Details of the Target
General Information of Target
Target ID | LDTP04570 | |||||
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Target Name | Coatomer subunit beta (COPB1) | |||||
Gene Name | COPB1 | |||||
Gene ID | 1315 | |||||
Synonyms |
COPB; Coatomer subunit beta; Beta-coat protein; Beta-COP |
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3D Structure | ||||||
Sequence |
MTAAENVCYTLINVPMDSEPPSEISLKNDLEKGDVKSKTEALKKVIIMILNGEKLPGLLM
TIIRFVLPLQDHTIKKLLLVFWEIVPKTTPDGRLLHEMILVCDAYRKDLQHPNEFIRGST LRFLCKLKEAELLEPLMPAIRACLEHRHSYVRRNAVLAIYTIYRNFEHLIPDAPELIHDF LVNEKDASCKRNAFMMLIHADQDRALDYLSTCIDQVQTFGDILQLVIVELIYKVCHANPS ERARFIRCIYNLLQSSSPAVKYEAAGTLVTLSSAPTAIKAAAQCYIDLIIKESDNNVKLI VLDRLIELKEHPAHERVLQDLVMDILRVLSTPDLEVRKKTLQLALDLVSSRNVEELVIVL KKEVIKTNNVSEHEDTDKYRQLLVRTLHSCSVRFPDMAANVIPVLMEFLSDNNEAAAADV LEFVREAIQRFDNLRMLIVEKMLEVFHAIKSVKIYRGALWILGEYCSTKEDIQSVMTEIR RSLGEIPIVESEIKKEAGELKPEEEITVGPVQKLVTEMGTYATQSALSSSRPTKKEEDRP PLRGFLLDGDFFVAASLATTLTKIALRYVALVQEKKKQNSFVAEAMLLMATILHLGKSSL PKKPITDDDVDRISLCLKVLSECSPLMNDIFNKECRQSLSHMLSAKLEEEKLSQKKESEK RNVTVQPDDPISFMQLTAKNEMNCKEDQFQLSLLAAMGNTQRKEAADPLASKLNKVTQLT GFSDPVYAEAYVHVNQYDIVLDVLVVNQTSDTLQNCTLELATLGDLKLVEKPSPLTLAPH DFANIKANVKVASTENGIIFGNIVYDVSGAASDRNCVVLSDIHIDIMDYIQPATCTDAEF RQMWAEFEWENKVTVNTNMVDLNDYLQHILKSTNMKCLTPEKALSGYCGFMAANLYARSI FGEDALANVSIEKPIHQGPDAAVTGHIRIRAKSQGMALSLGDKINLSQKKTSI |
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Target Bioclass |
Other
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Subcellular location |
Cytoplasm
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Function |
The coatomer is a cytosolic protein complex that binds to dilysine motifs and reversibly associates with Golgi non-clathrin-coated vesicles, which further mediate biosynthetic protein transport from the ER, via the Golgi up to the trans Golgi network. Coatomer complex is required for budding from Golgi membranes, and is essential for the retrograde Golgi-to-ER transport of dilysine-tagged proteins. In mammals, the coatomer can only be recruited by membranes associated to ADP-ribosylation factors (ARFs), which are small GTP-binding proteins; the complex also influences the Golgi structural integrity, as well as the processing, activity, and endocytic recycling of LDL receptors. Plays a functional role in facilitating the transport of kappa-type opioid receptor mRNAs into axons and enhances translation of these proteins. Required for limiting lipid storage in lipid droplets. Involved in lipid homeostasis by regulating the presence of perilipin family members PLIN2 and PLIN3 at the lipid droplet surface and promoting the association of adipocyte surface triglyceride lipase (PNPLA2) with the lipid droplet to mediate lipolysis. Involved in the Golgi disassembly and reassembly processes during cell cycle. Involved in autophagy by playing a role in early endosome function. Plays a role in organellar compartmentalization of secretory compartments including endoplasmic reticulum (ER)-Golgi intermediate compartment (ERGIC), Golgi, trans-Golgi network (TGN) and recycling endosomes, and in biosynthetic transport of CAV1. Promotes degradation of Nef cellular targets CD4 and MHC class I antigens by facilitating their trafficking to degradative compartments.
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Uniprot ID | ||||||
Ensemble ID | ||||||
HGNC ID | ||||||
ChEMBL ID |
Probe(s) Labeling This Target
ABPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
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m-APA Probe Info |
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13.75 | LDD0402 | [1] | |
A-EBA Probe Info |
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3.89 | LDD0215 | [2] | |
CY-1 Probe Info |
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66.28 | LDD0243 | [3] | |
CY4 Probe Info |
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39.64 | LDD0244 | [3] | |
TH211 Probe Info |
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Y379(20.00); Y521(20.00); Y896(16.76); Y887(12.94) | LDD0257 | [4] | |
TH216 Probe Info |
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Y896(9.65); Y521(6.10) | LDD0259 | [4] | |
YN-1 Probe Info |
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100.00 | LDD0444 | [5] | |
YN-4 Probe Info |
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100.00 | LDD0445 | [5] | |
1oxF11yne Probe Info |
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N.A. | LDD0193 | [6] | |
ONAyne Probe Info |
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K107(0.39); K190(0.49); K309(1.07); K712(0.95) | LDD0274 | [7] | |
BTD Probe Info |
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C143(2.45) | LDD1699 | [8] | |
Probe 1 Probe Info |
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Y568(18.26) | LDD3495 | [9] | |
JZ128-DTB Probe Info |
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N.A. | LDD0462 | [10] | |
DA-P3 Probe Info |
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7.76 | LDD0183 | [11] | |
AHL-Pu-1 Probe Info |
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C684(2.65); C623(2.12) | LDD0168 | [12] | |
HHS-482 Probe Info |
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Y521(1.02) | LDD0285 | [13] | |
HHS-475 Probe Info |
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Y887(0.77); Y521(0.84); Y160(0.95) | LDD0264 | [14] | |
HHS-465 Probe Info |
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Y521(10.00); Y887(10.00) | LDD2237 | [15] | |
DBIA Probe Info |
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C888(1.24); C623(0.98) | LDD0078 | [16] | |
5E-2FA Probe Info |
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H780(0.00); H916(0.00); H373(0.00) | LDD2235 | [17] | |
ATP probe Probe Info |
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K107(0.00); K703(0.00); K633(0.00); K712(0.00) | LDD0199 | [18] | |
4-Iodoacetamidophenylacetylene Probe Info |
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C284(0.00); C888(0.00); C248(0.00); C466(0.00) | LDD0038 | [19] | |
IA-alkyne Probe Info |
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C616(0.00); C623(0.00); C888(0.00); C248(0.00) | LDD0032 | [20] | |
Lodoacetamide azide Probe Info |
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C284(0.00); C888(0.00); C248(0.00); C466(0.00) | LDD0037 | [19] | |
ATP probe Probe Info |
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K128(0.00); K339(0.00) | LDD0035 | [21] | |
NAIA_4 Probe Info |
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C623(0.00); C635(0.00); C684(0.00); C888(0.00) | LDD2226 | [22] | |
TFBX Probe Info |
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N.A. | LDD0027 | [23] | |
WYneN Probe Info |
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N.A. | LDD0021 | [24] | |
WYneO Probe Info |
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N.A. | LDD0022 | [24] | |
aHNE Probe Info |
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N.A. | LDD0001 | [24] | |
Compound 10 Probe Info |
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N.A. | LDD2216 | [25] | |
ENE Probe Info |
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N.A. | LDD0006 | [24] | |
IPM Probe Info |
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C616(0.00); C623(0.00) | LDD0005 | [24] | |
NHS Probe Info |
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N.A. | LDD0010 | [24] | |
SF Probe Info |
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N.A. | LDD0028 | [26] | |
STPyne Probe Info |
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N.A. | LDD0009 | [24] | |
VSF Probe Info |
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C248(0.00); C684(0.00); C623(0.00) | LDD0007 | [24] | |
Phosphinate-6 Probe Info |
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C877(0.00); C684(0.00) | LDD0018 | [27] | |
1c-yne Probe Info |
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K771(0.00); K361(0.00); K128(0.00); K679(0.00) | LDD0228 | [28] | |
Acrolein Probe Info |
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C390(0.00); C235(0.00); C248(0.00); C143(0.00) | LDD0217 | [29] | |
Cinnamaldehyde Probe Info |
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N.A. | LDD0220 | [29] | |
Crotonaldehyde Probe Info |
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C616(0.00); C235(0.00) | LDD0219 | [29] | |
Methacrolein Probe Info |
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C390(0.00); C623(0.00); C143(0.00); C616(0.00) | LDD0218 | [29] | |
W1 Probe Info |
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C623(0.00); C102(0.00); C390(0.00); C284(0.00) | LDD0236 | [30] | |
AOyne Probe Info |
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5.30 | LDD0443 | [31] | |
NAIA_5 Probe Info |
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C284(0.00); C143(0.00); C212(0.00); C888(0.00) | LDD2223 | [22] |
PAL-AfBPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
---|---|---|---|---|---|
FFF probe12 Probe Info |
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12.23 | LDD0473 | [32] | |
FFF probe13 Probe Info |
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14.36 | LDD0475 | [32] | |
FFF probe14 Probe Info |
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20.00 | LDD0477 | [32] | |
FFF probe3 Probe Info |
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20.00 | LDD0464 | [32] | |
VE-P Probe Info |
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N.A. | LDD0396 | [33] | |
Alk-rapa Probe Info |
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3.42 | LDD0213 | [34] | |
DA-2 Probe Info |
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N.A. | LDD0071 | [35] |
Competitor(s) Related to This Target
Competitor ID | Name | Cell line | Binding Site(Ratio) | Interaction ID | Ref |
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LDCM0548 | 1-(4-(Benzo[d][1,3]dioxol-5-ylmethyl)piperazin-1-yl)-2-nitroethan-1-one | MDA-MB-231 | C684(0.81); C235(0.75); C390(0.36); C143(0.74) | LDD2142 | [8] |
LDCM0519 | 1-(6-methoxy-3,4-dihydroquinolin-1(2H)-yl)-2-nitroethan-1-one | MDA-MB-231 | C684(0.87); C877(0.78); C235(0.72); C143(0.98) | LDD2112 | [8] |
LDCM0502 | 1-(Cyanoacetyl)piperidine | MDA-MB-231 | C684(1.11); C877(0.75); C235(0.62); C390(0.51) | LDD2095 | [8] |
LDCM0537 | 2-Cyano-N,N-dimethylacetamide | MDA-MB-231 | C684(0.74); C877(0.99); C235(0.68); C390(1.11) | LDD2130 | [8] |
LDCM0524 | 2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide | MDA-MB-231 | C684(1.41); C877(1.48); C235(0.74); C390(1.19) | LDD2117 | [8] |
LDCM0558 | 2-Cyano-N-phenylacetamide | MDA-MB-231 | C684(1.46); C235(1.38); C390(1.55); C143(1.63) | LDD2152 | [8] |
LDCM0510 | 3-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-3-oxopropanenitrile | MDA-MB-231 | C684(0.72); C390(1.04); C143(1.13) | LDD2103 | [8] |
LDCM0539 | 3-(4-Isopropylpiperazin-1-yl)-3-oxopropanenitrile | MDA-MB-231 | C684(0.53); C235(0.66); C390(0.45); C143(0.47) | LDD2132 | [8] |
LDCM0538 | 4-(Cyanoacetyl)morpholine | MDA-MB-231 | C684(0.61); C877(0.77); C390(0.81); C143(0.40) | LDD2131 | [8] |
LDCM0025 | 4SU-RNA | HEK-293T | C684(2.65); C623(2.12) | LDD0168 | [12] |
LDCM0026 | 4SU-RNA+native RNA | HEK-293T | C684(3.41); C623(3.64) | LDD0169 | [12] |
LDCM0214 | AC1 | HCT 116 | C102(0.95); C235(0.97); C248(0.93); C284(1.04) | LDD0531 | [16] |
LDCM0215 | AC10 | HCT 116 | C102(1.00); C235(0.95); C248(0.92); C284(0.95) | LDD0532 | [16] |
LDCM0216 | AC100 | HCT 116 | C102(0.77); C235(1.24); C248(0.82); C284(0.84) | LDD0533 | [16] |
LDCM0217 | AC101 | HCT 116 | C102(0.72); C235(1.27); C248(0.73); C284(0.72) | LDD0534 | [16] |
LDCM0218 | AC102 | HCT 116 | C102(0.77); C235(1.13); C248(0.75); C284(0.78) | LDD0535 | [16] |
LDCM0219 | AC103 | HCT 116 | C102(0.75); C235(0.96); C248(0.69); C284(0.73) | LDD0536 | [16] |
LDCM0220 | AC104 | HCT 116 | C102(0.85); C235(1.24); C248(0.74); C284(0.80) | LDD0537 | [16] |
LDCM0221 | AC105 | HCT 116 | C102(0.79); C235(0.97); C248(0.79); C284(0.79) | LDD0538 | [16] |
LDCM0222 | AC106 | HCT 116 | C102(0.74); C235(1.14); C248(0.81); C284(0.77) | LDD0539 | [16] |
LDCM0223 | AC107 | HCT 116 | C102(0.83); C235(1.09); C248(0.71); C284(1.00) | LDD0540 | [16] |
LDCM0224 | AC108 | HCT 116 | C102(0.73); C235(1.48); C248(0.78); C284(0.92) | LDD0541 | [16] |
LDCM0225 | AC109 | HCT 116 | C102(0.81); C235(1.36); C248(0.73); C284(0.84) | LDD0542 | [16] |
LDCM0226 | AC11 | HCT 116 | C102(1.01); C235(0.90); C248(0.95); C284(0.87) | LDD0543 | [16] |
LDCM0227 | AC110 | HCT 116 | C102(0.76); C235(1.04); C248(0.72); C284(0.77) | LDD0544 | [16] |
LDCM0228 | AC111 | HCT 116 | C102(0.73); C235(1.09); C248(0.75); C284(0.76) | LDD0545 | [16] |
LDCM0229 | AC112 | HCT 116 | C102(0.73); C235(0.94); C248(0.67); C284(0.84) | LDD0546 | [16] |
LDCM0230 | AC113 | HCT 116 | C102(0.86); C235(1.21); C248(0.97); C284(0.90) | LDD0547 | [16] |
LDCM0231 | AC114 | HCT 116 | C102(0.97); C235(1.23); C248(0.91); C284(0.86) | LDD0548 | [16] |
LDCM0232 | AC115 | HCT 116 | C102(0.96); C235(1.01); C248(0.86); C284(1.01) | LDD0549 | [16] |
LDCM0233 | AC116 | HCT 116 | C102(0.91); C235(1.19); C248(0.92); C284(0.92) | LDD0550 | [16] |
LDCM0234 | AC117 | HCT 116 | C102(0.99); C235(1.06); C248(0.87); C284(0.86) | LDD0551 | [16] |
LDCM0235 | AC118 | HCT 116 | C102(1.00); C235(1.03); C248(0.91); C284(0.91) | LDD0552 | [16] |
LDCM0236 | AC119 | HCT 116 | C102(0.91); C235(1.33); C248(0.92); C284(0.90) | LDD0553 | [16] |
LDCM0237 | AC12 | HCT 116 | C102(0.96); C235(0.90); C248(1.00); C284(0.92) | LDD0554 | [16] |
LDCM0238 | AC120 | HCT 116 | C102(0.99); C235(1.33); C248(0.97); C284(0.90) | LDD0555 | [16] |
LDCM0239 | AC121 | HCT 116 | C102(0.91); C235(0.98); C248(0.91); C284(0.94) | LDD0556 | [16] |
LDCM0240 | AC122 | HCT 116 | C102(0.88); C235(1.27); C248(0.98); C284(0.93) | LDD0557 | [16] |
LDCM0241 | AC123 | HCT 116 | C102(0.97); C235(0.91); C248(0.85); C284(0.94) | LDD0558 | [16] |
LDCM0242 | AC124 | HCT 116 | C102(0.94); C235(1.22); C248(0.94); C284(0.92) | LDD0559 | [16] |
LDCM0243 | AC125 | HCT 116 | C102(0.82); C235(1.39); C248(0.91); C284(0.89) | LDD0560 | [16] |
LDCM0244 | AC126 | HCT 116 | C102(0.93); C235(1.20); C248(0.92); C284(0.97) | LDD0561 | [16] |
LDCM0245 | AC127 | HCT 116 | C102(0.92); C235(1.01); C248(0.86); C284(0.87) | LDD0562 | [16] |
LDCM0246 | AC128 | HCT 116 | C102(1.25); C235(0.91); C248(1.17); C284(0.96) | LDD0563 | [16] |
LDCM0247 | AC129 | HCT 116 | C102(0.93); C235(0.91); C248(1.09); C284(0.90) | LDD0564 | [16] |
LDCM0249 | AC130 | HCT 116 | C102(0.98); C235(0.73); C248(1.05); C284(1.09) | LDD0566 | [16] |
LDCM0250 | AC131 | HCT 116 | C102(0.93); C235(0.77); C248(0.94); C284(0.73) | LDD0567 | [16] |
LDCM0251 | AC132 | HCT 116 | C102(0.97); C235(0.95); C248(1.01); C284(0.93) | LDD0568 | [16] |
LDCM0252 | AC133 | HCT 116 | C102(1.03); C235(0.86); C248(0.97); C284(0.88) | LDD0569 | [16] |
LDCM0253 | AC134 | HCT 116 | C102(1.02); C235(0.81); C248(0.98); C284(1.08) | LDD0570 | [16] |
LDCM0254 | AC135 | HCT 116 | C102(1.04); C235(0.80); C248(1.04); C284(0.97) | LDD0571 | [16] |
LDCM0255 | AC136 | HCT 116 | C102(1.01); C235(0.97); C248(1.05); C284(0.92) | LDD0572 | [16] |
LDCM0256 | AC137 | HCT 116 | C102(1.01); C235(0.90); C248(1.03); C284(1.10) | LDD0573 | [16] |
LDCM0257 | AC138 | HCT 116 | C102(1.11); C235(0.79); C248(1.07); C284(1.00) | LDD0574 | [16] |
LDCM0258 | AC139 | HCT 116 | C102(0.98); C235(0.87); C248(1.01); C284(1.14) | LDD0575 | [16] |
LDCM0259 | AC14 | HCT 116 | C102(0.97); C235(0.90); C248(0.86); C284(0.89) | LDD0576 | [16] |
LDCM0260 | AC140 | HCT 116 | C102(1.08); C235(0.91); C248(1.03); C284(0.94) | LDD0577 | [16] |
LDCM0261 | AC141 | HCT 116 | C102(1.09); C235(0.87); C248(1.04); C284(1.06) | LDD0578 | [16] |
LDCM0262 | AC142 | HCT 116 | C102(0.94); C235(1.03); C248(1.00); C284(0.95) | LDD0579 | [16] |
LDCM0263 | AC143 | HCT 116 | C102(0.92); C235(0.75); C248(0.89); C284(0.74) | LDD0580 | [16] |
LDCM0264 | AC144 | HCT 116 | C284(0.72); C390(0.73); C248(0.87); C102(0.96) | LDD0581 | [16] |
LDCM0265 | AC145 | HCT 116 | C390(0.85); C235(0.89); C466(0.90); C284(0.93) | LDD0582 | [16] |
LDCM0266 | AC146 | HCT 116 | C284(0.70); C390(0.72); C102(0.88); C248(0.89) | LDD0583 | [16] |
LDCM0267 | AC147 | HCT 116 | C390(0.76); C466(0.88); C248(0.89); C235(0.92) | LDD0584 | [16] |
LDCM0268 | AC148 | HCT 116 | C284(0.76); C390(0.83); C466(0.97); C102(1.04) | LDD0585 | [16] |
LDCM0269 | AC149 | HCT 116 | C284(0.57); C390(0.78); C102(0.84); C248(0.89) | LDD0586 | [16] |
LDCM0270 | AC15 | HCT 116 | C235(0.85); C390(0.87); C248(0.89); C284(0.93) | LDD0587 | [16] |
LDCM0271 | AC150 | HCT 116 | C284(0.65); C390(0.83); C102(0.90); C235(0.90) | LDD0588 | [16] |
LDCM0272 | AC151 | HCT 116 | C284(0.74); C390(0.84); C235(0.88); C102(0.88) | LDD0589 | [16] |
LDCM0273 | AC152 | HCT 116 | C284(0.75); C390(0.82); C235(0.83); C248(0.93) | LDD0590 | [16] |
LDCM0274 | AC153 | HCT 116 | C284(0.74); C390(0.78); C102(0.99); C466(1.09) | LDD0591 | [16] |
LDCM0621 | AC154 | HCT 116 | C102(0.99); C235(0.90); C248(0.90); C284(0.64) | LDD2158 | [16] |
LDCM0622 | AC155 | HCT 116 | C102(0.93); C235(0.93); C248(0.91); C284(0.69) | LDD2159 | [16] |
LDCM0623 | AC156 | HCT 116 | C102(0.89); C235(0.92); C248(0.99); C284(0.88) | LDD2160 | [16] |
LDCM0624 | AC157 | HCT 116 | C102(0.86); C235(0.90); C248(0.94); C284(0.64) | LDD2161 | [16] |
LDCM0276 | AC17 | HCT 116 | C888(0.81); C248(0.91); C623(0.95); C102(0.98) | LDD0593 | [16] |
LDCM0277 | AC18 | HCT 116 | C248(0.89); C235(0.97); C102(1.05); C466(1.07) | LDD0594 | [16] |
LDCM0278 | AC19 | HCT 116 | C888(0.83); C248(0.87); C235(0.94); C284(0.96) | LDD0595 | [16] |
LDCM0279 | AC2 | HCT 116 | C888(0.65); C248(0.89); C390(0.96); C284(0.97) | LDD0596 | [16] |
LDCM0280 | AC20 | HCT 116 | C248(0.92); C235(0.98); C466(0.98); C102(1.02) | LDD0597 | [16] |
LDCM0281 | AC21 | HCT 116 | C248(0.89); C888(0.95); C235(1.00); C102(1.03) | LDD0598 | [16] |
LDCM0282 | AC22 | HCT 116 | C888(0.81); C248(0.98); C102(1.00); C235(1.04) | LDD0599 | [16] |
LDCM0283 | AC23 | HCT 116 | C248(0.93); C102(0.95); C888(0.96); C284(1.00) | LDD0600 | [16] |
LDCM0284 | AC24 | HCT 116 | C248(0.95); C623(0.97); C235(0.99); C102(1.01) | LDD0601 | [16] |
LDCM0285 | AC25 | HCT 116 | C390(0.74); C888(0.78); C235(0.92); C102(0.94) | LDD0602 | [16] |
LDCM0286 | AC26 | HCT 116 | C390(0.79); C888(0.83); C235(0.86); C248(0.88) | LDD0603 | [16] |
LDCM0287 | AC27 | HCT 116 | C390(0.78); C248(0.80); C235(0.83); C466(0.93) | LDD0604 | [16] |
LDCM0288 | AC28 | HCT 116 | C390(0.81); C235(0.83); C888(0.89); C102(0.91) | LDD0605 | [16] |
LDCM0289 | AC29 | HCT 116 | C390(0.73); C235(0.78); C248(0.86); C888(0.89) | LDD0606 | [16] |
LDCM0290 | AC3 | HCT 116 | C888(0.49); C248(0.93); C102(0.96); C466(1.00) | LDD0607 | [16] |
LDCM0291 | AC30 | HCT 116 | C390(0.73); C235(0.78); C248(0.90); C102(0.93) | LDD0608 | [16] |
LDCM0292 | AC31 | HCT 116 | C102(0.88); C248(0.88); C235(0.88); C390(0.89) | LDD0609 | [16] |
LDCM0293 | AC32 | HCT 116 | C390(0.72); C235(0.74); C248(0.83); C466(0.92) | LDD0610 | [16] |
LDCM0294 | AC33 | HCT 116 | C235(0.70); C248(0.80); C390(0.80); C466(0.85) | LDD0611 | [16] |
LDCM0295 | AC34 | HCT 116 | C235(0.76); C248(0.85); C466(0.89); C390(0.89) | LDD0612 | [16] |
LDCM0296 | AC35 | HCT 116 | C102(0.99); C284(1.05); C466(1.06); C248(1.09) | LDD0613 | [16] |
LDCM0297 | AC36 | HCT 116 | C235(0.87); C888(0.94); C284(0.95); C248(0.96) | LDD0614 | [16] |
LDCM0298 | AC37 | HCT 116 | C888(0.81); C102(0.94); C248(0.96); C284(0.99) | LDD0615 | [16] |
LDCM0299 | AC38 | HCT 116 | C888(0.74); C102(0.94); C248(0.95); C235(0.97) | LDD0616 | [16] |
LDCM0300 | AC39 | HCT 116 | C888(0.67); C102(0.96); C248(1.01); C235(1.06) | LDD0617 | [16] |
LDCM0301 | AC4 | HCT 116 | C888(0.54); C248(0.88); C390(0.95); C466(0.97) | LDD0618 | [16] |
LDCM0302 | AC40 | HCT 116 | C248(0.98); C235(1.01); C888(1.03); C390(1.05) | LDD0619 | [16] |
LDCM0303 | AC41 | HCT 116 | C102(0.89); C888(0.91); C390(0.91); C248(0.95) | LDD0620 | [16] |
LDCM0304 | AC42 | HCT 116 | C248(0.94); C235(0.98); C284(0.98); C466(1.02) | LDD0621 | [16] |
LDCM0305 | AC43 | HCT 116 | C248(0.93); C102(0.93); C888(0.95); C390(0.96) | LDD0622 | [16] |
LDCM0306 | AC44 | HCT 116 | C390(0.90); C248(0.94); C235(0.95); C888(1.00) | LDD0623 | [16] |
LDCM0307 | AC45 | HCT 116 | C390(0.84); C248(0.98); C235(1.02); C888(1.02) | LDD0624 | [16] |
LDCM0308 | AC46 | HCT 116 | C623(0.82); C888(0.89); C102(0.90); C390(0.93) | LDD0625 | [16] |
LDCM0309 | AC47 | HCT 116 | C623(0.77); C888(0.86); C248(0.97); C102(1.01) | LDD0626 | [16] |
LDCM0310 | AC48 | HCT 116 | C623(0.73); C888(0.82); C102(0.95); C390(0.99) | LDD0627 | [16] |
LDCM0311 | AC49 | HCT 116 | C248(1.04); C235(1.09); C623(1.10); C466(1.11) | LDD0628 | [16] |
LDCM0312 | AC5 | HCT 116 | C888(0.50); C248(0.90); C102(0.98); C390(0.99) | LDD0629 | [16] |
LDCM0313 | AC50 | HCT 116 | C623(0.94); C390(0.95); C248(1.01); C466(1.05) | LDD0630 | [16] |
LDCM0314 | AC51 | HCT 116 | C623(0.71); C102(0.89); C284(0.96); C466(0.98) | LDD0631 | [16] |
LDCM0315 | AC52 | HCT 116 | C623(0.74); C284(0.97); C102(0.98); C888(1.00) | LDD0632 | [16] |
LDCM0316 | AC53 | HCT 116 | C623(0.93); C390(0.94); C248(0.95); C466(0.97) | LDD0633 | [16] |
LDCM0317 | AC54 | HCT 116 | C623(0.90); C888(1.05); C235(1.05); C248(1.06) | LDD0634 | [16] |
LDCM0318 | AC55 | HCT 116 | C248(1.03); C390(1.04); C466(1.05); C235(1.08) | LDD0635 | [16] |
LDCM0319 | AC56 | HCT 116 | C390(1.11); C235(1.14); C248(1.14); C623(1.15) | LDD0636 | [16] |
LDCM0320 | AC57 | HCT 116 | C235(0.86); C248(0.88); C390(0.92); C102(0.95) | LDD0637 | [16] |
LDCM0321 | AC58 | HCT 116 | C235(0.82); C390(0.82); C248(0.84); C102(0.89) | LDD0638 | [16] |
LDCM0322 | AC59 | HCT 116 | C390(0.83); C235(0.88); C248(0.90); C466(0.95) | LDD0639 | [16] |
LDCM0323 | AC6 | HCT 116 | C284(0.75); C235(0.87); C248(0.89); C623(0.90) | LDD0640 | [16] |
LDCM0324 | AC60 | HCT 116 | C390(0.81); C248(0.82); C235(0.88); C102(0.90) | LDD0641 | [16] |
LDCM0325 | AC61 | HCT 116 | C248(0.86); C102(0.89); C390(0.89); C888(0.93) | LDD0642 | [16] |
LDCM0326 | AC62 | HCT 116 | C390(0.86); C235(0.86); C248(0.94); C466(0.98) | LDD0643 | [16] |
LDCM0327 | AC63 | HCT 116 | C390(0.83); C235(0.87); C102(0.89); C248(0.91) | LDD0644 | [16] |
LDCM0328 | AC64 | HCT 116 | C248(0.92); C390(0.95); C235(0.97); C888(0.98) | LDD0645 | [16] |
LDCM0329 | AC65 | HCT 116 | C888(0.82); C390(0.93); C248(0.95); C235(1.00) | LDD0646 | [16] |
LDCM0330 | AC66 | HCT 116 | C888(0.97); C248(0.98); C235(0.99); C390(1.01) | LDD0647 | [16] |
LDCM0331 | AC67 | HCT 116 | C235(0.89); C390(0.95); C248(0.98); C466(1.06) | LDD0648 | [16] |
LDCM0332 | AC68 | HCT 116 | C235(0.84); C390(0.95); C284(0.95); C623(1.02) | LDD0649 | [16] |
LDCM0333 | AC69 | HCT 116 | C284(0.95); C235(1.00); C623(1.02); C466(1.03) | LDD0650 | [16] |
LDCM0334 | AC7 | HCT 116 | C390(0.86); C235(0.91); C284(0.92); C102(0.96) | LDD0651 | [16] |
LDCM0335 | AC70 | HCT 116 | C284(0.87); C623(0.88); C466(0.93); C888(0.93) | LDD0652 | [16] |
LDCM0336 | AC71 | HCT 116 | C888(0.89); C623(0.91); C284(1.01); C248(1.01) | LDD0653 | [16] |
LDCM0337 | AC72 | HCT 116 | C390(0.91); C623(0.96); C248(0.97); C235(0.98) | LDD0654 | [16] |
LDCM0338 | AC73 | HCT 116 | C235(0.89); C390(0.92); C623(0.97); C466(1.06) | LDD0655 | [16] |
LDCM0339 | AC74 | HCT 116 | C623(0.86); C390(1.09); C235(1.09); C466(1.10) | LDD0656 | [16] |
LDCM0340 | AC75 | HCT 116 | C235(1.03); C623(1.03); C390(1.04); C466(1.13) | LDD0657 | [16] |
LDCM0341 | AC76 | HCT 116 | C888(0.96); C623(0.97); C466(1.04); C284(1.04) | LDD0658 | [16] |
LDCM0342 | AC77 | HCT 116 | C390(0.88); C235(0.96); C466(1.00); C248(1.00) | LDD0659 | [16] |
LDCM0343 | AC78 | HCT 116 | C284(0.87); C390(0.92); C888(0.92); C102(0.93) | LDD0660 | [16] |
LDCM0344 | AC79 | HCT 116 | C284(0.94); C466(0.95); C623(0.98); C888(1.00) | LDD0661 | [16] |
LDCM0345 | AC8 | HCT 116 | C390(0.95); C102(0.95); C623(0.98); C248(1.01) | LDD0662 | [16] |
LDCM0346 | AC80 | HCT 116 | C390(0.96); C102(0.99); C466(1.02); C623(1.03) | LDD0663 | [16] |
LDCM0347 | AC81 | HCT 116 | C466(0.97); C623(1.00); C102(1.01); C888(1.05) | LDD0664 | [16] |
LDCM0348 | AC82 | HCT 116 | C623(1.01); C390(1.14); C466(1.16); C235(1.27) | LDD0665 | [16] |
LDCM0349 | AC83 | HCT 116 | C466(0.69); C623(0.78); C235(0.80); C390(0.85) | LDD0666 | [16] |
LDCM0350 | AC84 | HCT 116 | C466(0.70); C623(0.76); C235(0.81); C248(0.89) | LDD0667 | [16] |
LDCM0351 | AC85 | HCT 116 | C466(0.67); C623(0.77); C235(0.85); C284(0.91) | LDD0668 | [16] |
LDCM0352 | AC86 | HCT 116 | C466(0.72); C888(0.82); C248(0.86); C623(0.87) | LDD0669 | [16] |
LDCM0353 | AC87 | HCT 116 | C888(0.76); C623(0.80); C284(0.85); C466(0.96) | LDD0670 | [16] |
LDCM0354 | AC88 | HCT 116 | C623(0.79); C888(0.88); C235(0.89); C284(0.90) | LDD0671 | [16] |
LDCM0355 | AC89 | HCT 116 | C623(0.67); C466(0.74); C390(0.80); C235(0.81) | LDD0672 | [16] |
LDCM0357 | AC90 | HCT 116 | C888(0.57); C623(0.73); C466(0.88); C102(1.00) | LDD0674 | [16] |
LDCM0358 | AC91 | HCT 116 | C623(0.68); C466(0.71); C235(0.87); C390(0.93) | LDD0675 | [16] |
LDCM0359 | AC92 | HCT 116 | C623(0.75); C235(0.84); C390(0.86); C888(0.93) | LDD0676 | [16] |
LDCM0360 | AC93 | HCT 116 | C466(0.71); C888(0.85); C235(0.86); C284(0.88) | LDD0677 | [16] |
LDCM0361 | AC94 | HCT 116 | C623(0.69); C466(0.69); C284(0.81); C248(0.92) | LDD0678 | [16] |
LDCM0362 | AC95 | HCT 116 | C284(0.68); C466(0.76); C235(0.79); C888(0.79) | LDD0679 | [16] |
LDCM0363 | AC96 | HCT 116 | C623(0.61); C466(0.76); C284(0.84); C888(0.88) | LDD0680 | [16] |
LDCM0364 | AC97 | HCT 116 | C466(0.68); C235(0.80); C623(0.80); C390(0.83) | LDD0681 | [16] |
LDCM0365 | AC98 | HCT 116 | C623(0.57); C248(0.70); C466(0.75); C284(0.84) | LDD0682 | [16] |
LDCM0366 | AC99 | HCT 116 | C623(0.74); C102(0.76); C284(0.84); C248(0.92) | LDD0683 | [16] |
LDCM0545 | Acetamide | MDA-MB-231 | C877(0.40); C235(0.37); C390(0.57); C143(0.45) | LDD2138 | [8] |
LDCM0520 | AKOS000195272 | MDA-MB-231 | C684(0.85); C235(1.20); C390(0.99); C143(0.93) | LDD2113 | [8] |
LDCM0248 | AKOS034007472 | HCT 116 | C102(0.99); C235(1.17); C248(0.98); C284(0.95) | LDD0565 | [16] |
LDCM0356 | AKOS034007680 | HCT 116 | C248(0.88); C466(0.88); C390(0.90); C284(0.94) | LDD0673 | [16] |
LDCM0275 | AKOS034007705 | HCT 116 | C235(0.81); C390(0.88); C248(0.92); C466(1.02) | LDD0592 | [16] |
LDCM0156 | Aniline | NCI-H1299 | C888(0.00); C684(0.00) | LDD0404 | [1] |
LDCM0020 | ARS-1620 | HCC44 | C888(1.24); C623(0.98) | LDD0078 | [16] |
LDCM0498 | BS-3668 | MDA-MB-231 | C877(0.57); C235(0.78); C390(0.68); C143(0.53) | LDD2091 | [8] |
LDCM0630 | CCW28-3 | 231MFP | C684(1.50) | LDD2214 | [36] |
LDCM0108 | Chloroacetamide | HeLa | H868(0.00); C102(0.00); C235(0.00); C623(0.00) | LDD0222 | [29] |
LDCM0632 | CL-Sc | Hep-G2 | C616(20.00); C466(4.18); C102(3.60); C616(2.14) | LDD2227 | [22] |
LDCM0367 | CL1 | HCT 116 | C623(0.92); C102(0.96); C390(0.96); C466(0.97) | LDD0684 | [16] |
LDCM0368 | CL10 | HCT 116 | C888(0.89); C466(0.89); C235(0.94); C102(0.96) | LDD0685 | [16] |
LDCM0369 | CL100 | HCT 116 | C888(0.58); C390(0.84); C248(0.91); C466(0.93) | LDD0686 | [16] |
LDCM0370 | CL101 | HCT 116 | C248(0.83); C284(0.87); C390(0.87); C466(0.88) | LDD0687 | [16] |
LDCM0371 | CL102 | HCT 116 | C248(0.88); C390(0.92); C466(0.93); C102(0.94) | LDD0688 | [16] |
LDCM0372 | CL103 | HCT 116 | C623(0.81); C390(0.83); C284(0.90); C102(0.92) | LDD0689 | [16] |
LDCM0373 | CL104 | HCT 116 | C623(0.83); C248(0.88); C102(0.92); C390(0.92) | LDD0690 | [16] |
LDCM0374 | CL105 | HCT 116 | C888(0.88); C248(0.89); C235(0.97); C466(0.99) | LDD0691 | [16] |
LDCM0375 | CL106 | HCT 116 | C248(0.96); C888(1.05); C466(1.11); C284(1.12) | LDD0692 | [16] |
LDCM0376 | CL107 | HCT 116 | C248(0.94); C235(1.02); C888(1.03); C466(1.07) | LDD0693 | [16] |
LDCM0377 | CL108 | HCT 116 | C248(0.97); C888(1.06); C466(1.14); C284(1.16) | LDD0694 | [16] |
LDCM0378 | CL109 | HCT 116 | C248(0.86); C235(0.89); C623(0.93); C102(0.94) | LDD0695 | [16] |
LDCM0379 | CL11 | HCT 116 | C102(1.07); C390(1.09); C466(1.14); C248(1.16) | LDD0696 | [16] |
LDCM0380 | CL110 | HCT 116 | C888(0.84); C248(0.85); C235(0.89); C284(1.02) | LDD0697 | [16] |
LDCM0381 | CL111 | HCT 116 | C623(0.85); C248(0.88); C888(0.93); C102(0.97) | LDD0698 | [16] |
LDCM0382 | CL112 | HCT 116 | C390(0.85); C102(0.96); C248(0.96); C888(0.97) | LDD0699 | [16] |
LDCM0383 | CL113 | HCT 116 | C390(0.79); C235(0.80); C248(0.92); C466(0.98) | LDD0700 | [16] |
LDCM0384 | CL114 | HCT 116 | C235(0.78); C390(0.80); C102(0.85); C248(0.87) | LDD0701 | [16] |
LDCM0385 | CL115 | HCT 116 | C235(0.76); C390(0.79); C248(0.81); C466(0.85) | LDD0702 | [16] |
LDCM0386 | CL116 | HCT 116 | C235(0.76); C390(0.78); C248(0.83); C466(0.86) | LDD0703 | [16] |
LDCM0387 | CL117 | HCT 116 | C235(1.00); C248(1.08); C888(1.27); C466(1.27) | LDD0704 | [16] |
LDCM0388 | CL118 | HCT 116 | C888(0.87); C390(0.88); C235(0.93); C248(0.96) | LDD0705 | [16] |
LDCM0389 | CL119 | HCT 116 | C390(0.90); C235(0.93); C888(0.97); C248(0.99) | LDD0706 | [16] |
LDCM0390 | CL12 | HCT 116 | C390(1.00); C466(1.03); C248(1.10); C102(1.11) | LDD0707 | [16] |
LDCM0391 | CL120 | HCT 116 | C888(0.72); C390(0.83); C248(0.95); C102(0.99) | LDD0708 | [16] |
LDCM0392 | CL121 | HCT 116 | C888(0.92); C248(0.98); C284(1.03); C466(1.04) | LDD0709 | [16] |
LDCM0393 | CL122 | HCT 116 | C623(0.82); C102(0.96); C248(0.96); C284(0.98) | LDD0710 | [16] |
LDCM0394 | CL123 | HCT 116 | C623(0.78); C390(0.97); C466(0.99); C102(1.01) | LDD0711 | [16] |
LDCM0395 | CL124 | HCT 116 | C235(0.97); C623(0.99); C248(0.99); C466(0.99) | LDD0712 | [16] |
LDCM0396 | CL125 | HCT 116 | C888(0.87); C235(0.94); C248(0.96); C390(0.97) | LDD0713 | [16] |
LDCM0397 | CL126 | HCT 116 | C102(0.87); C248(0.89); C390(0.91); C235(0.96) | LDD0714 | [16] |
LDCM0398 | CL127 | HCT 116 | C248(0.90); C102(0.92); C235(0.94); C390(0.95) | LDD0715 | [16] |
LDCM0399 | CL128 | HCT 116 | C248(0.86); C390(0.88); C235(0.94); C888(0.99) | LDD0716 | [16] |
LDCM0400 | CL13 | HCT 116 | C390(0.95); C248(0.96); C102(1.00); C284(1.01) | LDD0717 | [16] |
LDCM0401 | CL14 | HCT 116 | C102(0.82); C466(0.88); C235(0.91); C284(0.92) | LDD0718 | [16] |
LDCM0402 | CL15 | HCT 116 | C888(0.88); C284(0.89); C102(0.90); C466(0.91) | LDD0719 | [16] |
LDCM0403 | CL16 | HCT 116 | C390(0.86); C284(0.88); C102(0.88); C235(0.92) | LDD0720 | [16] |
LDCM0404 | CL17 | HCT 116 | C284(0.80); C102(0.88); C235(0.91); C248(0.94) | LDD0721 | [16] |
LDCM0405 | CL18 | HCT 116 | C102(0.81); C235(0.82); C284(0.84); C248(0.85) | LDD0722 | [16] |
LDCM0406 | CL19 | HCT 116 | C390(0.84); C466(0.87); C235(0.92); C248(0.92) | LDD0723 | [16] |
LDCM0407 | CL2 | HCT 116 | C390(0.89); C466(0.91); C888(0.92); C102(0.97) | LDD0724 | [16] |
LDCM0408 | CL20 | HCT 116 | C235(0.77); C390(0.84); C248(0.88); C284(0.89) | LDD0725 | [16] |
LDCM0409 | CL21 | HCT 116 | C235(0.81); C284(0.84); C466(0.91); C248(0.97) | LDD0726 | [16] |
LDCM0410 | CL22 | HCT 116 | C235(0.97); C390(0.99); C248(1.10); C466(1.12) | LDD0727 | [16] |
LDCM0411 | CL23 | HCT 116 | C235(0.86); C390(0.93); C248(0.94); C466(0.97) | LDD0728 | [16] |
LDCM0412 | CL24 | HCT 116 | C235(0.94); C390(0.96); C466(1.01); C248(1.06) | LDD0729 | [16] |
LDCM0413 | CL25 | HCT 116 | C102(1.09); C235(0.97); C248(0.98); C284(1.20) | LDD0730 | [16] |
LDCM0414 | CL26 | HCT 116 | C102(0.95); C235(0.84); C248(0.99); C284(0.91) | LDD0731 | [16] |
LDCM0415 | CL27 | HCT 116 | C102(0.96); C235(0.88); C248(0.91); C284(0.96) | LDD0732 | [16] |
LDCM0416 | CL28 | HCT 116 | C102(0.95); C235(0.85); C248(0.92); C284(0.94) | LDD0733 | [16] |
LDCM0417 | CL29 | HCT 116 | C102(0.95); C235(0.83); C248(0.88); C284(0.85) | LDD0734 | [16] |
LDCM0418 | CL3 | HCT 116 | C102(0.91); C235(0.95); C248(1.10); C284(0.94) | LDD0735 | [16] |
LDCM0419 | CL30 | HCT 116 | C102(0.91); C235(1.11); C248(1.00); C284(1.15) | LDD0736 | [16] |
LDCM0420 | CL31 | HCT 116 | C102(0.92); C235(0.98); C248(0.84); C284(1.01) | LDD0737 | [16] |
LDCM0421 | CL32 | HCT 116 | C102(0.86); C235(0.93); C248(0.77); C284(0.91) | LDD0738 | [16] |
LDCM0422 | CL33 | HCT 116 | C102(0.75); C235(0.77); C248(0.68); C284(0.80) | LDD0739 | [16] |
LDCM0423 | CL34 | HCT 116 | C102(1.10); C235(1.07); C248(0.78); C284(0.88) | LDD0740 | [16] |
LDCM0424 | CL35 | HCT 116 | C102(1.04); C235(0.88); C248(0.83); C284(0.93) | LDD0741 | [16] |
LDCM0425 | CL36 | HCT 116 | C102(1.03); C235(0.87); C248(0.74); C284(0.94) | LDD0742 | [16] |
LDCM0426 | CL37 | HCT 116 | C102(1.06); C235(0.84); C248(0.81); C284(0.88) | LDD0743 | [16] |
LDCM0428 | CL39 | HCT 116 | C102(1.01); C235(0.89); C248(0.84); C284(0.92) | LDD0745 | [16] |
LDCM0429 | CL4 | HCT 116 | C102(0.96); C235(0.89); C248(1.03); C284(0.95) | LDD0746 | [16] |
LDCM0430 | CL40 | HCT 116 | C102(1.03); C235(0.89); C248(0.83); C284(0.85) | LDD0747 | [16] |
LDCM0431 | CL41 | HCT 116 | C102(0.97); C235(0.90); C248(0.74); C284(0.95) | LDD0748 | [16] |
LDCM0432 | CL42 | HCT 116 | C102(1.31); C235(0.96); C248(1.01); C284(1.05) | LDD0749 | [16] |
LDCM0433 | CL43 | HCT 116 | C102(1.06); C235(0.93); C248(0.82); C284(1.03) | LDD0750 | [16] |
LDCM0434 | CL44 | HCT 116 | C102(0.93); C235(0.86); C248(0.77); C284(0.85) | LDD0751 | [16] |
LDCM0435 | CL45 | HCT 116 | C102(1.00); C235(0.92); C248(0.84); C284(0.96) | LDD0752 | [16] |
LDCM0436 | CL46 | HCT 116 | C102(0.91); C235(0.85); C248(1.00); C284(1.07) | LDD0753 | [16] |
LDCM0437 | CL47 | HCT 116 | C102(0.99); C235(0.80); C248(0.99); C284(1.15) | LDD0754 | [16] |
LDCM0438 | CL48 | HCT 116 | C102(0.92); C235(0.98); C248(1.04); C284(1.05) | LDD0755 | [16] |
LDCM0439 | CL49 | HCT 116 | C102(0.99); C235(0.91); C248(1.02); C284(0.95) | LDD0756 | [16] |
LDCM0440 | CL5 | HCT 116 | C102(1.04); C235(0.88); C248(1.10); C284(1.04) | LDD0757 | [16] |
LDCM0441 | CL50 | HCT 116 | C102(0.88); C235(0.87); C248(0.97); C284(0.96) | LDD0758 | [16] |
LDCM0442 | CL51 | HCT 116 | C102(0.99); C235(0.95); C248(0.99); C284(1.01) | LDD0759 | [16] |
LDCM0443 | CL52 | HCT 116 | C102(0.86); C235(0.92); C248(0.98); C284(1.04) | LDD0760 | [16] |
LDCM0444 | CL53 | HCT 116 | C102(0.92); C235(0.80); C248(0.92); C284(0.92) | LDD0761 | [16] |
LDCM0445 | CL54 | HCT 116 | C102(0.95); C235(0.93); C248(1.02); C284(0.96) | LDD0762 | [16] |
LDCM0446 | CL55 | HCT 116 | C102(0.95); C235(0.98); C248(1.10); C284(0.95) | LDD0763 | [16] |
LDCM0447 | CL56 | HCT 116 | C102(1.00); C235(0.90); C248(0.99); C284(0.97) | LDD0764 | [16] |
LDCM0448 | CL57 | HCT 116 | C102(0.91); C235(0.89); C248(0.94); C284(0.90) | LDD0765 | [16] |
LDCM0449 | CL58 | HCT 116 | C102(0.96); C235(0.94); C248(1.00); C284(1.06) | LDD0766 | [16] |
LDCM0450 | CL59 | HCT 116 | C102(0.99); C235(0.89); C248(0.98); C284(0.94) | LDD0767 | [16] |
LDCM0451 | CL6 | HCT 116 | C102(0.81); C235(0.92); C248(0.94); C284(0.83) | LDD0768 | [16] |
LDCM0452 | CL60 | HCT 116 | C102(0.92); C235(0.92); C248(1.06); C284(0.92) | LDD0769 | [16] |
LDCM0453 | CL61 | HCT 116 | C102(0.83); C235(1.03); C248(1.03); C284(0.76) | LDD0770 | [16] |
LDCM0454 | CL62 | HCT 116 | C102(0.87); C235(0.82); C248(1.01); C284(0.84) | LDD0771 | [16] |
LDCM0455 | CL63 | HCT 116 | C102(0.87); C235(0.78); C248(0.90); C284(0.70) | LDD0772 | [16] |
LDCM0456 | CL64 | HCT 116 | C102(0.87); C235(1.09); C248(0.85); C284(0.86) | LDD0773 | [16] |
LDCM0457 | CL65 | HCT 116 | C102(1.01); C235(1.09); C248(1.13); C284(0.94) | LDD0774 | [16] |
LDCM0458 | CL66 | HCT 116 | C102(1.04); C235(0.95); C248(1.04); C284(0.29) | LDD0775 | [16] |
LDCM0459 | CL67 | HCT 116 | C102(1.00); C235(0.96); C248(0.91); C284(0.84) | LDD0776 | [16] |
LDCM0460 | CL68 | HCT 116 | C102(0.91); C235(1.43); C248(0.93); C284(0.72) | LDD0777 | [16] |
LDCM0461 | CL69 | HCT 116 | C102(0.79); C235(0.78); C248(0.85); C284(0.67) | LDD0778 | [16] |
LDCM0462 | CL7 | HCT 116 | C102(1.05); C235(1.16); C248(1.05); C284(1.09) | LDD0779 | [16] |
LDCM0463 | CL70 | HCT 116 | C102(0.95); C235(1.09); C248(1.02); C284(0.89) | LDD0780 | [16] |
LDCM0464 | CL71 | HCT 116 | C102(0.94); C235(0.97); C248(1.01); C284(0.80) | LDD0781 | [16] |
LDCM0465 | CL72 | HCT 116 | C102(0.90); C235(0.96); C248(0.94); C284(0.73) | LDD0782 | [16] |
LDCM0466 | CL73 | HCT 116 | C102(0.91); C235(0.94); C248(0.96); C284(0.83) | LDD0783 | [16] |
LDCM0467 | CL74 | HCT 116 | C102(0.96); C235(0.85); C248(0.93); C284(0.87) | LDD0784 | [16] |
LDCM0469 | CL76 | HCT 116 | C102(0.95); C235(0.88); C248(0.96); C284(0.88) | LDD0786 | [16] |
LDCM0470 | CL77 | HCT 116 | C102(0.97); C235(0.82); C248(0.96); C284(0.87) | LDD0787 | [16] |
LDCM0471 | CL78 | HCT 116 | C102(1.05); C235(0.82); C248(1.00); C284(0.90) | LDD0788 | [16] |
LDCM0472 | CL79 | HCT 116 | C102(1.10); C235(0.77); C248(0.99); C284(0.89) | LDD0789 | [16] |
LDCM0473 | CL8 | HCT 116 | C102(0.94); C235(0.84); C248(1.03); C284(1.05) | LDD0790 | [16] |
LDCM0474 | CL80 | HCT 116 | C102(0.93); C235(0.93); C248(0.91); C284(0.86) | LDD0791 | [16] |
LDCM0475 | CL81 | HCT 116 | C102(1.05); C235(0.84); C248(0.95); C284(0.83) | LDD0792 | [16] |
LDCM0476 | CL82 | HCT 116 | C102(1.29); C235(1.00); C248(1.10); C284(1.03) | LDD0793 | [16] |
LDCM0477 | CL83 | HCT 116 | C102(1.22); C235(0.87); C248(1.06); C284(0.96) | LDD0794 | [16] |
LDCM0478 | CL84 | HCT 116 | C102(1.51); C235(1.15); C248(1.12); C284(1.23) | LDD0795 | [16] |
LDCM0479 | CL85 | HCT 116 | C102(0.99); C235(0.92); C248(0.98); C284(0.87) | LDD0796 | [16] |
LDCM0480 | CL86 | HCT 116 | C102(1.04); C235(1.06); C248(1.05); C284(0.96) | LDD0797 | [16] |
LDCM0481 | CL87 | HCT 116 | C102(1.10); C235(0.91); C248(0.99); C284(0.93) | LDD0798 | [16] |
LDCM0482 | CL88 | HCT 116 | C102(1.16); C235(0.95); C248(1.05); C284(0.98) | LDD0799 | [16] |
LDCM0483 | CL89 | HCT 116 | C102(1.78); C235(1.00); C248(1.22); C284(1.44) | LDD0800 | [16] |
LDCM0484 | CL9 | HCT 116 | C102(0.96); C235(1.01); C248(1.23); C284(0.97) | LDD0801 | [16] |
LDCM0485 | CL90 | HCT 116 | C102(1.02); C235(0.90); C248(1.02); C284(0.92) | LDD0802 | [16] |
LDCM0486 | CL91 | HCT 116 | C102(0.90); C235(0.91); C248(0.91); C284(0.94) | LDD0803 | [16] |
LDCM0487 | CL92 | HCT 116 | C102(1.03); C235(0.91); C248(0.90); C284(0.90) | LDD0804 | [16] |
LDCM0488 | CL93 | HCT 116 | C102(0.99); C235(0.98); C248(0.97); C284(1.06) | LDD0805 | [16] |
LDCM0489 | CL94 | HCT 116 | C102(0.95); C235(0.84); C248(0.80); C284(0.91) | LDD0806 | [16] |
LDCM0490 | CL95 | HCT 116 | C102(0.95); C235(0.85); C248(0.84); C284(0.97) | LDD0807 | [16] |
LDCM0491 | CL96 | HCT 116 | C102(1.02); C235(0.88); C248(0.90); C284(0.94) | LDD0808 | [16] |
LDCM0492 | CL97 | HCT 116 | C102(0.95); C235(0.90); C248(0.86); C284(0.92) | LDD0809 | [16] |
LDCM0493 | CL98 | HCT 116 | C102(0.99); C235(0.91); C248(0.84); C284(1.04) | LDD0810 | [16] |
LDCM0494 | CL99 | HCT 116 | C102(1.04); C235(1.00); C248(0.91); C284(1.16) | LDD0811 | [16] |
LDCM0191 | Compound 21 | HEK-293T | 8.47 | LDD0508 | [32] |
LDCM0190 | Compound 34 | HEK-293T | 10.81 | LDD0510 | [32] |
LDCM0192 | Compound 35 | HEK-293T | 6.04 | LDD0509 | [32] |
LDCM0193 | Compound 36 | HEK-293T | 10.10 | LDD0511 | [32] |
LDCM0634 | CY-0357 | Hep-G2 | C888(1.73); C235(1.13); C623(0.75) | LDD2228 | [22] |
LDCM0495 | E2913 | HEK-293T | C235(0.98); C102(0.94); C888(0.97); C248(0.96) | LDD1698 | [37] |
LDCM0213 | Electrophilic fragment 2 | MDA-MB-231 | C877(14.05); C235(4.70); C390(4.18); C248(3.70) | LDD1702 | [8] |
LDCM0031 | Epigallocatechin gallate | HEK-293T | 7.76 | LDD0183 | [11] |
LDCM0625 | F8 | Ramos | C390(1.25); C623(0.78); C888(1.34); C616(0.94) | LDD2187 | [38] |
LDCM0572 | Fragment10 | Ramos | C390(0.86); C623(0.56); C616(0.98) | LDD2189 | [38] |
LDCM0573 | Fragment11 | Ramos | C623(11.88); C616(3.80); 0.33; C684(0.12) | LDD2190 | [38] |
LDCM0574 | Fragment12 | Ramos | C390(0.98); C623(0.56); C616(0.48); 1.35 | LDD2191 | [38] |
LDCM0575 | Fragment13 | Ramos | C390(0.95); C623(0.57); C616(0.66); C684(1.32) | LDD2192 | [38] |
LDCM0576 | Fragment14 | Ramos | C390(2.75); C102(0.48); C623(0.91); C888(1.59) | LDD2193 | [38] |
LDCM0579 | Fragment20 | Ramos | C390(1.15); C623(0.62); C616(0.49); 1.15 | LDD2194 | [38] |
LDCM0580 | Fragment21 | Ramos | C390(1.08); C623(0.62); C616(0.46); 1.62 | LDD2195 | [38] |
LDCM0582 | Fragment23 | Ramos | C390(0.68); C623(1.11); C684(0.31) | LDD2196 | [38] |
LDCM0578 | Fragment27 | Ramos | C390(0.85); C623(0.61); C616(0.88); 2.22 | LDD2197 | [38] |
LDCM0586 | Fragment28 | Ramos | C390(0.48); C623(1.44); C616(0.29); 0.72 | LDD2198 | [38] |
LDCM0588 | Fragment30 | Ramos | C390(1.15); C623(0.72); C616(0.81); 0.81 | LDD2199 | [38] |
LDCM0589 | Fragment31 | Ramos | C390(1.05); C623(0.73); C684(0.84) | LDD2200 | [38] |
LDCM0590 | Fragment32 | Ramos | C390(0.78); C623(0.42); C616(0.54); 1.29 | LDD2201 | [38] |
LDCM0468 | Fragment33 | HCT 116 | C102(0.88); C235(1.04); C248(0.93); C284(0.72) | LDD0785 | [16] |
LDCM0596 | Fragment38 | Ramos | C390(1.21); C623(0.51); C684(1.09) | LDD2203 | [38] |
LDCM0566 | Fragment4 | Ramos | C390(1.26); C102(0.85); C623(0.88); C888(0.68) | LDD2184 | [38] |
LDCM0427 | Fragment51 | HCT 116 | C102(1.23); C235(0.97); C248(0.98); C284(1.09) | LDD0744 | [16] |
LDCM0610 | Fragment52 | Ramos | C623(0.72) | LDD2204 | [38] |
LDCM0614 | Fragment56 | Ramos | C390(1.06); C623(0.65); C616(0.69); C684(0.61) | LDD2205 | [38] |
LDCM0569 | Fragment7 | Ramos | C390(1.33); C102(0.82); C623(0.93); C888(1.05) | LDD2186 | [38] |
LDCM0571 | Fragment9 | Ramos | C390(0.92); C623(0.51); C616(0.43); C684(1.13) | LDD2188 | [38] |
LDCM0116 | HHS-0101 | DM93 | Y887(0.77); Y521(0.84); Y160(0.95) | LDD0264 | [14] |
LDCM0117 | HHS-0201 | DM93 | Y887(0.73); Y521(0.78); Y160(0.89) | LDD0265 | [14] |
LDCM0118 | HHS-0301 | DM93 | Y887(0.39); Y521(0.80); Y160(1.00) | LDD0266 | [14] |
LDCM0119 | HHS-0401 | DM93 | Y887(0.79); Y521(0.84); Y160(1.19) | LDD0267 | [14] |
LDCM0120 | HHS-0701 | DM93 | Y887(0.66); Y521(0.71); Y160(0.99) | LDD0268 | [14] |
LDCM0107 | IAA | HeLa | C623(0.00); H373(0.00); C616(0.00); C390(0.00) | LDD0221 | [29] |
LDCM0123 | JWB131 | DM93 | Y521(1.02) | LDD0285 | [13] |
LDCM0124 | JWB142 | DM93 | Y521(0.69) | LDD0286 | [13] |
LDCM0125 | JWB146 | DM93 | Y521(1.03) | LDD0287 | [13] |
LDCM0126 | JWB150 | DM93 | Y521(2.98) | LDD0288 | [13] |
LDCM0127 | JWB152 | DM93 | Y521(2.17) | LDD0289 | [13] |
LDCM0128 | JWB198 | DM93 | Y521(0.86) | LDD0290 | [13] |
LDCM0129 | JWB202 | DM93 | Y521(0.54) | LDD0291 | [13] |
LDCM0130 | JWB211 | DM93 | Y521(0.89) | LDD0292 | [13] |
LDCM0179 | JZ128 | PC-3 | N.A. | LDD0462 | [10] |
LDCM0022 | KB02 | HCT 116 | C248(2.06); C466(1.96); C102(1.63); C390(1.51) | LDD0080 | [16] |
LDCM0023 | KB03 | HCT 116 | C248(4.86); C466(3.06); C102(2.82); C390(2.98) | LDD0081 | [16] |
LDCM0024 | KB05 | HCT 116 | C248(4.64); C466(3.30); C102(2.62); C390(2.17) | LDD0082 | [16] |
LDCM0509 | N-(4-bromo-3,5-dimethylphenyl)-2-nitroacetamide | MDA-MB-231 | C684(0.87); C235(0.95); C390(1.57); C143(1.41) | LDD2102 | [8] |
LDCM0528 | N-(4-bromophenyl)-2-cyano-N-phenylacetamide | MDA-MB-231 | C684(0.67); C877(0.58); C235(0.65); C390(0.90) | LDD2121 | [8] |
LDCM0109 | NEM | HeLa | H199(0.00); H373(0.00); H926(0.00) | LDD0223 | [29] |
LDCM0496 | Nucleophilic fragment 11a | MDA-MB-231 | C684(0.74); C235(0.54); C390(0.99); C143(0.67) | LDD2089 | [8] |
LDCM0497 | Nucleophilic fragment 11b | MDA-MB-231 | C684(1.04); C390(1.16) | LDD2090 | [8] |
LDCM0499 | Nucleophilic fragment 12b | MDA-MB-231 | C684(0.67); C235(0.73); C390(1.14); C143(1.58) | LDD2092 | [8] |
LDCM0500 | Nucleophilic fragment 13a | MDA-MB-231 | C684(0.91); C235(0.66); C390(1.35); C143(1.29) | LDD2093 | [8] |
LDCM0501 | Nucleophilic fragment 13b | MDA-MB-231 | C684(1.37); C235(0.93); C390(2.19); C143(2.40) | LDD2094 | [8] |
LDCM0503 | Nucleophilic fragment 14b | MDA-MB-231 | C684(1.40); C877(0.18); C235(1.80); C390(0.17) | LDD2096 | [8] |
LDCM0504 | Nucleophilic fragment 15a | MDA-MB-231 | C235(1.82); C390(1.02); C143(1.38) | LDD2097 | [8] |
LDCM0505 | Nucleophilic fragment 15b | MDA-MB-231 | C684(0.72); C235(0.94); C390(0.83); C143(1.23) | LDD2098 | [8] |
LDCM0506 | Nucleophilic fragment 16a | MDA-MB-231 | C684(1.01); C235(1.24); C390(1.42); C143(1.42) | LDD2099 | [8] |
LDCM0507 | Nucleophilic fragment 16b | MDA-MB-231 | C684(1.10); C235(0.99); C390(0.34); C143(0.96) | LDD2100 | [8] |
LDCM0508 | Nucleophilic fragment 17a | MDA-MB-231 | C684(0.81); C235(0.72); C390(1.40); C143(0.93) | LDD2101 | [8] |
LDCM0511 | Nucleophilic fragment 18b | MDA-MB-231 | C684(1.06); C143(0.57) | LDD2104 | [8] |
LDCM0512 | Nucleophilic fragment 19a | MDA-MB-231 | C684(1.20); C877(4.24); C235(0.88); C390(1.39) | LDD2105 | [8] |
LDCM0513 | Nucleophilic fragment 19b | MDA-MB-231 | C684(1.17); C390(0.63); C143(0.63); C623(0.55) | LDD2106 | [8] |
LDCM0514 | Nucleophilic fragment 20a | MDA-MB-231 | C684(1.07); C235(1.02); C390(1.10); C143(0.99) | LDD2107 | [8] |
LDCM0515 | Nucleophilic fragment 20b | MDA-MB-231 | C684(0.79); C877(1.01); C235(0.85); C390(0.50) | LDD2108 | [8] |
LDCM0516 | Nucleophilic fragment 21a | MDA-MB-231 | C684(0.82); C877(1.38); C235(0.33); C390(0.60) | LDD2109 | [8] |
LDCM0517 | Nucleophilic fragment 21b | MDA-MB-231 | C684(2.24); C390(1.00) | LDD2110 | [8] |
LDCM0518 | Nucleophilic fragment 22a | MDA-MB-231 | C684(1.37); C235(0.93); C390(1.39); C143(1.02) | LDD2111 | [8] |
LDCM0521 | Nucleophilic fragment 23b | MDA-MB-231 | C877(1.28); C235(0.87); C390(0.97); C143(1.16) | LDD2114 | [8] |
LDCM0522 | Nucleophilic fragment 24a | MDA-MB-231 | C684(0.51); C235(0.38); C390(0.58); C143(0.61) | LDD2115 | [8] |
LDCM0523 | Nucleophilic fragment 24b | MDA-MB-231 | C684(1.48); C877(0.38); C143(0.62) | LDD2116 | [8] |
LDCM0525 | Nucleophilic fragment 25b | MDA-MB-231 | C684(1.88); C877(0.30); C390(0.32); C143(0.62) | LDD2118 | [8] |
LDCM0526 | Nucleophilic fragment 26a | MDA-MB-231 | C684(2.51); C235(1.26); C390(1.94); C143(1.96) | LDD2119 | [8] |
LDCM0527 | Nucleophilic fragment 26b | MDA-MB-231 | C684(0.82); C877(1.12); C235(0.55); C390(0.69) | LDD2120 | [8] |
LDCM0529 | Nucleophilic fragment 27b | MDA-MB-231 | C684(1.66); C877(0.28); C235(2.27); C143(0.49) | LDD2122 | [8] |
LDCM0530 | Nucleophilic fragment 28a | MDA-MB-231 | C684(0.86); C877(0.81); C235(0.64); C390(0.90) | LDD2123 | [8] |
LDCM0531 | Nucleophilic fragment 28b | MDA-MB-231 | C684(1.44); C877(0.29); C235(2.20); C143(0.44) | LDD2124 | [8] |
LDCM0532 | Nucleophilic fragment 29a | MDA-MB-231 | C684(1.00); C877(0.42); C235(0.59); C390(0.94) | LDD2125 | [8] |
LDCM0533 | Nucleophilic fragment 29b | MDA-MB-231 | C684(1.51); C877(0.42); C390(0.13); C143(0.49) | LDD2126 | [8] |
LDCM0534 | Nucleophilic fragment 30a | MDA-MB-231 | C684(1.27); C877(1.34); C235(0.95); C390(1.23) | LDD2127 | [8] |
LDCM0535 | Nucleophilic fragment 30b | MDA-MB-231 | C684(0.91); C235(1.06); C390(0.91); C143(0.56) | LDD2128 | [8] |
LDCM0536 | Nucleophilic fragment 31 | MDA-MB-231 | C684(0.85); C235(0.85); C390(1.50); C143(1.15) | LDD2129 | [8] |
LDCM0540 | Nucleophilic fragment 35 | MDA-MB-231 | C684(0.52); C235(0.59); C390(0.78); C143(0.63) | LDD2133 | [8] |
LDCM0541 | Nucleophilic fragment 36 | MDA-MB-231 | C684(0.40); C235(0.77); C390(0.48); C143(0.66) | LDD2134 | [8] |
LDCM0542 | Nucleophilic fragment 37 | MDA-MB-231 | C684(0.77); C235(1.23); C390(1.99); C143(1.58) | LDD2135 | [8] |
LDCM0543 | Nucleophilic fragment 38 | MDA-MB-231 | C684(1.28); C235(0.97); C390(1.70); C143(1.43) | LDD2136 | [8] |
LDCM0544 | Nucleophilic fragment 39 | MDA-MB-231 | C684(1.06); C235(0.83); C390(0.96); C143(1.11) | LDD2137 | [8] |
LDCM0211 | Nucleophilic fragment 3b | MDA-MB-231 | C390(4.10); C143(3.83); C235(2.42); C684(2.06) | LDD1700 | [8] |
LDCM0546 | Nucleophilic fragment 40 | MDA-MB-231 | C684(0.95); C877(0.88); C235(0.73); C390(0.95) | LDD2140 | [8] |
LDCM0547 | Nucleophilic fragment 41 | MDA-MB-231 | C684(0.82); C877(0.96); C235(0.99); C143(0.75) | LDD2141 | [8] |
LDCM0549 | Nucleophilic fragment 43 | MDA-MB-231 | C684(1.07); C877(0.52); C235(0.59); C390(0.56) | LDD2143 | [8] |
LDCM0550 | Nucleophilic fragment 5a | MDA-MB-231 | C684(2.95); C235(1.75); C390(1.91); C143(2.14) | LDD2144 | [8] |
LDCM0551 | Nucleophilic fragment 5b | MDA-MB-231 | C684(9.41); C390(1.25) | LDD2145 | [8] |
LDCM0552 | Nucleophilic fragment 6a | MDA-MB-231 | C684(1.00); C877(0.50); C235(0.79); C390(1.14) | LDD2146 | [8] |
LDCM0553 | Nucleophilic fragment 6b | MDA-MB-231 | C684(3.21); C390(1.91); C143(1.56) | LDD2147 | [8] |
LDCM0554 | Nucleophilic fragment 7a | MDA-MB-231 | C684(0.50); C235(0.39); C390(0.47) | LDD2148 | [8] |
LDCM0555 | Nucleophilic fragment 7b | MDA-MB-231 | C684(2.27); C877(0.31); C390(0.06); C143(0.50) | LDD2149 | [8] |
LDCM0556 | Nucleophilic fragment 8a | MDA-MB-231 | C877(0.35); C235(0.58); C390(0.60); C143(0.38) | LDD2150 | [8] |
LDCM0557 | Nucleophilic fragment 8b | MDA-MB-231 | C684(4.53); C877(0.39); C390(0.21); C143(0.51) | LDD2151 | [8] |
LDCM0559 | Nucleophilic fragment 9b | MDA-MB-231 | C684(1.22); C877(4.92); C390(1.50); C143(2.56) | LDD2153 | [8] |
LDCM0627 | NUDT7-COV-1 | HEK-293T | C888(1.13) | LDD2206 | [39] |
LDCM0628 | OTUB2-COV-1 | HEK-293T | C684(1.32); C888(0.78) | LDD2207 | [39] |
LDCM0131 | RA190 | MM1.R | C888(1.06) | LDD0304 | [40] |
LDCM0090 | Rapamycin | JHH-7 | 3.42 | LDD0213 | [34] |
LDCM0021 | THZ1 | HCT 116 | C888(1.30); C235(1.01); C248(1.06) | LDD2173 | [16] |
LDCM0111 | W14 | Hep-G2 | C623(6.92) | LDD0238 | [30] |
The Interaction Atlas With This Target
The Protein(s) Related To This Target
Enzyme
Protein name | Family | Uniprot ID | |||
---|---|---|---|---|---|
GTP-binding protein 4 (GTPBP4) | OBG GTPase family | Q9BZE4 | |||
E3 ubiquitin-protein ligase TRIM37 (TRIM37) | TRIM/RBCC family | O94972 |
Transporter and channel
Other
References