General Information of Target

Target ID LDTP11199
Target Name DCN1-like protein 5 (DCUN1D5)
Gene Name DCUN1D5
Gene ID 84259
Synonyms
SCCRO5; DCN1-like protein 5; DCNL5; DCUN1 domain-containing protein 5; Defective in cullin neddylation protein 1-like protein 5; Squamous cell carcinoma-related oncogene 5
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MAFWCQRDSYAREFTTTVVSCCPAELQTEGSNGKKEVLSGFQVVLEDTVLFPEGGGQPDD
RGTINDISVLRVTRRGEQADHFTQTPLDPGSQVLVRVDWERRFDHMQQHSGQHLITAVAD
HLFKLKTTSWELGRFRSAIELDTPSMTAEQVAAIEQSVNEKIRDRLPVNVRELSLDDPEV
EQVSGRGLPDDHAGPIRVVNIEGVDSNMCCGTHVSNLSDLQVIKILGTEKGKKNRTNLIF
LSGNRVLKWMERSHGTEKALTALLKCGAEDHVEAVKKLQNSTKILQKNNLNLLRDLAVHI
AHSLRNSPDWGGVVILHRKEGDSEFMNIIANEIGSEETLLFLTVGDEKGGGLFLLAGPPA
SVETLGPRVAEVLEGKGAGKKGRFQGKATKMSRRMEAQALLQDYISTQSAKE
Target Bioclass
Enzyme
Subcellular location
Nucleus
Function
Contributes to the neddylation of all cullins by transferring NEDD8 from N-terminally acetylated NEDD8-conjugating E2s enzyme to different cullin C-terminal domain-RBX complexes which is necessary for the activation of cullin-RING E3 ubiquitin ligases (CRLs). May play a role in DNA damage response and may participate in cell proliferation and anchorage-independent cell growth.
Uniprot ID
Q9BTE7
Ensemble ID
ENST00000260247.10
HGNC ID
HGNC:28409
ChEMBL ID
CHEMBL4295937

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 22 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
m-APA
 Probe Info 
15.00  LDD0402  [1]
Alkylaryl probe 1
 Probe Info 
6.00  LDD0385  [2]
Jackson_1
 Probe Info 
20.00  LDD0122  [3]
C-Sul
 Probe Info 
6.15  LDD0066  [4]
TH211
 Probe Info 
Y144(20.00)  LDD0257  [5]
STPyne
 Probe Info 
K124(9.43); K139(0.92)  LDD0277  [6]
JZ128-DTB
 Probe Info 
N.A.  LDD0462  [7]
BTD
 Probe Info 
C25(0.38)  LDD2116  [8]
EA-probe
 Probe Info 
N.A.  LDD0440  [9]
DBIA
 Probe Info 
C115(6.00); C51(2.58); C117(1.12)  LDD0080  [10]
ATP probe
 Probe Info 
K139(0.00); K8(0.00)  LDD0199  [11]
N1
 Probe Info 
E119(0.00); K120(0.00)  LDD0245  [12]
IA-alkyne
 Probe Info 
N.A.  LDD0162  [13]
Lodoacetamide azide
 Probe Info 
N.A.  LDD0037  [14]
WYneN
 Probe Info 
N.A.  LDD0021  [15]
ENE
 Probe Info 
N.A.  LDD0006  [15]
IPM
 Probe Info 
C117(0.00); C115(0.00); C31(0.00)  LDD0005  [15]
NHS
 Probe Info 
N.A.  LDD0010  [15]
TFBX
 Probe Info 
N.A.  LDD0148  [16]
VSF
 Probe Info 
N.A.  LDD0007  [15]
Ox-W18
 Probe Info 
N.A.  LDD2175  [17]
AOyne
 Probe Info 
15.00  LDD0443  [18]
PAL-AfBPP Probe
Click To Hide/Show 30 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
C003
 Probe Info 
13.00  LDD1713  [19]
C004
 Probe Info 
5.70  LDD1714  [19]
C022
 Probe Info 
15.78  LDD1728  [19]
C049
 Probe Info 
5.06  LDD1747  [19]
C055
 Probe Info 
13.83  LDD1752  [19]
C094
 Probe Info 
34.54  LDD1785  [19]
C106
 Probe Info 
30.27  LDD1793  [19]
C159
 Probe Info 
54.95  LDD1839  [19]
C160
 Probe Info 
7.84  LDD1840  [19]
C161
 Probe Info 
9.92  LDD1841  [19]
C187
 Probe Info 
20.25  LDD1865  [19]
C191
 Probe Info 
11.08  LDD1868  [19]
C193
 Probe Info 
20.68  LDD1869  [19]
C201
 Probe Info 
29.04  LDD1877  [19]
C213
 Probe Info 
36.76  LDD1887  [19]
C233
 Probe Info 
12.91  LDD1906  [19]
C249
 Probe Info 
12.13  LDD1922  [19]
C264
 Probe Info 
28.44  LDD1935  [19]
C278
 Probe Info 
89.88  LDD1948  [19]
C280
 Probe Info 
12.82  LDD1950  [19]
C282
 Probe Info 
99.73  LDD1952  [19]
C284
 Probe Info 
38.85  LDD1954  [19]
C350
 Probe Info 
30.70  LDD2011  [19]
C362
 Probe Info 
41.93  LDD2023  [19]
C364
 Probe Info 
21.86  LDD2025  [19]
C382
 Probe Info 
8.82  LDD2041  [19]
C386
 Probe Info 
6.96  LDD2045  [19]
C403
 Probe Info 
23.59  LDD2061  [19]
C413
 Probe Info 
21.86  LDD2069  [19]
Alk-rapa
 Probe Info 
6.22  LDD0213  [20]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0214  AC1 HCT 116 C115(1.00); C117(0.93); C51(0.63)  LDD0531  [10]
 LDCM0215  AC10 HCT 116 C115(0.74); C117(0.74); C51(0.79)  LDD0532  [10]
 LDCM0216  AC100 HCT 116 C115(0.56); C117(0.59); C51(0.42)  LDD0533  [10]
 LDCM0217  AC101 HCT 116 C115(0.52); C117(0.56); C51(0.52)  LDD0534  [10]
 LDCM0218  AC102 HCT 116 C115(0.57); C117(0.59); C51(0.48)  LDD0535  [10]
 LDCM0219  AC103 HCT 116 C115(0.44); C117(0.47); C51(0.34)  LDD0536  [10]
 LDCM0220  AC104 HCT 116 C115(0.52); C117(0.55); C51(0.41)  LDD0537  [10]
 LDCM0221  AC105 HCT 116 C115(0.43); C117(0.46); C51(0.38)  LDD0538  [10]
 LDCM0222  AC106 HCT 116 C115(0.48); C117(0.50); C51(0.41)  LDD0539  [10]
 LDCM0223  AC107 HCT 116 C115(0.52); C117(0.52); C51(0.36)  LDD0540  [10]
 LDCM0224  AC108 HCT 116 C115(0.60); C117(0.67); C51(0.77)  LDD0541  [10]
 LDCM0225  AC109 HCT 116 C115(0.64); C117(0.68); C51(0.65)  LDD0542  [10]
 LDCM0226  AC11 HCT 116 C115(0.70); C117(0.70); C51(0.84)  LDD0543  [10]
 LDCM0227  AC110 HCT 116 C115(0.51); C117(0.57); C51(0.47)  LDD0544  [10]
 LDCM0228  AC111 HCT 116 C115(0.55); C117(0.57); C51(0.52)  LDD0545  [10]
 LDCM0229  AC112 HCT 116 C115(0.44); C117(0.49); C51(0.39)  LDD0546  [10]
 LDCM0230  AC113 HCT 116 C115(0.93); C117(0.93)  LDD0547  [10]
 LDCM0231  AC114 HCT 116 C115(0.66); C117(0.65)  LDD0548  [10]
 LDCM0232  AC115 HCT 116 C115(0.59); C117(0.59)  LDD0549  [10]
 LDCM0233  AC116 HCT 116 C115(0.56); C117(0.56)  LDD0550  [10]
 LDCM0234  AC117 HCT 116 C115(0.72); C117(0.73)  LDD0551  [10]
 LDCM0235  AC118 HCT 116 C115(0.78); C117(0.78)  LDD0552  [10]
 LDCM0236  AC119 HCT 116 C115(0.73); C117(0.74)  LDD0553  [10]
 LDCM0237  AC12 HCT 116 C115(0.95); C117(0.95); C51(0.96)  LDD0554  [10]
 LDCM0238  AC120 HCT 116 C115(0.65); C117(0.63)  LDD0555  [10]
 LDCM0239  AC121 HCT 116 C115(0.94); C117(0.95)  LDD0556  [10]
 LDCM0240  AC122 HCT 116 C115(0.89); C117(0.87)  LDD0557  [10]
 LDCM0241  AC123 HCT 116 C115(1.00); C117(1.03)  LDD0558  [10]
 LDCM0242  AC124 HCT 116 C115(0.92); C117(0.92)  LDD0559  [10]
 LDCM0243  AC125 HCT 116 C115(0.77); C117(0.75)  LDD0560  [10]
 LDCM0244  AC126 HCT 116 C115(0.69); C117(0.69)  LDD0561  [10]
 LDCM0245  AC127 HCT 116 C115(0.70); C117(0.70)  LDD0562  [10]
 LDCM0246  AC128 HCT 116 C115(1.26); C117(1.28)  LDD0563  [10]
 LDCM0247  AC129 HCT 116 C115(1.30); C117(1.20)  LDD0564  [10]
 LDCM0249  AC130 HCT 116 C115(1.04); C117(1.09)  LDD0566  [10]
 LDCM0250  AC131 HCT 116 C115(1.29); C117(1.20)  LDD0567  [10]
 LDCM0251  AC132 HCT 116 C115(1.21); C117(1.21)  LDD0568  [10]
 LDCM0252  AC133 HCT 116 C115(1.07); C117(1.07)  LDD0569  [10]
 LDCM0253  AC134 HCT 116 C115(0.94); C117(1.07)  LDD0570  [10]
 LDCM0254  AC135 HCT 116 C115(1.02); C117(1.05)  LDD0571  [10]
 LDCM0255  AC136 HCT 116 C115(0.95); C117(1.08)  LDD0572  [10]
 LDCM0256  AC137 HCT 116 C115(1.04); C117(1.07)  LDD0573  [10]
 LDCM0257  AC138 HCT 116 C115(0.90); C117(0.95)  LDD0574  [10]
 LDCM0258  AC139 HCT 116 C115(0.93); C117(1.07)  LDD0575  [10]
 LDCM0259  AC14 HCT 116 C115(0.76); C117(0.76); C51(0.72)  LDD0576  [10]
 LDCM0260  AC140 HCT 116 C115(0.89); C117(1.06)  LDD0577  [10]
 LDCM0261  AC141 HCT 116 C115(0.86); C117(1.02)  LDD0578  [10]
 LDCM0262  AC142 HCT 116 C115(1.33); C117(1.26)  LDD0579  [10]
 LDCM0263  AC143 HCT 116 C115(0.91); C117(0.91); C51(1.05)  LDD0580  [10]
 LDCM0264  AC144 HCT 116 C115(0.63); C117(0.64); C51(0.65)  LDD0581  [10]
 LDCM0265  AC145 HCT 116 C51(0.69); C117(0.86); C115(0.90)  LDD0582  [10]
 LDCM0266  AC146 HCT 116 C115(0.68); C117(0.68); C51(0.73)  LDD0583  [10]
 LDCM0267  AC147 HCT 116 C51(0.60); C117(0.67); C115(0.74)  LDD0584  [10]
 LDCM0268  AC148 HCT 116 C51(0.50); C115(0.70); C117(0.73)  LDD0585  [10]
 LDCM0269  AC149 HCT 116 C51(0.49); C115(0.61); C117(0.61)  LDD0586  [10]
 LDCM0270  AC15 HCT 116 C115(0.70); C117(0.70); C51(0.74)  LDD0587  [10]
 LDCM0271  AC150 HCT 116 C117(0.80); C115(0.80); C51(0.90)  LDD0588  [10]
 LDCM0272  AC151 HCT 116 C115(0.72); C117(0.75); C51(1.01)  LDD0589  [10]
 LDCM0273  AC152 HCT 116 C115(0.60); C51(0.62); C117(0.62)  LDD0590  [10]
 LDCM0274  AC153 HCT 116 C51(0.48); C115(0.67); C117(0.68)  LDD0591  [10]
 LDCM0621  AC154 HCT 116 C115(0.72); C117(0.72); C51(0.52)  LDD2158  [10]
 LDCM0622  AC155 HCT 116 C115(0.63); C117(0.64); C51(0.57)  LDD2159  [10]
 LDCM0623  AC156 HCT 116 C115(0.96); C117(0.97); C51(0.89)  LDD2160  [10]
 LDCM0624  AC157 HCT 116 C115(1.02); C117(1.02); C51(1.21)  LDD2161  [10]
 LDCM0276  AC17 HCT 116 C117(0.80); C115(0.84); C51(0.91)  LDD0593  [10]
 LDCM0277  AC18 HCT 116 C51(0.58); C117(0.69); C115(0.70)  LDD0594  [10]
 LDCM0278  AC19 HCT 116 C117(0.77); C115(0.77); C51(0.79)  LDD0595  [10]
 LDCM0279  AC2 HCT 116 C51(0.54); C115(0.83); C117(0.84)  LDD0596  [10]
 LDCM0280  AC20 HCT 116 C115(0.81); C117(0.81); C51(0.83)  LDD0597  [10]
 LDCM0281  AC21 HCT 116 C51(0.73); C117(0.83); C115(0.84)  LDD0598  [10]
 LDCM0282  AC22 HCT 116 C115(0.95); C117(0.96); C51(1.11)  LDD0599  [10]
 LDCM0283  AC23 HCT 116 C51(0.80); C117(0.95); C115(0.96)  LDD0600  [10]
 LDCM0284  AC24 HCT 116 C115(0.92); C117(0.93); C51(1.09)  LDD0601  [10]
 LDCM0285  AC25 HCT 116 C115(0.80); C117(0.86); C51(0.86)  LDD0602  [10]
 LDCM0286  AC26 HCT 116 C51(0.61); C115(0.66); C117(0.81)  LDD0603  [10]
 LDCM0287  AC27 HCT 116 C115(0.59); C51(0.60); C117(0.71)  LDD0604  [10]
 LDCM0288  AC28 HCT 116 C51(0.53); C115(0.59); C117(0.70)  LDD0605  [10]
 LDCM0289  AC29 HCT 116 C115(0.57); C117(0.68); C51(0.74)  LDD0606  [10]
 LDCM0290  AC3 HCT 116 C51(0.85); C117(0.96); C115(1.05)  LDD0607  [10]
 LDCM0291  AC30 HCT 116 C115(0.53); C117(0.60); C51(0.72)  LDD0608  [10]
 LDCM0292  AC31 HCT 116 C51(0.61); C115(0.62); C117(0.72)  LDD0609  [10]
 LDCM0293  AC32 HCT 116 C51(0.45); C115(0.48); C117(0.61)  LDD0610  [10]
 LDCM0294  AC33 HCT 116 C51(0.49); C115(0.52); C117(0.60)  LDD0611  [10]
 LDCM0295  AC34 HCT 116 C51(0.50); C115(0.51); C117(0.62)  LDD0612  [10]
 LDCM0296  AC35 HCT 116 C51(0.57); C117(1.25); C115(1.32)  LDD0613  [10]
 LDCM0297  AC36 HCT 116 C51(0.74); C117(1.09); C115(1.17)  LDD0614  [10]
 LDCM0298  AC37 HCT 116 C51(1.00); C117(1.01); C115(1.12)  LDD0615  [10]
 LDCM0299  AC38 HCT 116 C51(0.75); C115(0.98); C117(0.98)  LDD0616  [10]
 LDCM0300  AC39 HCT 116 C51(0.81); C115(0.98); C117(1.05)  LDD0617  [10]
 LDCM0301  AC4 HCT 116 C51(0.61); C117(0.82); C115(0.88)  LDD0618  [10]
 LDCM0302  AC40 HCT 116 C117(0.92); C115(0.93); C51(0.98)  LDD0619  [10]
 LDCM0303  AC41 HCT 116 C115(0.98); C117(0.99); C51(1.03)  LDD0620  [10]
 LDCM0304  AC42 HCT 116 C115(0.92); C51(0.97); C117(0.97)  LDD0621  [10]
 LDCM0305  AC43 HCT 116 C51(0.78); C115(0.92); C117(0.98)  LDD0622  [10]
 LDCM0306  AC44 HCT 116 C51(0.93); C117(0.97); C115(0.99)  LDD0623  [10]
 LDCM0307  AC45 HCT 116 C51(0.80); C117(0.98); C115(0.99)  LDD0624  [10]
 LDCM0308  AC46 HCT 116 C51(0.88); C115(0.98); C117(1.00)  LDD0625  [10]
 LDCM0309  AC47 HCT 116 C51(0.93); C117(0.93); C115(0.95)  LDD0626  [10]
 LDCM0310  AC48 HCT 116 C51(1.17); C117(1.20); C115(1.25)  LDD0627  [10]
 LDCM0311  AC49 HCT 116 C115(0.89); C117(0.97); C51(1.02)  LDD0628  [10]
 LDCM0312  AC5 HCT 116 C51(0.42); C117(0.84); C115(0.88)  LDD0629  [10]
 LDCM0313  AC50 HCT 116 C51(0.81); C115(0.91); C117(0.95)  LDD0630  [10]
 LDCM0314  AC51 HCT 116 C117(1.21); C115(1.39); C51(1.85)  LDD0631  [10]
 LDCM0315  AC52 HCT 116 C51(0.92); C115(0.97); C117(0.98)  LDD0632  [10]
 LDCM0316  AC53 HCT 116 C51(0.83); C115(0.93); C117(0.96)  LDD0633  [10]
 LDCM0317  AC54 HCT 116 C51(0.81); C115(0.92); C117(0.93)  LDD0634  [10]
 LDCM0318  AC55 HCT 116 C51(0.86); C117(0.94); C115(0.97)  LDD0635  [10]
 LDCM0319  AC56 HCT 116 C51(1.05); C117(1.06); C115(1.07)  LDD0636  [10]
 LDCM0320  AC57 HCT 116 C117(0.67); C115(0.67); C51(1.04)  LDD0637  [10]
 LDCM0321  AC58 HCT 116 C115(0.61); C117(0.62); C51(1.14)  LDD0638  [10]
 LDCM0322  AC59 HCT 116 C117(0.55); C115(0.56); C51(0.98)  LDD0639  [10]
 LDCM0323  AC6 HCT 116 C115(0.67); C117(0.67); C51(0.70)  LDD0640  [10]
 LDCM0324  AC60 HCT 116 C117(0.59); C115(0.60); C51(1.08)  LDD0641  [10]
 LDCM0325  AC61 HCT 116 C115(0.76); C117(0.77); C51(1.07)  LDD0642  [10]
 LDCM0326  AC62 HCT 116 C117(0.61); C115(0.64); C51(1.18)  LDD0643  [10]
 LDCM0327  AC63 HCT 116 C117(0.62); C115(0.65); C51(1.54)  LDD0644  [10]
 LDCM0328  AC64 HCT 116 C117(0.61); C115(0.64); C51(1.01)  LDD0645  [10]
 LDCM0329  AC65 HCT 116 C115(0.62); C117(0.63); C51(1.16)  LDD0646  [10]
 LDCM0330  AC66 HCT 116 C115(0.63); C117(0.64); C51(1.37)  LDD0647  [10]
 LDCM0331  AC67 HCT 116 C117(0.60); C115(0.61); C51(0.98)  LDD0648  [10]
 LDCM0332  AC68 HCT 116 C115(0.96); C117(0.96); C51(1.04)  LDD0649  [10]
 LDCM0333  AC69 HCT 116 C51(0.76); C117(1.06); C115(1.06)  LDD0650  [10]
 LDCM0334  AC7 HCT 116 C115(0.81); C117(0.81); C51(0.89)  LDD0651  [10]
 LDCM0335  AC70 HCT 116 C51(0.85); C115(1.03); C117(1.03)  LDD0652  [10]
 LDCM0336  AC71 HCT 116 C51(0.97); C115(1.15); C117(1.19)  LDD0653  [10]
 LDCM0337  AC72 HCT 116 C51(0.82); C115(0.83); C117(0.88)  LDD0654  [10]
 LDCM0338  AC73 HCT 116 C115(0.97); C117(1.05); C51(1.12)  LDD0655  [10]
 LDCM0339  AC74 HCT 116 C51(0.93); C115(1.08); C117(1.13)  LDD0656  [10]
 LDCM0340  AC75 HCT 116 C115(1.06); C117(1.12); C51(1.55)  LDD0657  [10]
 LDCM0341  AC76 HCT 116 C115(0.94); C117(0.94); C51(1.12)  LDD0658  [10]
 LDCM0342  AC77 HCT 116 C51(0.93); C115(0.99); C117(1.01)  LDD0659  [10]
 LDCM0343  AC78 HCT 116 C51(1.01); C117(1.12); C115(1.12)  LDD0660  [10]
 LDCM0344  AC79 HCT 116 C51(0.87); C115(0.95); C117(1.03)  LDD0661  [10]
 LDCM0345  AC8 HCT 116 C115(0.68); C117(0.68); C51(0.86)  LDD0662  [10]
 LDCM0346  AC80 HCT 116 C51(0.80); C117(0.94); C115(0.97)  LDD0663  [10]
 LDCM0347  AC81 HCT 116 C51(0.84); C115(1.23); C117(1.24)  LDD0664  [10]
 LDCM0348  AC82 HCT 116 C51(0.91); C115(1.18); C117(1.20)  LDD0665  [10]
 LDCM0349  AC83 HCT 116 C51(0.23); C115(0.51); C117(0.54)  LDD0666  [10]
 LDCM0350  AC84 HCT 116 C51(0.23); C115(0.51); C117(0.53)  LDD0667  [10]
 LDCM0351  AC85 HCT 116 C51(0.24); C115(0.55); C117(0.56)  LDD0668  [10]
 LDCM0352  AC86 HCT 116 C51(0.40); C115(0.56); C117(0.59)  LDD0669  [10]
 LDCM0353  AC87 HCT 116 C51(0.47); C115(0.79); C117(0.81)  LDD0670  [10]
 LDCM0354  AC88 HCT 116 C51(0.27); C115(0.62); C117(0.66)  LDD0671  [10]
 LDCM0355  AC89 HCT 116 C51(0.27); C115(0.52); C117(0.55)  LDD0672  [10]
 LDCM0357  AC90 HCT 116 C51(0.33); C115(0.95); C117(1.00)  LDD0674  [10]
 LDCM0358  AC91 HCT 116 C51(0.25); C117(0.51); C115(0.52)  LDD0675  [10]
 LDCM0359  AC92 HCT 116 C51(0.24); C115(0.50); C117(0.53)  LDD0676  [10]
 LDCM0360  AC93 HCT 116 C51(0.21); C115(0.54); C117(0.54)  LDD0677  [10]
 LDCM0361  AC94 HCT 116 C51(0.26); C117(0.68); C115(0.75)  LDD0678  [10]
 LDCM0362  AC95 HCT 116 C51(0.32); C115(0.66); C117(0.68)  LDD0679  [10]
 LDCM0363  AC96 HCT 116 C51(0.32); C117(0.62); C115(0.66)  LDD0680  [10]
 LDCM0364  AC97 HCT 116 C51(0.24); C115(0.45); C117(0.47)  LDD0681  [10]
 LDCM0365  AC98 HCT 116 C51(0.34); C115(0.48); C117(0.51)  LDD0682  [10]
 LDCM0366  AC99 HCT 116 C51(0.56); C117(0.62); C115(0.62)  LDD0683  [10]
 LDCM0248  AKOS034007472 HCT 116 C115(0.93); C117(0.93); C51(1.15)  LDD0565  [10]
 LDCM0356  AKOS034007680 HCT 116 C115(0.76); C117(0.76); C51(0.93)  LDD0673  [10]
 LDCM0275  AKOS034007705 HCT 116 C115(0.58); C117(0.58); C51(0.68)  LDD0592  [10]
 LDCM0156  Aniline NCI-H1299 12.30  LDD0403  [1]
 LDCM0102  BDHI 8 Jurkat C115(18.43); C117(18.43)  LDD0204  [21]
 LDCM0367  CL1 HCT 116 C117(1.05); C115(1.12); C51(1.65)  LDD0684  [10]
 LDCM0368  CL10 HCT 116 C51(0.76); C115(0.84); C117(0.85)  LDD0685  [10]
 LDCM0369  CL100 HCT 116 C51(0.59); C117(0.78); C115(0.78)  LDD0686  [10]
 LDCM0370  CL101 HCT 116 C115(0.65); C117(0.65); C51(0.84)  LDD0687  [10]
 LDCM0371  CL102 HCT 116 C115(0.81); C117(0.81); C51(0.93)  LDD0688  [10]
 LDCM0372  CL103 HCT 116 C115(0.80); C117(0.80); C51(0.93)  LDD0689  [10]
 LDCM0373  CL104 HCT 116 C115(0.82); C117(0.82); C51(0.92)  LDD0690  [10]
 LDCM0374  CL105 HCT 116 C51(0.64); C117(0.74); C115(0.76)  LDD0691  [10]
 LDCM0375  CL106 HCT 116 C51(0.59); C117(0.83); C115(0.86)  LDD0692  [10]
 LDCM0376  CL107 HCT 116 C51(0.56); C117(0.69); C115(0.73)  LDD0693  [10]
 LDCM0377  CL108 HCT 116 C51(0.57); C117(0.68); C115(0.73)  LDD0694  [10]
 LDCM0378  CL109 HCT 116 C51(0.66); C117(0.67); C115(0.68)  LDD0695  [10]
 LDCM0379  CL11 HCT 116 C115(0.89); C117(0.89); C51(1.07)  LDD0696  [10]
 LDCM0380  CL110 HCT 116 C51(0.56); C117(0.73); C115(0.73)  LDD0697  [10]
 LDCM0381  CL111 HCT 116 C117(0.71); C115(0.71); C51(0.74)  LDD0698  [10]
 LDCM0382  CL112 HCT 116 C115(0.91); C117(0.95); C51(1.32)  LDD0699  [10]
 LDCM0383  CL113 HCT 116 C115(0.50); C51(0.54); C117(0.62)  LDD0700  [10]
 LDCM0384  CL114 HCT 116 C115(0.57); C117(0.65); C51(0.69)  LDD0701  [10]
 LDCM0385  CL115 HCT 116 C115(0.55); C117(0.67); C51(0.76)  LDD0702  [10]
 LDCM0386  CL116 HCT 116 C115(0.61); C117(0.72); C51(0.77)  LDD0703  [10]
 LDCM0387  CL117 HCT 116 C51(0.72); C115(1.07); C117(1.12)  LDD0704  [10]
 LDCM0388  CL118 HCT 116 C115(0.96); C117(0.97); C51(1.14)  LDD0705  [10]
 LDCM0389  CL119 HCT 116 C51(0.69); C117(0.98); C115(0.98)  LDD0706  [10]
 LDCM0390  CL12 HCT 116 C115(0.81); C51(0.82); C117(0.86)  LDD0707  [10]
 LDCM0391  CL120 HCT 116 C51(0.90); C117(1.03); C115(1.04)  LDD0708  [10]
 LDCM0392  CL121 HCT 116 C51(0.84); C117(0.89); C115(1.26)  LDD0709  [10]
 LDCM0393  CL122 HCT 116 C115(0.99); C51(1.00); C117(1.00)  LDD0710  [10]
 LDCM0394  CL123 HCT 116 C51(0.79); C115(0.92); C117(0.94)  LDD0711  [10]
 LDCM0395  CL124 HCT 116 C51(0.81); C115(0.87); C117(0.94)  LDD0712  [10]
 LDCM0396  CL125 HCT 116 C115(0.81); C117(0.85); C51(1.07)  LDD0713  [10]
 LDCM0397  CL126 HCT 116 C115(0.62); C117(0.64); C51(1.14)  LDD0714  [10]
 LDCM0398  CL127 HCT 116 C115(0.66); C117(0.67); C51(1.69)  LDD0715  [10]
 LDCM0399  CL128 HCT 116 C117(0.60); C115(0.60); C51(1.20)  LDD0716  [10]
 LDCM0400  CL13 HCT 116 C51(0.76); C115(0.87); C117(0.90)  LDD0717  [10]
 LDCM0401  CL14 HCT 116 C51(0.76); C117(0.86); C115(0.88)  LDD0718  [10]
 LDCM0402  CL15 HCT 116 C115(0.92); C117(0.93); C51(0.98)  LDD0719  [10]
 LDCM0403  CL16 HCT 116 C115(0.85); C117(0.88); C51(0.92)  LDD0720  [10]
 LDCM0404  CL17 HCT 116 C115(0.79); C51(0.85); C117(0.85)  LDD0721  [10]
 LDCM0405  CL18 HCT 116 C51(0.69); C115(0.81); C117(0.87)  LDD0722  [10]
 LDCM0406  CL19 HCT 116 C51(0.70); C115(0.78); C117(0.87)  LDD0723  [10]
 LDCM0407  CL2 HCT 116 C117(1.00); C115(1.07); C51(1.44)  LDD0724  [10]
 LDCM0408  CL20 HCT 116 C115(0.61); C51(0.62); C117(0.77)  LDD0725  [10]
 LDCM0409  CL21 HCT 116 C51(0.60); C115(0.66); C117(0.78)  LDD0726  [10]
 LDCM0410  CL22 HCT 116 C115(0.73); C51(0.79); C117(0.88)  LDD0727  [10]
 LDCM0411  CL23 HCT 116 C115(0.66); C117(0.73); C51(0.82)  LDD0728  [10]
 LDCM0412  CL24 HCT 116 C51(0.58); C115(0.67); C117(0.78)  LDD0729  [10]
 LDCM0413  CL25 HCT 116 C115(0.66); C117(0.75); C51(0.63)  LDD0730  [10]
 LDCM0414  CL26 HCT 116 C115(0.69); C117(0.76); C51(0.65)  LDD0731  [10]
 LDCM0415  CL27 HCT 116 C115(0.73); C117(0.85); C51(0.75)  LDD0732  [10]
 LDCM0416  CL28 HCT 116 C115(0.62); C117(0.70); C51(0.61)  LDD0733  [10]
 LDCM0417  CL29 HCT 116 C115(0.64); C117(0.75); C51(0.62)  LDD0734  [10]
 LDCM0418  CL3 HCT 116 C115(1.01); C117(0.97); C51(1.12)  LDD0735  [10]
 LDCM0419  CL30 HCT 116 C115(0.83); C117(0.91); C51(0.92)  LDD0736  [10]
 LDCM0420  CL31 HCT 116 C115(0.77); C117(0.78); C51(0.62)  LDD0737  [10]
 LDCM0421  CL32 HCT 116 C115(0.77); C117(0.79); C51(0.62)  LDD0738  [10]
 LDCM0422  CL33 HCT 116 C115(0.73); C117(0.81); C51(0.59)  LDD0739  [10]
 LDCM0423  CL34 HCT 116 C115(0.63); C117(0.71); C51(0.54)  LDD0740  [10]
 LDCM0424  CL35 HCT 116 C115(0.61); C117(0.64); C51(0.47)  LDD0741  [10]
 LDCM0425  CL36 HCT 116 C115(0.68); C117(0.71); C51(0.56)  LDD0742  [10]
 LDCM0426  CL37 HCT 116 C115(0.72); C117(0.76); C51(0.60)  LDD0743  [10]
 LDCM0428  CL39 HCT 116 C115(0.62); C117(0.66); C51(0.46)  LDD0745  [10]
 LDCM0429  CL4 HCT 116 C115(0.95); C117(0.92); C51(1.05)  LDD0746  [10]
 LDCM0430  CL40 HCT 116 C115(0.65); C117(0.64); C51(0.50)  LDD0747  [10]
 LDCM0431  CL41 HCT 116 C115(0.59); C117(0.65); C51(0.57)  LDD0748  [10]
 LDCM0432  CL42 HCT 116 C115(0.82); C117(0.79); C51(0.61)  LDD0749  [10]
 LDCM0433  CL43 HCT 116 C115(0.61); C117(0.68); C51(0.54)  LDD0750  [10]
 LDCM0434  CL44 HCT 116 C115(0.73); C117(0.77); C51(0.56)  LDD0751  [10]
 LDCM0435  CL45 HCT 116 C115(0.69); C117(0.69); C51(0.59)  LDD0752  [10]
 LDCM0436  CL46 HCT 116 C115(1.19); C117(1.20); C51(1.70)  LDD0753  [10]
 LDCM0437  CL47 HCT 116 C115(1.11); C117(1.14); C51(1.40)  LDD0754  [10]
 LDCM0438  CL48 HCT 116 C115(1.23); C117(1.27); C51(1.64)  LDD0755  [10]
 LDCM0439  CL49 HCT 116 C115(0.91); C117(0.87); C51(1.08)  LDD0756  [10]
 LDCM0440  CL5 HCT 116 C115(0.91); C117(0.92); C51(1.14)  LDD0757  [10]
 LDCM0441  CL50 HCT 116 C115(1.05); C117(1.11); C51(1.51)  LDD0758  [10]
 LDCM0442  CL51 HCT 116 C115(1.09); C117(1.08); C51(1.61)  LDD0759  [10]
 LDCM0443  CL52 HCT 116 C115(1.04); C117(1.11); C51(1.42)  LDD0760  [10]
 LDCM0444  CL53 HCT 116 C115(1.03); C117(1.11); C51(1.51)  LDD0761  [10]
 LDCM0445  CL54 HCT 116 C115(1.15); C117(1.22); C51(1.43)  LDD0762  [10]
 LDCM0446  CL55 HCT 116 C115(1.21); C117(1.22); C51(1.53)  LDD0763  [10]
 LDCM0447  CL56 HCT 116 C115(0.90); C117(0.95); C51(1.02)  LDD0764  [10]
 LDCM0448  CL57 HCT 116 C115(1.04); C117(1.09); C51(1.47)  LDD0765  [10]
 LDCM0449  CL58 HCT 116 C115(1.07); C117(1.13); C51(1.45)  LDD0766  [10]
 LDCM0450  CL59 HCT 116 C115(1.00); C117(1.02); C51(1.17)  LDD0767  [10]
 LDCM0451  CL6 HCT 116 C115(0.94); C117(0.91); C51(1.26)  LDD0768  [10]
 LDCM0452  CL60 HCT 116 C115(0.90); C117(0.96); C51(1.19)  LDD0769  [10]
 LDCM0453  CL61 HCT 116 C115(0.83); C117(0.93); C51(0.86)  LDD0770  [10]
 LDCM0454  CL62 HCT 116 C115(0.84); C117(0.82); C51(0.78)  LDD0771  [10]
 LDCM0455  CL63 HCT 116 C115(0.73); C117(0.77); C51(0.73)  LDD0772  [10]
 LDCM0456  CL64 HCT 116 C115(0.64); C117(0.70); C51(0.59)  LDD0773  [10]
 LDCM0457  CL65 HCT 116 C115(0.84); C117(0.90); C51(0.69)  LDD0774  [10]
 LDCM0458  CL66 HCT 116 C115(0.67); C117(0.78); C51(0.53)  LDD0775  [10]
 LDCM0459  CL67 HCT 116 C115(0.66); C117(0.72); C51(0.56)  LDD0776  [10]
 LDCM0460  CL68 HCT 116 C115(0.70); C117(0.81); C51(0.64)  LDD0777  [10]
 LDCM0461  CL69 HCT 116 C115(0.83); C117(0.92); C51(0.80)  LDD0778  [10]
 LDCM0462  CL7 HCT 116 C115(0.85); C117(0.86); C51(0.86)  LDD0779  [10]
 LDCM0463  CL70 HCT 116 C115(0.77); C117(0.83); C51(0.70)  LDD0780  [10]
 LDCM0464  CL71 HCT 116 C115(0.72); C117(0.75); C51(0.62)  LDD0781  [10]
 LDCM0465  CL72 HCT 116 C115(0.82); C117(0.93); C51(0.89)  LDD0782  [10]
 LDCM0466  CL73 HCT 116 C115(0.69); C117(0.75); C51(0.69)  LDD0783  [10]
 LDCM0467  CL74 HCT 116 C115(0.71); C117(0.76); C51(0.66)  LDD0784  [10]
 LDCM0469  CL76 HCT 116 C115(0.93); C117(0.94)  LDD0786  [10]
 LDCM0470  CL77 HCT 116 C115(0.89); C117(0.88)  LDD0787  [10]
 LDCM0471  CL78 HCT 116 C115(0.79); C117(0.77)  LDD0788  [10]
 LDCM0472  CL79 HCT 116 C115(0.73); C117(0.75)  LDD0789  [10]
 LDCM0473  CL8 HCT 116 C115(0.76); C117(0.82); C51(0.75)  LDD0790  [10]
 LDCM0474  CL80 HCT 116 C115(0.99); C117(0.97)  LDD0791  [10]
 LDCM0475  CL81 HCT 116 C115(0.87); C117(0.87)  LDD0792  [10]
 LDCM0476  CL82 HCT 116 C115(0.89); C117(0.88)  LDD0793  [10]
 LDCM0477  CL83 HCT 116 C115(0.82); C117(0.80)  LDD0794  [10]
 LDCM0478  CL84 HCT 116 C115(0.81); C117(0.79)  LDD0795  [10]
 LDCM0479  CL85 HCT 116 C115(0.79); C117(0.78)  LDD0796  [10]
 LDCM0480  CL86 HCT 116 C115(0.93); C117(0.92)  LDD0797  [10]
 LDCM0481  CL87 HCT 116 C115(0.87); C117(0.87)  LDD0798  [10]
 LDCM0482  CL88 HCT 116 C115(0.88); C117(0.87)  LDD0799  [10]
 LDCM0483  CL89 HCT 116 C115(0.91); C117(0.87)  LDD0800  [10]
 LDCM0484  CL9 HCT 116 C115(0.80); C117(0.83); C51(0.77)  LDD0801  [10]
 LDCM0485  CL90 HCT 116 C115(1.12); C117(1.10)  LDD0802  [10]
 LDCM0486  CL91 HCT 116 C115(0.90); C117(0.93); C51(0.75)  LDD0803  [10]
 LDCM0487  CL92 HCT 116 C115(0.92); C117(0.93); C51(0.73)  LDD0804  [10]
 LDCM0488  CL93 HCT 116 C115(1.00); C117(0.91); C51(0.57)  LDD0805  [10]
 LDCM0489  CL94 HCT 116 C115(0.87); C117(0.82); C51(0.52)  LDD0806  [10]
 LDCM0490  CL95 HCT 116 C115(0.80); C117(0.79); C51(0.53)  LDD0807  [10]
 LDCM0491  CL96 HCT 116 C115(0.75); C117(0.79); C51(0.64)  LDD0808  [10]
 LDCM0492  CL97 HCT 116 C115(0.78); C117(0.78); C51(0.52)  LDD0809  [10]
 LDCM0493  CL98 HCT 116 C115(0.73); C117(0.75); C51(0.51)  LDD0810  [10]
 LDCM0494  CL99 HCT 116 C115(0.85); C117(0.81); C51(0.59)  LDD0811  [10]
 LDCM0495  E2913 HEK-293T C51(0.92); C74(0.85); C117(0.89)  LDD1698  [22]
 LDCM0175  Ethacrynic acid HeLa N.A.  LDD0440  [9]
 LDCM0625  F8 Ramos 0.99  LDD2187  [23]
 LDCM0573  Fragment11 Ramos 0.50  LDD2190  [23]
 LDCM0575  Fragment13 Ramos 1.39  LDD2192  [23]
 LDCM0576  Fragment14 Ramos 1.10  LDD2193  [23]
 LDCM0580  Fragment21 Ramos 1.61  LDD2195  [23]
 LDCM0578  Fragment27 Ramos 0.78  LDD2197  [23]
 LDCM0586  Fragment28 Ramos 0.98  LDD2198  [23]
 LDCM0588  Fragment30 Ramos 1.23  LDD2199  [23]
 LDCM0589  Fragment31 Ramos 2.03  LDD2200  [23]
 LDCM0468  Fragment33 HCT 116 C115(0.67); C117(0.77); C51(0.57)  LDD0785  [10]
 LDCM0596  Fragment38 Ramos 1.07  LDD2203  [23]
 LDCM0427  Fragment51 HCT 116 C115(0.81); C117(0.81); C51(0.60)  LDD0744  [10]
 LDCM0610  Fragment52 Ramos 5.10  LDD2204  [23]
 LDCM0614  Fragment56 Ramos 1.21  LDD2205  [23]
 LDCM0179  JZ128 PC-3 N.A.  LDD0462  [7]
 LDCM0022  KB02 HCT 116 C115(6.00); C51(2.58); C117(1.12)  LDD0080  [10]
 LDCM0023  KB03 HCT 116 C115(7.94); C51(1.76); C117(1.21)  LDD0081  [10]
 LDCM0024  KB05 HCT 116 C115(3.29); C51(2.15); C117(1.17)  LDD0082  [10]
 LDCM0523  Nucleophilic fragment 24b MDA-MB-231 C25(0.38)  LDD2116  [8]
 LDCM0525  Nucleophilic fragment 25b MDA-MB-231 C25(0.35)  LDD2118  [8]
 LDCM0529  Nucleophilic fragment 27b MDA-MB-231 C25(0.26)  LDD2122  [8]
 LDCM0533  Nucleophilic fragment 29b MDA-MB-231 C25(0.37)  LDD2126  [8]
 LDCM0535  Nucleophilic fragment 30b MDA-MB-231 C25(1.09)  LDD2128  [8]
 LDCM0555  Nucleophilic fragment 7b MDA-MB-231 C25(0.33)  LDD2149  [8]
 LDCM0559  Nucleophilic fragment 9b MDA-MB-231 C25(0.65)  LDD2153  [8]
 LDCM0627  NUDT7-COV-1 HEK-293T C31(0.69); C51(0.68); C115(0.56)  LDD2206  [24]
 LDCM0628  OTUB2-COV-1 HEK-293T C51(1.69); C31(0.69)  LDD2207  [24]
 LDCM0090  Rapamycin JHH-7 6.22  LDD0213  [20]

The Interaction Atlas With This Target

The Protein(s) Related To This Target

Enzyme
Click To Hide/Show 2 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Kallikrein-6 (KLK6) Peptidase S1 family Q92876
E3 ubiquitin-protein ligase LNX (LNX1) . Q8TBB1
Other
Click To Hide/Show 4 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Cytoplasmic dynein 1 heavy chain 1 (DYNC1H1) Dynein heavy chain family Q14204
Checkpoint protein HUS1 (HUS1) HUS1 family O60921
PRKCA-binding protein (PICK1) . Q9NRD5
Puratrophin-1 (PLEKHG4) . Q58EX7

References

1 Quantitative and Site-Specific Chemoproteomic Profiling of Targets of Acrolein. Chem Res Toxicol. 2019 Mar 18;32(3):467-473. doi: 10.1021/acs.chemrestox.8b00343. Epub 2019 Jan 15.
2 Hydrazines as versatile chemical biology probes and drug-discovery tools for cofactor-dependent enzymes. bioRxiv, 2020-06.
3 Appendage and Scaffold Diverse Fully Functionalized Small-Molecule Probes via a Minimalist Terminal Alkyne-Aliphatic Diazirine Isocyanide. J Org Chem. 2018 Sep 21;83(18):11245-11253. doi: 10.1021/acs.joc.8b01831. Epub 2018 Aug 31.
4 Low-Toxicity Sulfonium-Based Probes for Cysteine-Specific Profiling in Live Cells. Anal Chem. 2022 Mar 15;94(10):4366-4372. doi: 10.1021/acs.analchem.1c05129. Epub 2022 Mar 4.
5 Chemoproteomic profiling of kinases in live cells using electrophilic sulfonyl triazole probes. Chem Sci. 2021 Jan 21;12(9):3295-3307. doi: 10.1039/d0sc06623k.
6 A Paal-Knorr agent for chemoproteomic profiling of targets of isoketals in cells. Chem Sci. 2021 Oct 15;12(43):14557-14563. doi: 10.1039/d1sc02230j. eCollection 2021 Nov 10.
Mass spectrometry data entry: PXD028270
7 A Chemoproteomic Strategy for Direct and Proteome-Wide Covalent Inhibitor Target-Site Identification. J Am Chem Soc. 2019 Jan 9;141(1):191-203. doi: 10.1021/jacs.8b07911. Epub 2018 Dec 20.
8 Nucleophilic covalent ligand discovery for the cysteine redoxome. Nat Chem Biol. 2023 Nov;19(11):1309-1319. doi: 10.1038/s41589-023-01330-5. Epub 2023 May 29.
Mass spectrometry data entry: PXD039908 , PXD029761
9 Chemoproteomic Profiling Reveals Ethacrynic Acid Targets Adenine Nucleotide Translocases to Impair Mitochondrial Function. Mol Pharm. 2018 Jun 4;15(6):2413-2422. doi: 10.1021/acs.molpharmaceut.8b00250. Epub 2018 May 15.
10 Reimagining high-throughput profiling of reactive cysteines for cell-based screening of large electrophile libraries. Nat Biotechnol. 2021 May;39(5):630-641. doi: 10.1038/s41587-020-00778-3. Epub 2021 Jan 4.
11 Targeted Proteomic Approaches for Proteome-Wide Characterizations of the AMP-Binding Capacities of Kinases. J Proteome Res. 2022 Aug 5;21(8):2063-2070. doi: 10.1021/acs.jproteome.2c00225. Epub 2022 Jul 12.
12 Cyclopropenone, Cyclopropeniminium Ion, and Cyclopropenethione as Novel Electrophilic Warheads for Potential Target Discovery of Triple-Negative Breast Cancer. J Med Chem. 2023 Feb 23;66(4):2851-2864. doi: 10.1021/acs.jmedchem.2c01889. Epub 2023 Feb 10.
13 SP3-FAIMS Chemoproteomics for High-Coverage Profiling of the Human Cysteinome*. Chembiochem. 2021 May 14;22(10):1841-1851. doi: 10.1002/cbic.202000870. Epub 2021 Feb 18.
Mass spectrometry data entry: PXD023056 , PXD023059 , PXD023058 , PXD023057 , PXD023060
14 Enhancing Cysteine Chemoproteomic Coverage through Systematic Assessment of Click Chemistry Product Fragmentation. Anal Chem. 2022 Mar 8;94(9):3800-3810. doi: 10.1021/acs.analchem.1c04402. Epub 2022 Feb 23.
Mass spectrometry data entry: PXD028853
15 A modification-centric assessment tool for the performance of chemoproteomic probes. Nat Chem Biol. 2022 Aug;18(8):904-912. doi: 10.1038/s41589-022-01074-8. Epub 2022 Jul 21.
Mass spectrometry data entry: PXD027758 , PXD027755 , PXD027760 , PXD027762 , PXD027756 , PXD027591 , PXD007149 , PXD030064 , PXD032392 , PXD027789 , PXD027767 , PXD027764
16 Chemoproteomic Profiling by Cysteine Fluoroalkylation Reveals Myrocin G as an Inhibitor of the Nonhomologous End Joining DNA Repair Pathway. J Am Chem Soc. 2021 Dec 8;143(48):20332-20342. doi: 10.1021/jacs.1c09724. Epub 2021 Nov 24.
Mass spectrometry data entry: PXD029255
17 Oxidative cyclization reagents reveal tryptophan cation- interactions. Nature. 2024 Mar;627(8004):680-687. doi: 10.1038/s41586-024-07140-6. Epub 2024 Mar 6.
Mass spectrometry data entry: PXD001377 , PXD005252
18 Chemoproteomic profiling of targets of lipid-derived electrophiles by bioorthogonal aminooxy probe. Redox Biol. 2017 Aug;12:712-718. doi: 10.1016/j.redox.2017.04.001. Epub 2017 Apr 5.
19 Large-scale chemoproteomics expedites ligand discovery and predicts ligand behavior in cells. Science. 2024 Apr 26;384(6694):eadk5864. doi: 10.1126/science.adk5864. Epub 2024 Apr 26.
Mass spectrometry data entry: PXD041587
20 Rapamycin targets STAT3 and impacts c-Myc to suppress tumor growth. Cell Chem Biol. 2022 Mar 17;29(3):373-385.e6. doi: 10.1016/j.chembiol.2021.10.006. Epub 2021 Oct 26.
21 Covalent Inhibition by a Natural Product-Inspired Latent Electrophile. J Am Chem Soc. 2023 May 24;145(20):11097-11109. doi: 10.1021/jacs.3c00598. Epub 2023 May 15.
22 Accelerating multiplexed profiling of protein-ligand interactions: High-throughput plate-based reactive cysteine profiling with minimal input. Cell Chem Biol. 2024 Mar 21;31(3):565-576.e4. doi: 10.1016/j.chembiol.2023.11.015. Epub 2023 Dec 19.
Mass spectrometry data entry: PXD044402
23 Site-specific quantitative cysteine profiling with data-independent acquisition-based mass spectrometry. Methods Enzymol. 2023;679:295-322. doi: 10.1016/bs.mie.2022.07.037. Epub 2022 Sep 7.
Mass spectrometry data entry: PXD027578
24 Rapid Covalent-Probe Discovery by Electrophile-Fragment Screening. J Am Chem Soc. 2019 Jun 5;141(22):8951-8968. doi: 10.1021/jacs.9b02822. Epub 2019 May 22.