Details of the Target

General Information of Target

Target ID LDTP17247
Target Name 5'-nucleotidase domain-containing protein 1 (NT5DC1)
Gene Name NT5DC1
Gene ID 221294
Synonyms
NT5C2L1; 5'-nucleotidase domain-containing protein 1; EC 3.1.3.-
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MLCASFLGLGLSVAIVGPTFQDLATNVNRNISSLSFIFVGRALGYLSGSVIGGFLVDVMN
YFLLLGISMSATTVGLYLVPFCKTAILLTVMMSIFGVSIGILDTGGNVLILAIWGDKGAP
HMQALHFSFALGAFLAPLLAKLALGPTASAENHTESDFHPALNQSSDADSEALFGVPNDK
NLLWAYAVIGTYMFLVSVIFFCLFLKNSSKQEKARASAETFRRAKYHNALLCLLFLFFFF
YVGAEVTYGSYVFSFATTHAGMKESEAAGLNSIFWGTFAACRGLAIFFATCLQPGTMIVL
SNIGSLTSSLFLVLFDKNPICLWIATSVYGASMATTFPSGVSWIEQYTTIHGKSAAFFVI
GASLGEMAIPAVIGILQGKYPDLPVVLYTSLGASIATGILFPVLYKLATSPLDRQRKEDR
KSEDQKALLSSSGLNEYEEENEEEDAEKWNEMDFEMIETNDTMRHSIIETSRSSLTEPTA
EVYNQYPSNALVFESSPFNTGSAHVKHLPETRTKGTNV
Target Bioclass
Enzyme
Family
5'(3')-deoxyribonucleotidase family
Uniprot ID
Q5TFE4
Ensemble ID
ENST00000319550.9
HGNC ID
HGNC:21556
ChEMBL ID
CHEMBL4295852

Target Site Mutations in Different Cell Lines

Cell line Mutation details Probe for labeling this protein in this cell
769P SNV: p.I162M DBIA    Probe Info 
JM1 SNV: p.L17V DBIA    Probe Info 
MOLT4 Deletion: p.T155HfsTer8 IA-alkyne    Probe Info 
NCIH1703 SNV: p.K373E DBIA    Probe Info 
OVK18 SNV: p.P56T DBIA    Probe Info 
RL952 Deletion: p.F379LfsTer74 DBIA    Probe Info 

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 34 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
m-APA
 Probe Info  		15.00  LDD0402  [1]
TH211
 Probe Info  		Y170(8.88)  LDD0257  [2]
TH214
 Probe Info  		Y310(20.00)  LDD0258  [2]
YN-1
 Probe Info  		100.00  LDD0444  [3]
STPyne
 Probe Info  		K307(2.94)  LDD0277  [4]
Johansson_61
 Probe Info  		_(20.00)  LDD1487  [5]
YY4-yne
 Probe Info  		3.45  LDD0400  [6]
AHL-Pu-1
 Probe Info  		C179(2.03)  LDD0169  [7]
HHS-475
 Probe Info  		Y124(0.46)  LDD0264  [8]
DBIA
 Probe Info  		C119(1.64)  LDD0078  [9]
ATP probe
 Probe Info  		K202(0.00); K109(0.00)  LDD0199  [10]
4-Iodoacetamidophenylacetylene
 Probe Info  		C179(0.00); C119(0.00); C226(0.00); C197(0.00)  LDD0038  [11]
IA-alkyne
 Probe Info  		N.A.  LDD0032  [12]
Lodoacetamide azide
 Probe Info  		C179(0.00); C119(0.00); C139(0.00); C226(0.00)  LDD0037  [11]
BTD
 Probe Info  		N.A.  LDD0004  [13]
JW-RF-010
 Probe Info  		N.A.  LDD0026  [14]
NAIA_4
 Probe Info  		C119(0.00); C179(0.00)  LDD2226  [15]
TFBX
 Probe Info  		N.A.  LDD0027  [14]
WYneN
 Probe Info  		N.A.  LDD0021  [13]
WYneO
 Probe Info  		N.A.  LDD0022  [13]
aHNE
 Probe Info  		N.A.  LDD0001  [13]
Compound 10
 Probe Info  		C119(0.00); C179(0.00)  LDD2216  [16]
Compound 11
 Probe Info  		C119(0.00); C179(0.00)  LDD2213  [16]
ENE
 Probe Info  		N.A.  LDD0006  [13]
IPM
 Probe Info  		N.A.  LDD0005  [13]
PF-06672131
 Probe Info  		N.A.  LDD0017  [17]
Phosphinate-6
 Probe Info  		N.A.  LDD0018  [18]
1c-yne
 Probe Info  		K171(0.00); K434(0.00)  LDD0228  [19]
Acrolein
 Probe Info  		C119(0.00); C179(0.00)  LDD0217  [20]
Methacrolein
 Probe Info  		C119(0.00); C179(0.00)  LDD0218  [20]
W1
 Probe Info  		C62(0.00); C63(0.00); C197(0.00); C119(0.00)  LDD0236  [21]
AOyne
 Probe Info  		15.00  LDD0443  [22]
NAIA_5
 Probe Info  		C179(0.00); C226(0.00); C230(0.00); C139(0.00)  LDD2223  [15]
HHS-482
 Probe Info  		Y124(0.98)  LDD2239  [23]
PAL-AfBPP Probe
Click To Hide/Show 18 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
C017
 Probe Info  		9.78  LDD1725  [24]
C130
 Probe Info  		7.11  LDD1812  [24]
C147
 Probe Info  		30.06  LDD1829  [24]
C160
 Probe Info  		7.21  LDD1840  [24]
C161
 Probe Info  		11.24  LDD1841  [24]
C205
 Probe Info  		5.35  LDD1880  [24]
C212
 Probe Info  		5.28  LDD1886  [24]
C243
 Probe Info  		49.52  LDD1916  [24]
C367
 Probe Info  		26.54  LDD2028  [24]
C383
 Probe Info  		28.44  LDD2042  [24]
C430
 Probe Info  		5.94  LDD2085  [24]
FFF probe11
 Probe Info  		11.61  LDD0472  [25]
FFF probe13
 Probe Info  		12.96  LDD0475  [25]
FFF probe2
 Probe Info  		13.22  LDD0463  [25]
FFF probe3
 Probe Info  		14.78  LDD0465  [25]
STS-2
 Probe Info  		N.A.  LDD0139  [26]
VE-P
 Probe Info  		N.A.  LDD0396  [27]
OEA-DA
 Probe Info  		3.19  LDD0046  [28]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0524  2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide MDA-MB-231 C119(1.00); C197(0.56)  LDD2117  [29]
 LDCM0026  4SU-RNA+native RNA HEK-293T C179(2.03)  LDD0169  [7]
 LDCM0214  AC1 HCT 116 C119(1.13); C179(0.95)  LDD0531  [9]
 LDCM0215  AC10 HCT 116 C119(1.04); C179(1.15); C63(1.34)  LDD0532  [9]
 LDCM0216  AC100 HCT 116 C119(1.12); C179(0.96); C62(0.69)  LDD0533  [9]
 LDCM0217  AC101 HCT 116 C119(1.06); C179(1.01); C62(0.71)  LDD0534  [9]
 LDCM0218  AC102 HCT 116 C119(1.02); C179(1.22); C62(0.75)  LDD0535  [9]
 LDCM0219  AC103 HCT 116 C119(1.34); C179(1.23); C62(0.70)  LDD0536  [9]
 LDCM0220  AC104 HCT 116 C119(1.15); C179(1.09); C62(0.86)  LDD0537  [9]
 LDCM0221  AC105 HCT 116 C119(1.18); C179(1.23); C62(0.71)  LDD0538  [9]
 LDCM0222  AC106 HCT 116 C119(1.19); C179(1.19); C62(0.66)  LDD0539  [9]
 LDCM0223  AC107 HCT 116 C119(1.38); C179(1.14); C62(0.82)  LDD0540  [9]
 LDCM0224  AC108 HCT 116 C119(0.93); C179(1.05); C62(0.63)  LDD0541  [9]
 LDCM0225  AC109 HCT 116 C119(0.98); C179(0.89); C62(0.94)  LDD0542  [9]
 LDCM0226  AC11 HCT 116 C119(1.08); C179(1.22); C63(1.39)  LDD0543  [9]
 LDCM0227  AC110 HCT 116 C119(0.98); C179(0.95); C62(0.67)  LDD0544  [9]
 LDCM0228  AC111 HCT 116 C119(1.14); C179(1.00); C62(0.55)  LDD0545  [9]
 LDCM0229  AC112 HCT 116 C119(1.23); C179(1.17); C62(0.56)  LDD0546  [9]
 LDCM0230  AC113 HCT 116 C119(1.11); C179(0.90)  LDD0547  [9]
 LDCM0231  AC114 HCT 116 C119(1.35); C179(1.13)  LDD0548  [9]
 LDCM0232  AC115 HCT 116 C119(1.48); C179(1.11)  LDD0549  [9]
 LDCM0233  AC116 HCT 116 C119(1.92); C179(1.01)  LDD0550  [9]
 LDCM0234  AC117 HCT 116 C119(1.33); C179(1.10)  LDD0551  [9]
 LDCM0235  AC118 HCT 116 C119(1.24); C179(1.18)  LDD0552  [9]
 LDCM0236  AC119 HCT 116 C119(1.16); C179(1.18)  LDD0553  [9]
 LDCM0237  AC12 HCT 116 C119(0.97); C179(1.09); C63(1.67)  LDD0554  [9]
 LDCM0238  AC120 HCT 116 C119(1.50); C179(1.18)  LDD0555  [9]
 LDCM0239  AC121 HCT 116 C119(1.20); C179(0.93)  LDD0556  [9]
 LDCM0240  AC122 HCT 116 C119(1.10); C179(1.23)  LDD0557  [9]
 LDCM0241  AC123 HCT 116 C119(1.11); C179(0.98)  LDD0558  [9]
 LDCM0242  AC124 HCT 116 C119(1.22); C179(0.96)  LDD0559  [9]
 LDCM0243  AC125 HCT 116 C119(1.21); C179(1.17)  LDD0560  [9]
 LDCM0244  AC126 HCT 116 C119(1.54); C179(1.17)  LDD0561  [9]
 LDCM0245  AC127 HCT 116 C119(1.63); C179(1.06)  LDD0562  [9]
 LDCM0246  AC128 HCT 116 C119(1.18); C179(0.92); C63(1.29)  LDD0563  [9]
 LDCM0247  AC129 HCT 116 C119(0.98); C179(1.03); C63(1.08)  LDD0564  [9]
 LDCM0249  AC130 HCT 116 C119(1.12); C179(1.10); C63(1.16)  LDD0566  [9]
 LDCM0250  AC131 HCT 116 C119(1.04); C179(1.31); C63(1.08)  LDD0567  [9]
 LDCM0251  AC132 HCT 116 C119(1.03); C179(1.47); C63(1.03)  LDD0568  [9]
 LDCM0252  AC133 HCT 116 C119(1.04); C179(1.11); C63(1.05)  LDD0569  [9]
 LDCM0253  AC134 HCT 116 C119(1.22); C179(1.19); C63(0.97)  LDD0570  [9]
 LDCM0254  AC135 HCT 116 C119(1.07); C179(1.14); C63(1.06)  LDD0571  [9]
 LDCM0255  AC136 HCT 116 C119(1.19); C179(1.08); C63(0.80)  LDD0572  [9]
 LDCM0256  AC137 HCT 116 C119(1.12); C179(1.35); C63(1.02)  LDD0573  [9]
 LDCM0257  AC138 HCT 116 C119(1.22); C179(1.45); C63(0.63)  LDD0574  [9]
 LDCM0258  AC139 HCT 116 C119(1.19); C179(1.55); C63(0.84)  LDD0575  [9]
 LDCM0259  AC14 HCT 116 C119(0.91); C179(1.18); C63(1.47)  LDD0576  [9]
 LDCM0260  AC140 HCT 116 C119(1.39); C179(1.46); C63(0.72)  LDD0577  [9]
 LDCM0261  AC141 HCT 116 C119(1.22); C179(1.41); C63(0.72)  LDD0578  [9]
 LDCM0262  AC142 HCT 116 C119(0.96); C179(1.21); C63(0.91)  LDD0579  [9]
 LDCM0263  AC143 HCT 116 C119(1.12); C179(1.15)  LDD0580  [9]
 LDCM0264  AC144 HCT 116 C179(1.15); C119(1.36)  LDD0581  [9]
 LDCM0265  AC145 HCT 116 C179(1.14); C119(1.20)  LDD0582  [9]
 LDCM0266  AC146 HCT 116 C179(1.14); C119(1.41)  LDD0583  [9]
 LDCM0267  AC147 HCT 116 C179(0.96); C119(1.48)  LDD0584  [9]
 LDCM0268  AC148 HCT 116 C179(1.18); C119(1.79)  LDD0585  [9]
 LDCM0269  AC149 HCT 116 C179(1.22); C119(1.54)  LDD0586  [9]
 LDCM0270  AC15 HCT 116 C119(1.05); C179(1.14); C63(1.23)  LDD0587  [9]
 LDCM0271  AC150 HCT 116 C179(1.06); C119(1.20)  LDD0588  [9]
 LDCM0272  AC151 HCT 116 C119(1.07); C179(1.18)  LDD0589  [9]
 LDCM0273  AC152 HCT 116 C179(1.18); C119(1.35)  LDD0590  [9]
 LDCM0274  AC153 HCT 116 C179(1.37); C119(2.04)  LDD0591  [9]
 LDCM0621  AC154 HCT 116 C119(1.26); C179(1.15)  LDD2158  [9]
 LDCM0622  AC155 HCT 116 C119(1.16); C179(1.19)  LDD2159  [9]
 LDCM0623  AC156 HCT 116 C119(1.06); C179(1.16)  LDD2160  [9]
 LDCM0624  AC157 HCT 116 C119(0.99); C179(1.26)  LDD2161  [9]
 LDCM0276  AC17 HCT 116 C179(1.10); C119(1.14)  LDD0593  [9]
 LDCM0277  AC18 HCT 116 C179(1.06); C119(1.30)  LDD0594  [9]
 LDCM0278  AC19 HCT 116 C119(1.00); C179(1.30)  LDD0595  [9]
 LDCM0279  AC2 HCT 116 C179(0.95); C119(1.07)  LDD0596  [9]
 LDCM0280  AC20 HCT 116 C119(1.10); C179(1.20)  LDD0597  [9]
 LDCM0281  AC21 HCT 116 C179(1.12); C119(1.24)  LDD0598  [9]
 LDCM0282  AC22 HCT 116 C179(1.07); C119(1.08)  LDD0599  [9]
 LDCM0283  AC23 HCT 116 C179(1.16); C119(1.30)  LDD0600  [9]
 LDCM0284  AC24 HCT 116 C179(0.95); C119(1.04)  LDD0601  [9]
 LDCM0285  AC25 HCT 116 C63(0.89); C179(0.93); C119(0.96); C62(0.96)  LDD0602  [9]
 LDCM0286  AC26 HCT 116 C62(0.50); C63(0.67); C179(0.98); C119(1.06)  LDD0603  [9]
 LDCM0287  AC27 HCT 116 C62(0.61); C63(0.90); C119(1.06); C179(1.11)  LDD0604  [9]
 LDCM0288  AC28 HCT 116 C62(0.49); C63(0.66); C179(1.05); C119(1.21)  LDD0605  [9]
 LDCM0289  AC29 HCT 116 C62(0.38); C63(0.52); C179(1.06); C119(1.19)  LDD0606  [9]
 LDCM0290  AC3 HCT 116 C119(1.00); C179(1.06)  LDD0607  [9]
 LDCM0291  AC30 HCT 116 C62(0.42); C63(0.52); C119(1.12); C179(1.24)  LDD0608  [9]
 LDCM0292  AC31 HCT 116 C62(0.47); C63(0.66); C119(1.03); C179(1.10)  LDD0609  [9]
 LDCM0293  AC32 HCT 116 C62(0.42); C63(0.55); C179(1.33); C119(1.47)  LDD0610  [9]
 LDCM0294  AC33 HCT 116 C62(0.92); C63(1.07); C179(1.09); C119(1.19)  LDD0611  [9]
 LDCM0295  AC34 HCT 116 C62(0.75); C63(0.97); C179(1.18); C119(1.46)  LDD0612  [9]
 LDCM0296  AC35 HCT 116 C119(0.89); C179(0.90)  LDD0613  [9]
 LDCM0297  AC36 HCT 116 C119(0.92); C179(0.93)  LDD0614  [9]
 LDCM0298  AC37 HCT 116 C119(0.85); C179(0.99)  LDD0615  [9]
 LDCM0299  AC38 HCT 116 C119(0.95); C179(0.98)  LDD0616  [9]
 LDCM0300  AC39 HCT 116 C179(1.01); C119(1.02)  LDD0617  [9]
 LDCM0301  AC4 HCT 116 C179(1.01); C119(1.21)  LDD0618  [9]
 LDCM0302  AC40 HCT 116 C179(1.11); C119(1.15)  LDD0619  [9]
 LDCM0303  AC41 HCT 116 C119(0.94); C179(1.03)  LDD0620  [9]
 LDCM0304  AC42 HCT 116 C179(1.03); C119(1.08)  LDD0621  [9]
 LDCM0305  AC43 HCT 116 C119(0.97); C179(1.05)  LDD0622  [9]
 LDCM0306  AC44 HCT 116 C119(0.95); C179(1.18)  LDD0623  [9]
 LDCM0307  AC45 HCT 116 C119(1.04); C179(1.17)  LDD0624  [9]
 LDCM0308  AC46 HCT 116 C62(0.49); C179(1.02); C119(1.14)  LDD0625  [9]
 LDCM0309  AC47 HCT 116 C62(0.80); C179(1.06); C119(1.08)  LDD0626  [9]
 LDCM0310  AC48 HCT 116 C62(0.60); C179(0.98); C119(0.99)  LDD0627  [9]
 LDCM0311  AC49 HCT 116 C62(0.61); C179(1.27); C119(1.32)  LDD0628  [9]
 LDCM0312  AC5 HCT 116 C179(1.07); C119(1.24)  LDD0629  [9]
 LDCM0313  AC50 HCT 116 C62(0.53); C179(1.22); C119(1.39)  LDD0630  [9]
 LDCM0314  AC51 HCT 116 C62(0.60); C119(0.86); C179(0.87)  LDD0631  [9]
 LDCM0315  AC52 HCT 116 C62(0.60); C119(1.01); C179(1.03)  LDD0632  [9]
 LDCM0316  AC53 HCT 116 C62(1.00); C179(1.20); C119(1.66)  LDD0633  [9]
 LDCM0317  AC54 HCT 116 C62(0.65); C119(1.11); C179(1.11)  LDD0634  [9]
 LDCM0318  AC55 HCT 116 C179(1.24); C62(1.25); C119(1.30)  LDD0635  [9]
 LDCM0319  AC56 HCT 116 C62(0.77); C179(1.27); C119(1.42)  LDD0636  [9]
 LDCM0320  AC57 HCT 116 C62(1.06); C119(1.22); C179(1.25)  LDD0637  [9]
 LDCM0321  AC58 HCT 116 C62(1.01); C179(1.34); C119(1.36)  LDD0638  [9]
 LDCM0322  AC59 HCT 116 C62(1.03); C119(1.55); C179(1.75)  LDD0639  [9]
 LDCM0323  AC6 HCT 116 C63(0.88); C119(1.16); C179(1.16)  LDD0640  [9]
 LDCM0324  AC60 HCT 116 C62(1.19); C179(1.55); C119(1.78)  LDD0641  [9]
 LDCM0325  AC61 HCT 116 C62(0.81); C119(1.19); C179(1.51)  LDD0642  [9]
 LDCM0326  AC62 HCT 116 C62(0.94); C119(1.35); C179(1.39)  LDD0643  [9]
 LDCM0327  AC63 HCT 116 C62(0.89); C119(1.38); C179(1.49)  LDD0644  [9]
 LDCM0328  AC64 HCT 116 C119(1.33); C62(1.36); C179(1.66)  LDD0645  [9]
 LDCM0329  AC65 HCT 116 C62(0.88); C119(1.31); C179(1.43)  LDD0646  [9]
 LDCM0330  AC66 HCT 116 C62(0.85); C119(1.27); C179(1.40)  LDD0647  [9]
 LDCM0331  AC67 HCT 116 C62(0.82); C119(1.47); C179(1.98)  LDD0648  [9]
 LDCM0332  AC68 HCT 116 C62(0.66); C63(0.75); C179(0.97); C119(1.07)  LDD0649  [9]
 LDCM0333  AC69 HCT 116 C62(0.59); C63(0.70); C179(0.93); C119(1.20)  LDD0650  [9]
 LDCM0334  AC7 HCT 116 C63(1.04); C179(1.06); C119(1.10)  LDD0651  [9]
 LDCM0335  AC70 HCT 116 C63(0.48); C62(0.51); C179(0.83); C119(1.29)  LDD0652  [9]
 LDCM0336  AC71 HCT 116 C179(0.77); C62(0.81); C63(0.94); C119(1.15)  LDD0653  [9]
 LDCM0337  AC72 HCT 116 C62(0.62); C63(0.62); C179(1.01); C119(1.24)  LDD0654  [9]
 LDCM0338  AC73 HCT 116 C63(0.47); C62(0.47); C179(1.23); C119(1.64)  LDD0655  [9]
 LDCM0339  AC74 HCT 116 C62(0.64); C63(0.75); C179(1.14); C119(1.58)  LDD0656  [9]
 LDCM0340  AC75 HCT 116 C62(0.41); C63(0.42); C179(1.29); C119(1.78)  LDD0657  [9]
 LDCM0341  AC76 HCT 116 C62(0.90); C179(1.01); C63(1.04); C119(1.31)  LDD0658  [9]
 LDCM0342  AC77 HCT 116 C62(0.57); C63(0.60); C179(1.00); C119(1.30)  LDD0659  [9]
 LDCM0343  AC78 HCT 116 C62(0.60); C63(0.69); C179(1.00); C119(1.06)  LDD0660  [9]
 LDCM0344  AC79 HCT 116 C62(0.62); C63(0.62); C179(1.03); C119(1.35)  LDD0661  [9]
 LDCM0345  AC8 HCT 116 C63(1.00); C119(1.21); C179(1.27)  LDD0662  [9]
 LDCM0346  AC80 HCT 116 C62(0.79); C63(0.94); C179(1.04); C119(1.07)  LDD0663  [9]
 LDCM0347  AC81 HCT 116 C62(0.45); C63(0.53); C179(0.99); C119(1.18)  LDD0664  [9]
 LDCM0348  AC82 HCT 116 C62(0.49); C63(0.62); C179(1.24); C119(1.57)  LDD0665  [9]
 LDCM0349  AC83 HCT 116 C179(1.67); C119(1.92)  LDD0666  [9]
 LDCM0350  AC84 HCT 116 C119(1.39); C179(1.44)  LDD0667  [9]
 LDCM0351  AC85 HCT 116 C179(1.23); C119(1.36)  LDD0668  [9]
 LDCM0352  AC86 HCT 116 C179(1.02); C119(1.40)  LDD0669  [9]
 LDCM0353  AC87 HCT 116 C119(1.05); C179(1.23)  LDD0670  [9]
 LDCM0354  AC88 HCT 116 C179(0.92); C119(1.23)  LDD0671  [9]
 LDCM0355  AC89 HCT 116 C119(1.17); C179(1.39)  LDD0672  [9]
 LDCM0357  AC90 HCT 116 C119(0.96); C179(1.23)  LDD0674  [9]
 LDCM0358  AC91 HCT 116 C119(1.51); C179(1.55)  LDD0675  [9]
 LDCM0359  AC92 HCT 116 C179(1.44); C119(1.52)  LDD0676  [9]
 LDCM0360  AC93 HCT 116 C179(1.11); C119(1.16)  LDD0677  [9]
 LDCM0361  AC94 HCT 116 C179(1.01); C119(1.21)  LDD0678  [9]
 LDCM0362  AC95 HCT 116 C179(1.12); C119(1.36)  LDD0679  [9]
 LDCM0363  AC96 HCT 116 C179(1.19); C119(1.35)  LDD0680  [9]
 LDCM0364  AC97 HCT 116 C179(1.08); C119(1.61)  LDD0681  [9]
 LDCM0365  AC98 HCT 116 C62(0.57); C179(1.15); C119(1.32)  LDD0682  [9]
 LDCM0366  AC99 HCT 116 C62(0.64); C179(0.89); C119(1.12)  LDD0683  [9]
 LDCM0248  AKOS034007472 HCT 116 C119(0.94); C179(1.09); C63(1.24)  LDD0565  [9]
 LDCM0356  AKOS034007680 HCT 116 C119(1.13); C179(1.27); C63(1.32)  LDD0673  [9]
 LDCM0275  AKOS034007705 HCT 116 C63(0.83); C119(1.38); C179(1.51)  LDD0592  [9]
 LDCM0156  Aniline NCI-H1299 11.83  LDD0403  [1]
 LDCM0020  ARS-1620 HCC44 C119(1.64)  LDD0078  [9]
 LDCM0200  BPK-25 T cell C119(4.88)  LDD0529  [30]
 LDCM0630  CCW28-3 231MFP C119(1.37)  LDD2214  [31]
 LDCM0108  Chloroacetamide HeLa C179(0.00); C119(0.00); C10(0.00); C22(0.00)  LDD0222  [20]
 LDCM0632  CL-Sc Hep-G2 C179(1.09); C119(0.89)  LDD2227  [15]
 LDCM0367  CL1 HCT 116 C63(0.48); C179(1.15); C119(1.53)  LDD0684  [9]
 LDCM0368  CL10 HCT 116 C63(0.30); C179(1.01); C119(3.60)  LDD0685  [9]
 LDCM0369  CL100 HCT 116 C179(1.04); C119(1.23)  LDD0686  [9]
 LDCM0370  CL101 HCT 116 C63(0.89); C179(1.00); C119(1.21)  LDD0687  [9]
 LDCM0371  CL102 HCT 116 C179(1.01); C63(1.07); C119(1.89)  LDD0688  [9]
 LDCM0372  CL103 HCT 116 C179(0.67); C63(1.15); C119(1.21)  LDD0689  [9]
 LDCM0373  CL104 HCT 116 C63(1.07); C119(1.12); C179(1.14)  LDD0690  [9]
 LDCM0374  CL105 HCT 116 C179(0.99); C119(1.35)  LDD0691  [9]
 LDCM0375  CL106 HCT 116 C179(1.23); C119(1.40)  LDD0692  [9]
 LDCM0376  CL107 HCT 116 C119(1.27); C179(1.39)  LDD0693  [9]
 LDCM0377  CL108 HCT 116 C179(1.40); C119(1.43)  LDD0694  [9]
 LDCM0378  CL109 HCT 116 C179(1.35); C119(1.36)  LDD0695  [9]
 LDCM0379  CL11 HCT 116 C63(0.33); C179(0.79); C119(1.87)  LDD0696  [9]
 LDCM0380  CL110 HCT 116 C179(1.05); C119(1.61)  LDD0697  [9]
 LDCM0381  CL111 HCT 116 C179(0.80); C119(2.42)  LDD0698  [9]
 LDCM0382  CL112 HCT 116 C62(0.84); C179(0.96); C63(1.21); C119(1.39)  LDD0699  [9]
 LDCM0383  CL113 HCT 116 C62(0.35); C63(0.55); C179(1.22); C119(1.42)  LDD0700  [9]
 LDCM0384  CL114 HCT 116 C62(0.34); C63(0.54); C179(0.90); C119(2.54)  LDD0701  [9]
 LDCM0385  CL115 HCT 116 C62(0.69); C63(0.74); C179(1.01); C119(1.54)  LDD0702  [9]
 LDCM0386  CL116 HCT 116 C62(0.86); C63(0.97); C179(1.14); C119(1.15)  LDD0703  [9]
 LDCM0387  CL117 HCT 116 C179(1.33); C119(1.54)  LDD0704  [9]
 LDCM0388  CL118 HCT 116 C179(1.03); C119(1.10)  LDD0705  [9]
 LDCM0389  CL119 HCT 116 C119(1.02); C179(1.10)  LDD0706  [9]
 LDCM0390  CL12 HCT 116 C63(0.50); C179(0.80); C119(1.69)  LDD0707  [9]
 LDCM0391  CL120 HCT 116 C119(0.93); C179(1.02)  LDD0708  [9]
 LDCM0392  CL121 HCT 116 C119(0.63); C62(0.72); C179(0.84)  LDD0709  [9]
 LDCM0393  CL122 HCT 116 C62(0.59); C179(1.01); C119(1.29)  LDD0710  [9]
 LDCM0394  CL123 HCT 116 C62(0.68); C179(0.87); C119(2.43)  LDD0711  [9]
 LDCM0395  CL124 HCT 116 C62(0.61); C179(1.21); C119(1.73)  LDD0712  [9]
 LDCM0396  CL125 HCT 116 C62(0.98); C119(1.12); C179(1.36)  LDD0713  [9]
 LDCM0397  CL126 HCT 116 C119(1.17); C62(1.20); C179(1.32)  LDD0714  [9]
 LDCM0398  CL127 HCT 116 C62(1.02); C179(1.10); C119(1.37)  LDD0715  [9]
 LDCM0399  CL128 HCT 116 C179(1.15); C62(1.19); C119(1.21)  LDD0716  [9]
 LDCM0400  CL13 HCT 116 C63(0.34); C179(0.83); C119(1.78)  LDD0717  [9]
 LDCM0401  CL14 HCT 116 C63(0.36); C179(0.79); C119(1.62)  LDD0718  [9]
 LDCM0402  CL15 HCT 116 C63(0.23); C179(0.59); C119(2.18)  LDD0719  [9]
 LDCM0403  CL16 HCT 116 C179(1.07); C119(1.10)  LDD0720  [9]
 LDCM0404  CL17 HCT 116 C179(0.77); C119(2.08)  LDD0721  [9]
 LDCM0405  CL18 HCT 116 C179(1.03); C119(1.05)  LDD0722  [9]
 LDCM0406  CL19 HCT 116 C179(0.91); C119(1.10)  LDD0723  [9]
 LDCM0407  CL2 HCT 116 C63(0.59); C179(1.04); C119(1.10)  LDD0724  [9]
 LDCM0408  CL20 HCT 116 C179(1.06); C119(1.10)  LDD0725  [9]
 LDCM0409  CL21 HCT 116 C179(0.80); C119(1.89)  LDD0726  [9]
 LDCM0410  CL22 HCT 116 C179(1.02); C119(1.31)  LDD0727  [9]
 LDCM0411  CL23 HCT 116 C119(1.04); C179(1.15)  LDD0728  [9]
 LDCM0412  CL24 HCT 116 C179(1.08); C119(1.18)  LDD0729  [9]
 LDCM0413  CL25 HCT 116 C119(2.46); C179(0.92)  LDD0730  [9]
 LDCM0414  CL26 HCT 116 C119(1.11); C179(1.02)  LDD0731  [9]
 LDCM0415  CL27 HCT 116 C119(1.04); C179(0.98)  LDD0732  [9]
 LDCM0416  CL28 HCT 116 C119(1.16); C179(1.04)  LDD0733  [9]
 LDCM0417  CL29 HCT 116 C119(1.13); C179(1.08)  LDD0734  [9]
 LDCM0418  CL3 HCT 116 C119(1.10); C179(0.95); C63(0.78)  LDD0735  [9]
 LDCM0419  CL30 HCT 116 C119(0.98); C179(1.10)  LDD0736  [9]
 LDCM0420  CL31 HCT 116 C119(1.16); C179(1.00)  LDD0737  [9]
 LDCM0421  CL32 HCT 116 C119(1.08); C179(0.98)  LDD0738  [9]
 LDCM0422  CL33 HCT 116 C119(1.37); C179(1.01)  LDD0739  [9]
 LDCM0423  CL34 HCT 116 C119(1.10); C179(0.83)  LDD0740  [9]
 LDCM0424  CL35 HCT 116 C119(1.18); C179(0.92)  LDD0741  [9]
 LDCM0425  CL36 HCT 116 C119(1.37); C179(0.80)  LDD0742  [9]
 LDCM0426  CL37 HCT 116 C119(1.07); C179(0.92)  LDD0743  [9]
 LDCM0428  CL39 HCT 116 C119(1.12); C179(0.95)  LDD0745  [9]
 LDCM0429  CL4 HCT 116 C119(1.48); C179(0.97); C63(0.60)  LDD0746  [9]
 LDCM0430  CL40 HCT 116 C119(2.30); C179(0.74)  LDD0747  [9]
 LDCM0431  CL41 HCT 116 C119(1.34); C179(0.75)  LDD0748  [9]
 LDCM0432  CL42 HCT 116 C119(1.05); C179(0.98)  LDD0749  [9]
 LDCM0433  CL43 HCT 116 C119(1.27); C179(0.82)  LDD0750  [9]
 LDCM0434  CL44 HCT 116 C119(1.13); C179(0.79)  LDD0751  [9]
 LDCM0435  CL45 HCT 116 C119(1.58); C179(0.69)  LDD0752  [9]
 LDCM0436  CL46 HCT 116 C119(1.13); C179(1.00); C62(0.95); C63(0.95)  LDD0753  [9]
 LDCM0437  CL47 HCT 116 C119(1.13); C179(0.96); C62(0.91); C63(0.91)  LDD0754  [9]
 LDCM0438  CL48 HCT 116 C119(0.97); C179(1.00); C62(0.82); C63(0.82)  LDD0755  [9]
 LDCM0439  CL49 HCT 116 C119(1.01); C179(0.96); C62(0.86); C63(0.86)  LDD0756  [9]
 LDCM0440  CL5 HCT 116 C119(1.07); C179(0.86); C63(0.41)  LDD0757  [9]
 LDCM0441  CL50 HCT 116 C119(1.18); C179(0.63); C62(1.04); C63(1.04)  LDD0758  [9]
 LDCM0442  CL51 HCT 116 C119(1.04); C179(0.83); C62(1.06); C63(1.06)  LDD0759  [9]
 LDCM0443  CL52 HCT 116 C119(1.03); C179(0.98); C62(0.68); C63(0.68)  LDD0760  [9]
 LDCM0444  CL53 HCT 116 C119(1.50); C179(0.93); C62(1.42); C63(1.42)  LDD0761  [9]
 LDCM0445  CL54 HCT 116 C119(1.26); C179(0.56); C62(0.96); C63(0.96)  LDD0762  [9]
 LDCM0446  CL55 HCT 116 C119(1.09); C179(0.88); C62(0.71); C63(0.71)  LDD0763  [9]
 LDCM0447  CL56 HCT 116 C119(1.11); C179(1.07); C62(0.74); C63(0.74)  LDD0764  [9]
 LDCM0448  CL57 HCT 116 C119(2.04); C179(0.84); C62(0.71); C63(0.71)  LDD0765  [9]
 LDCM0449  CL58 HCT 116 C119(1.00); C179(0.96); C62(1.23); C63(1.23)  LDD0766  [9]
 LDCM0450  CL59 HCT 116 C119(0.97); C179(0.97); C62(0.87); C63(0.87)  LDD0767  [9]
 LDCM0451  CL6 HCT 116 C119(2.19); C179(0.99); C63(0.40)  LDD0768  [9]
 LDCM0452  CL60 HCT 116 C119(1.29); C179(0.86); C62(0.75); C63(0.75)  LDD0769  [9]
 LDCM0453  CL61 HCT 116 C119(1.27); C179(1.12); C62(0.95); C63(1.02)  LDD0770  [9]
 LDCM0454  CL62 HCT 116 C119(1.28); C179(1.04); C62(0.90); C63(0.91)  LDD0771  [9]
 LDCM0455  CL63 HCT 116 C119(1.52); C179(1.02); C62(0.83); C63(0.92)  LDD0772  [9]
 LDCM0456  CL64 HCT 116 C119(1.71); C179(1.00); C62(0.85); C63(0.98)  LDD0773  [9]
 LDCM0457  CL65 HCT 116 C119(1.39); C179(1.16); C62(0.91); C63(0.92)  LDD0774  [9]
 LDCM0458  CL66 HCT 116 C119(1.96); C179(1.45); C62(0.50); C63(0.69)  LDD0775  [9]
 LDCM0459  CL67 HCT 116 C119(1.46); C179(1.33); C62(0.69); C63(0.81)  LDD0776  [9]
 LDCM0460  CL68 HCT 116 C119(1.59); C179(1.14); C62(0.46); C63(0.67)  LDD0777  [9]
 LDCM0461  CL69 HCT 116 C119(1.66); C179(1.06); C62(0.52); C63(0.61)  LDD0778  [9]
 LDCM0462  CL7 HCT 116 C119(1.33); C179(0.83); C63(0.61)  LDD0779  [9]
 LDCM0463  CL70 HCT 116 C119(1.37); C179(0.95); C62(0.50); C63(0.58)  LDD0780  [9]
 LDCM0464  CL71 HCT 116 C119(1.81); C179(1.14); C62(0.82); C63(0.81)  LDD0781  [9]
 LDCM0465  CL72 HCT 116 C119(1.21); C179(1.09); C62(0.82); C63(0.96)  LDD0782  [9]
 LDCM0466  CL73 HCT 116 C119(7.69); C179(0.73); C62(0.88); C63(1.04)  LDD0783  [9]
 LDCM0467  CL74 HCT 116 C119(1.53); C179(1.15); C62(0.69); C63(0.78)  LDD0784  [9]
 LDCM0469  CL76 HCT 116 C119(1.06); C179(1.03); C62(0.46); C63(0.46)  LDD0786  [9]
 LDCM0470  CL77 HCT 116 C119(1.50); C179(0.68); C62(0.77); C63(0.77)  LDD0787  [9]
 LDCM0471  CL78 HCT 116 C119(1.19); C179(1.09); C62(0.64); C63(0.64)  LDD0788  [9]
 LDCM0472  CL79 HCT 116 C119(1.39); C179(1.20); C62(0.54); C63(0.54)  LDD0789  [9]
 LDCM0473  CL8 HCT 116 C119(3.02); C179(0.89); C63(0.34)  LDD0790  [9]
 LDCM0474  CL80 HCT 116 C119(1.07); C179(1.04); C62(0.41); C63(0.41)  LDD0791  [9]
 LDCM0475  CL81 HCT 116 C119(1.21); C179(1.06); C62(0.84); C63(0.84)  LDD0792  [9]
 LDCM0476  CL82 HCT 116 C119(1.44); C179(1.20); C62(0.35); C63(0.35)  LDD0793  [9]
 LDCM0477  CL83 HCT 116 C119(1.61); C179(1.33); C62(0.38); C63(0.38)  LDD0794  [9]
 LDCM0478  CL84 HCT 116 C119(1.96); C179(1.46); C62(0.27); C63(0.27)  LDD0795  [9]
 LDCM0479  CL85 HCT 116 C119(1.30); C179(1.12); C62(0.64); C63(0.64)  LDD0796  [9]
 LDCM0480  CL86 HCT 116 C119(1.21); C179(1.02); C62(0.79); C63(0.79)  LDD0797  [9]
 LDCM0481  CL87 HCT 116 C119(1.46); C179(1.08); C62(0.76); C63(0.76)  LDD0798  [9]
 LDCM0482  CL88 HCT 116 C119(1.37); C179(1.17); C62(0.45); C63(0.45)  LDD0799  [9]
 LDCM0483  CL89 HCT 116 C119(1.71); C179(1.65); C62(0.15); C63(0.15)  LDD0800  [9]
 LDCM0484  CL9 HCT 116 C119(1.65); C179(0.86); C63(0.61)  LDD0801  [9]
 LDCM0485  CL90 HCT 116 C119(1.99); C179(0.78); C62(0.92); C63(0.92)  LDD0802  [9]
 LDCM0486  CL91 HCT 116 C119(1.14); C179(1.11)  LDD0803  [9]
 LDCM0487  CL92 HCT 116 C119(1.42); C179(0.89)  LDD0804  [9]
 LDCM0488  CL93 HCT 116 C119(1.31); C179(0.90)  LDD0805  [9]
 LDCM0489  CL94 HCT 116 C119(1.76); C179(0.92)  LDD0806  [9]
 LDCM0490  CL95 HCT 116 C119(2.14); C179(0.83)  LDD0807  [9]
 LDCM0491  CL96 HCT 116 C119(1.31); C179(0.93)  LDD0808  [9]
 LDCM0492  CL97 HCT 116 C119(1.48); C179(1.08)  LDD0809  [9]
 LDCM0493  CL98 HCT 116 C119(1.39); C179(1.10)  LDD0810  [9]
 LDCM0494  CL99 HCT 116 C119(1.23); C179(1.04)  LDD0811  [9]
 LDCM0634  CY-0357 Hep-G2 C119(0.70)  LDD2228  [15]
 LDCM0495  E2913 HEK-293T C119(1.18); C197(1.03); C179(1.01); C139(1.04)  LDD1698  [32]
 LDCM0213  Electrophilic fragment 2 MDA-MB-231 C119(5.30)  LDD1702  [29]
 LDCM0201  EV-3 T cell C119(5.30)  LDD0515  [30]
 LDCM0202  EV-93 T cell C119(9.36)  LDD0514  [30]
 LDCM0625  F8 Ramos C179(1.31); C119(2.75); C197(1.24)  LDD2187  [33]
 LDCM0572  Fragment10 MDA-MB-231 C119(20.00)  LDD1389  [5]
 LDCM0573  Fragment11 MDA-MB-231 C119(20.00)  LDD1391  [5]
 LDCM0574  Fragment12 MDA-MB-231 C119(20.00)  LDD1393  [5]
 LDCM0575  Fragment13 MDA-MB-231 C119(1.48)  LDD1395  [5]
 LDCM0576  Fragment14 MDA-MB-231 C119(2.05)  LDD1397  [5]
 LDCM0577  Fragment15 Ramos C119(6.83)  LDD1400  [5]
 LDCM0579  Fragment20 Ramos C119(20.00)  LDD1403  [5]
 LDCM0580  Fragment21 MDA-MB-231 C119(1.19)  LDD1404  [5]
 LDCM0581  Fragment22 MDA-MB-231 C119(1.67)  LDD1406  [5]
 LDCM0582  Fragment23 Ramos C119(1.26)  LDD1409  [5]
 LDCM0583  Fragment24 Ramos C119(1.48)  LDD1410  [5]
 LDCM0584  Fragment25 MDA-MB-231 C119(0.93)  LDD1411  [5]
 LDCM0585  Fragment26 Ramos C119(0.96)  LDD1412  [5]
 LDCM0578  Fragment27 MDA-MB-231 C119(0.81)  LDD1401  [5]
 LDCM0586  Fragment28 MDA-MB-231 C119(1.18)  LDD1415  [5]
 LDCM0587  Fragment29 MDA-MB-231 C119(1.21)  LDD1417  [5]
 LDCM0588  Fragment30 MDA-MB-231 C119(1.68)  LDD1419  [5]
 LDCM0589  Fragment31 MDA-MB-231 C119(3.25)  LDD1421  [5]
 LDCM0590  Fragment32 MDA-MB-231 C119(10.82)  LDD1423  [5]
 LDCM0468  Fragment33 HCT 116 C119(1.51); C179(1.11); C62(0.79); C63(0.92)  LDD0785  [9]
 LDCM0592  Fragment34 MDA-MB-231 C119(0.88)  LDD1427  [5]
 LDCM0593  Fragment35 Ramos C119(1.14)  LDD1430  [5]
 LDCM0595  Fragment37 Ramos C119(0.98)  LDD1432  [5]
 LDCM0596  Fragment38 MDA-MB-231 C119(3.23)  LDD1433  [5]
 LDCM0597  Fragment39 MDA-MB-231 C119(3.81)  LDD1435  [5]
 LDCM0566  Fragment4 MDA-MB-231 C119(8.66)  LDD1378  [5]
 LDCM0598  Fragment40 Ramos C119(1.31)  LDD1437  [5]
 LDCM0599  Fragment41 MDA-MB-231 C119(1.19)  LDD1438  [5]
 LDCM0600  Fragment42 Ramos C119(0.90)  LDD1440  [5]
 LDCM0601  Fragment43 MDA-MB-231 C119(3.43)  LDD1441  [5]
 LDCM0602  Fragment44 MDA-MB-231 C119(1.37)  LDD1443  [5]
 LDCM0603  Fragment45 MDA-MB-231 C119(20.00)  LDD1444  [5]
 LDCM0604  Fragment46 MDA-MB-231 C119(0.84)  LDD1445  [5]
 LDCM0605  Fragment47 MDA-MB-231 C119(1.09)  LDD1446  [5]
 LDCM0607  Fragment49 MDA-MB-231 C119(5.58)  LDD1448  [5]
 LDCM0427  Fragment51 HCT 116 C119(1.66); C179(0.67)  LDD0744  [9]
 LDCM0610  Fragment52 MDA-MB-231 C119(1.06)  LDD1452  [5]
 LDCM0611  Fragment53 MDA-MB-231 C119(1.13)  LDD1454  [5]
 LDCM0612  Fragment54 MDA-MB-231 C119(1.14)  LDD1456  [5]
 LDCM0613  Fragment55 MDA-MB-231 C119(1.02)  LDD1457  [5]
 LDCM0614  Fragment56 MDA-MB-231 C119(1.15)  LDD1458  [5]
 LDCM0615  Fragment63-R Jurkat _(20.00)  LDD1487  [5]
 LDCM0617  Fragment63-S Jurkat _(20.00)  LDD1490  [5]
 LDCM0569  Fragment7 Ramos C179(1.93); C119(12.39); C197(0.67)  LDD2186  [33]
 LDCM0570  Fragment8 MDA-MB-231 C119(20.00)  LDD1385  [5]
 LDCM0571  Fragment9 MDA-MB-231 C119(20.00)  LDD1387  [5]
 LDCM0116  HHS-0101 DM93 Y124(0.46)  LDD0264  [8]
 LDCM0117  HHS-0201 DM93 Y124(0.78)  LDD0265  [8]
 LDCM0118  HHS-0301 DM93 Y124(1.71)  LDD0266  [8]
 LDCM0119  HHS-0401 DM93 Y124(1.05)  LDD0267  [8]
 LDCM0120  HHS-0701 DM93 Y124(1.40)  LDD0268  [8]
 LDCM0022  KB02 HCT 116 C119(7.65)  LDD0080  [9]
 LDCM0023  KB03 HCT 116 C119(3.85)  LDD0081  [9]
 LDCM0024  KB05 HCT 116 C119(7.57)  LDD0082  [9]
 LDCM0169  KB63 Ramos 12.29  LDD0432  [34]
 LDCM0109  NEM HeLa N.A.  LDD0224  [20]
 LDCM0512  Nucleophilic fragment 19a MDA-MB-231 C119(1.62)  LDD2105  [29]
 LDCM0514  Nucleophilic fragment 20a MDA-MB-231 C197(0.99)  LDD2107  [29]
 LDCM0516  Nucleophilic fragment 21a MDA-MB-231 C197(1.00)  LDD2109  [29]
 LDCM0518  Nucleophilic fragment 22a MDA-MB-231 C197(1.24)  LDD2111  [29]
 LDCM0522  Nucleophilic fragment 24a MDA-MB-231 C197(0.55)  LDD2115  [29]
 LDCM0530  Nucleophilic fragment 28a MDA-MB-231 C197(0.98)  LDD2123  [29]
 LDCM0532  Nucleophilic fragment 29a MDA-MB-231 C119(0.57)  LDD2125  [29]
 LDCM0534  Nucleophilic fragment 30a MDA-MB-231 C197(1.17)  LDD2127  [29]
 LDCM0536  Nucleophilic fragment 31 MDA-MB-231 C119(0.97)  LDD2129  [29]
 LDCM0542  Nucleophilic fragment 37 MDA-MB-231 C197(0.85)  LDD2135  [29]
 LDCM0543  Nucleophilic fragment 38 MDA-MB-231 C197(1.40)  LDD2136  [29]
 LDCM0544  Nucleophilic fragment 39 MDA-MB-231 C197(1.04)  LDD2137  [29]
 LDCM0546  Nucleophilic fragment 40 MDA-MB-231 C119(0.96); C197(0.87)  LDD2140  [29]
 LDCM0550  Nucleophilic fragment 5a MDA-MB-231 C197(1.05)  LDD2144  [29]
 LDCM0552  Nucleophilic fragment 6a MDA-MB-231 C197(0.98)  LDD2146  [29]
 LDCM0627  NUDT7-COV-1 HEK-293T C179(0.25); C119(0.07)  LDD2206  [35]
 LDCM0628  OTUB2-COV-1 HEK-293T C179(0.92); C119(0.67)  LDD2207  [35]
 LDCM0131  RA190 MM1.R C119(1.82)  LDD0304  [36]
 LDCM0021  THZ1 HCT 116 C119(1.11); C179(0.89)  LDD2173  [9]
 LDCM0112  W16 Hep-G2 C119(1.39)  LDD0239  [21]
 LDCM0154  YY4 T cell 3.45  LDD0400  [6]

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