Details of the Target

General Information of Target

Target ID LDTP06302
Target Name Arf-GAP with coiled-coil, ANK repeat and PH domain-containing protein 2 (ACAP2)
Gene Name ACAP2
Gene ID 23527
Synonyms
CENTB2; KIAA0041; Arf-GAP with coiled-coil, ANK repeat and PH domain-containing protein 2; Centaurin-beta-2; Cnt-b2
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MKMTVDFEECLKDSPRFRAALEEVEGDVAELELKLDKLVKLCIAMIDTGKAFCVANKQFM
NGIRDLAQYSSNDAVVETSLTKFSDSLQEMINFHTILFDQTQRSIKAQLQNFVKEDLRKF
KDAKKQFEKVSEEKENALVKNAQVQRNKQHEVEEATNILTATRKCFRHIALDYVLQINVL
QSKRRSEILKSMLSFMYAHLAFFHQGYDLFSELGPYMKDLGAQLDRLVVDAAKEKREMEQ
KHSTIQQKDFSSDDSKLEYNVDAANGIVMEGYLFKRASNAFKTWNRRWFSIQNNQLVYQK
KFKDNPTVVVEDLRLCTVKHCEDIERRFCFEVVSPTKSCMLQADSEKLRQAWIKAVQTSI
ATAYREKGDESEKLDKKSSPSTGSLDSGNESKEKLLKGESALQRVQCIPGNASCCDCGLA
DPRWASINLGITLCIECSGIHRSLGVHFSKVRSLTLDTWEPELLKLMCELGNDVINRVYE
ANVEKMGIKKPQPGQRQEKEAYIRAKYVERKFVDKYSISLSPPEQQKKFVSKSSEEKRLS
ISKFGPGDQVRASAQSSVRSNDSGIQQSSDDGRESLPSTVSANSLYEPEGERQDSSMFLD
SKHLNPGLQLYRASYEKNLPKMAEALAHGADVNWANSEENKATPLIQAVLGGSLVTCEFL
LQNGANVNQRDVQGRGPLHHATVLGHTGQVCLFLKRGANQHATDEEGKDPLSIAVEAANA
DIVTLLRLARMNEEMRESEGLYGQPGDETYQDIFRDFSQMASNNPEKLNRFQQDSQKF
Target Bioclass
Other
Subcellular location
Endosome membrane
Function GTPase-activating protein (GAP) for ADP ribosylation factor 6 (ARF6).
Uniprot ID
Q15057
Ensemble ID
ENST00000326793.11
HGNC ID
HGNC:16469

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 16 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
m-APA
 Probe Info  		13.31  LDD0402  [1]
EN219-alkyne
 Probe Info  		5.75  LDD0297  [2]
Probe 1
 Probe Info  		Y586(12.44); Y750(15.12)  LDD3495  [3]
BTD
 Probe Info  		C53(2.56)  LDD1700  [4]
AHL-Pu-1
 Probe Info  		C468(2.04)  LDD0169  [5]
DBIA
 Probe Info  		C53(4.69)  LDD0204  [6]
IPM
 Probe Info  		C53(1.59)  LDD1701  [4]
4-Iodoacetamidophenylacetylene
 Probe Info  		C329(0.00); C321(0.00); C42(0.00); C53(0.00)  LDD0038  [7]
IA-alkyne
 Probe Info  		C329(0.00); C42(0.00); C10(0.00); C339(0.00)  LDD0036  [7]
Lodoacetamide azide
 Probe Info  		C329(0.00); C10(0.00); C339(0.00); C53(0.00)  LDD0037  [7]
NAIA_4
 Probe Info  		C414(0.00); C407(0.00)  LDD2226  [8]
STPyne
 Probe Info  		N.A.  LDD0009  [9]
TFBX
 Probe Info  		C53(0.00); C468(0.00)  LDD0148  [10]
Acrolein
 Probe Info  		N.A.  LDD0217  [11]
AOyne
 Probe Info  		15.00  LDD0443  [12]
NAIA_5
 Probe Info  		C657(0.00); C329(0.00); C321(0.00); C339(0.00)  LDD2223  [8]
PAL-AfBPP Probe
Click To Hide/Show 5 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
C147
 Probe Info  		6.54  LDD1829  [13]
C156
 Probe Info  		6.02  LDD1836  [13]
C159
 Probe Info  		12.04  LDD1839  [13]
C160
 Probe Info  		9.85  LDD1840  [13]
VE-P
 Probe Info  		N.A.  LDD0396  [14]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0026  4SU-RNA+native RNA HEK-293T C468(2.04)  LDD0169  [5]
 LDCM0214  AC1 HCT 116 C321(0.72); C329(1.76); C407(0.89); C414(0.84)  LDD0531  [15]
 LDCM0215  AC10 HCT 116 C321(0.87); C329(1.09); C407(1.16); C414(1.17)  LDD0532  [15]
 LDCM0216  AC100 HCT 116 C321(0.62); C329(0.67); C407(0.73); C414(0.77)  LDD0533  [15]
 LDCM0217  AC101 HCT 116 C321(0.67); C329(0.79); C407(0.82); C414(0.83)  LDD0534  [15]
 LDCM0218  AC102 HCT 116 C321(0.61); C329(0.66); C407(0.70); C414(0.73)  LDD0535  [15]
 LDCM0219  AC103 HCT 116 C321(0.68); C329(0.74); C407(0.85); C414(0.92)  LDD0536  [15]
 LDCM0220  AC104 HCT 116 C321(0.62); C329(0.65); C407(0.70); C414(0.76)  LDD0537  [15]
 LDCM0221  AC105 HCT 116 C321(0.63); C329(0.75); C407(0.80); C414(0.85)  LDD0538  [15]
 LDCM0222  AC106 HCT 116 C321(0.63); C329(0.66); C407(0.74); C414(0.89)  LDD0539  [15]
 LDCM0223  AC107 HCT 116 C321(0.69); C329(0.65); C407(0.74); C414(0.87)  LDD0540  [15]
 LDCM0224  AC108 HCT 116 C321(0.84); C329(0.76); C407(0.80); C414(0.79)  LDD0541  [15]
 LDCM0225  AC109 HCT 116 C321(0.61); C329(0.96); C407(0.94); C414(0.85)  LDD0542  [15]
 LDCM0226  AC11 HCT 116 C321(0.88); C329(1.27); C407(0.95); C414(0.96)  LDD0543  [15]
 LDCM0227  AC110 HCT 116 C321(0.67); C329(0.86); C407(0.77); C414(0.79)  LDD0544  [15]
 LDCM0228  AC111 HCT 116 C321(0.60); C329(0.63); C407(0.76); C414(0.77)  LDD0545  [15]
 LDCM0229  AC112 HCT 116 C321(0.60); C329(0.75); C407(0.83); C414(0.91)  LDD0546  [15]
 LDCM0230  AC113 HCT 116 C321(1.11); C329(0.98); C407(0.88); C414(1.01)  LDD0547  [15]
 LDCM0231  AC114 HCT 116 C321(0.99); C329(0.82); C407(0.80); C414(1.06)  LDD0548  [15]
 LDCM0232  AC115 HCT 116 C321(1.03); C329(0.85); C407(0.68); C414(1.00)  LDD0549  [15]
 LDCM0233  AC116 HCT 116 C321(1.01); C329(0.83); C407(0.70); C414(1.13)  LDD0550  [15]
 LDCM0234  AC117 HCT 116 C321(0.82); C329(0.86); C407(0.80); C414(0.78)  LDD0551  [15]
 LDCM0235  AC118 HCT 116 C321(0.96); C329(0.92); C407(0.94); C414(0.96)  LDD0552  [15]
 LDCM0236  AC119 HCT 116 C321(0.94); C329(0.85); C407(0.79); C414(1.19)  LDD0553  [15]
 LDCM0237  AC12 HCT 116 C321(0.85); C329(1.24); C407(1.16); C414(1.06)  LDD0554  [15]
 LDCM0238  AC120 HCT 116 C321(1.07); C329(0.90); C407(0.79); C414(1.09)  LDD0555  [15]
 LDCM0239  AC121 HCT 116 C321(0.73); C329(0.96); C407(0.88); C414(0.87)  LDD0556  [15]
 LDCM0240  AC122 HCT 116 C321(0.91); C329(1.11); C407(0.73); C414(0.91)  LDD0557  [15]
 LDCM0241  AC123 HCT 116 C321(0.74); C329(1.08); C407(0.89); C414(0.61)  LDD0558  [15]
 LDCM0242  AC124 HCT 116 C321(0.77); C329(0.88); C407(1.10); C414(1.15)  LDD0559  [15]
 LDCM0243  AC125 HCT 116 C321(0.99); C329(0.93); C407(0.69); C414(1.40)  LDD0560  [15]
 LDCM0244  AC126 HCT 116 C321(1.05); C329(0.96); C407(0.75); C414(1.25)  LDD0561  [15]
 LDCM0245  AC127 HCT 116 C321(0.89); C329(0.87); C407(0.73); C414(1.40)  LDD0562  [15]
 LDCM0246  AC128 HCT 116 C321(1.11); C329(1.09); C407(1.27); C414(1.26)  LDD0563  [15]
 LDCM0247  AC129 HCT 116 C321(1.18); C329(0.84); C407(1.26); C414(1.15)  LDD0564  [15]
 LDCM0249  AC130 HCT 116 C321(1.09); C329(0.98); C407(1.24); C414(1.20)  LDD0566  [15]
 LDCM0250  AC131 HCT 116 C321(0.99); C329(0.73); C407(1.02); C414(0.94)  LDD0567  [15]
 LDCM0251  AC132 HCT 116 C321(1.26); C329(1.01); C407(1.26); C414(1.17)  LDD0568  [15]
 LDCM0252  AC133 HCT 116 C321(1.10); C329(1.05); C407(1.10); C414(1.06)  LDD0569  [15]
 LDCM0253  AC134 HCT 116 C321(1.00); C329(0.97); C407(1.14); C414(1.13)  LDD0570  [15]
 LDCM0254  AC135 HCT 116 C321(1.13); C329(1.00); C407(1.24); C414(1.32)  LDD0571  [15]
 LDCM0255  AC136 HCT 116 C321(1.10); C329(1.14); C407(1.21); C414(1.12)  LDD0572  [15]
 LDCM0256  AC137 HCT 116 C321(0.95); C329(1.19); C407(1.15); C414(1.14)  LDD0573  [15]
 LDCM0257  AC138 HCT 116 C321(1.02); C329(1.04); C407(1.12); C414(1.00)  LDD0574  [15]
 LDCM0258  AC139 HCT 116 C321(1.05); C329(1.14); C407(1.29); C414(1.26)  LDD0575  [15]
 LDCM0259  AC14 HCT 116 C321(0.94); C329(1.17); C407(0.92); C414(0.94)  LDD0576  [15]
 LDCM0260  AC140 HCT 116 C321(1.12); C329(1.08); C407(1.36); C414(1.20)  LDD0577  [15]
 LDCM0261  AC141 HCT 116 C321(1.08); C329(1.00); C407(1.20); C414(1.18)  LDD0578  [15]
 LDCM0262  AC142 HCT 116 C321(1.15); C329(1.15); C407(1.12); C414(1.05)  LDD0579  [15]
 LDCM0263  AC143 HCT 116 C329(0.81); C407(1.07); C414(1.47); C415(0.76)  LDD0580  [15]
 LDCM0264  AC144 HCT 116 C329(0.86); C417(0.87); C415(0.99); C53(1.10)  LDD0581  [15]
 LDCM0265  AC145 HCT 116 C415(0.87); C329(0.88); C53(1.04); C407(1.21)  LDD0582  [15]
 LDCM0266  AC146 HCT 116 C417(0.59); C329(0.76); C53(1.05); C407(1.15)  LDD0583  [15]
 LDCM0267  AC147 HCT 116 C329(0.96); C415(1.03); C417(1.20); C407(1.24)  LDD0584  [15]
 LDCM0268  AC148 HCT 116 C329(0.79); C417(0.84); C415(1.03); C407(1.06)  LDD0585  [15]
 LDCM0269  AC149 HCT 116 C417(0.43); C329(0.76); C415(1.10); C407(1.21)  LDD0586  [15]
 LDCM0270  AC15 HCT 116 C321(0.87); C53(0.98); C407(0.99); C329(1.02)  LDD0587  [15]
 LDCM0271  AC150 HCT 116 C417(0.65); C329(0.79); C415(0.97); C53(1.43)  LDD0588  [15]
 LDCM0272  AC151 HCT 116 C417(0.69); C329(0.85); C53(1.05); C415(1.20)  LDD0589  [15]
 LDCM0273  AC152 HCT 116 C417(0.63); C329(0.82); C53(1.01); C407(1.16)  LDD0590  [15]
 LDCM0274  AC153 HCT 116 C417(0.36); C329(0.68); C415(1.26); C407(1.27)  LDD0591  [15]
 LDCM0621  AC154 HCT 116 C329(0.69); C407(1.29); C414(1.54); C415(1.08)  LDD2158  [15]
 LDCM0622  AC155 HCT 116 C329(0.65); C407(1.29); C414(1.60); C415(1.36)  LDD2159  [15]
 LDCM0623  AC156 HCT 116 C329(0.81); C407(1.15); C414(1.37); C415(1.10)  LDD2160  [15]
 LDCM0624  AC157 HCT 116 C329(0.75); C407(1.26); C414(1.69); C415(1.19)  LDD2161  [15]
 LDCM0276  AC17 HCT 116 C53(0.79); C329(0.85); C417(0.88); C414(0.97)  LDD0593  [15]
 LDCM0277  AC18 HCT 116 C329(0.76); C53(0.89); C417(0.99); C468(1.03)  LDD0594  [15]
 LDCM0278  AC19 HCT 116 C417(0.83); C329(0.89); C53(0.89); C414(1.01)  LDD0595  [15]
 LDCM0279  AC2 HCT 116 C321(0.73); C407(0.99); C417(1.00); C414(1.01)  LDD0596  [15]
 LDCM0280  AC20 HCT 116 C407(0.84); C329(0.84); C414(0.90); C321(0.92)  LDD0597  [15]
 LDCM0281  AC21 HCT 116 C329(0.76); C53(0.84); C407(0.90); C414(0.90)  LDD0598  [15]
 LDCM0282  AC22 HCT 116 C321(0.74); C53(0.85); C407(0.93); C329(0.98)  LDD0599  [15]
 LDCM0283  AC23 HCT 116 C321(0.66); C329(0.85); C407(0.92); C414(0.95)  LDD0600  [15]
 LDCM0284  AC24 HCT 116 C53(0.73); C321(0.74); C407(0.89); C329(0.93)  LDD0601  [15]
 LDCM0285  AC25 HCT 116 C417(0.84); C415(0.86); C468(0.89); C329(0.91)  LDD0602  [15]
 LDCM0286  AC26 HCT 116 C468(0.77); C329(0.80); C417(0.85); C415(0.86)  LDD0603  [15]
 LDCM0287  AC27 HCT 116 C468(0.67); C329(0.72); C417(0.75); C415(0.79)  LDD0604  [15]
 LDCM0288  AC28 HCT 116 C468(0.72); C329(0.79); C415(0.86); C414(0.88)  LDD0605  [15]
 LDCM0289  AC29 HCT 116 C468(0.64); C329(0.70); C417(0.76); C415(0.77)  LDD0606  [15]
 LDCM0290  AC3 HCT 116 C321(0.79); C417(0.85); C415(0.86); C414(0.89)  LDD0607  [15]
 LDCM0291  AC30 HCT 116 C329(0.66); C468(0.80); C415(0.82); C407(0.85)  LDD0608  [15]
 LDCM0292  AC31 HCT 116 C329(0.74); C415(0.81); C468(0.82); C417(0.83)  LDD0609  [15]
 LDCM0293  AC32 HCT 116 C321(0.63); C329(0.67); C417(0.78); C468(0.85)  LDD0610  [15]
 LDCM0294  AC33 HCT 116 C321(0.46); C417(0.77); C329(0.77); C415(0.79)  LDD0611  [15]
 LDCM0295  AC34 HCT 116 C321(0.44); C329(0.72); C468(0.72); C53(0.94)  LDD0612  [15]
 LDCM0296  AC35 HCT 116 C53(0.86); C407(0.94); C321(0.97); C468(1.05)  LDD0613  [15]
 LDCM0297  AC36 HCT 116 C407(0.88); C53(0.92); C321(1.05); C414(1.05)  LDD0614  [15]
 LDCM0298  AC37 HCT 116 C407(0.84); C414(0.91); C417(0.92); C415(0.93)  LDD0615  [15]
 LDCM0299  AC38 HCT 116 C407(0.96); C321(0.96); C53(0.96); C415(0.96)  LDD0616  [15]
 LDCM0300  AC39 HCT 116 C321(0.90); C53(1.06); C417(1.08); C407(1.12)  LDD0617  [15]
 LDCM0301  AC4 HCT 116 C321(0.81); C415(0.83); C417(0.83); C414(0.97)  LDD0618  [15]
 LDCM0302  AC40 HCT 116 C329(0.99); C321(1.00); C407(1.01); C414(1.05)  LDD0619  [15]
 LDCM0303  AC41 HCT 116 C321(0.86); C415(0.86); C329(0.94); C53(0.99)  LDD0620  [15]
 LDCM0304  AC42 HCT 116 C321(0.81); C53(0.90); C468(0.97); C329(1.01)  LDD0621  [15]
 LDCM0305  AC43 HCT 116 C321(0.84); C329(0.96); C53(1.01); C468(1.02)  LDD0622  [15]
 LDCM0306  AC44 HCT 116 C407(0.91); C329(0.92); C53(0.96); C321(0.98)  LDD0623  [15]
 LDCM0307  AC45 HCT 116 C415(0.96); C329(0.96); C321(1.00); C414(1.01)  LDD0624  [15]
 LDCM0308  AC46 HCT 116 C53(0.94); C329(0.97); C468(0.98); C407(1.00)  LDD0625  [15]
 LDCM0309  AC47 HCT 116 C468(0.87); C53(0.97); C329(0.99); C417(1.11)  LDD0626  [15]
 LDCM0310  AC48 HCT 116 C407(1.00); C468(1.00); C53(1.04); C329(1.05)  LDD0627  [15]
 LDCM0311  AC49 HCT 116 C53(0.87); C329(0.90); C321(0.92); C417(1.01)  LDD0628  [15]
 LDCM0312  AC5 HCT 116 C417(0.85); C321(0.86); C53(0.99); C414(1.07)  LDD0629  [15]
 LDCM0313  AC50 HCT 116 C53(0.85); C417(0.88); C321(0.88); C468(0.92)  LDD0630  [15]
 LDCM0314  AC51 HCT 116 C468(0.80); C53(0.92); C321(0.99); C329(1.01)  LDD0631  [15]
 LDCM0315  AC52 HCT 116 C329(0.88); C53(0.90); C468(0.90); C321(0.93)  LDD0632  [15]
 LDCM0316  AC53 HCT 116 C53(0.91); C468(0.93); C417(1.04); C329(1.05)  LDD0633  [15]
 LDCM0317  AC54 HCT 116 C417(0.85); C53(0.87); C415(0.90); C321(0.90)  LDD0634  [15]
 LDCM0318  AC55 HCT 116 C53(0.91); C468(1.01); C321(1.01); C329(1.06)  LDD0635  [15]
 LDCM0319  AC56 HCT 116 C321(0.85); C417(0.97); C53(0.97); C468(1.03)  LDD0636  [15]
 LDCM0320  AC57 HCT 116 C414(0.91); C407(0.97); C53(1.01); C329(1.09)  LDD0637  [15]
 LDCM0321  AC58 HCT 116 C329(0.92); C415(1.01); C53(1.07); C417(1.08)  LDD0638  [15]
 LDCM0322  AC59 HCT 116 C329(0.94); C53(1.00); C414(1.01); C407(1.05)  LDD0639  [15]
 LDCM0323  AC6 HCT 116 C407(0.83); C321(0.94); C329(0.95); C417(1.00)  LDD0640  [15]
 LDCM0324  AC60 HCT 116 C407(0.86); C329(0.87); C53(0.93); C414(0.99)  LDD0641  [15]
 LDCM0325  AC61 HCT 116 C407(0.79); C53(0.85); C329(0.94); C414(0.95)  LDD0642  [15]
 LDCM0326  AC62 HCT 116 C329(0.87); C468(0.98); C53(0.98); C414(1.09)  LDD0643  [15]
 LDCM0327  AC63 HCT 116 C414(0.78); C407(0.82); C329(0.95); C415(0.98)  LDD0644  [15]
 LDCM0328  AC64 HCT 116 C329(0.92); C414(0.98); C407(1.05); C53(1.08)  LDD0645  [15]
 LDCM0329  AC65 HCT 116 C329(0.87); C53(0.93); C407(1.04); C415(1.12)  LDD0646  [15]
 LDCM0330  AC66 HCT 116 C329(0.92); C407(0.94); C415(0.99); C414(1.07)  LDD0647  [15]
 LDCM0331  AC67 HCT 116 C329(0.84); C415(1.03); C53(1.08); C407(1.09)  LDD0648  [15]
 LDCM0332  AC68 HCT 116 C407(0.90); C414(0.90); C329(0.99); C415(1.00)  LDD0649  [15]
 LDCM0333  AC69 HCT 116 C414(1.02); C415(1.06); C329(1.06); C417(1.11)  LDD0650  [15]
 LDCM0334  AC7 HCT 116 C321(0.92); C329(1.02); C468(1.04); C414(1.06)  LDD0651  [15]
 LDCM0335  AC70 HCT 116 C414(0.94); C329(0.95); C415(0.98); C417(1.01)  LDD0652  [15]
 LDCM0336  AC71 HCT 116 C407(1.03); C329(1.10); C414(1.21); C415(1.24)  LDD0653  [15]
 LDCM0337  AC72 HCT 116 C414(0.94); C329(0.99); C407(1.04); C415(1.26)  LDD0654  [15]
 LDCM0338  AC73 HCT 116 C407(1.01); C414(1.13); C329(1.19); C415(1.19)  LDD0655  [15]
 LDCM0339  AC74 HCT 116 C414(1.14); C407(1.15); C329(1.22); C415(1.33)  LDD0656  [15]
 LDCM0340  AC75 HCT 116 C414(0.90); C407(0.94); C415(1.14); C329(1.22)  LDD0657  [15]
 LDCM0341  AC76 HCT 116 C407(0.97); C414(1.03); C329(1.04); C415(1.28)  LDD0658  [15]
 LDCM0342  AC77 HCT 116 C407(0.89); C329(0.98); C414(1.01); C415(1.23)  LDD0659  [15]
 LDCM0343  AC78 HCT 116 C407(0.88); C414(1.09); C415(1.10); C329(1.12)  LDD0660  [15]
 LDCM0344  AC79 HCT 116 C407(1.00); C329(1.06); C414(1.07); C415(1.32)  LDD0661  [15]
 LDCM0345  AC8 HCT 116 C407(0.83); C417(0.85); C414(0.93); C321(0.93)  LDD0662  [15]
 LDCM0346  AC80 HCT 116 C329(1.02); C407(1.11); C415(1.12); C414(1.13)  LDD0663  [15]
 LDCM0347  AC81 HCT 116 C414(1.01); C415(1.10); C407(1.12); C329(1.14)  LDD0664  [15]
 LDCM0348  AC82 HCT 116 C407(0.90); C414(1.00); C415(1.21); C329(1.37)  LDD0665  [15]
 LDCM0349  AC83 HCT 116 C329(0.75); C414(0.86); C407(0.88); C468(0.90)  LDD0666  [15]
 LDCM0350  AC84 HCT 116 C329(0.72); C468(0.78); C414(0.79); C407(0.83)  LDD0667  [15]
 LDCM0351  AC85 HCT 116 C329(0.71); C468(0.74); C414(0.81); C407(0.85)  LDD0668  [15]
 LDCM0352  AC86 HCT 116 C329(0.69); C468(0.75); C407(0.79); C414(0.81)  LDD0669  [15]
 LDCM0353  AC87 HCT 116 C468(0.79); C329(0.93); C407(0.98); C53(1.02)  LDD0670  [15]
 LDCM0354  AC88 HCT 116 C407(0.73); C414(0.74); C329(0.77); C468(0.81)  LDD0671  [15]
 LDCM0355  AC89 HCT 116 C329(0.72); C407(0.75); C414(0.80); C468(0.89)  LDD0672  [15]
 LDCM0357  AC90 HCT 116 C468(0.82); C415(0.96); C329(1.01); C414(1.01)  LDD0674  [15]
 LDCM0358  AC91 HCT 116 C468(0.67); C329(0.72); C407(0.74); C414(0.82)  LDD0675  [15]
 LDCM0359  AC92 HCT 116 C329(0.75); C414(0.79); C407(0.80); C468(0.87)  LDD0676  [15]
 LDCM0360  AC93 HCT 116 C329(0.71); C415(0.79); C414(0.80); C407(0.84)  LDD0677  [15]
 LDCM0361  AC94 HCT 116 C468(0.75); C329(0.77); C407(1.08); C53(1.09)  LDD0678  [15]
 LDCM0362  AC95 HCT 116 C415(0.82); C468(0.83); C414(0.92); C407(0.93)  LDD0679  [15]
 LDCM0363  AC96 HCT 116 C329(0.71); C414(0.86); C407(0.87); C468(0.92)  LDD0680  [15]
 LDCM0364  AC97 HCT 116 C329(0.70); C407(0.74); C414(0.76); C468(0.78)  LDD0681  [15]
 LDCM0365  AC98 HCT 116 C321(0.65); C53(0.66); C415(0.72); C407(0.84)  LDD0682  [15]
 LDCM0366  AC99 HCT 116 C321(0.64); C468(0.71); C415(0.72); C53(0.79)  LDD0683  [15]
 LDCM0248  AKOS034007472 HCT 116 C321(0.90); C329(1.22); C407(0.96); C414(1.18)  LDD0565  [15]
 LDCM0356  AKOS034007680 HCT 116 C53(0.95); C321(0.98); C407(1.05); C417(1.16)  LDD0673  [15]
 LDCM0275  AKOS034007705 HCT 116 C407(0.90); C415(0.91); C321(0.92); C417(0.92)  LDD0592  [15]
 LDCM0102  BDHI 8 Jurkat C53(4.69)  LDD0204  [6]
 LDCM0108  Chloroacetamide HeLa N.A.  LDD0222  [11]
 LDCM0632  CL-Sc Hep-G2 C691(20.00)  LDD2227  [8]
 LDCM0367  CL1 HCT 116 C407(0.89); C414(0.89); C415(0.90); C468(0.93)  LDD0684  [15]
 LDCM0368  CL10 HCT 116 C414(0.91); C329(0.98); C415(0.99); C407(1.00)  LDD0685  [15]
 LDCM0369  CL100 HCT 116 C417(0.69); C321(0.71); C414(0.79); C415(0.83)  LDD0686  [15]
 LDCM0370  CL101 HCT 116 C407(0.82); C417(0.91); C321(0.94); C329(0.98)  LDD0687  [15]
 LDCM0371  CL102 HCT 116 C53(0.97); C415(1.02); C407(1.03); C321(1.05)  LDD0688  [15]
 LDCM0372  CL103 HCT 116 C414(0.97); C407(1.00); C321(1.00); C53(1.03)  LDD0689  [15]
 LDCM0373  CL104 HCT 116 C407(0.88); C321(0.96); C414(0.97); C417(1.01)  LDD0690  [15]
 LDCM0374  CL105 HCT 116 C329(0.76); C417(0.79); C414(0.91); C53(0.94)  LDD0691  [15]
 LDCM0375  CL106 HCT 116 C329(0.85); C417(0.98); C53(1.05); C414(1.19)  LDD0692  [15]
 LDCM0376  CL107 HCT 116 C329(0.70); C53(0.87); C407(1.06); C321(1.07)  LDD0693  [15]
 LDCM0377  CL108 HCT 116 C329(0.84); C53(0.91); C417(1.01); C414(1.05)  LDD0694  [15]
 LDCM0378  CL109 HCT 116 C417(0.65); C321(0.71); C329(0.73); C414(0.75)  LDD0695  [15]
 LDCM0379  CL11 HCT 116 C407(0.89); C321(0.99); C414(1.00); C329(1.06)  LDD0696  [15]
 LDCM0380  CL110 HCT 116 C321(0.67); C417(0.77); C329(0.78); C414(0.84)  LDD0697  [15]
 LDCM0381  CL111 HCT 116 C329(0.77); C407(0.78); C321(0.79); C414(0.81)  LDD0698  [15]
 LDCM0382  CL112 HCT 116 C468(0.60); C329(0.83); C417(0.85); C415(0.94)  LDD0699  [15]
 LDCM0383  CL113 HCT 116 C321(0.53); C329(0.63); C417(0.72); C415(0.76)  LDD0700  [15]
 LDCM0384  CL114 HCT 116 C321(0.50); C329(0.68); C468(0.75); C417(0.77)  LDD0701  [15]
 LDCM0385  CL115 HCT 116 C321(0.55); C329(0.65); C415(0.80); C417(0.81)  LDD0702  [15]
 LDCM0386  CL116 HCT 116 C321(0.47); C329(0.79); C468(0.85); C415(0.87)  LDD0703  [15]
 LDCM0387  CL117 HCT 116 C321(1.05); C407(1.09); C415(1.10); C417(1.10)  LDD0704  [15]
 LDCM0388  CL118 HCT 116 C468(1.00); C407(1.01); C321(1.01); C329(1.06)  LDD0705  [15]
 LDCM0389  CL119 HCT 116 C321(0.91); C407(0.95); C329(0.95); C53(1.02)  LDD0706  [15]
 LDCM0390  CL12 HCT 116 C414(1.04); C407(1.04); C321(1.08); C329(1.08)  LDD0707  [15]
 LDCM0391  CL120 HCT 116 C321(0.86); C53(0.90); C415(0.91); C329(0.96)  LDD0708  [15]
 LDCM0392  CL121 HCT 116 C53(0.83); C329(0.85); C468(0.95); C414(1.00)  LDD0709  [15]
 LDCM0393  CL122 HCT 116 C53(0.83); C321(0.92); C329(0.96); C468(1.03)  LDD0710  [15]
 LDCM0394  CL123 HCT 116 C468(0.82); C417(0.84); C415(0.84); C53(0.90)  LDD0711  [15]
 LDCM0395  CL124 HCT 116 C415(0.91); C53(0.92); C417(0.93); C329(0.94)  LDD0712  [15]
 LDCM0396  CL125 HCT 116 C53(0.84); C329(0.89); C468(0.90); C415(1.00)  LDD0713  [15]
 LDCM0397  CL126 HCT 116 C329(0.86); C415(0.91); C468(0.95); C53(0.96)  LDD0714  [15]
 LDCM0398  CL127 HCT 116 C329(0.85); C407(0.87); C414(0.92); C468(0.96)  LDD0715  [15]
 LDCM0399  CL128 HCT 116 C407(0.79); C53(0.87); C415(0.88); C414(0.92)  LDD0716  [15]
 LDCM0400  CL13 HCT 116 C321(0.89); C414(0.94); C407(1.01); C329(1.04)  LDD0717  [15]
 LDCM0401  CL14 HCT 116 C321(0.87); C329(0.95); C414(0.96); C415(1.05)  LDD0718  [15]
 LDCM0402  CL15 HCT 116 C407(0.91); C414(0.95); C321(1.01); C329(1.03)  LDD0719  [15]
 LDCM0403  CL16 HCT 116 C415(0.52); C417(0.52); C329(0.85); C321(0.85)  LDD0720  [15]
 LDCM0404  CL17 HCT 116 C415(0.65); C417(0.65); C321(0.89); C53(1.02)  LDD0721  [15]
 LDCM0405  CL18 HCT 116 C415(0.72); C417(0.72); C407(0.78); C414(0.78)  LDD0722  [15]
 LDCM0406  CL19 HCT 116 C415(0.66); C417(0.66); C407(0.85); C414(0.85)  LDD0723  [15]
 LDCM0407  CL2 HCT 116 C468(0.98); C417(1.00); C415(1.02); C321(1.03)  LDD0724  [15]
 LDCM0408  CL20 HCT 116 C415(0.50); C417(0.50); C407(0.89); C414(0.89)  LDD0725  [15]
 LDCM0409  CL21 HCT 116 C415(0.56); C417(0.56); C329(0.99); C53(1.11)  LDD0726  [15]
 LDCM0410  CL22 HCT 116 C415(0.61); C417(0.61); C407(1.02); C414(1.02)  LDD0727  [15]
 LDCM0411  CL23 HCT 116 C415(0.55); C417(0.55); C407(0.68); C414(0.68)  LDD0728  [15]
 LDCM0412  CL24 HCT 116 C415(0.52); C417(0.52); C407(0.76); C414(0.76)  LDD0729  [15]
 LDCM0413  CL25 HCT 116 C321(1.00); C329(0.79); C407(0.79); C414(0.79)  LDD0730  [15]
 LDCM0414  CL26 HCT 116 C321(0.93); C329(0.79); C407(1.12); C414(1.12)  LDD0731  [15]
 LDCM0415  CL27 HCT 116 C321(1.26); C329(1.01); C407(0.85); C414(0.85)  LDD0732  [15]
 LDCM0416  CL28 HCT 116 C321(1.19); C329(0.85); C407(0.87); C414(0.87)  LDD0733  [15]
 LDCM0417  CL29 HCT 116 C321(1.12); C329(0.97); C407(0.76); C414(0.76)  LDD0734  [15]
 LDCM0418  CL3 HCT 116 C321(1.00); C329(1.01); C407(1.13); C414(0.88)  LDD0735  [15]
 LDCM0419  CL30 HCT 116 C321(1.03); C329(0.90); C407(0.99); C414(0.99)  LDD0736  [15]
 LDCM0420  CL31 HCT 116 C321(1.01); C407(0.82); C414(0.66); C415(0.81)  LDD0737  [15]
 LDCM0421  CL32 HCT 116 C321(1.18); C407(1.02); C414(1.13); C415(1.20)  LDD0738  [15]
 LDCM0422  CL33 HCT 116 C321(0.94); C407(0.97); C414(0.81); C415(0.80)  LDD0739  [15]
 LDCM0423  CL34 HCT 116 C321(1.09); C407(0.98); C414(1.01); C415(0.99)  LDD0740  [15]
 LDCM0424  CL35 HCT 116 C321(0.94); C407(1.12); C414(1.12); C415(0.78)  LDD0741  [15]
 LDCM0425  CL36 HCT 116 C321(1.15); C407(0.96); C414(0.82); C415(0.85)  LDD0742  [15]
 LDCM0426  CL37 HCT 116 C321(1.05); C407(1.02); C414(0.93); C415(0.84)  LDD0743  [15]
 LDCM0428  CL39 HCT 116 C321(1.05); C407(1.03); C414(1.29); C415(1.11)  LDD0745  [15]
 LDCM0429  CL4 HCT 116 C321(1.00); C329(0.99); C407(1.16); C414(0.98)  LDD0746  [15]
 LDCM0430  CL40 HCT 116 C321(0.99); C407(0.85); C414(0.77); C415(0.71)  LDD0747  [15]
 LDCM0431  CL41 HCT 116 C321(0.97); C407(0.95); C414(0.88); C415(0.97)  LDD0748  [15]
 LDCM0432  CL42 HCT 116 C321(0.94); C407(1.12); C414(1.04); C415(1.01)  LDD0749  [15]
 LDCM0433  CL43 HCT 116 C321(1.08); C407(0.95); C414(0.89); C415(0.95)  LDD0750  [15]
 LDCM0434  CL44 HCT 116 C321(1.04); C407(1.02); C414(0.85); C415(0.92)  LDD0751  [15]
 LDCM0435  CL45 HCT 116 C321(1.01); C407(1.14); C414(1.14); C415(0.94)  LDD0752  [15]
 LDCM0436  CL46 HCT 116 C321(0.95); C329(1.07); C407(1.85); C414(1.23)  LDD0753  [15]
 LDCM0437  CL47 HCT 116 C321(0.85); C329(0.97); C407(0.81); C414(0.86)  LDD0754  [15]
 LDCM0438  CL48 HCT 116 C321(1.27); C329(1.05); C407(1.01); C414(1.06)  LDD0755  [15]
 LDCM0439  CL49 HCT 116 C321(1.56); C329(1.05); C407(1.48); C414(1.26)  LDD0756  [15]
 LDCM0440  CL5 HCT 116 C321(1.11); C329(1.00); C407(1.10); C414(1.05)  LDD0757  [15]
 LDCM0441  CL50 HCT 116 C321(0.87); C329(1.08); C407(1.19); C414(1.02)  LDD0758  [15]
 LDCM0442  CL51 HCT 116 C321(0.89); C329(1.09); C407(0.94); C414(1.23)  LDD0759  [15]
 LDCM0443  CL52 HCT 116 C321(1.01); C329(1.02); C407(0.89); C414(0.82)  LDD0760  [15]
 LDCM0444  CL53 HCT 116 C321(0.70); C329(0.85); C407(1.27); C414(1.03)  LDD0761  [15]
 LDCM0445  CL54 HCT 116 C321(0.93); C329(1.03); C407(1.14); C414(1.11)  LDD0762  [15]
 LDCM0446  CL55 HCT 116 C321(0.87); C329(1.06); C407(0.88); C414(1.00)  LDD0763  [15]
 LDCM0447  CL56 HCT 116 C321(0.92); C329(0.98); C407(0.93); C414(0.94)  LDD0764  [15]
 LDCM0448  CL57 HCT 116 C321(0.82); C329(0.94); C407(1.21); C414(1.11)  LDD0765  [15]
 LDCM0449  CL58 HCT 116 C321(0.95); C329(1.10); C407(0.74); C414(0.90)  LDD0766  [15]
 LDCM0450  CL59 HCT 116 C321(1.15); C329(0.99); C407(1.19); C414(1.46)  LDD0767  [15]
 LDCM0451  CL6 HCT 116 C321(1.03); C329(1.10); C407(0.82); C414(0.91)  LDD0768  [15]
 LDCM0452  CL60 HCT 116 C321(1.06); C329(1.02); C407(1.02); C414(0.97)  LDD0769  [15]
 LDCM0453  CL61 HCT 116 C329(0.99); C407(1.11); C414(1.05); C415(0.92)  LDD0770  [15]
 LDCM0454  CL62 HCT 116 C329(0.92); C407(1.06); C414(1.08); C415(0.87)  LDD0771  [15]
 LDCM0455  CL63 HCT 116 C329(0.92); C407(1.17); C414(1.00); C415(0.89)  LDD0772  [15]
 LDCM0456  CL64 HCT 116 C329(0.80); C407(1.15); C414(1.05); C415(1.02)  LDD0773  [15]
 LDCM0457  CL65 HCT 116 C329(0.99); C407(1.33); C414(1.09); C415(1.00)  LDD0774  [15]
 LDCM0458  CL66 HCT 116 C329(0.92); C407(1.15); C414(1.07); C415(0.89)  LDD0775  [15]
 LDCM0459  CL67 HCT 116 C329(0.95); C407(1.02); C414(1.07); C415(1.15)  LDD0776  [15]
 LDCM0460  CL68 HCT 116 C329(0.98); C407(1.10); C414(1.24); C415(1.76)  LDD0777  [15]
 LDCM0461  CL69 HCT 116 C329(1.25); C407(0.81); C414(1.04); C415(1.03)  LDD0778  [15]
 LDCM0462  CL7 HCT 116 C321(0.97); C329(1.06); C407(1.04); C414(1.02)  LDD0779  [15]
 LDCM0463  CL70 HCT 116 C329(1.01); C407(0.91); C414(0.94); C415(0.95)  LDD0780  [15]
 LDCM0464  CL71 HCT 116 C329(0.85); C407(1.26); C414(1.15); C415(1.19)  LDD0781  [15]
 LDCM0465  CL72 HCT 116 C329(1.04); C407(0.90); C414(1.11); C415(1.20)  LDD0782  [15]
 LDCM0466  CL73 HCT 116 C329(0.85); C407(1.08); C414(1.07); C415(1.02)  LDD0783  [15]
 LDCM0467  CL74 HCT 116 C329(0.87); C407(1.05); C414(1.11); C415(1.19)  LDD0784  [15]
 LDCM0469  CL76 HCT 116 C321(1.05); C407(0.99); C414(0.94); C415(0.89)  LDD0786  [15]
 LDCM0470  CL77 HCT 116 C321(0.89); C407(0.84); C414(0.79); C415(0.77)  LDD0787  [15]
 LDCM0471  CL78 HCT 116 C321(1.06); C407(0.85); C414(0.76); C415(0.87)  LDD0788  [15]
 LDCM0472  CL79 HCT 116 C321(1.12); C407(0.89); C414(0.85); C415(0.85)  LDD0789  [15]
 LDCM0473  CL8 HCT 116 C321(1.01); C329(0.93); C407(1.02); C414(1.02)  LDD0790  [15]
 LDCM0474  CL80 HCT 116 C321(1.06); C407(1.05); C414(0.95); C415(1.11)  LDD0791  [15]
 LDCM0475  CL81 HCT 116 C321(0.94); C407(1.37); C414(1.19); C415(1.02)  LDD0792  [15]
 LDCM0476  CL82 HCT 116 C321(1.11); C407(0.99); C414(0.96); C415(0.79)  LDD0793  [15]
 LDCM0477  CL83 HCT 116 C321(1.09); C407(1.03); C414(1.07); C415(0.95)  LDD0794  [15]
 LDCM0478  CL84 HCT 116 C321(1.19); C407(0.91); C414(0.92); C415(0.94)  LDD0795  [15]
 LDCM0479  CL85 HCT 116 C321(1.03); C407(0.82); C414(0.81); C415(0.91)  LDD0796  [15]
 LDCM0480  CL86 HCT 116 C321(0.95); C407(0.99); C414(1.04); C415(0.90)  LDD0797  [15]
 LDCM0481  CL87 HCT 116 C321(1.09); C407(1.36); C414(1.27); C415(1.00)  LDD0798  [15]
 LDCM0482  CL88 HCT 116 C321(1.09); C407(1.22); C414(1.28); C415(0.80)  LDD0799  [15]
 LDCM0483  CL89 HCT 116 C321(1.20); C407(1.04); C414(1.07); C415(1.00)  LDD0800  [15]
 LDCM0484  CL9 HCT 116 C321(0.98); C329(0.95); C407(1.11); C414(1.01)  LDD0801  [15]
 LDCM0485  CL90 HCT 116 C321(0.94); C407(1.18); C414(1.12); C415(0.99)  LDD0802  [15]
 LDCM0486  CL91 HCT 116 C321(0.91); C329(1.02); C407(0.81); C414(0.91)  LDD0803  [15]
 LDCM0487  CL92 HCT 116 C321(0.81); C329(0.92); C407(0.69); C414(0.74)  LDD0804  [15]
 LDCM0488  CL93 HCT 116 C321(1.02); C329(1.29); C407(1.01); C414(0.81)  LDD0805  [15]
 LDCM0489  CL94 HCT 116 C321(0.97); C329(1.48); C407(0.68); C414(0.80)  LDD0806  [15]
 LDCM0490  CL95 HCT 116 C321(0.83); C329(0.96); C407(1.00); C414(1.05)  LDD0807  [15]
 LDCM0491  CL96 HCT 116 C321(1.03); C329(1.08); C407(1.00); C414(0.75)  LDD0808  [15]
 LDCM0492  CL97 HCT 116 C321(0.91); C329(1.06); C407(0.88); C414(0.76)  LDD0809  [15]
 LDCM0493  CL98 HCT 116 C321(0.98); C329(1.50); C407(0.72); C414(0.85)  LDD0810  [15]
 LDCM0494  CL99 HCT 116 C321(0.84); C329(1.62); C407(0.79); C414(0.80)  LDD0811  [15]
 LDCM0495  E2913 HEK-293T C321(1.08); C329(0.86); C468(1.00); C407(1.12)  LDD1698  [16]
 LDCM0213  Electrophilic fragment 2 MDA-MB-231 C53(1.63)  LDD1702  [4]
 LDCM0100  EN219 231MFP 4.17  LDD0298  [2]
 LDCM0625  F8 Ramos C468(0.77); C53(1.33); C42(0.65)  LDD2187  [17]
 LDCM0572  Fragment10 Ramos C468(1.06); C53(1.41)  LDD2189  [17]
 LDCM0573  Fragment11 Ramos C468(0.15); C53(0.66); C42(0.76)  LDD2190  [17]
 LDCM0574  Fragment12 Ramos C468(1.57); C53(1.87)  LDD2191  [17]
 LDCM0575  Fragment13 Ramos C468(1.04); C53(0.91)  LDD2192  [17]
 LDCM0576  Fragment14 Ramos C468(0.88); C53(0.73); C42(0.56)  LDD2193  [17]
 LDCM0579  Fragment20 Ramos C468(0.99); C53(1.90)  LDD2194  [17]
 LDCM0580  Fragment21 Ramos C468(1.23)  LDD2195  [17]
 LDCM0582  Fragment23 Ramos C468(1.18); C53(1.15)  LDD2196  [17]
 LDCM0578  Fragment27 Ramos C468(1.03); C53(0.90)  LDD2197  [17]
 LDCM0586  Fragment28 Ramos C468(0.82); C53(0.84)  LDD2198  [17]
 LDCM0588  Fragment30 Ramos C468(1.73); C53(0.86)  LDD2199  [17]
 LDCM0589  Fragment31 Ramos C468(1.09); C53(0.89)  LDD2200  [17]
 LDCM0590  Fragment32 Ramos C468(0.85); C53(0.89)  LDD2201  [17]
 LDCM0468  Fragment33 HCT 116 C329(0.92); C407(1.01); C414(0.94); C415(1.05)  LDD0785  [15]
 LDCM0596  Fragment38 Ramos C468(0.88); C53(0.95)  LDD2203  [17]
 LDCM0566  Fragment4 Ramos C468(0.78); C53(2.46); C42(1.01)  LDD2184  [17]
 LDCM0427  Fragment51 HCT 116 C321(0.98); C407(1.04); C414(1.19); C415(0.94)  LDD0744  [15]
 LDCM0610  Fragment52 Ramos C468(1.28); C53(1.11)  LDD2204  [17]
 LDCM0614  Fragment56 Ramos C468(1.20); C53(0.80)  LDD2205  [17]
 LDCM0569  Fragment7 Ramos C468(0.64); C53(1.32); C42(0.62)  LDD2186  [17]
 LDCM0571  Fragment9 Ramos C468(0.98)  LDD2188  [17]
 LDCM0022  KB02 HEK-293T C321(0.94); C53(1.04); C329(0.89); C468(1.01)  LDD1492  [16]
 LDCM0023  KB03 HEK-293T C321(1.00); C53(1.02); C329(1.08); C468(0.95)  LDD1497  [16]
 LDCM0024  KB05 SKMEL24 C468(3.20)  LDD3323  [18]
 LDCM0518  Nucleophilic fragment 22a MDA-MB-231 C53(1.28)  LDD2111  [4]
 LDCM0536  Nucleophilic fragment 31 MDA-MB-231 C53(2.19)  LDD2129  [4]
 LDCM0211  Nucleophilic fragment 3b MDA-MB-231 C53(2.56)  LDD1700  [4]
 LDCM0554  Nucleophilic fragment 7a MDA-MB-231 C53(0.66)  LDD2148  [4]

References

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Mass spectrometry data entry: PXD039908 , PXD029761
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Mass spectrometry data entry: PXD044625
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Mass spectrometry data entry: PXD028853
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Mass spectrometry data entry: PXD041264
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Mass spectrometry data entry: PXD027758 , PXD027755 , PXD027760 , PXD027762 , PXD027756 , PXD027591 , PXD007149 , PXD030064 , PXD032392 , PXD027789 , PXD027767 , PXD027764
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Mass spectrometry data entry: PXD029255
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Mass spectrometry data entry: PXD041587
14 Pharmacological Targeting of Vacuolar H(+)-ATPase via Subunit V1G Combats Multidrug-Resistant Cancer. Cell Chem Biol. 2020 Nov 19;27(11):1359-1370.e8. doi: 10.1016/j.chembiol.2020.06.011. Epub 2020 Jul 9.
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Mass spectrometry data entry: PXD044402
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Mass spectrometry data entry: PXD027578
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Mass spectrometry data entry: PXD047840