCT 116 C70(1.13)  LDD0801  [6]
 LDCM0485  CL90 PaTu 8988t C70(1.00)  LDD1364  [6]
 LDCM0486  CL91 HCT 116 C70(1.28)  LDD0803  [6]
 LDCM0487  CL92 HCT 116 C70(1.24)  LDD0804  [6]
 LDCM0488  CL93 HCT 116 C70(1.45)  LDD0805  [6]
 LDCM0489  CL94 HCT 116 C70(1.51)  LDD0806  [6]
 LDCM0490  CL95 HCT 116 C70(1.41)  LDD0807  [6]
 LDCM0491  CL96 HCT 116 C70(1.63)  LDD0808  [6]
 LDCM0492  CL97 HCT 116 C70(1.27)  LDD0809  [6]
 LDCM0493  CL98 HCT 116 C70(1.21)  LDD0810  [6]
 LDCM0494  CL99 HCT 116 C70(1.20)  LDD0811  [6]
 LDCM0495  E2913 HEK-293T C70(0.95)  LDD1698  [18]
 LDCM0625  F8 Ramos C159(1.53)  LDD2187  [19]
 LDCM0573  Fragment11 Ramos C159(1.28)  LDD2190  [19]
 LDCM0575  Fragment13 Ramos C159(1.11)  LDD2192  [19]
 LDCM0576  Fragment14 Ramos C159(11.26)  LDD2193  [19]
 LDCM0580  Fragment21 Ramos C159(1.22)  LDD2195  [19]
 LDCM0582  Fragment23 Ramos C159(0.48)  LDD2196  [19]
 LDCM0578  Fragment27 Ramos C159(0.78)  LDD2197  [19]
 LDCM0586  Fragment28 Ramos C159(0.98)  LDD2198  [19]
 LDCM0588  Fragment30 Ramos C159(1.35)  LDD2199  [19]
 LDCM0589  Fragment31 Ramos C159(0.98)  LDD2200  [19]
 LDCM0468  Fragment33 HCT 116 C70(1.31)  LDD0785  [6]
 LDCM0427  Fragment51 HCT 116 C70(0.85)  LDD0744  [6]
 LDCM0614  Fragment56 Ramos C159(1.09)  LDD2205  [19]
 LDCM0022  KB02 HEK-293T C70(0.78)  LDD1492  [18]
 LDCM0023  KB03 HEK-293T C70(0.97)  LDD1497  [18]
 LDCM0024  KB05 HMCB C70(1.57)  LDD3312  [20]
 LDCM0497  Nucleophilic fragment 11b MDA-MB-231 C159(1.16)  LDD2090  [4]
 LDCM0499  Nucleophilic fragment 12b MDA-MB-231 C159(1.05)  LDD2092  [4]
 LDCM0500  Nucleophilic fragment 13a MDA-MB-231 C159(1.03)  LDD2093  [4]
 LDCM0504  Nucleophilic fragment 15a MDA-MB-231 C159(0.40)  LDD2097  [4]
 LDCM0506  Nucleophilic fragment 16a MDA-MB-231 C159(0.76)  LDD2099  [4]
 LDCM0514  Nucleophilic fragment 20a MDA-MB-231 C159(0.78)  LDD2107  [4]
 LDCM0526  Nucleophilic fragment 26a MDA-MB-231 C159(1.31)  LDD2119  [4]
 LDCM0543  Nucleophilic fragment 38 MDA-MB-231 C159(0.76)  LDD2136  [4]
 LDCM0546  Nucleophilic fragment 40 MDA-MB-231 C159(0.65)  LDD2140  [4]
 LDCM0547  Nucleophilic fragment 41 MDA-MB-231 C159(1.61)  LDD2141  [4]
 LDCM0556  Nucleophilic fragment 8a MDA-MB-231 C159(0.54)  LDD2150  [4]
 LDCM0559  Nucleophilic fragment 9b MDA-MB-231 C159(1.21)  LDD2153  [4]
 LDCM0627  NUDT7-COV-1 HEK-293T C70(1.07)  LDD2206  [21]
 LDCM0628  OTUB2-COV-1 HEK-293T C70(1.14); C159(0.66)  LDD2207  [21]
 LDCM0131  RA190 MM1.R C159(1.51); C70(0.60)  LDD0304  [22]

References

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Mass spectrometry data entry: PXD028270
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Mass spectrometry data entry: PXD039908 , PXD029761
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Mass spectrometry data entry: PXD044625
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Mass spectrometry data entry: PXD028853
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Mass spectrometry data entry: PXD029255
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Mass spectrometry data entry: PXD027758 , PXD027755 , PXD027760 , PXD027762 , PXD027756 , PXD027591 , PXD007149 , PXD030064 , PXD032392 , PXD027789 , PXD027767 , PXD027764
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Mass spectrometry data entry: PXD041264
14 Large-scale chemoproteomics expedites ligand discovery and predicts ligand behavior in cells. Science. 2024 Apr 26;384(6694):eadk5864. doi: 10.1126/science.adk5864. Epub 2024 Apr 26.
Mass spectrometry data entry: PXD041587
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Mass spectrometry data entry: PXD025652
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Mass spectrometry data entry: PXD007570
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Mass spectrometry data entry: PXD044402
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Mass spectrometry data entry: PXD027578
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Mass spectrometry data entry: PXD047840
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