Details of the Competitor

General Information of Competitor

Competitor ID
LDCM0102
Competitor Name
BDHI 8
Structure
2D MOL
Ro5 Violations (Lipinski): 0 Molecular Weight (mw) 405.092
Lipid-water partition coefficient (xlogp) 4.16
Rotatable Bond Count (rotbonds) 2
Hydrogen Bond Donor Count (hbonddonor) 1
Hydrogen Bond Acceptor Count (hbondacc) 3
Chemical Identifiers
Formula
C12H7BrF6N2O2
Canonical SMILES
O=C(Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C1CC(Br)=NO1
InChI
InChI=1S/C12H7BrF6N2O2/c13-9-4-8(23-21-9)10(22)20-7-2-5(11(14,15)16)1-6(3-7)12(17,18)19/h1-3,8H,4H2,(H,20,22)
InChIKey
PDHWJQDCCMPLCN-UHFFFAOYSA-N

The Competitor Interaction Atlas

Probe(s) Related This Competitor

ABPP Probe
Click To Hide/Show 1 Probe Related to This Competitor
Probe Name Structure Concentration Cell-system Ref
DBIA
 Probe Info  		50 mM Human T acute lymphoblastic leukemia cell lysate (Jurkat) [1]

Target(s) List of this Competitor

97 Enzyme Competed by This Competitor
Target Name Target ID Binding Ratio Interaction ID
2-amino-3-ketobutyrate coenzyme A ligase, mitochondrial (GCAT) LDTP01268 34.90  LDD0204 
2-hydroxyacyl-CoA lyase 2 (ILVBL) LDTP00032 10.99  LDD0204 
2-oxoglutarate dehydrogenase complex component E1 (OGDH) LDTP05341 4.20  LDD0204 
26S proteasome non-ATPase regulatory subunit 13 (PSMD13) LDTP13667 5.32  LDD0204 
Actin, cytoplasmic 1 (ACTB) LDTP04876 1,125.59; 1,125.59  LDD0204 
Archaemetzincin-2 (AMZ2) LDTP17590 9.42  LDD0204 
ATP-dependent 6-phosphofructokinase, platelet type (PFKP) LDTP05314 4.14  LDD0204 
ATP-dependent RNA helicase DHX33 (DHX33) LDTP11991 11.01  LDD0204 
C-1-tetrahydrofolate synthase, cytoplasmic (MTHFD1) LDTP02580 4.47; 4.47; 4.82  LDD0204 
Cell cycle checkpoint control protein RAD9A (RAD9A) LDTP10929 5.21  LDD0204 
Centromere-associated protein E (CENPE) LDTP05343 14.67  LDD0204 
Chromosome-associated kinesin KIF4A (KIF4A) LDTP01539 4.38  LDD0204 
Cleavage and polyadenylation specificity factor subunit 3 (CPSF3) LDTP13449 18.80  LDD0204 
DCN1-like protein 5 (DCUN1D5) LDTP11199 18.43; 18.43  LDD0204 
DNA dC->dU-editing enzyme APOBEC-3C (APOBEC3C) LDTP12539 30.67  LDD0204 
DNA replication licensing factor MCM6 (MCM6) LDTP06150 34.45; 34.45  LDD0204 
DNA topoisomerase 3-beta-1 (TOP3B) LDTP01732 13.65  LDD0204 
DNA-binding protein SMUBP-2 (IGHMBP2) LDTP03862 4.62  LDD0204 
DNA-dependent protein kinase catalytic subunit (PRKDC) LDTP05136 26.99; 26.99  LDD0204 
DNA-directed RNA polymerase I subunit RPA43 (POLR1F) LDTP14904 11.84  LDD0204 
DNA-directed RNA polymerase, mitochondrial (POLRMT) LDTP00267 6.81  LDD0204 
DnaJ homolog subfamily C member 10 (DNAJC10) LDTP08590 7.78  LDD0204 
E3 SUMO-protein ligase ZBED1 (ZBED1) LDTP01746 6.68  LDD0204 
E3 ubiquitin-protein ligase CHIP (STUB1) LDTP13655 13.47  LDD0204 
E3 ubiquitin-protein ligase HUWE1 (HUWE1) LDTP08135 8.27  LDD0204 
E3 ubiquitin-protein ligase LRSAM1 (LRSAM1) LDTP07672 15.86  LDD0204 
E3 ubiquitin-protein ligase Mdm2 (MDM2) LDTP05267 8.80  LDD0204 
E3 ubiquitin-protein ligase RNF8 (RNF8) LDTP01390 19.10  LDD0204 
E3 ubiquitin-protein ligase UHRF2 (UHRF2) LDTP10698 8.42  LDD0204 
Electron transfer flavoprotein subunit beta (ETFB) LDTP03849 8.66  LDD0204 
Endoribonuclease Dicer (DICER1) LDTP13733 5.39  LDD0204 
Eukaryotic translation initiation factor 2-alpha kinase 1 (EIF2AK1) LDTP11083 4.57  LDD0204 
Exonuclease 1 (EXO1) LDTP13751 5.06  LDD0204 
Exosome complex component MTR3 (EXOSC6) LDTP07054 18.22  LDD0204 
Exosome complex component RRP43 (EXOSC8) LDTP10110 10.60  LDD0204 
FAD synthase (FLAD1) LDTP09200 5.02  LDD0204 
Farnesyl pyrophosphate synthase (FDPS) LDTP02721 16.89  LDD0204 
FAST kinase domain-containing protein 1, mitochondrial (FASTKD1) LDTP06919 4.59  LDD0204 
Fatty acid synthase (FASN) LDTP04243 14.17; 14.17  LDD0204 
Glucose 1,6-bisphosphate synthase (PGM2L1) LDTP07561 5.47  LDD0204 
Glutaminase kidney isoform, mitochondrial (GLS) LDTP01465 42.16; 17.75  LDD0204 
GTPase IMAP family member 2 (GIMAP2) LDTP13219 8.51  LDD0204 
Helicase MOV-10 (MOV10) LDTP12233 6.75  LDD0204 
Histidine--tRNA ligase, cytoplasmic (HARS1) LDTP02602 23.58  LDD0204 
Histone deacetylase 1 (HDAC1) LDTP05918 5.29  LDD0204 
Histone deacetylase 3 (HDAC3) LDTP00622 6.23  LDD0204 
Histone deacetylase 8 (HDAC8) LDTP11433 6.10  LDD0204 
Histone-lysine N-methyltransferase EZH2 (EZH2) LDTP06502 6.73  LDD0204 
Histone-lysine N-methyltransferase, H3 lysine-36 specific (NSD1) LDTP10531 10.69  LDD0204 
Inositol-trisphosphate 3-kinase B (ITPKB) LDTP03409 10.60  LDD0204 
Isocitrate dehydrogenase [NAD] subunit beta, mitochondrial (IDH3B) LDTP00885 4.10  LDD0204 
Kinesin-like protein KIF11 (KIF11) LDTP04519 31.33; 31.33; 8.48  LDD0204 
Kinesin-like protein KIF2A (KIF2A) LDTP00188 24.35; 24.35  LDD0204 
Kynurenine--oxoglutarate transaminase 3 (KYAT3) LDTP07763 10.08  LDD0204 
Lanosterol synthase (LSS) LDTP04183 10.46  LDD0204 
Lymphoid-specific helicase (HELLS) LDTP12552 42.74  LDD0204 
Lysine-specific demethylase 5C (KDM5C) LDTP03939 21.22; 21.22  LDD0204 
Methionine aminopeptidase 1 (METAP1) LDTP04565 4.74  LDD0204 
Mitotic checkpoint serine/threonine-protein kinase BUB1 (BUB1) LDTP00837 18.67  LDD0204 
Monofunctional C1-tetrahydrofolate synthase, mitochondrial (MTHFD1L) LDTP07651 6.75  LDD0204 
N-acetyltransferase ESCO1 (ESCO1) LDTP06971 17.07  LDD0204 
NADH dehydrogenase iron-sulfur protein 2, mitochondrial (NDUFS2) LDTP01168 14.98  LDD0204 
NK-tumor recognition protein (NKTR) LDTP03536 11.60  LDD0204 
Non-receptor tyrosine-protein kinase TYK2 (TYK2) LDTP03497 13.34  LDD0204 
Nuclear receptor-binding protein (NRBP1) LDTP13313 17.34  LDD0204 
Peptide-N(4)-(N-acetyl-beta-glucosaminyl)asparagine amidase (NGLY1) LDTP10429 17.89; 17.89  LDD0204 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform (PIK3CB) LDTP03979 13.22  LDD0204 
Polyribonucleotide nucleotidyltransferase 1, mitochondrial (PNPT1) LDTP09390 5.31  LDD0204 
Probable E3 ubiquitin-protein ligase HERC1 (HERC1) LDTP06461 29.38  LDD0204 
Proteasome subunit beta type-3 (PSMB3) LDTP04284 4.08  LDD0204 
Protein mono-ADP-ribosyltransferase PARP9 (PARP9) LDTP08610 8.23  LDD0204 
Protein NDRG3 (NDRG3) LDTP18530 25.17  LDD0204 
Protein O-GlcNAcase (OGA) LDTP00988 4.97  LDD0204 
Ras-related protein Rab-22A (RAB22A) LDTP13513 14.13  LDD0204 
Regulator of telomere elongation helicase 1 (RTEL1) LDTP12878 22.60  LDD0204 
Ribonuclease P protein subunit p38 (RPP38) LDTP05099 19.92  LDD0204 
RNA cytidine acetyltransferase (NAT10) LDTP11690 7.37; 7.37  LDD0204 
Selenocysteine-specific elongation factor (EEFSEC) LDTP14723 16.30  LDD0204 
Separin (ESPL1) LDTP06175 4.26  LDD0204 
Serine hydroxymethyltransferase, mitochondrial (SHMT2) LDTP03689 4.44  LDD0204 
Serine/threonine-protein kinase 16 (STK16) LDTP01298 6.93  LDD0204 
Serine/threonine-protein kinase MARK2 (MARK2) LDTP07930 13.77  LDD0204 
Serine/threonine-protein phosphatase 2A regulatory subunit B'' subunit beta (PPP2R3B) LDTP14142 6.68  LDD0204 
Serine/threonine-protein phosphatase PP1-beta catalytic subunit (PPP1CB) LDTP04960 4.43  LDD0204 
Short/branched chain specific acyl-CoA dehydrogenase, mitochondrial (ACADSB) LDTP04072 5.28  LDD0204 
Signal recognition particle subunit SRP54 (SRP54) LDTP04890 19.78  LDD0204 
Sterol-4-alpha-carboxylate 3-dehydrogenase, decarboxylating (NSDHL) LDTP06455 15.31  LDD0204 
T-cell differentiation antigen CD6 (CD6) LDTP03524 5.52  LDD0204 
Transcription activator BRG1 (SMARCA4) LDTP04422 5.25  LDD0204 
tRNA N6-adenosine threonylcarbamoyltransferase, mitochondrial (OSGEPL1) LDTP11913 11.98  LDD0204 
Tubulin alpha-4A chain (TUBA4A) LDTP05075 50.09  LDD0204 
Tyrosine-protein kinase Blk (BLK) LDTP04414 17.88  LDD0204 
Tyrosine-protein phosphatase non-receptor type 9 (PTPN9) LDTP04046 5.33  LDD0204 
Ubiquitin-protein ligase E3A (UBE3A) LDTP05446 10.65  LDD0204 
Ubiquitin-protein ligase E3B (UBE3B) LDTP15246 4.96  LDD0204 
Unconventional myosin-VI (MYO6) LDTP13609 5.60  LDD0204 
WW domain-containing oxidoreductase (WWOX) LDTP12888 5.72  LDD0204 
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⏷ Show the Full List of 97 Enzyme
18 Transporter and channel Competed by This Competitor
Target Name Target ID Binding Ratio Interaction ID
AP-4 complex subunit beta-1 (AP4B1) LDTP14232 5.19  LDD0204 
Apoptotic protease-activating factor 1 (APAF1) LDTP00411 5.44; 21.44  LDD0204 
Cell division cycle protein 20 homolog (CDC20) LDTP05662 6.62; 14.86  LDD0204 
Importin-11 (IPO11) LDTP13322 7.78  LDD0204 
Importin-5 (IPO5) LDTP00266 4.36; 4.36; 4.44  LDD0204 
Intraflagellar transport protein 122 homolog (IFT122) LDTP12176 9.68  LDD0204 
Intraflagellar transport protein 88 homolog (IFT88) LDTP05747 32.19  LDD0204 
Microtubule-actin cross-linking factor 1, isoforms 1/2/3/4/5 (MACF1) LDTP13698 4.82  LDD0204 
Nuclear envelope pore membrane protein POM 121C (POM121C) LDTP00127 22.10  LDD0204 
Nuclear pore complex protein Nup133 (NUP133) LDTP09579 22.54  LDD0204 
Nuclear pore complex protein Nup153 (NUP153) LDTP04309 15.04; 15.04  LDD0204 
Nuclear pore complex protein Nup160 (NUP160) LDTP05642 6.13  LDD0204 
Protein mago nashi homolog (MAGOH) LDTP04920 9.35  LDD0204 
Small ribosomal subunit protein RACK1 (RACK1) LDTP05057 6.47; 6.47  LDD0204 
SUN domain-containing protein 2 (SUN2) LDTP13256 20.31  LDD0204 
T-complex protein 1 subunit delta (CCT4) LDTP04391 12.89  LDD0204 
Thioredoxin-interacting protein (TXNIP) LDTP11873 11.35  LDD0204 
THO complex subunit 2 (THOC2) LDTP09279 15.17  LDD0204 
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⏷ Show the Full List of 18 Transporter and channel
11 Transcription factor Competed by This Competitor
Target Name Target ID Binding Ratio Interaction ID
Basic helix-loop-helix ARNT-like protein 2 (BMAL2) LDTP09732 7.52  LDD0204 
CCAAT/enhancer-binding protein zeta (CEBPZ) LDTP14809 5.90  LDD0204 
Forkhead box protein K1 (FOXK1) LDTP05201 7.96  LDD0204 
Leucine-rich repeat flightless-interacting protein 1 (LRRFIP1) LDTP06748 12.85; 12.85  LDD0204 
Myb-related protein B (MYBL2) LDTP02485 7.15  LDD0204 
NF-kappa-B-repressing factor (NKRF) LDTP00576 14.31; 15.78  LDD0204 
Nuclear receptor subfamily 2 group C member 2 (NR2C2) LDTP04228 21.50  LDD0204 
Transcription factor E2F4 (E2F4) LDTP06519 4.18  LDD0204 
Uncharacterized protein C8orf76 (C8orf76) LDTP19877 18.97  LDD0204 
Zinc finger and BTB domain-containing protein 11 (ZBTB11) LDTP14540 22.28  LDD0204 
Zinc finger protein 687 (ZNF687) LDTP08771 8.80  LDD0204 
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⏷ Show the Full List of 11 Transcription factor
98 Other Competed by This Competitor
Target Name Target ID Binding Ratio Interaction ID
Actin-like protein 6A (ACTL6A) LDTP01756 6.56  LDD0204 
Actin-related protein 5 (ACTR5) LDTP12095 26.64  LDD0204 
Activating signal cointegrator 1 complex subunit 2 (ASCC2) LDTP11766 4.87  LDD0204 
Ankyrin repeat and KH domain-containing protein 1 (ANKHD1) LDTP08573 24.56  LDD0204 
Ankyrin repeat and LEM domain-containing protein 2 (ANKLE2) LDTP08364 13.97  LDD0204 
Ankyrin repeat and SOCS box protein 1 (ASB1) LDTP14096 5.01  LDD0204 
Ankyrin repeat domain-containing protein 12 (ANKRD12) LDTP07652 11.97  LDD0204 
Arf-GAP with coiled-coil, ANK repeat and PH domain-containing protein 2 (ACAP2) LDTP06302 4.69  LDD0204 
Arf-GAP with SH3 domain, ANK repeat and PH domain-containing protein 2 (ASAP2) LDTP00688 14.52  LDD0204 
Armadillo repeat-containing protein 6 (ARMC6) LDTP15101 6.27  LDD0204 
BLOC-2 complex member HPS3 (HPS3) LDTP09994 4.75  LDD0204 
Centromere protein F (CENPF) LDTP04258 15.13  LDD0204 
Centrosomal protein of 76 kDa (CEP76) LDTP09308 9.36  LDD0204 
Cleavage and polyadenylation specificity factor subunit 1 (CPSF1) LDTP05626 8.97; 13.69  LDD0204 
CLIP-associating protein 1 (CLASP1) LDTP08062 12.47  LDD0204 
CLIP-associating protein 2 (CLASP2) LDTP01129 24.61  LDD0204 
Coilin (COIL) LDTP03853 5.21  LDD0204 
Condensin complex subunit 1 (NCAPD2) LDTP06281 37.59  LDD0204 
Condensin complex subunit 3 (NCAPG) LDTP11040 8.61; 8.61  LDD0204 
Conserved oligomeric Golgi complex subunit 2 (COG2) LDTP06201 13.70  LDD0204 
Constitutive coactivator of PPAR-gamma-like protein 1 (FAM120A) LDTP12883 14.21; 14.21  LDD0204 
Corepressor interacting with RBPJ 1 (CIR1) LDTP08354 23.04  LDD0204 
cTAGE family member 2 (CTAGE1) LDTP18264 14.01  LDD0204 
CUGBP Elav-like family member 1 (CELF1) LDTP09913 4.03  LDD0204 
Cytoplasmic polyadenylation element-binding protein 1 (CPEB1) LDTP11521 6.50  LDD0204 
DNA mismatch repair protein Mlh1 (MLH1) LDTP03902 4.24  LDD0204 
DNA topoisomerase 2-binding protein 1 (TOPBP1) LDTP09791 5.62  LDD0204 
Dynein axonemal assembly factor 5 (DNAAF5) LDTP08387 4.61  LDD0204 
E3 ubiquitin-protein ligase RNFT2 (RNFT2) LDTP15719 14.60  LDD0204 
Elongator complex protein 6 (ELP6) LDTP05607 13.95  LDD0204 
Eukaryotic translation initiation factor 4 gamma 3 (EIF4G3) LDTP00766 14.07  LDD0204 
Fanconi anemia group I protein (FANCI) LDTP12680 26.29  LDD0204 
Gamma-parvin (PARVG) LDTP12183 49.13  LDD0204 
GRIP and coiled-coil domain-containing protein 2 (GCC2) LDTP08543 13.04  LDD0204 
HEAT repeat-containing protein 5B (HEATR5B) LDTP13038 7.01  LDD0204 
Heterogeneous nuclear ribonucleoprotein U (HNRNPU) LDTP05259 33.36; 4.49  LDD0204 
Integrator complex subunit 1 (INTS1) LDTP08785 4.83  LDD0204 
Integrator complex subunit 3 (INTS3) LDTP07333 16.18  LDD0204 
Integrator complex subunit 4 (INTS4) LDTP10402 21.75; 24.32  LDD0204 
Kelch-like protein 26 (KLHL26) LDTP14946 4.49  LDD0204 
Kinesin-associated protein 3 (KIFAP3) LDTP09902 36.23  LDD0204 
La-related protein 4B (LARP4B) LDTP09820 4.38  LDD0204 
Large ribosomal subunit protein eL36 (RPL36) LDTP14012 4.00  LDD0204 
Large ribosomal subunit protein uL14 (RPL23) LDTP05008 7.62  LDD0204 
Large ribosomal subunit protein uL22 (RPL17) LDTP02961 4.68  LDD0204 
MAD2L1-binding protein (MAD2L1BP) LDTP06276 17.44  LDD0204 
Mediator of RNA polymerase II transcription subunit 16 (MED16) LDTP13924 4.12  LDD0204 
Midasin (MDN1) LDTP12619 23.74  LDD0204 
Multiple myeloma tumor-associated protein 2 (MMTAG2) LDTP11223 10.48  LDD0204 
Next to BRCA1 gene 1 protein (NBR1) LDTP06159 10.28  LDD0204 
Nonsense-mediated mRNA decay factor SMG8 (SMG8) LDTP09112 6.84  LDD0204 
Nucleotide-binding oligomerization domain-containing protein 1 (NOD1) LDTP13795 15.99  LDD0204 
Origin recognition complex subunit 5 (ORC5) LDTP00900 4.60  LDD0204 
PH and SEC7 domain-containing protein 3 (PSD3) LDTP12831 21.41  LDD0204 
PH-interacting protein (PHIP) LDTP09660 24.45  LDD0204 
PHD finger protein 6 (PHF6) LDTP08552 6.56; 6.56  LDD0204 
Phosducin-like protein (PDCL) LDTP05846 7.99  LDD0204 
Pleckstrin homology domain-containing family A member 2 (PLEKHA2) LDTP12155 12.17  LDD0204 
Programmed cell death protein 2 (PDCD2) LDTP06525 13.73  LDD0204 
Proteasome assembly chaperone 1 (PSMG1) LDTP01608 6.93  LDD0204 
Protein asteroid homolog 1 (ASTE1) LDTP19259 16.62  LDD0204 
Protein C12orf4 (C12orf4) LDTP18456 19.06  LDD0204 
Protein C19orf12 (C19orf12) LDTP12592 7.80  LDD0204 
Protein CIP2A (CIP2A) LDTP09383 4.61  LDD0204 
Protein MMS22-like (MMS22L) LDTP07814 4.38; 19.25  LDD0204 
Protein pelota homolog (PELO) LDTP11138 11.70  LDD0204 
Protein RRP5 homolog (PDCD11) LDTP06186 4.20  LDD0204 
Putative rhophilin-2-like protein RHPN2P1 (RHPN2P1) LDTP18877 18.40  LDD0204 
RAB6A-GEF complex partner protein 2 (RGP1) LDTP09790 7.49  LDD0204 
Raftlin (RFTN1) LDTP06193 9.96  LDD0204 
RAS guanyl-releasing protein 1 (RASGRP1) LDTP01550 4.37  LDD0204 
Rho GTPase-activating protein 19 (ARHGAP19) LDTP06256 10.68  LDD0204 
Rho GTPase-activating protein 9 (ARHGAP9) LDTP11128 4.40  LDD0204 
Rho guanine nucleotide exchange factor 1 (ARHGEF1) LDTP09917 4.49  LDD0204 
Rho guanine nucleotide exchange factor 6 (ARHGEF6) LDTP06299 7.13  LDD0204 
Ribosomal RNA processing protein 1 homolog B (RRP1B) LDTP06182 4.41  LDD0204 
RNA polymerase II-associated protein 1 (RPAP1) LDTP11327 4.12  LDD0204 
RNA-binding protein 43 (RBM43) LDTP19567 8.32  LDD0204 
Rotatin (RTTN) LDTP08303 6.54  LDD0204 
RRP15-like protein (RRP15) LDTP18570 14.29  LDD0204 
Serine/arginine-rich splicing factor 3 (SRSF3) LDTP05197 5.99  LDD0204 
Small ribosomal subunit protein uS7 (RPS5) LDTP04110 5.50  LDD0204 
Spermatid perinuclear RNA-binding protein (STRBP) LDTP10815 4.41  LDD0204 
Stalled ribosome sensor GCN1 (GCN1) LDTP09821 16.94; 10.51  LDD0204 
Sterile alpha motif domain-containing protein 1 (SAMD1) LDTP07638 15.33  LDD0204 
Symplekin (SYMPK) LDTP09878 6.09  LDD0204 
Telomere length regulation protein TEL2 homolog (TELO2) LDTP14072 26.46; 6.76  LDD0204 
Telomeric repeat-binding factor 2 (TERF2) LDTP06412 27.15  LDD0204 
Tetratricopeptide repeat protein 21B (TTC21B) LDTP08073 9.49  LDD0204 
Tetratricopeptide repeat protein 27 (TTC27) LDTP19505 18.68; 18.68  LDD0204 
Transcription initiation factor TFIID subunit 2 (TAF2) LDTP07517 8.95  LDD0204 
Translation initiation factor eIF2B subunit delta (EIF2B4) LDTP13318 4.16  LDD0204 
Transmembrane protein 209 (TMEM209) LDTP18272 7.14  LDD0204 
Transport and Golgi organization protein 6 homolog (TANGO6) LDTP18348 13.71  LDD0204 
Ubiquitin-ribosomal protein eS31 fusion protein (RPS27A) LDTP05033 4.63; 4.63; 4.63  LDD0204 
WD repeat domain-containing protein 83 (WDR83) LDTP11141 11.71  LDD0204 
Wings apart-like protein homolog (WAPL) LDTP08094 21.22  LDD0204 
Zinc finger ZZ-type and EF-hand domain-containing protein 1 (ZZEF1) LDTP00687 13.01; 4.46  LDD0204 
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⏷ Show the Full List of 98 Other

Full Information of The Labelling Profiles of This Competitor

Quantification: Probe vs (Probe+Competitor)
  
Experiment 1 Reporting the Labelling Profiles of This Probe
REF [1]
Probe concentration 50 mM
Quantitative Method TMT
Competitor Name BDHI 8
Competitor Concentration 50 mM
In Vitro Experiment Model Model Type
Cell lysate
Derived Tissue
Bone marrow
Disease Model T acute lymphoblastic leukemia [ICD-11:2A90]
Model Name Human T acute lymphoblastic leukemia cell lysate (Jurkat)
Interaction Atlas ID  LDD0204  Download The Altas

References

1 Covalent Inhibition by a Natural Product-Inspired Latent Electrophile. J Am Chem Soc. 2023 May 24;145(20):11097-11109. doi: 10.1021/jacs.3c00598. Epub 2023 May 15.