Details of the Target

General Information of Target

Target ID LDTP06366
Target Name Poly(rC)-binding protein 1 (PCBP1)
Gene Name PCBP1
Gene ID 5093
Synonyms
Poly(rC)-binding protein 1; Alpha-CP1; Heterogeneous nuclear ribonucleoprotein E1; hnRNP E1; Nucleic acid-binding protein SUB2.3
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MDAGVTESGLNVTLTIRLLMHGKEVGSIIGKKGESVKRIREESGARINISEGNCPERIIT
LTGPTNAIFKAFAMIIDKLEEDINSSMTNSTAASRPPVTLRLVVPATQCGSLIGKGGCKI
KEIRESTGAQVQVAGDMLPNSTERAITIAGVPQSVTECVKQICLVMLETLSQSPQGRVMT
IPYQPMPASSPVICAGGQDRCSDAAGYPHATHDLEGPPLDAYSIQGQHTISPLDLAKLNQ
VARQQSHFAMMHGGTGFAGIDSSSPEVKGYWASLDASTQTTHELTIPNNLIGCIIGRQGA
NINEIRQMSGAQIKIANPVEGSSGRQVTITGSAASISLAQYLINARLSSEKGMGCS
Target Bioclass
Other
Subcellular location
Nucleus
Function
Single-stranded nucleic acid binding protein that binds preferentially to oligo dC. Together with PCBP2, required for erythropoiesis, possibly by regulating mRNA splicing.; (Microbial infection) In case of infection by poliovirus, plays a role in initiation of viral RNA replication in concert with the viral protein 3CD.
Uniprot ID
Q15365
Ensemble ID
ENST00000303577.7
HGNC ID
HGNC:8647
ChEMBL ID
CHEMBL4295825

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 64 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
m-APA
 Probe Info  		15.00  LDD0402  [1]
P1
 Probe Info  		10.00  LDD0448  [2]
P2
 Probe Info  		10.00  LDD0449  [2]
P3
 Probe Info  		10.00  LDD0450  [2]
P8
 Probe Info  		1.69  LDD0451  [2]
A-EBA
 Probe Info  		4.73  LDD0215  [3]
11RK72
 Probe Info  		3.01  LDD0327  [4]
11RK73
 Probe Info  		2.97  LDD0328  [4]
DAyne
 Probe Info  		5.10  LDD0261  [5]
CHEMBL5175495
 Probe Info  		5.80  LDD0196  [6]
CY-1
 Probe Info  		19.28  LDD0243  [7]
CY4
 Probe Info  		5.41  LDD0244  [7]
W1
 Probe Info  		17.21  LDD0235  [8]
TH211
 Probe Info  		Y183(20.00); Y341(5.40)  LDD0260  [9]
TH216
 Probe Info  		Y183(9.21); Y341(7.72)  LDD0259  [9]
YN-1
 Probe Info  		2.36  LDD0444  [10]
YN-4
 Probe Info  		100.00  LDD0445  [10]
ONAyne
 Probe Info  		K115(0.94)  LDD0274  [11]
BTD
 Probe Info  		C54(8.76)  LDD1699  [12]
AZ-9
 Probe Info  		E304(0.98); E56(1.00); D199(1.36)  LDD2208  [13]
OPA-S-S-alkyne
 Probe Info  		K314(1.71)  LDD3494  [14]
JZ128-DTB
 Probe Info  		C109(0.00); C54(0.00)  LDD0462  [15]
THZ1-DTB
 Probe Info  		C109(1.06); C54(1.05)  LDD0460  [15]
AHL-Pu-1
 Probe Info  		C194(2.59)  LDD0169  [16]
Alkyne-RA190
 Probe Info  		2.01  LDD0299  [17]
EA-probe
 Probe Info  		N.A.  LDD0440  [18]
HHS-482
 Probe Info  		Y183(1.07); Y270(1.24); Y341(1.03)  LDD0285  [19]
HHS-475
 Probe Info  		Y222(0.71); Y183(0.81); Y341(0.85); Y270(0.93)  LDD0264  [20]
HHS-465
 Probe Info  		Y183(10.00); Y207(10.00); Y270(8.38); Y341(7.78)  LDD2237  [21]
DBIA
 Probe Info  		C194(1.06)  LDD0078  [22]
5E-2FA
 Probe Info  		H252(0.00); H247(0.00)  LDD2235  [23]
AMP probe
 Probe Info  		N.A.  LDD0200  [24]
ATP probe
 Probe Info  		K23(0.00); K31(0.00); K32(0.00); K115(0.00)  LDD0199  [24]
4-Iodoacetamidophenylacetylene
 Probe Info  		C158(0.00); C201(0.00); C293(0.00); C54(0.00)  LDD0038  [25]
IA-alkyne
 Probe Info  		C54(0.00); C194(0.00); C158(0.00); C109(0.00)  LDD0032  [26]
IPIAA_H
 Probe Info  		C158(0.00); C54(0.00)  LDD0030  [27]
IPIAA_L
 Probe Info  		C293(0.00); C201(0.00); C163(0.00); C158(0.00)  LDD0031  [27]
Lodoacetamide azide
 Probe Info  		C158(0.00); C201(0.00); C293(0.00); C54(0.00)  LDD0037  [25]
ATP probe
 Probe Info  		N.A.  LDD0035  [28]
JW-RF-010
 Probe Info  		C163(0.00); C54(0.00); C158(0.00); C118(0.00)  LDD0026  [29]
NAIA_4
 Probe Info  		C54(0.00); C109(0.00); C118(0.00); C158(0.00)  LDD2226  [30]
TFBX
 Probe Info  		C201(0.00); C109(0.00); C355(0.00); C158(0.00)  LDD0027  [29]
WYneC
 Probe Info  		N.A.  LDD0014  [31]
WYneN
 Probe Info  		C194(0.00); C54(0.00); C109(0.00)  LDD0021  [31]
WYneO
 Probe Info  		C54(0.00); C194(0.00); C109(0.00); C158(0.00)  LDD0022  [31]
DA-P3
 Probe Info  		N.A.  LDD0178  [32]
aHNE
 Probe Info  		C201(0.00); C194(0.00)  LDD0001  [31]
Compound 10
 Probe Info  		C109(0.00); C158(0.00); C194(0.00); C201(0.00)  LDD2216  [33]
Compound 11
 Probe Info  		C109(0.00); C158(0.00); C194(0.00); C201(0.00)  LDD2213  [33]
ENE
 Probe Info  		C194(0.00); C109(0.00); C158(0.00); C54(0.00)  LDD0006  [31]
IPM
 Probe Info  		C54(0.00); C194(0.00); C109(0.00)  LDD0005  [31]
NHS
 Probe Info  		K23(0.00); K314(0.00)  LDD0010  [31]
PF-06672131
 Probe Info  		C54(0.00); C109(0.00); C158(0.00); C194(0.00)  LDD0017  [34]
PPMS
 Probe Info  		C194(0.00); C54(0.00); C158(0.00); C109(0.00)  LDD0008  [31]
SF
 Probe Info  		K31(0.00); K32(0.00); Y341(0.00)  LDD0028  [35]
STPyne
 Probe Info  		K160(0.00); K115(0.00)  LDD0009  [31]
VSF
 Probe Info  		C158(0.00); C54(0.00); C194(0.00)  LDD0007  [31]
Phosphinate-6
 Probe Info  		C194(0.00); C54(0.00); C118(0.00); C109(0.00)  LDD0018  [36]
1c-yne
 Probe Info  		K78(0.00); K160(0.00); K314(0.00)  LDD0228  [37]
Acrolein
 Probe Info  		C194(0.00); C163(0.00); C158(0.00); C109(0.00)  LDD0217  [38]
Cinnamaldehyde
 Probe Info  		N.A.  LDD0220  [38]
Crotonaldehyde
 Probe Info  		C158(0.00); C109(0.00)  LDD0219  [38]
Methacrolein
 Probe Info  		C109(0.00); C194(0.00)  LDD0218  [38]
NAIA_5
 Probe Info  		C163(0.00); C158(0.00); C201(0.00); C118(0.00)  LDD2223  [30]
PAL-AfBPP Probe
Click To Hide/Show 10 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
FFF probe11
 Probe Info  		5.80  LDD0472  [39]
FFF probe13
 Probe Info  		10.50  LDD0475  [39]
FFF probe2
 Probe Info  		9.53  LDD0463  [39]
FFF probe3
 Probe Info  		12.63  LDD0464  [39]
FFF probe4
 Probe Info  		20.00  LDD0466  [39]
STS-2
 Probe Info  		N.A.  LDD0138  [40]
VE-P
 Probe Info  		N.A.  LDD0396  [41]
BD-F
 Probe Info  		A345(0.00); N344(0.00)  LDD0024  [42]
OEA-DA
 Probe Info  		3.20  LDD0046  [43]
STS-1
 Probe Info  		N.A.  LDD0068  [44]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0548  1-(4-(Benzo[d][1,3]dioxol-5-ylmethyl)piperazin-1-yl)-2-nitroethan-1-one MDA-MB-231 C109(0.44)  LDD2142  [12]
 LDCM0519  1-(6-methoxy-3,4-dihydroquinolin-1(2H)-yl)-2-nitroethan-1-one MDA-MB-231 C158(0.73)  LDD2112  [12]
 LDCM0502  1-(Cyanoacetyl)piperidine MDA-MB-231 C158(0.76); C109(0.58)  LDD2095  [12]
 LDCM0537  2-Cyano-N,N-dimethylacetamide MDA-MB-231 C158(1.00); C109(0.83)  LDD2130  [12]
 LDCM0524  2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide MDA-MB-231 C158(0.96); C109(0.71); C194(0.83)  LDD2117  [12]
 LDCM0558  2-Cyano-N-phenylacetamide MDA-MB-231 C158(0.90); C109(1.02)  LDD2152  [12]
 LDCM0539  3-(4-Isopropylpiperazin-1-yl)-3-oxopropanenitrile MDA-MB-231 C158(0.54); C109(0.39); C201(0.71)  LDD2132  [12]
 LDCM0538  4-(Cyanoacetyl)morpholine MDA-MB-231 C158(0.88); C109(0.61)  LDD2131  [12]
 LDCM0025  4SU-RNA DM93 C201(2.50); C194(2.28)  LDD0170  [16]
 LDCM0026  4SU-RNA+native RNA HEK-293T C194(2.59)  LDD0169  [16]
 LDCM0214  AC1 HCT 116 C109(1.24); C118(1.29); C158(0.71); C163(0.84)  LDD0531  [22]
 LDCM0215  AC10 HCT 116 C109(1.30); C118(1.44); C158(1.00); C194(0.66)  LDD0532  [22]
 LDCM0216  AC100 HCT 116 C109(0.79); C118(0.58); C158(0.82); C194(0.86)  LDD0533  [22]
 LDCM0217  AC101 HCT 116 C109(0.81); C118(0.75); C158(0.77); C194(0.84)  LDD0534  [22]
 LDCM0218  AC102 HCT 116 C109(0.90); C118(0.93); C158(0.81); C194(0.82)  LDD0535  [22]
 LDCM0219  AC103 HCT 116 C109(0.98); C118(1.09); C158(0.79); C194(1.10)  LDD0536  [22]
 LDCM0220  AC104 HCT 116 C109(0.95); C118(0.93); C158(0.82); C194(1.01)  LDD0537  [22]
 LDCM0221  AC105 HCT 116 C109(1.30); C118(1.70); C158(0.77); C194(0.88)  LDD0538  [22]
 LDCM0222  AC106 HCT 116 C109(0.67); C118(0.35); C158(0.80); C194(0.86)  LDD0539  [22]
 LDCM0223  AC107 HCT 116 C109(0.77); C118(0.65); C158(0.78); C194(0.92)  LDD0540  [22]
 LDCM0224  AC108 HCT 116 C109(0.95); C118(0.72); C158(0.84); C194(0.83)  LDD0541  [22]
 LDCM0225  AC109 HCT 116 C109(1.79); C118(2.52); C158(0.82); C194(0.81)  LDD0542  [22]
 LDCM0226  AC11 HCT 116 C109(2.81); C118(3.90); C158(0.92); C194(0.81)  LDD0543  [22]
 LDCM0227  AC110 HCT 116 C109(0.96); C118(0.93); C158(0.83); C194(0.96)  LDD0544  [22]
 LDCM0228  AC111 HCT 116 C109(1.06); C118(0.85); C158(0.77); C194(1.17)  LDD0545  [22]
 LDCM0229  AC112 HCT 116 C109(0.91); C118(0.78); C158(0.78); C194(1.10)  LDD0546  [22]
 LDCM0230  AC113 HCT 116 C109(1.03); C118(0.94); C158(0.85); C163(0.88)  LDD0547  [22]
 LDCM0231  AC114 HCT 116 C109(1.10); C118(1.27); C158(0.84); C163(0.89)  LDD0548  [22]
 LDCM0232  AC115 HCT 116 C109(1.15); C118(0.81); C158(0.89); C163(0.93)  LDD0549  [22]
 LDCM0233  AC116 HCT 116 C109(1.08); C118(1.00); C158(0.86); C163(0.86)  LDD0550  [22]
 LDCM0234  AC117 HCT 116 C109(1.07); C118(1.06); C158(0.84); C163(0.92)  LDD0551  [22]
 LDCM0235  AC118 HCT 116 C109(1.07); C118(1.14); C158(0.87); C163(1.04)  LDD0552  [22]
 LDCM0236  AC119 HCT 116 C109(1.07); C118(1.33); C158(0.88); C163(0.88)  LDD0553  [22]
 LDCM0237  AC12 HCT 116 C109(1.72); C118(2.13); C158(1.00); C194(0.74)  LDD0554  [22]
 LDCM0238  AC120 HCT 116 C109(1.06); C118(0.18); C158(0.96); C163(1.09)  LDD0555  [22]
 LDCM0239  AC121 HCT 116 C109(1.05); C118(1.04); C158(0.95); C163(1.16)  LDD0556  [22]
 LDCM0240  AC122 HCT 116 C109(1.14); C118(1.19); C158(0.87); C163(1.00)  LDD0557  [22]
 LDCM0241  AC123 HCT 116 C109(1.20); C118(1.12); C158(0.89); C163(0.86)  LDD0558  [22]
 LDCM0242  AC124 HCT 116 C109(1.02); C118(0.54); C158(0.96); C163(0.86)  LDD0559  [22]
 LDCM0243  AC125 HCT 116 C109(1.03); C118(0.30); C158(0.91); C163(0.95)  LDD0560  [22]
 LDCM0244  AC126 HCT 116 C109(1.17); C118(0.84); C158(0.99); C163(0.93)  LDD0561  [22]
 LDCM0245  AC127 HCT 116 C109(1.17); C118(0.85); C158(0.89); C163(0.80)  LDD0562  [22]
 LDCM0246  AC128 HCT 116 C109(1.15); C118(1.12); C158(1.04); C194(0.75)  LDD0563  [22]
 LDCM0247  AC129 HCT 116 C109(0.94); C118(0.89); C158(0.94); C194(0.91)  LDD0564  [22]
 LDCM0249  AC130 HCT 116 C109(0.94); C118(0.82); C158(0.98); C194(0.72)  LDD0566  [22]
 LDCM0250  AC131 HCT 116 C109(0.99); C118(1.05); C158(0.91); C194(2.20)  LDD0567  [22]
 LDCM0251  AC132 HCT 116 C109(0.97); C118(0.96); C158(1.07); C194(0.41)  LDD0568  [22]
 LDCM0252  AC133 HCT 116 C109(1.06); C118(1.10); C158(1.00); C194(0.43)  LDD0569  [22]
 LDCM0253  AC134 HCT 116 C109(1.05); C118(1.05); C158(0.96); C194(0.56)  LDD0570  [22]
 LDCM0254  AC135 HCT 116 C109(0.96); C118(0.85); C158(0.98); C194(0.38)  LDD0571  [22]
 LDCM0255  AC136 HCT 116 C109(0.96); C118(0.82); C158(0.94); C194(0.46)  LDD0572  [22]
 LDCM0256  AC137 HCT 116 C109(1.18); C118(1.23); C158(1.00); C194(0.43)  LDD0573  [22]
 LDCM0257  AC138 HCT 116 C109(1.06); C118(0.88); C158(0.97); C194(0.38)  LDD0574  [22]
 LDCM0258  AC139 HCT 116 C109(0.99); C118(0.84); C158(0.89); C194(0.47)  LDD0575  [22]
 LDCM0259  AC14 HCT 116 C109(1.41); C118(1.73); C158(0.90); C194(0.99)  LDD0576  [22]
 LDCM0260  AC140 HCT 116 C109(1.06); C118(0.96); C158(0.99); C194(0.44)  LDD0577  [22]
 LDCM0261  AC141 HCT 116 C109(0.95); C118(0.79); C158(0.99); C194(0.44)  LDD0578  [22]
 LDCM0262  AC142 HCT 116 C109(0.87); C118(0.75); C158(0.92); C194(0.34)  LDD0579  [22]
 LDCM0263  AC143 HCT 116 C118(0.74); C194(0.81); C158(0.88); C109(0.94)  LDD0580  [22]
 LDCM0264  AC144 HCT 116 C118(0.72); C158(0.84); C109(0.99); C194(1.32)  LDD0581  [22]
 LDCM0265  AC145 HCT 116 C118(0.65); C194(0.79); C158(0.85); C109(0.93)  LDD0582  [22]
 LDCM0266  AC146 HCT 116 C118(0.75); C158(0.79); C194(0.84); C109(0.91)  LDD0583  [22]
 LDCM0267  AC147 HCT 116 C118(0.67); C158(0.86); C194(0.94); C109(1.01)  LDD0584  [22]
 LDCM0268  AC148 HCT 116 C118(0.76); C158(0.91); C194(1.10); C109(1.13)  LDD0585  [22]
 LDCM0269  AC149 HCT 116 C118(0.77); C158(0.83); C194(0.87); C109(0.97)  LDD0586  [22]
 LDCM0270  AC15 HCT 116 C194(0.89); C158(0.94); C109(1.69); C118(2.25)  LDD0587  [22]
 LDCM0271  AC150 HCT 116 C118(0.61); C109(0.86); C158(0.86); C194(0.86)  LDD0588  [22]
 LDCM0272  AC151 HCT 116 C118(0.66); C109(0.88); C158(0.90); C194(1.07)  LDD0589  [22]
 LDCM0273  AC152 HCT 116 C118(0.48); C158(0.87); C109(0.95); C194(0.98)  LDD0590  [22]
 LDCM0274  AC153 HCT 116 C118(0.51); C158(0.95); C109(1.20); C194(1.50)  LDD0591  [22]
 LDCM0621  AC154 HCT 116 C109(0.93); C118(0.69); C158(0.86); C194(1.13)  LDD2158  [22]
 LDCM0622  AC155 HCT 116 C109(0.97); C118(0.74); C158(0.88); C194(1.83)  LDD2159  [22]
 LDCM0623  AC156 HCT 116 C109(0.91); C118(0.75); C158(0.92); C194(1.53)  LDD2160  [22]
 LDCM0624  AC157 HCT 116 C109(0.87); C118(0.65); C158(0.89); C194(2.50)  LDD2161  [22]
 LDCM0276  AC17 HCT 116 C118(0.74); C109(0.88); C158(0.96); C194(1.25)  LDD0593  [22]
 LDCM0277  AC18 HCT 116 C118(0.68); C194(0.80); C158(0.85); C293(0.92)  LDD0594  [22]
 LDCM0278  AC19 HCT 116 C158(0.90); C293(0.97); C109(1.05); C118(1.12)  LDD0595  [22]
 LDCM0279  AC2 HCT 116 C194(0.51); C158(0.80); C163(0.91); C118(0.97)  LDD0596  [22]
 LDCM0280  AC20 HCT 116 C158(0.93); C118(1.02); C109(1.04); C194(1.21)  LDD0597  [22]
 LDCM0281  AC21 HCT 116 C118(0.78); C109(0.94); C158(0.95); C293(1.18)  LDD0598  [22]
 LDCM0282  AC22 HCT 116 C293(0.91); C118(0.98); C158(1.00); C194(1.07)  LDD0599  [22]
 LDCM0283  AC23 HCT 116 C158(0.89); C118(1.03); C109(1.09); C194(1.11)  LDD0600  [22]
 LDCM0284  AC24 HCT 116 C158(0.95); C109(1.06); C118(1.11); C293(1.28)  LDD0601  [22]
 LDCM0285  AC25 HCT 116 C158(0.91); C293(1.03); C109(1.10); C194(1.31)  LDD0602  [22]
 LDCM0286  AC26 HCT 116 C158(0.84); C293(0.94); C109(1.03); C194(1.14)  LDD0603  [22]
 LDCM0287  AC27 HCT 116 C158(0.77); C293(1.10); C109(1.19); C194(1.36)  LDD0604  [22]
 LDCM0288  AC28 HCT 116 C158(0.87); C293(1.23); C194(1.35); C109(1.36)  LDD0605  [22]
 LDCM0289  AC29 HCT 116 C158(0.87); C293(0.97); C194(1.19); C109(1.22)  LDD0606  [22]
 LDCM0290  AC3 HCT 116 C194(0.42); C158(0.85); C163(0.87); C109(1.09)  LDD0607  [22]
 LDCM0291  AC30 HCT 116 C158(0.84); C109(1.15); C194(1.21); C118(1.40)  LDD0608  [22]
 LDCM0292  AC31 HCT 116 C158(0.81); C194(0.90); C293(1.07); C109(1.27)  LDD0609  [22]
 LDCM0293  AC32 HCT 116 C158(0.82); C194(1.03); C293(1.13); C109(1.45)  LDD0610  [22]
 LDCM0294  AC33 HCT 116 C158(0.81); C293(0.99); C109(1.31); C194(1.42)  LDD0611  [22]
 LDCM0295  AC34 HCT 116 C158(0.88); C293(1.25); C109(1.60); C194(1.67)  LDD0612  [22]
 LDCM0296  AC35 HCT 116 C293(0.94); C109(0.96); C158(0.96); C194(1.06)  LDD0613  [22]
 LDCM0297  AC36 HCT 116 C293(0.82); C194(0.87); C158(0.98); C109(1.01)  LDD0614  [22]
 LDCM0298  AC37 HCT 116 C293(0.71); C194(0.85); C158(0.94); C109(0.99)  LDD0615  [22]
 LDCM0299  AC38 HCT 116 C194(0.89); C109(0.98); C158(1.01); C293(1.01)  LDD0616  [22]
 LDCM0300  AC39 HCT 116 C194(0.74); C293(1.01); C109(1.06); C158(1.08)  LDD0617  [22]
 LDCM0301  AC4 HCT 116 C194(0.41); C158(0.75); C163(0.97); C109(1.07)  LDD0618  [22]
 LDCM0302  AC40 HCT 116 C194(0.98); C293(0.99); C158(1.01); C109(1.10)  LDD0619  [22]
 LDCM0303  AC41 HCT 116 C194(0.79); C293(0.89); C158(1.01); C109(1.11)  LDD0620  [22]
 LDCM0304  AC42 HCT 116 C194(0.82); C293(0.91); C158(1.01); C109(1.08)  LDD0621  [22]
 LDCM0305  AC43 HCT 116 C194(0.76); C293(0.79); C158(0.98); C109(1.04)  LDD0622  [22]
 LDCM0306  AC44 HCT 116 C194(0.70); C293(0.89); C158(1.06); C109(1.06)  LDD0623  [22]
 LDCM0307  AC45 HCT 116 C194(0.79); C293(0.87); C158(1.08); C109(1.20)  LDD0624  [22]
 LDCM0308  AC46 HCT 116 C293(0.94); C194(0.98); C158(1.00); C109(1.04)  LDD0625  [22]
 LDCM0309  AC47 HCT 116 C158(0.95); C293(1.00); C194(1.06); C109(1.12)  LDD0626  [22]
 LDCM0310  AC48 HCT 116 C194(0.83); C158(0.95); C293(1.01); C109(1.18)  LDD0627  [22]
 LDCM0311  AC49 HCT 116 C293(0.85); C158(0.99); C194(1.00); C109(1.64)  LDD0628  [22]
 LDCM0312  AC5 HCT 116 C194(0.31); C158(0.76); C163(0.89); C109(1.26)  LDD0629  [22]
 LDCM0313  AC50 HCT 116 C293(0.97); C158(0.98); C194(1.25); C109(1.30)  LDD0630  [22]
 LDCM0314  AC51 HCT 116 C293(0.78); C158(0.91); C194(1.06); C109(1.32)  LDD0631  [22]
 LDCM0315  AC52 HCT 116 C293(0.76); C158(0.95); C194(1.13); C109(1.45)  LDD0632  [22]
 LDCM0316  AC53 HCT 116 C293(0.85); C158(0.90); C194(1.01); C109(1.39)  LDD0633  [22]
 LDCM0317  AC54 HCT 116 C293(0.82); C194(1.02); C158(1.07); C109(1.35)  LDD0634  [22]
 LDCM0318  AC55 HCT 116 C293(0.91); C158(0.97); C194(1.07); C109(1.34)  LDD0635  [22]
 LDCM0319  AC56 HCT 116 C293(1.00); C158(1.04); C194(1.20); C109(1.72)  LDD0636  [22]
 LDCM0320  AC57 HCT 116 C194(0.53); C118(0.80); C158(0.82); C293(0.84)  LDD0637  [22]
 LDCM0321  AC58 HCT 116 C194(0.68); C118(0.71); C158(0.79); C109(0.99)  LDD0638  [22]
 LDCM0322  AC59 HCT 116 C194(0.55); C158(0.84); C118(0.89); C109(1.08)  LDD0639  [22]
 LDCM0323  AC6 HCT 116 C194(0.78); C158(0.94); C109(1.22); C118(1.24)  LDD0640  [22]
 LDCM0324  AC60 HCT 116 C194(0.54); C158(0.77); C118(0.92); C109(1.03)  LDD0641  [22]
 LDCM0325  AC61 HCT 116 C194(0.47); C118(0.71); C158(0.85); C109(0.95)  LDD0642  [22]
 LDCM0326  AC62 HCT 116 C118(0.45); C194(0.55); C158(0.81); C293(0.96)  LDD0643  [22]
 LDCM0327  AC63 HCT 116 C194(0.68); C293(0.80); C118(0.83); C158(0.83)  LDD0644  [22]
 LDCM0328  AC64 HCT 116 C194(0.58); C158(0.83); C118(0.92); C109(1.12)  LDD0645  [22]
 LDCM0329  AC65 HCT 116 C194(0.47); C158(0.87); C118(1.05); C293(1.13)  LDD0646  [22]
 LDCM0330  AC66 HCT 116 C194(0.52); C158(0.85); C293(1.15); C109(1.27)  LDD0647  [22]
 LDCM0331  AC67 HCT 116 C194(0.51); C158(0.80); C118(1.03); C293(1.17)  LDD0648  [22]
 LDCM0332  AC68 HCT 116 C118(0.90); C194(0.97); C109(0.99); C158(1.03)  LDD0649  [22]
 LDCM0333  AC69 HCT 116 C118(0.89); C109(0.98); C163(1.04); C158(1.11)  LDD0650  [22]
 LDCM0334  AC7 HCT 116 C194(0.68); C158(0.88); C109(1.60); C118(1.98)  LDD0651  [22]
 LDCM0335  AC70 HCT 116 C118(0.92); C194(0.99); C158(1.00); C109(1.02)  LDD0652  [22]
 LDCM0336  AC71 HCT 116 C118(0.86); C194(0.91); C109(0.93); C163(1.01)  LDD0653  [22]
 LDCM0337  AC72 HCT 116 C118(0.87); C109(0.97); C158(1.07); C163(1.29)  LDD0654  [22]
 LDCM0338  AC73 HCT 116 C163(1.02); C118(1.04); C158(1.11); C109(1.16)  LDD0655  [22]
 LDCM0339  AC74 HCT 116 C163(0.84); C118(0.98); C109(1.10); C194(1.10)  LDD0656  [22]
 LDCM0340  AC75 HCT 116 C118(1.13); C158(1.21); C109(1.22); C163(1.26)  LDD0657  [22]
 LDCM0341  AC76 HCT 116 C118(0.80); C109(0.94); C158(1.03); C194(1.10)  LDD0658  [22]
 LDCM0342  AC77 HCT 116 C118(0.84); C109(1.01); C158(1.10); C163(1.25)  LDD0659  [22]
 LDCM0343  AC78 HCT 116 C118(0.82); C163(0.90); C109(0.96); C158(1.04)  LDD0660  [22]
 LDCM0344  AC79 HCT 116 C118(0.85); C109(0.98); C158(1.01); C194(1.09)  LDD0661  [22]
 LDCM0345  AC8 HCT 116 C194(0.76); C158(0.94); C109(1.76); C118(2.35)  LDD0662  [22]
 LDCM0346  AC80 HCT 116 C118(0.69); C109(0.90); C163(1.05); C158(1.11)  LDD0663  [22]
 LDCM0347  AC81 HCT 116 C118(0.39); C109(0.71); C194(1.00); C158(1.14)  LDD0664  [22]
 LDCM0348  AC82 HCT 116 C118(1.01); C163(1.01); C194(1.07); C158(1.15)  LDD0665  [22]
 LDCM0349  AC83 HCT 116 C158(1.01); C194(1.16); C109(1.32); C118(1.67)  LDD0666  [22]
 LDCM0350  AC84 HCT 116 C158(1.09); C194(1.18); C109(1.66); C118(2.27)  LDD0667  [22]
 LDCM0351  AC85 HCT 116 C158(0.94); C194(1.00); C109(1.62); C118(2.37)  LDD0668  [22]
 LDCM0352  AC86 HCT 116 C158(0.96); C194(1.12); C109(1.13); C118(1.60)  LDD0669  [22]
 LDCM0353  AC87 HCT 116 C158(1.00); C109(1.24); C194(1.28); C118(1.94)  LDD0670  [22]
 LDCM0354  AC88 HCT 116 C158(1.02); C109(1.24); C194(1.39); C118(1.79)  LDD0671  [22]
 LDCM0355  AC89 HCT 116 C158(0.94); C109(1.25); C194(1.56); C118(1.61)  LDD0672  [22]
 LDCM0357  AC90 HCT 116 C158(1.03); C194(1.05); C109(1.21); C118(1.76)  LDD0674  [22]
 LDCM0358  AC91 HCT 116 C158(1.03); C109(1.58); C194(1.77); C118(2.35)  LDD0675  [22]
 LDCM0359  AC92 HCT 116 C158(0.99); C109(1.54); C194(1.74); C118(2.03)  LDD0676  [22]
 LDCM0360  AC93 HCT 116 C158(1.00); C109(1.50); C194(1.58); C118(2.29)  LDD0677  [22]
 LDCM0361  AC94 HCT 116 C158(0.95); C109(1.46); C194(1.53); C118(2.16)  LDD0678  [22]
 LDCM0362  AC95 HCT 116 C158(0.86); C109(1.20); C194(1.53); C118(2.02)  LDD0679  [22]
 LDCM0363  AC96 HCT 116 C158(0.93); C109(1.32); C194(1.60); C118(1.99)  LDD0680  [22]
 LDCM0364  AC97 HCT 116 C158(0.92); C109(1.33); C194(1.57); C118(1.66)  LDD0681  [22]
 LDCM0365  AC98 HCT 116 C194(0.70); C158(0.75); C118(0.88); C109(0.93)  LDD0682  [22]
 LDCM0366  AC99 HCT 116 C194(0.83); C158(0.84); C118(0.86); C109(0.88)  LDD0683  [22]
 LDCM0545  Acetamide MDA-MB-231 C109(0.49)  LDD2138  [12]
 LDCM0520  AKOS000195272 MDA-MB-231 C158(0.84); C109(0.66)  LDD2113  [12]
 LDCM0248  AKOS034007472 HCT 116 C109(1.87); C118(2.53); C158(1.02); C194(0.70)  LDD0565  [22]
 LDCM0356  AKOS034007680 HCT 116 C194(0.68); C158(0.92); C109(1.57); C118(2.00)  LDD0673  [22]
 LDCM0275  AKOS034007705 HCT 116 C194(0.86); C158(1.01); C109(2.13); C118(2.81)  LDD0592  [22]
 LDCM0156  Aniline NCI-H1299 12.05  LDD0403  [1]
 LDCM0020  ARS-1620 HCC44 C194(1.06)  LDD0078  [22]
 LDCM0498  BS-3668 MDA-MB-231 C158(0.97)  LDD2091  [12]
 LDCM0630  CCW28-3 231MFP C109(1.64); C194(1.41); C293(1.24)  LDD2214  [45]
 LDCM0108  Chloroacetamide HeLa C158(0.00); C163(0.00); C194(0.00); C109(0.00)  LDD0222  [38]
 LDCM0632  CL-Sc Hep-G2 C163(20.00); C109(0.98); C201(0.86); C54(0.83)  LDD2227  [30]
 LDCM0367  CL1 HCT 116 C163(0.96); C158(1.02); C109(1.04); C194(1.18)  LDD0684  [22]
 LDCM0368  CL10 HCT 116 C158(0.86); C194(0.98); C163(1.14); C109(1.15)  LDD0685  [22]
 LDCM0369  CL100 HCT 116 C194(0.52); C158(0.75); C163(0.91); C109(1.37)  LDD0686  [22]
 LDCM0370  CL101 HCT 116 C158(0.88); C109(1.57); C194(1.66); C118(2.09)  LDD0687  [22]
 LDCM0371  CL102 HCT 116 C158(0.95); C109(1.61); C118(2.03); C194(2.10)  LDD0688  [22]
 LDCM0372  CL103 HCT 116 C158(0.86); C194(1.48); C109(1.79); C118(2.42)  LDD0689  [22]
 LDCM0373  CL104 HCT 116 C158(0.91); C194(1.46); C109(1.49); C118(1.90)  LDD0690  [22]
 LDCM0374  CL105 HCT 116 C194(0.66); C158(0.91); C293(1.06); C109(1.23)  LDD0691  [22]
 LDCM0375  CL106 HCT 116 C194(0.84); C158(0.92); C109(1.31); C293(1.33)  LDD0692  [22]
 LDCM0376  CL107 HCT 116 C194(0.67); C158(0.91); C293(1.16); C109(1.25)  LDD0693  [22]
 LDCM0377  CL108 HCT 116 C194(0.75); C158(0.97); C109(1.18); C293(1.25)  LDD0694  [22]
 LDCM0378  CL109 HCT 116 C158(0.85); C194(0.99); C109(1.22); C293(1.24)  LDD0695  [22]
 LDCM0379  CL11 HCT 116 C158(1.07); C194(1.08); C163(1.27); C109(1.52)  LDD0696  [22]
 LDCM0380  CL110 HCT 116 C158(0.79); C194(0.87); C293(1.07); C109(1.25)  LDD0697  [22]
 LDCM0381  CL111 HCT 116 C158(0.84); C194(0.91); C293(1.04); C109(1.28)  LDD0698  [22]
 LDCM0382  CL112 HCT 116 C158(0.94); C293(0.98); C109(1.21); C194(1.61)  LDD0699  [22]
 LDCM0383  CL113 HCT 116 C158(0.79); C293(1.15); C194(1.27); C109(1.69)  LDD0700  [22]
 LDCM0384  CL114 HCT 116 C293(0.83); C158(0.83); C194(1.19); C109(1.51)  LDD0701  [22]
 LDCM0385  CL115 HCT 116 C158(0.80); C293(1.08); C194(1.29); C109(1.40)  LDD0702  [22]
 LDCM0386  CL116 HCT 116 C158(0.87); C293(0.97); C194(1.03); C109(1.23)  LDD0703  [22]
 LDCM0387  CL117 HCT 116 C293(1.03); C158(1.19); C194(1.26); C109(1.37)  LDD0704  [22]
 LDCM0388  CL118 HCT 116 C194(0.71); C158(0.97); C109(1.01); C293(1.06)  LDD0705  [22]
 LDCM0389  CL119 HCT 116 C118(0.81); C194(0.82); C293(0.94); C158(0.98)  LDD0706  [22]
 LDCM0390  CL12 HCT 116 C158(1.04); C109(1.20); C118(1.28); C194(1.34)  LDD0707  [22]
 LDCM0391  CL120 HCT 116 C293(0.71); C194(0.77); C158(0.99); C109(1.09)  LDD0708  [22]
 LDCM0392  CL121 HCT 116 C158(0.99); C293(1.15); C194(1.46); C109(1.56)  LDD0709  [22]
 LDCM0393  CL122 HCT 116 C293(0.64); C194(0.86); C158(0.95); C109(1.14)  LDD0710  [22]
 LDCM0394  CL123 HCT 116 C158(0.81); C293(0.97); C194(1.24); C109(1.45)  LDD0711  [22]
 LDCM0395  CL124 HCT 116 C293(0.95); C158(0.98); C194(1.19); C109(1.52)  LDD0712  [22]
 LDCM0396  CL125 HCT 116 C194(0.54); C118(0.77); C293(0.83); C158(0.90)  LDD0713  [22]
 LDCM0397  CL126 HCT 116 C194(0.55); C118(0.67); C158(0.82); C109(0.89)  LDD0714  [22]
 LDCM0398  CL127 HCT 116 C194(0.59); C293(0.82); C158(0.83); C118(0.83)  LDD0715  [22]
 LDCM0399  CL128 HCT 116 C194(0.59); C158(0.84); C118(0.99); C109(1.06)  LDD0716  [22]
 LDCM0400  CL13 HCT 116 C158(0.92); C109(1.09); C194(1.17); C163(1.18)  LDD0717  [22]
 LDCM0401  CL14 HCT 116 C118(0.72); C158(0.81); C109(0.91); C163(1.03)  LDD0718  [22]
 LDCM0402  CL15 HCT 116 C158(0.90); C163(0.95); C194(1.03); C109(1.09)  LDD0719  [22]
 LDCM0403  CL16 HCT 116 C158(0.98); C194(1.04); C163(1.07); C293(1.16)  LDD0720  [22]
 LDCM0404  CL17 HCT 116 C158(0.81); C194(0.92); C163(1.01); C293(1.04)  LDD0721  [22]
 LDCM0405  CL18 HCT 116 C158(0.82); C163(0.99); C194(1.08); C293(1.12)  LDD0722  [22]
 LDCM0406  CL19 HCT 116 C158(0.85); C194(0.93); C163(1.04); C109(1.09)  LDD0723  [22]
 LDCM0407  CL2 HCT 116 C158(1.04); C109(1.05); C163(1.06); C194(1.09)  LDD0724  [22]
 LDCM0408  CL20 HCT 116 C158(0.73); C109(1.04); C194(1.07); C293(1.08)  LDD0725  [22]
 LDCM0409  CL21 HCT 116 C158(0.72); C194(0.92); C293(1.04); C163(1.06)  LDD0726  [22]
 LDCM0410  CL22 HCT 116 C158(0.85); C194(1.05); C293(1.26); C163(1.27)  LDD0727  [22]
 LDCM0411  CL23 HCT 116 C158(0.83); C118(0.87); C109(0.95); C163(1.01)  LDD0728  [22]
 LDCM0412  CL24 HCT 116 C158(0.86); C194(1.03); C293(1.13); C163(1.20)  LDD0729  [22]
 LDCM0413  CL25 HCT 116 C109(1.90); C118(2.15); C158(0.69); C163(0.97)  LDD0730  [22]
 LDCM0414  CL26 HCT 116 C109(1.51); C118(1.69); C158(0.80); C163(1.07)  LDD0731  [22]
 LDCM0415  CL27 HCT 116 C109(1.44); C118(1.64); C158(0.81); C163(1.08)  LDD0732  [22]
 LDCM0416  CL28 HCT 116 C109(1.48); C118(1.97); C158(0.89); C163(1.01)  LDD0733  [22]
 LDCM0417  CL29 HCT 116 C109(1.14); C118(1.20); C158(0.76); C163(1.04)  LDD0734  [22]
 LDCM0418  CL3 HCT 116 C109(1.05); C118(1.27); C158(0.90); C163(1.13)  LDD0735  [22]
 LDCM0419  CL30 HCT 116 C109(0.96); C118(0.98); C158(0.75); C163(1.02)  LDD0736  [22]
 LDCM0420  CL31 HCT 116 C109(0.96); C118(1.10); C158(0.77); C194(0.95)  LDD0737  [22]
 LDCM0421  CL32 HCT 116 C109(0.99); C118(0.83); C158(0.75); C194(0.80)  LDD0738  [22]
 LDCM0422  CL33 HCT 116 C109(1.04); C118(1.15); C158(0.57); C194(1.10)  LDD0739  [22]
 LDCM0423  CL34 HCT 116 C109(1.02); C118(1.30); C158(0.78); C194(0.95)  LDD0740  [22]
 LDCM0424  CL35 HCT 116 C109(1.11); C118(1.25); C158(0.80); C194(1.58)  LDD0741  [22]
 LDCM0425  CL36 HCT 116 C109(1.02); C118(1.25); C158(0.69); C194(1.12)  LDD0742  [22]
 LDCM0426  CL37 HCT 116 C109(1.41); C118(2.06); C158(0.82); C194(1.40)  LDD0743  [22]
 LDCM0428  CL39 HCT 116 C109(1.01); C118(0.55); C158(0.87); C194(1.08)  LDD0745  [22]
 LDCM0429  CL4 HCT 116 C109(0.90); C118(1.08); C158(0.93); C163(1.07)  LDD0746  [22]
 LDCM0430  CL40 HCT 116 C109(1.14); C118(1.16); C158(0.69); C194(1.35)  LDD0747  [22]
 LDCM0431  CL41 HCT 116 C109(1.12); C118(1.75); C158(0.71); C194(1.21)  LDD0748  [22]
 LDCM0432  CL42 HCT 116 C109(1.87); C118(2.25); C158(0.81); C194(1.13)  LDD0749  [22]
 LDCM0433  CL43 HCT 116 C109(1.12); C118(1.19); C158(0.87); C194(1.68)  LDD0750  [22]
 LDCM0434  CL44 HCT 116 C109(1.05); C118(1.12); C158(0.81); C194(1.45)  LDD0751  [22]
 LDCM0435  CL45 HCT 116 C109(1.16); C118(1.37); C158(0.70); C194(1.01)  LDD0752  [22]
 LDCM0436  CL46 HCT 116 C109(1.55); C118(1.98); C158(1.05); C163(1.30)  LDD0753  [22]
 LDCM0437  CL47 HCT 116 C109(1.54); C118(1.88); C158(1.08); C163(1.05)  LDD0754  [22]
 LDCM0438  CL48 HCT 116 C109(0.89); C118(1.05); C158(1.07); C163(1.06)  LDD0755  [22]
 LDCM0439  CL49 HCT 116 C109(1.45); C118(1.75); C158(0.96); C163(0.88)  LDD0756  [22]
 LDCM0440  CL5 HCT 116 C109(0.91); C118(0.90); C158(1.01); C163(1.06)  LDD0757  [22]
 LDCM0441  CL50 HCT 116 C109(1.69); C118(2.13); C158(1.01); C163(1.27)  LDD0758  [22]
 LDCM0442  CL51 HCT 116 C109(1.31); C118(1.61); C158(1.07); C163(1.06)  LDD0759  [22]
 LDCM0443  CL52 HCT 116 C109(1.91); C118(2.34); C158(0.99); C163(0.90)  LDD0760  [22]
 LDCM0444  CL53 HCT 116 C109(2.11); C118(2.55); C158(0.96); C163(0.97)  LDD0761  [22]
 LDCM0445  CL54 HCT 116 C109(2.29); C118(3.10); C158(0.93); C163(0.97)  LDD0762  [22]
 LDCM0446  CL55 HCT 116 C109(2.17); C118(2.77); C158(1.08); C163(0.82)  LDD0763  [22]
 LDCM0447  CL56 HCT 116 C109(1.96); C118(2.40); C158(1.12); C163(0.81)  LDD0764  [22]
 LDCM0448  CL57 HCT 116 C109(1.56); C118(2.03); C158(1.04); C163(1.04)  LDD0765  [22]
 LDCM0449  CL58 HCT 116 C109(1.72); C118(2.20); C158(1.10); C163(1.37)  LDD0766  [22]
 LDCM0450  CL59 HCT 116 C109(1.74); C118(2.13); C158(1.07); C163(1.10)  LDD0767  [22]
 LDCM0451  CL6 HCT 116 C109(1.22); C118(1.63); C158(0.90); C163(1.14)  LDD0768  [22]
 LDCM0452  CL60 HCT 116 C109(1.60); C118(1.91); C158(1.02); C163(0.87)  LDD0769  [22]
 LDCM0453  CL61 HCT 116 C109(0.89); C118(0.77); C158(0.92); C163(1.05)  LDD0770  [22]
 LDCM0454  CL62 HCT 116 C109(0.99); C118(0.92); C158(0.93); C163(0.78)  LDD0771  [22]
 LDCM0455  CL63 HCT 116 C109(0.98); C118(0.93); C158(0.88); C163(1.04)  LDD0772  [22]
 LDCM0456  CL64 HCT 116 C109(1.15); C118(1.26); C158(0.88); C163(0.79)  LDD0773  [22]
 LDCM0457  CL65 HCT 116 C109(0.94); C118(0.84); C158(0.97); C163(0.96)  LDD0774  [22]
 LDCM0458  CL66 HCT 116 C109(0.95); C118(0.77); C158(0.91); C163(1.30)  LDD0775  [22]
 LDCM0459  CL67 HCT 116 C109(0.93); C118(0.73); C158(1.08); C163(1.29)  LDD0776  [22]
 LDCM0460  CL68 HCT 116 C109(0.95); C118(0.92); C158(0.87); C163(1.01)  LDD0777  [22]
 LDCM0461  CL69 HCT 116 C109(1.05); C118(1.20); C158(0.83); C163(0.77)  LDD0778  [22]
 LDCM0462  CL7 HCT 116 C109(1.11); C118(1.28); C158(1.04); C163(1.47)  LDD0779  [22]
 LDCM0463  CL70 HCT 116 C109(1.09); C118(1.10); C158(0.85); C163(1.26)  LDD0780  [22]
 LDCM0464  CL71 HCT 116 C109(0.95); C118(0.75); C158(0.92); C163(0.86)  LDD0781  [22]
 LDCM0465  CL72 HCT 116 C109(1.01); C118(0.91); C158(0.98); C163(0.83)  LDD0782  [22]
 LDCM0466  CL73 HCT 116 C109(1.01); C118(1.04); C158(0.82); C163(1.04)  LDD0783  [22]
 LDCM0467  CL74 HCT 116 C109(0.98); C118(0.89); C158(0.88); C163(0.84)  LDD0784  [22]
 LDCM0469  CL76 HCT 116 C109(1.06); C118(1.28); C158(0.80); C163(1.25)  LDD0786  [22]
 LDCM0470  CL77 HCT 116 C109(1.05); C118(1.20); C158(0.65); C163(0.86)  LDD0787  [22]
 LDCM0471  CL78 HCT 116 C109(1.09); C118(1.02); C158(0.80); C163(0.94)  LDD0788  [22]
 LDCM0472  CL79 HCT 116 C109(1.08); C118(0.91); C158(0.84); C163(1.21)  LDD0789  [22]
 LDCM0473  CL8 HCT 116 C109(1.69); C118(2.58); C158(0.94); C163(1.11)  LDD0790  [22]
 LDCM0474  CL80 HCT 116 C109(0.84); C118(0.43); C158(0.94); C163(1.04)  LDD0791  [22]
 LDCM0475  CL81 HCT 116 C109(1.21); C118(1.61); C158(0.81); C163(1.21)  LDD0792  [22]
 LDCM0476  CL82 HCT 116 C109(1.28); C118(1.55); C158(0.96); C163(1.36)  LDD0793  [22]
 LDCM0477  CL83 HCT 116 C109(1.31); C118(1.63); C158(0.74); C163(1.24)  LDD0794  [22]
 LDCM0478  CL84 HCT 116 C109(1.20); C118(0.96); C158(0.82); C163(1.20)  LDD0795  [22]
 LDCM0479  CL85 HCT 116 C109(1.12); C118(0.84); C158(0.70); C163(0.96)  LDD0796  [22]
 LDCM0480  CL86 HCT 116 C109(1.13); C118(1.01); C158(0.84); C163(1.38)  LDD0797  [22]
 LDCM0481  CL87 HCT 116 C109(1.11); C118(1.08); C158(0.78); C163(1.14)  LDD0798  [22]
 LDCM0482  CL88 HCT 116 C109(1.17); C118(0.99); C158(0.80); C163(1.28)  LDD0799  [22]
 LDCM0483  CL89 HCT 116 C109(1.45); C118(1.26); C158(0.86); C163(1.14)  LDD0800  [22]
 LDCM0484  CL9 HCT 116 C109(0.90); C118(0.59); C158(0.91); C163(1.22)  LDD0801  [22]
 LDCM0485  CL90 HCT 116 C109(1.03); C118(1.30); C158(0.62); C163(0.76)  LDD0802  [22]
 LDCM0486  CL91 HCT 116 C109(1.04); C118(1.03); C158(0.80); C163(0.72)  LDD0803  [22]
 LDCM0487  CL92 HCT 116 C109(1.10); C118(1.25); C158(0.78); C163(0.99)  LDD0804  [22]
 LDCM0488  CL93 HCT 116 C109(1.06); C118(1.23); C158(0.76); C163(0.93)  LDD0805  [22]
 LDCM0489  CL94 HCT 116 C109(1.58); C118(2.14); C158(0.66); C163(0.87)  LDD0806  [22]
 LDCM0490  CL95 HCT 116 C109(1.67); C118(2.23); C158(0.69); C163(0.80)  LDD0807  [22]
 LDCM0491  CL96 HCT 116 C109(1.00); C118(1.05); C158(0.73); C163(0.80)  LDD0808  [22]
 LDCM0492  CL97 HCT 116 C109(0.98); C118(1.06); C158(0.77); C163(0.83)  LDD0809  [22]
 LDCM0493  CL98 HCT 116 C109(1.20); C118(1.28); C158(0.78); C163(0.93)  LDD0810  [22]
 LDCM0494  CL99 HCT 116 C109(1.11); C118(1.05); C158(0.80); C163(0.84)  LDD0811  [22]
 LDCM0634  CY-0357 Hep-G2 C293(1.65); C54(1.03); C194(0.61); C109(0.53)  LDD2228  [30]
 LDCM0495  E2913 HEK-293T C194(0.99); C201(0.95); C109(0.90); C158(0.94)  LDD1698  [46]
 LDCM0213  Electrophilic fragment 2 MDA-MB-231 C109(2.19); C201(1.18); C194(1.14); C158(0.42)  LDD1702  [12]
 LDCM0175  Ethacrynic acid HeLa N.A.  LDD0440  [18]
 LDCM0625  F8 Ramos C109(1.07); C158(0.85); 1.06; C194(1.31)  LDD2187  [47]
 LDCM0572  Fragment10 MDA-MB-231 C109(0.88); C194(3.87)  LDD1389  [48]
 LDCM0573  Fragment11 MDA-MB-231 C109(1.02); C194(2.25)  LDD1391  [48]
 LDCM0574  Fragment12 MDA-MB-231 C109(1.14); C194(1.28)  LDD1393  [48]
 LDCM0575  Fragment13 MDA-MB-231 C109(0.87); C194(1.61)  LDD1395  [48]
 LDCM0576  Fragment14 MDA-MB-231 C109(1.12); C194(2.21)  LDD1397  [48]
 LDCM0577  Fragment15 MDA-MB-231 C109(1.06); C194(0.96)  LDD1399  [48]
 LDCM0579  Fragment20 MDA-MB-231 C109(1.10); C194(2.34)  LDD1402  [48]
 LDCM0580  Fragment21 MDA-MB-231 C109(0.59); C194(1.28)  LDD1404  [48]
 LDCM0581  Fragment22 MDA-MB-231 C109(1.00); C194(2.41)  LDD1406  [48]
 LDCM0582  Fragment23 MDA-MB-231 C109(1.84); C194(4.99)  LDD1408  [48]
 LDCM0583  Fragment24 Ramos C109(0.95); C194(1.40)  LDD1410  [48]
 LDCM0584  Fragment25 MDA-MB-231 C109(0.77); C194(0.70)  LDD1411  [48]
 LDCM0585  Fragment26 Ramos C109(0.86); C194(1.04)  LDD1412  [48]
 LDCM0578  Fragment27 MDA-MB-231 C109(0.90); C194(0.95)  LDD1401  [48]
 LDCM0586  Fragment28 MDA-MB-231 C109(0.84); C194(0.95)  LDD1415  [48]
 LDCM0587  Fragment29 MDA-MB-231 C109(1.17); C194(1.56)  LDD1417  [48]
 LDCM0588  Fragment30 MDA-MB-231 C109(0.60); C194(1.74)  LDD1419  [48]
 LDCM0589  Fragment31 MDA-MB-231 C109(1.66); C194(1.42)  LDD1421  [48]
 LDCM0590  Fragment32 MDA-MB-231 C109(0.90); C194(2.34)  LDD1423  [48]
 LDCM0468  Fragment33 HCT 116 C109(0.86); C118(0.71); C158(0.92); C163(1.12)  LDD0785  [22]
 LDCM0592  Fragment34 MDA-MB-231 C109(0.60); C194(1.21)  LDD1427  [48]
 LDCM0593  Fragment35 MDA-MB-231 C109(0.90)  LDD1429  [48]
 LDCM0594  Fragment36 MDA-MB-231 C109(1.22); C194(2.05)  LDD1431  [48]
 LDCM0595  Fragment37 Ramos C109(0.73); C194(1.03)  LDD1432  [48]
 LDCM0596  Fragment38 MDA-MB-231 C109(0.87); C194(1.02)  LDD1433  [48]
 LDCM0597  Fragment39 MDA-MB-231 C109(0.78); C194(1.24)  LDD1435  [48]
 LDCM0566  Fragment4 MDA-MB-231 C109(0.68); C194(2.42)  LDD1378  [48]
 LDCM0598  Fragment40 MDA-MB-231 C109(0.71)  LDD1436  [48]
 LDCM0599  Fragment41 MDA-MB-231 C109(0.70); C194(1.19)  LDD1438  [48]
 LDCM0600  Fragment42 Ramos C109(0.76); C194(1.18)  LDD1440  [48]
 LDCM0601  Fragment43 MDA-MB-231 C109(0.73); C194(1.53)  LDD1441  [48]
 LDCM0602  Fragment44 MDA-MB-231 C109(0.80); C194(0.93)  LDD1443  [48]
 LDCM0603  Fragment45 MDA-MB-231 C109(2.98); C194(4.71)  LDD1444  [48]
 LDCM0604  Fragment46 MDA-MB-231 C109(0.85); C194(1.40)  LDD1445  [48]
 LDCM0605  Fragment47 MDA-MB-231 C109(1.06); C194(1.91)  LDD1446  [48]
 LDCM0606  Fragment48 MDA-MB-231 C109(1.08); C194(1.11)  LDD1447  [48]
 LDCM0607  Fragment49 MDA-MB-231 C109(3.58); C194(2.67)  LDD1448  [48]
 LDCM0608  Fragment50 MDA-MB-231 C109(1.06); C194(3.29)  LDD1449  [48]
 LDCM0427  Fragment51 HCT 116 C109(1.43); C118(1.76); C158(0.77); C194(1.28)  LDD0744  [22]
 LDCM0610  Fragment52 MDA-MB-231 C109(0.92); C194(1.56)  LDD1452  [48]
 LDCM0611  Fragment53 MDA-MB-231 C109(0.80); C194(1.13)  LDD1454  [48]
 LDCM0612  Fragment54 MDA-MB-231 C109(1.04); C194(1.27)  LDD1456  [48]
 LDCM0613  Fragment55 MDA-MB-231 C109(0.71); C194(1.10)  LDD1457  [48]
 LDCM0614  Fragment56 MDA-MB-231 C109(0.93); C194(1.25)  LDD1458  [48]
 LDCM0568  Fragment6 MDA-MB-231 C109(1.34)  LDD1382  [48]
 LDCM0569  Fragment7 MDA-MB-231 C109(0.74); C194(1.91)  LDD1383  [48]
 LDCM0570  Fragment8 MDA-MB-231 C109(0.86); C194(3.33)  LDD1385  [48]
 LDCM0571  Fragment9 MDA-MB-231 C109(0.88); C194(2.73)  LDD1387  [48]
 LDCM0116  HHS-0101 DM93 Y222(0.71); Y183(0.81); Y341(0.85); Y270(0.93)  LDD0264  [20]
 LDCM0117  HHS-0201 DM93 Y183(0.72); Y270(0.76); Y341(0.79); Y222(1.51)  LDD0265  [20]
 LDCM0118  HHS-0301 DM93 Y222(0.07); Y270(0.72); Y341(0.79); Y183(0.81)  LDD0266  [20]
 LDCM0119  HHS-0401 DM93 Y207(0.35); Y270(0.72); Y341(0.85); Y183(0.86)  LDD0267  [20]
 LDCM0120  HHS-0701 DM93 Y270(0.84); Y341(0.88); Y183(0.98); Y222(1.30)  LDD0268  [20]
 LDCM0107  IAA HeLa C163(0.00); C158(0.00); C109(0.00)  LDD0221  [38]
 LDCM0123  JWB131 DM93 Y183(1.07); Y270(1.24); Y341(1.03)  LDD0285  [19]
 LDCM0124  JWB142 DM93 Y183(0.81); Y270(0.79); Y341(0.81)  LDD0286  [19]
 LDCM0125  JWB146 DM93 Y183(1.05); Y270(1.45); Y341(1.07)  LDD0287  [19]
 LDCM0126  JWB150 DM93 Y183(3.76); Y270(2.48); Y341(2.84)  LDD0288  [19]
 LDCM0127  JWB152 DM93 Y183(2.60); Y270(2.06); Y341(2.04)  LDD0289  [19]
 LDCM0128  JWB198 DM93 Y183(0.65); Y270(1.91); Y341(1.58)  LDD0290  [19]
 LDCM0129  JWB202 DM93 Y183(0.83); Y270(0.37); Y341(0.64)  LDD0291  [19]
 LDCM0130  JWB211 DM93 Y183(0.90); Y270(1.04); Y341(1.06)  LDD0292  [19]
 LDCM0179  JZ128 PC-3 C109(0.00); C54(0.00)  LDD0462  [15]
 LDCM0022  KB02 HCT 116 C194(3.02); C163(1.84); C158(1.25)  LDD0080  [22]
 LDCM0023  KB03 HCT 116 C194(1.57); C163(2.16); C158(1.91)  LDD0081  [22]
 LDCM0024  KB05 HCT 116 C194(1.99); C163(1.63); C158(1.25)  LDD0082  [22]
 LDCM0509  N-(4-bromo-3,5-dimethylphenyl)-2-nitroacetamide MDA-MB-231 C158(1.16); C109(1.13)  LDD2102  [12]
 LDCM0528  N-(4-bromophenyl)-2-cyano-N-phenylacetamide MDA-MB-231 C158(0.84); C109(0.57)  LDD2121  [12]
 LDCM0109  NEM HeLa C109(0.00); H247(0.00); H228(0.00)  LDD0223  [38]
 LDCM0496  Nucleophilic fragment 11a MDA-MB-231 C158(0.85); C109(0.60); C194(0.50)  LDD2089  [12]
 LDCM0497  Nucleophilic fragment 11b MDA-MB-231 C158(0.98)  LDD2090  [12]
 LDCM0499  Nucleophilic fragment 12b MDA-MB-231 C109(1.09)  LDD2092  [12]
 LDCM0500  Nucleophilic fragment 13a MDA-MB-231 C158(0.81); C109(0.94)  LDD2093  [12]
 LDCM0501  Nucleophilic fragment 13b MDA-MB-231 C158(1.46); C109(1.37)  LDD2094  [12]
 LDCM0504  Nucleophilic fragment 15a MDA-MB-231 C158(1.02); C109(0.60)  LDD2097  [12]
 LDCM0505  Nucleophilic fragment 15b MDA-MB-231 C158(0.85); C109(0.45)  LDD2098  [12]
 LDCM0506  Nucleophilic fragment 16a MDA-MB-231 C158(1.24); C194(0.95)  LDD2099  [12]
 LDCM0507  Nucleophilic fragment 16b MDA-MB-231 C158(0.54); C109(0.44)  LDD2100  [12]
 LDCM0508  Nucleophilic fragment 17a MDA-MB-231 C158(0.91); C109(0.91)  LDD2101  [12]
 LDCM0511  Nucleophilic fragment 18b MDA-MB-231 C158(0.38); C109(0.47)  LDD2104  [12]
 LDCM0512  Nucleophilic fragment 19a MDA-MB-231 C158(1.11); C109(1.52)  LDD2105  [12]
 LDCM0513  Nucleophilic fragment 19b MDA-MB-231 C158(0.44); C109(0.62)  LDD2106  [12]
 LDCM0514  Nucleophilic fragment 20a MDA-MB-231 C158(0.86); C109(0.79); C194(0.81)  LDD2107  [12]
 LDCM0515  Nucleophilic fragment 20b MDA-MB-231 C158(0.48); C109(0.40)  LDD2108  [12]
 LDCM0516  Nucleophilic fragment 21a MDA-MB-231 C158(0.74); C109(0.68)  LDD2109  [12]
 LDCM0517  Nucleophilic fragment 21b MDA-MB-231 C158(0.73); C109(1.39)  LDD2110  [12]
 LDCM0518  Nucleophilic fragment 22a MDA-MB-231 C158(1.04); C109(0.75); C194(1.15)  LDD2111  [12]
 LDCM0521  Nucleophilic fragment 23b MDA-MB-231 C158(0.34); C109(0.68)  LDD2114  [12]
 LDCM0522  Nucleophilic fragment 24a MDA-MB-231 C109(0.47)  LDD2115  [12]
 LDCM0523  Nucleophilic fragment 24b MDA-MB-231 C109(0.42); C54(0.79)  LDD2116  [12]
 LDCM0525  Nucleophilic fragment 25b MDA-MB-231 C109(0.39)  LDD2118  [12]
 LDCM0526  Nucleophilic fragment 26a MDA-MB-231 C158(2.13); C109(2.60); C54(2.45)  LDD2119  [12]
 LDCM0527  Nucleophilic fragment 26b MDA-MB-231 C158(0.79); C109(0.74)  LDD2120  [12]
 LDCM0529  Nucleophilic fragment 27b MDA-MB-231 C109(0.43)  LDD2122  [12]
 LDCM0530  Nucleophilic fragment 28a MDA-MB-231 C109(0.71); C194(0.96)  LDD2123  [12]
 LDCM0531  Nucleophilic fragment 28b MDA-MB-231 C158(0.48); C109(0.38)  LDD2124  [12]
 LDCM0532  Nucleophilic fragment 29a MDA-MB-231 C158(0.81); C109(0.64); C194(0.94)  LDD2125  [12]
 LDCM0533  Nucleophilic fragment 29b MDA-MB-231 C158(0.62); C109(0.42)  LDD2126  [12]
 LDCM0534  Nucleophilic fragment 30a MDA-MB-231 C158(0.85); C109(0.74)  LDD2127  [12]
 LDCM0535  Nucleophilic fragment 30b MDA-MB-231 C109(0.76)  LDD2128  [12]
 LDCM0536  Nucleophilic fragment 31 MDA-MB-231 C158(0.94); C109(0.87); C54(0.95)  LDD2129  [12]
 LDCM0540  Nucleophilic fragment 35 MDA-MB-231 C158(0.57); C109(0.59)  LDD2133  [12]
 LDCM0541  Nucleophilic fragment 36 MDA-MB-231 C109(0.49); C194(0.65)  LDD2134  [12]
 LDCM0542  Nucleophilic fragment 37 MDA-MB-231 C158(1.30); C109(0.95)  LDD2135  [12]
 LDCM0543  Nucleophilic fragment 38 MDA-MB-231 C158(1.01); C109(0.94); C194(1.28)  LDD2136  [12]
 LDCM0544  Nucleophilic fragment 39 MDA-MB-231 C158(0.85); C109(0.75); C194(0.88)  LDD2137  [12]
 LDCM0211  Nucleophilic fragment 3b MDA-MB-231 C109(1.80)  LDD1700  [12]
 LDCM0546  Nucleophilic fragment 40 MDA-MB-231 C158(0.69); C109(0.51); C194(0.68)  LDD2140  [12]
 LDCM0547  Nucleophilic fragment 41 MDA-MB-231 C158(0.67); C109(0.67)  LDD2141  [12]
 LDCM0549  Nucleophilic fragment 43 MDA-MB-231 C158(0.84); C109(0.69)  LDD2143  [12]
 LDCM0550  Nucleophilic fragment 5a MDA-MB-231 C158(3.31); C109(3.35)  LDD2144  [12]
 LDCM0551  Nucleophilic fragment 5b MDA-MB-231 C158(1.91)  LDD2145  [12]
 LDCM0552  Nucleophilic fragment 6a MDA-MB-231 C158(0.99); C109(0.69); C54(0.83)  LDD2146  [12]
 LDCM0553  Nucleophilic fragment 6b MDA-MB-231 C158(2.05); C109(1.95)  LDD2147  [12]
 LDCM0554  Nucleophilic fragment 7a MDA-MB-231 C158(0.30); C109(0.48); C194(0.55)  LDD2148  [12]
 LDCM0555  Nucleophilic fragment 7b MDA-MB-231 C109(0.54)  LDD2149  [12]
 LDCM0556  Nucleophilic fragment 8a MDA-MB-231 C158(0.82); C109(0.41)  LDD2150  [12]
 LDCM0559  Nucleophilic fragment 9b MDA-MB-231 C158(1.79); C109(1.73)  LDD2153  [12]
 LDCM0627  NUDT7-COV-1 HEK-293T C293(0.91); C118(0.75)  LDD2206  [49]
 LDCM0628  OTUB2-COV-1 HEK-293T C118(1.16); C109(1.10); C355(1.09); C194(1.05)  LDD2207  [49]
 LDCM0029  Quercetin HEK-293T 4.23  LDD0181  [32]
 LDCM0131  RA190 MM1.R 2.01  LDD0299  [17]
 LDCM0170  Structure8 Ramos 8.38  LDD0433  [50]
 LDCM0021  THZ1 HeLa S3 C109(1.06); C54(1.05)  LDD0460  [15]
 LDCM0110  W12 Hep-G2 C109(10.87); C194(16.53)  LDD0237  [8]
 LDCM0111  W14 Hep-G2 C109(9.72); C194(16.70)  LDD0238  [8]
 LDCM0113  W17 Hep-G2 C109(3.85); C194(7.44)  LDD0240  [8]

The Interaction Atlas With This Target

The Protein(s) Related To This Target

Enzyme
Click To Hide/Show 2 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Serine/threonine-protein kinase PAK 1 (PAK1) STE Ser/Thr protein kinase family Q13153
Peptidyl-prolyl cis-trans isomerase G (PPIG) . Q13427
Transcription factor
Click To Hide/Show 3 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Krueppel-like factor 1 (KLF1) Krueppel C2H2-type zinc-finger protein family Q13351
THAP domain-containing protein 11 (THAP11) THAP11 family Q96EK4
TSC22 domain family protein 4 (TSC22D4) TSC-22/Dip/Bun family Q9Y3Q8
Other
Click To Hide/Show 12 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Poly(U)-binding-splicing factor PUF60 (PUF60) RRM half pint family Q9UHX1
Insulin-like growth factor 2 mRNA-binding protein 3 (IGF2BP3) RRM IMP/VICKZ family O00425
U1 small nuclear ribonucleoprotein A (SNRPA) RRM U1 A/B'' family P09012
RNA-binding protein 39 (RBM39) Splicing factor SR family Q14498
KH domain-containing RNA-binding protein QKI (QKI) . Q96PU8
Poly(rC)-binding protein 2 (PCBP2) . Q15366
Polypyrimidine tract-binding protein 1 (PTBP1) . P26599
Pre-mRNA-processing-splicing factor 8 (PRPF8) . Q6P2Q9
RNA-binding protein 3 (RBM3) . P98179
RNA-binding protein with multiple splicing 2 (RBPMS2) . Q6ZRY4
WW domain-binding protein 11 (WBP11) . Q9Y2W2
Zinc finger protein 830 (ZNF830) . Q96NB3

References

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Mass spectrometry data entry: PXD028270
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Mass spectrometry data entry: PXD042377
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Mass spectrometry data entry: PXD029255
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Mass spectrometry data entry: PXD041264
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