Details of the Target

General Information of Target

Target ID LDTP12831
Target Name PH and SEC7 domain-containing protein 3 (PSD3)
Gene Name PSD3
Gene ID 23362
Synonyms
EFA6D; EFA6R; HCA67; KIAA0942; PH and SEC7 domain-containing protein 3; Epididymis tissue protein Li 20mP; Exchange factor for ADP-ribosylation factor guanine nucleotide factor 6 D; Exchange factor for ARF6 D; Hepatocellular carcinoma-associated antigen 67; Pleckstrin homology and SEC7 domain-containing protein 3
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MAEIIQERIEDRLPELEQLERIGLFSHAEIKAIIKKASDLEYKIQRRTLFKEDFINYVQY
EINLLELIQRRRTRIGYSFKKDEIENSIVHRVQGVFQRASAKWKDDVQLWLSYVAFCKKW
ATKTRLSKVFSAMLAIHSNKPALWIMAAKWEMEDRLSSESARQLFLRALRFHPECPKLYK
EYFRMELMHAEKLRKEKEEFEKASMDVENPDYSEEILKGELAWIIYKNSVSIIKGAEFHV
SLLSIAQLFDFAKDLQKEIYDDLQALHTDDPLTWDYVARRELEIESQTEEQPTTKQAKAV
EVGRKEERCCAVYEEAVKTLPTEAMWKCYITFCLERFTKKSNSGFLRGKRLERTMTVFRK
AHELKLLSECQYKQLSVSLLCYNFLREALEVAVAGTELFRDSGTMWQLKLQVLIESKSPD
IAMLFEEAFVHLKPQVCLPLWISWAEWSEGAKSQEDTEAVFKKALLAVIGADSVTLKNKY
LDWAYRSGGYKKARAVFKSLQESRPFSVDFFRKMIQFEKEQESCNMANIREYYERALREF
GSADSDLWMDYMKEELNHPLGRPENCGQIYWRAMKMLQGESAEAFVAKHAMHQTGHL
Target Bioclass
Other
Subcellular location
Cell membrane
Function Guanine nucleotide exchange factor for ARF6.
Uniprot ID
Q9NYI0
Ensemble ID
ENST00000286485.12
HGNC ID
HGNC:19093

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 6 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
STPyne
 Probe Info  		K28(10.00); K605(10.00)  LDD0277  [1]
DBIA
 Probe Info  		C284(21.41)  LDD0204  [2]
IA-alkyne
 Probe Info  		N.A.  LDD0162  [3]
NAIA_4
 Probe Info  		N.A.  LDD2226  [4]
IPM
 Probe Info  		N.A.  LDD0147  [5]
Phosphinate-6
 Probe Info  		N.A.  LDD0018  [6]
PAL-AfBPP Probe
Click To Hide/Show 1 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
STS-2
 Probe Info  		N.A.  LDD0139  [7]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0214  AC1 HCT 116 C284(0.84)  LDD0531  [8]
 LDCM0215  AC10 HCT 116 C284(0.84)  LDD0532  [8]
 LDCM0226  AC11 HCT 116 C284(0.96)  LDD0543  [8]
 LDCM0230  AC113 HCT 116 C284(0.93)  LDD0547  [8]
 LDCM0231  AC114 HCT 116 C284(0.85)  LDD0548  [8]
 LDCM0232  AC115 HCT 116 C284(1.02)  LDD0549  [8]
 LDCM0233  AC116 HCT 116 C284(0.94)  LDD0550  [8]
 LDCM0234  AC117 HCT 116 C284(0.89)  LDD0551  [8]
 LDCM0235  AC118 HCT 116 C284(0.86)  LDD0552  [8]
 LDCM0236  AC119 HCT 116 C284(0.98)  LDD0553  [8]
 LDCM0237  AC12 HCT 116 C284(0.88)  LDD0554  [8]
 LDCM0238  AC120 HCT 116 C284(0.72)  LDD0555  [8]
 LDCM0239  AC121 HCT 116 C284(0.78)  LDD0556  [8]
 LDCM0240  AC122 HCT 116 C284(0.79)  LDD0557  [8]
 LDCM0241  AC123 HCT 116 C284(0.71)  LDD0558  [8]
 LDCM0242  AC124 HCT 116 C284(0.77)  LDD0559  [8]
 LDCM0243  AC125 HCT 116 C284(0.72)  LDD0560  [8]
 LDCM0244  AC126 HCT 116 C284(0.84)  LDD0561  [8]
 LDCM0245  AC127 HCT 116 C284(0.84)  LDD0562  [8]
 LDCM0259  AC14 HCT 116 C284(0.87)  LDD0576  [8]
 LDCM0263  AC143 HCT 116 C284(1.17)  LDD0580  [8]
 LDCM0264  AC144 HCT 116 C284(0.83)  LDD0581  [8]
 LDCM0265  AC145 HCT 116 C284(0.73)  LDD0582  [8]
 LDCM0266  AC146 HCT 116 C284(0.87)  LDD0583  [8]
 LDCM0267  AC147 HCT 116 C284(0.87)  LDD0584  [8]
 LDCM0268  AC148 HCT 116 C284(0.72)  LDD0585  [8]
 LDCM0269  AC149 HCT 116 C284(0.84)  LDD0586  [8]
 LDCM0270  AC15 HCT 116 C284(0.89)  LDD0587  [8]
 LDCM0271  AC150 HCT 116 C284(0.90)  LDD0588  [8]
 LDCM0272  AC151 HCT 116 C284(0.85)  LDD0589  [8]
 LDCM0273  AC152 HCT 116 C284(0.88)  LDD0590  [8]
 LDCM0274  AC153 HCT 116 C284(0.89)  LDD0591  [8]
 LDCM0621  AC154 HCT 116 C284(1.11)  LDD2158  [8]
 LDCM0622  AC155 HCT 116 C284(0.87)  LDD2159  [8]
 LDCM0623  AC156 HCT 116 C284(1.01)  LDD2160  [8]
 LDCM0624  AC157 HCT 116 C284(0.82)  LDD2161  [8]
 LDCM0276  AC17 HEK-293T C284(1.06)  LDD1515  [9]
 LDCM0277  AC18 HEK-293T C284(1.01)  LDD1516  [9]
 LDCM0278  AC19 HEK-293T C284(1.53)  LDD1517  [9]
 LDCM0279  AC2 HCT 116 C284(0.94)  LDD0596  [8]
 LDCM0280  AC20 HEK-293T C284(0.99)  LDD1519  [9]
 LDCM0281  AC21 HEK-293T C284(0.97)  LDD1520  [9]
 LDCM0282  AC22 HEK-293T C284(1.01)  LDD1521  [9]
 LDCM0283  AC23 HEK-293T C284(0.97)  LDD1522  [9]
 LDCM0284  AC24 HEK-293T C284(1.05)  LDD1523  [9]
 LDCM0285  AC25 HEK-293T C284(1.06)  LDD1524  [9]
 LDCM0286  AC26 HEK-293T C284(0.96)  LDD1525  [9]
 LDCM0287  AC27 HEK-293T C284(1.01)  LDD1526  [9]
 LDCM0288  AC28 HEK-293T C284(0.99)  LDD1527  [9]
 LDCM0289  AC29 HEK-293T C284(1.06)  LDD1528  [9]
 LDCM0290  AC3 HCT 116 C284(0.89)  LDD0607  [8]
 LDCM0291  AC30 HEK-293T C284(0.92)  LDD1530  [9]
 LDCM0292  AC31 HEK-293T C284(0.93)  LDD1531  [9]
 LDCM0293  AC32 HEK-293T C284(1.03)  LDD1532  [9]
 LDCM0294  AC33 HEK-293T C284(1.10)  LDD1533  [9]
 LDCM0295  AC34 HEK-293T C284(0.99)  LDD1534  [9]
 LDCM0296  AC35 HCT 116 C284(1.42)  LDD0613  [8]
 LDCM0297  AC36 HCT 116 C284(1.36)  LDD0614  [8]
 LDCM0298  AC37 HCT 116 C284(1.40)  LDD0615  [8]
 LDCM0299  AC38 HCT 116 C284(1.59)  LDD0616  [8]
 LDCM0300  AC39 HCT 116 C284(1.32)  LDD0617  [8]
 LDCM0301  AC4 HCT 116 C284(0.88)  LDD0618  [8]
 LDCM0302  AC40 HCT 116 C284(1.57)  LDD0619  [8]
 LDCM0303  AC41 HCT 116 C284(1.18)  LDD0620  [8]
 LDCM0304  AC42 HCT 116 C284(1.23)  LDD0621  [8]
 LDCM0305  AC43 HCT 116 C284(1.15)  LDD0622  [8]
 LDCM0306  AC44 HCT 116 C284(1.19)  LDD0623  [8]
 LDCM0307  AC45 HCT 116 C284(1.42)  LDD0624  [8]
 LDCM0308  AC46 HCT 116 C284(1.05)  LDD0625  [8]
 LDCM0309  AC47 HCT 116 C284(0.91)  LDD0626  [8]
 LDCM0310  AC48 HCT 116 C284(1.03)  LDD0627  [8]
 LDCM0311  AC49 HCT 116 C284(1.19)  LDD0628  [8]
 LDCM0312  AC5 HCT 116 C284(0.82)  LDD0629  [8]
 LDCM0313  AC50 HCT 116 C284(1.00)  LDD0630  [8]
 LDCM0314  AC51 HCT 116 C284(0.95)  LDD0631  [8]
 LDCM0315  AC52 HCT 116 C284(0.98)  LDD0632  [8]
 LDCM0316  AC53 HCT 116 C284(1.17)  LDD0633  [8]
 LDCM0317  AC54 HCT 116 C284(0.85)  LDD0634  [8]
 LDCM0318  AC55 HCT 116 C284(1.16)  LDD0635  [8]
 LDCM0319  AC56 HCT 116 C284(1.25)  LDD0636  [8]
 LDCM0320  AC57 HCT 116 C284(1.18)  LDD0637  [8]
 LDCM0321  AC58 HCT 116 C284(0.96)  LDD0638  [8]
 LDCM0322  AC59 HCT 116 C284(1.26)  LDD0639  [8]
 LDCM0323  AC6 HCT 116 C284(1.05)  LDD0640  [8]
 LDCM0324  AC60 HCT 116 C284(1.21)  LDD0641  [8]
 LDCM0325  AC61 HCT 116 C284(0.97)  LDD0642  [8]
 LDCM0326  AC62 HCT 116 C284(1.52)  LDD0643  [8]
 LDCM0327  AC63 HCT 116 C284(1.42)  LDD0644  [8]
 LDCM0328  AC64 HCT 116 C284(1.40)  LDD0645  [8]
 LDCM0329  AC65 HCT 116 C284(1.26)  LDD0646  [8]
 LDCM0330  AC66 HCT 116 C284(0.83)  LDD0647  [8]
 LDCM0331  AC67 HCT 116 C284(1.23)  LDD0648  [8]
 LDCM0332  AC68 HCT 116 C284(0.81)  LDD0649  [8]
 LDCM0333  AC69 HCT 116 C284(0.68)  LDD0650  [8]
 LDCM0334  AC7 HCT 116 C284(0.95)  LDD0651  [8]
 LDCM0335  AC70 HCT 116 C284(0.91)  LDD0652  [8]
 LDCM0336  AC71 HCT 116 C284(0.90)  LDD0653  [8]
 LDCM0337  AC72 HCT 116 C284(0.86)  LDD0654  [8]
 LDCM0338  AC73 HCT 116 C284(0.95)  LDD0655  [8]
 LDCM0339  AC74 HCT 116 C284(0.82)  LDD0656  [8]
 LDCM0340  AC75 HCT 116 C284(1.12)  LDD0657  [8]
 LDCM0341  AC76 HCT 116 C284(1.06)  LDD0658  [8]
 LDCM0342  AC77 HCT 116 C284(0.84)  LDD0659  [8]
 LDCM0343  AC78 HCT 116 C284(0.99)  LDD0660  [8]
 LDCM0344  AC79 HCT 116 C284(0.99)  LDD0661  [8]
 LDCM0345  AC8 HCT 116 C284(0.99)  LDD0662  [8]
 LDCM0346  AC80 HCT 116 C284(1.01)  LDD0663  [8]
 LDCM0347  AC81 HCT 116 C284(0.98)  LDD0664  [8]
 LDCM0348  AC82 HCT 116 C284(1.09)  LDD0665  [8]
 LDCM0248  AKOS034007472 HCT 116 C284(0.95)  LDD0565  [8]
 LDCM0356  AKOS034007680 HCT 116 C284(1.07)  LDD0673  [8]
 LDCM0275  AKOS034007705 HCT 116 C284(0.98)  LDD0592  [8]
 LDCM0020  ARS-1620 HCC44 C242(1.42); C248(1.42); C260(1.42); C284(0.98)  LDD2171  [8]
 LDCM0102  BDHI 8 Jurkat C284(21.41)  LDD0204  [2]
 LDCM0367  CL1 HEK-293T C284(1.01)  LDD1571  [9]
 LDCM0368  CL10 HEK-293T C284(1.18)  LDD1572  [9]
 LDCM0369  CL100 HCT 116 C284(0.84)  LDD0686  [8]
 LDCM0370  CL101 HCT 116 C284(0.90)  LDD0687  [8]
 LDCM0371  CL102 HCT 116 C284(0.99)  LDD0688  [8]
 LDCM0372  CL103 HCT 116 C284(0.88)  LDD0689  [8]
 LDCM0373  CL104 HCT 116 C284(0.90)  LDD0690  [8]
 LDCM0374  CL105 HEK-293T C284(1.03)  LDD1578  [9]
 LDCM0375  CL106 HEK-293T C284(0.98)  LDD1579  [9]
 LDCM0376  CL107 HEK-293T C284(0.96); C895(0.98)  LDD1580  [9]
 LDCM0377  CL108 HEK-293T C284(0.88)  LDD1581  [9]
 LDCM0378  CL109 HEK-293T C284(1.01)  LDD1582  [9]
 LDCM0379  CL11 HEK-293T C284(1.07)  LDD1583  [9]
 LDCM0380  CL110 HEK-293T C284(1.09)  LDD1584  [9]
 LDCM0381  CL111 HEK-293T C284(1.04); C895(0.98)  LDD1585  [9]
 LDCM0382  CL112 HEK-293T C284(1.00)  LDD1586  [9]
 LDCM0383  CL113 HEK-293T C284(1.06)  LDD1587  [9]
 LDCM0384  CL114 HEK-293T C284(0.98)  LDD1588  [9]
 LDCM0385  CL115 HEK-293T C284(1.05); C895(0.69)  LDD1589  [9]
 LDCM0386  CL116 HEK-293T C284(0.92)  LDD1590  [9]
 LDCM0387  CL117 HCT 116 C284(1.32)  LDD0704  [8]
 LDCM0388  CL118 HCT 116 C284(1.22)  LDD0705  [8]
 LDCM0389  CL119 HCT 116 C284(1.73)  LDD0706  [8]
 LDCM0390  CL12 HEK-293T C284(1.03)  LDD1594  [9]
 LDCM0391  CL120 HCT 116 C284(1.43)  LDD0708  [8]
 LDCM0392  CL121 HCT 116 C284(1.00)  LDD0709  [8]
 LDCM0393  CL122 HCT 116 C284(1.01)  LDD0710  [8]
 LDCM0394  CL123 HCT 116 C284(0.88)  LDD0711  [8]
 LDCM0395  CL124 HCT 116 C284(1.07)  LDD0712  [8]
 LDCM0396  CL125 HCT 116 C284(1.13)  LDD0713  [8]
 LDCM0397  CL126 HCT 116 C284(1.00)  LDD0714  [8]
 LDCM0398  CL127 HCT 116 C284(1.06)  LDD0715  [8]
 LDCM0399  CL128 HCT 116 C284(1.19)  LDD0716  [8]
 LDCM0400  CL13 HEK-293T C284(1.03)  LDD1604  [9]
 LDCM0401  CL14 HEK-293T C284(0.95)  LDD1605  [9]
 LDCM0402  CL15 HEK-293T C284(1.05); C895(0.88)  LDD1606  [9]
 LDCM0403  CL16 HEK-293T C284(0.86)  LDD1607  [9]
 LDCM0404  CL17 HEK-293T C284(1.20)  LDD1608  [9]
 LDCM0405  CL18 HEK-293T C284(1.02)  LDD1609  [9]
 LDCM0406  CL19 HEK-293T C284(1.00)  LDD1610  [9]
 LDCM0407  CL2 HEK-293T C284(1.07)  LDD1611  [9]
 LDCM0408  CL20 HEK-293T C284(1.02)  LDD1612  [9]
 LDCM0409  CL21 HEK-293T C284(1.03)  LDD1613  [9]
 LDCM0410  CL22 HEK-293T C284(1.09)  LDD1614  [9]
 LDCM0411  CL23 HEK-293T C284(1.06)  LDD1615  [9]
 LDCM0412  CL24 HEK-293T C284(0.97)  LDD1616  [9]
 LDCM0413  CL25 HEK-293T C284(1.00)  LDD1617  [9]
 LDCM0414  CL26 HEK-293T C284(0.95)  LDD1618  [9]
 LDCM0415  CL27 HEK-293T C284(1.00); C895(0.77)  LDD1619  [9]
 LDCM0416  CL28 HEK-293T C284(0.95)  LDD1620  [9]
 LDCM0417  CL29 HEK-293T C284(1.10)  LDD1621  [9]
 LDCM0418  CL3 HEK-293T C284(0.99); C895(0.91)  LDD1622  [9]
 LDCM0419  CL30 HEK-293T C284(1.00)  LDD1623  [9]
 LDCM0420  CL31 HCT 116 C284(1.03)  LDD0737  [8]
 LDCM0421  CL32 HCT 116 C284(1.06)  LDD0738  [8]
 LDCM0422  CL33 HCT 116 C284(1.17)  LDD0739  [8]
 LDCM0423  CL34 HCT 116 C284(1.33)  LDD0740  [8]
 LDCM0424  CL35 HCT 116 C284(1.08)  LDD0741  [8]
 LDCM0425  CL36 HCT 116 C284(1.21)  LDD0742  [8]
 LDCM0426  CL37 HCT 116 C284(1.24)  LDD0743  [8]
 LDCM0428  CL39 HCT 116 C284(1.26)  LDD0745  [8]
 LDCM0429  CL4 HEK-293T C284(0.86)  LDD1633  [9]
 LDCM0430  CL40 HCT 116 C284(1.93)  LDD0747  [8]
 LDCM0431  CL41 HCT 116 C284(1.09)  LDD0748  [8]
 LDCM0432  CL42 HCT 116 C284(1.12)  LDD0749  [8]
 LDCM0433  CL43 HCT 116 C284(1.20)  LDD0750  [8]
 LDCM0434  CL44 HCT 116 C284(1.23)  LDD0751  [8]
 LDCM0435  CL45 HCT 116 C284(1.16)  LDD0752  [8]
 LDCM0436  CL46 HEK-293T C284(1.14)  LDD1640  [9]
 LDCM0437  CL47 HEK-293T C284(1.01)  LDD1641  [9]
 LDCM0438  CL48 HEK-293T C284(1.00)  LDD1642  [9]
 LDCM0439  CL49 HEK-293T C284(0.98)  LDD1643  [9]
 LDCM0440  CL5 HEK-293T C284(1.09)  LDD1644  [9]
 LDCM0441  CL50 HEK-293T C284(1.09)  LDD1645  [9]
 LDCM0443  CL52 HEK-293T C284(0.99)  LDD1646  [9]
 LDCM0444  CL53 HEK-293T C284(1.13)  LDD1647  [9]
 LDCM0445  CL54 HEK-293T C284(1.00)  LDD1648  [9]
 LDCM0446  CL55 HEK-293T C284(1.05)  LDD1649  [9]
 LDCM0447  CL56 HEK-293T C284(1.09)  LDD1650  [9]
 LDCM0448  CL57 HEK-293T C284(1.11)  LDD1651  [9]
 LDCM0449  CL58 HEK-293T C284(1.02)  LDD1652  [9]
 LDCM0450  CL59 HEK-293T C284(1.09)  LDD1653  [9]
 LDCM0451  CL6 HEK-293T C284(1.08)  LDD1654  [9]
 LDCM0452  CL60 HEK-293T C284(1.01)  LDD1655  [9]
 LDCM0453  CL61 HCT 116 C284(0.99)  LDD0770  [8]
 LDCM0454  CL62 HCT 116 C284(1.01)  LDD0771  [8]
 LDCM0455  CL63 HCT 116 C284(0.84)  LDD0772  [8]
 LDCM0456  CL64 HCT 116 C284(0.86)  LDD0773  [8]
 LDCM0457  CL65 HCT 116 C284(0.88)  LDD0774  [8]
 LDCM0458  CL66 HCT 116 C284(0.92)  LDD0775  [8]
 LDCM0459  CL67 HCT 116 C284(0.92)  LDD0776  [8]
 LDCM0460  CL68 HCT 116 C284(0.83)  LDD0777  [8]
 LDCM0461  CL69 HCT 116 C284(1.12)  LDD0778  [8]
 LDCM0462  CL7 HEK-293T C284(1.00)  LDD1665  [9]
 LDCM0463  CL70 HCT 116 C284(0.76)  LDD0780  [8]
 LDCM0464  CL71 HCT 116 C284(0.83)  LDD0781  [8]
 LDCM0465  CL72 HCT 116 C284(1.02)  LDD0782  [8]
 LDCM0466  CL73 HCT 116 C284(0.84)  LDD0783  [8]
 LDCM0467  CL74 HCT 116 C284(1.02)  LDD0784  [8]
 LDCM0469  CL76 HCT 116 C284(0.83)  LDD0786  [8]
 LDCM0470  CL77 HCT 116 C284(0.74)  LDD0787  [8]
 LDCM0471  CL78 HCT 116 C284(0.87)  LDD0788  [8]
 LDCM0472  CL79 HCT 116 C284(1.02)  LDD0789  [8]
 LDCM0473  CL8 HEK-293T C284(1.09)  LDD1676  [9]
 LDCM0474  CL80 HCT 116 C284(0.84)  LDD0791  [8]
 LDCM0475  CL81 HCT 116 C284(0.79)  LDD0792  [8]
 LDCM0476  CL82 HCT 116 C284(0.70)  LDD0793  [8]
 LDCM0477  CL83 HCT 116 C284(0.80)  LDD0794  [8]
 LDCM0478  CL84 HCT 116 C284(0.76)  LDD0795  [8]
 LDCM0479  CL85 HCT 116 C284(0.81)  LDD0796  [8]
 LDCM0480  CL86 HCT 116 C284(0.99)  LDD0797  [8]
 LDCM0481  CL87 HCT 116 C284(0.76)  LDD0798  [8]
 LDCM0482  CL88 HCT 116 C284(0.76)  LDD0799  [8]
 LDCM0483  CL89 HCT 116 C284(0.95)  LDD0800  [8]
 LDCM0484  CL9 HEK-293T C284(0.95)  LDD1687  [9]
 LDCM0485  CL90 HCT 116 C284(0.83)  LDD0802  [8]
 LDCM0486  CL91 HCT 116 C284(0.94)  LDD0803  [8]
 LDCM0487  CL92 HCT 116 C284(0.95)  LDD0804  [8]
 LDCM0488  CL93 HCT 116 C284(0.85)  LDD0805  [8]
 LDCM0489  CL94 HCT 116 C284(1.05)  LDD0806  [8]
 LDCM0490  CL95 HCT 116 C284(0.96)  LDD0807  [8]
 LDCM0491  CL96 HCT 116 C284(0.99)  LDD0808  [8]
 LDCM0492  CL97 HCT 116 C284(0.97)  LDD0809  [8]
 LDCM0493  CL98 HCT 116 C284(0.94)  LDD0810  [8]
 LDCM0494  CL99 HCT 116 C284(0.81)  LDD0811  [8]
 LDCM0495  E2913 HEK-293T C284(1.06); C895(0.83)  LDD1698  [9]
 LDCM0468  Fragment33 HCT 116 C284(0.89)  LDD0785  [8]
 LDCM0427  Fragment51 HCT 116 C284(1.55)  LDD0744  [8]
 LDCM0022  KB02 HEK-293T C284(0.99)  LDD1492  [9]
 LDCM0023  KB03 HEK-293T C284(0.99)  LDD1497  [9]
 LDCM0024  KB05 COLO792 C284(2.54)  LDD3310  [10]
 LDCM0021  THZ1 HCT 116 C242(1.42); C248(1.42); C260(1.42); C284(0.98)  LDD2173  [8]

References

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Mass spectrometry data entry: PXD028270
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Mass spectrometry data entry: PXD023056 , PXD023059 , PXD023058 , PXD023057 , PXD023060
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Mass spectrometry data entry: PXD041264
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Mass spectrometry data entry: PXD029255
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Mass spectrometry data entry: PXD033004
7 Design and synthesis of minimalist terminal alkyne-containing diazirine photo-crosslinkers and their incorporation into kinase inhibitors for cell- and tissue-based proteome profiling. Angew Chem Int Ed Engl. 2013 Aug 12;52(33):8551-6. doi: 10.1002/anie.201300683. Epub 2013 Jun 10.
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9 Accelerating multiplexed profiling of protein-ligand interactions: High-throughput plate-based reactive cysteine profiling with minimal input. Cell Chem Biol. 2024 Mar 21;31(3):565-576.e4. doi: 10.1016/j.chembiol.2023.11.015. Epub 2023 Dec 19.
Mass spectrometry data entry: PXD044402
10 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840