Details of the Target

General Information of Target

Target ID LDTP04571
Target Name Coatomer subunit alpha (COPA)
Gene Name COPA
Gene ID 1314
Synonyms
Coatomer subunit alpha; Alpha-coat protein; Alpha-COP; HEP-COP; HEPCOP) [Cleaved into: Xenin; Xenopsin-related peptide; Proxenin]
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MLTKFETKSARVKGLSFHPKRPWILTSLHNGVIQLWDYRMCTLIDKFDEHDGPVRGIDFH
KQQPLFVSGGDDYKIKVWNYKLRRCLFTLLGHLDYIRTTFFHHEYPWILSASDDQTIRVW
NWQSRTCVCVLTGHNHYVMCAQFHPTEDLVVSASLDQTVRVWDISGLRKKNLSPGAVESD
VRGITGVDLFGTTDAVVKHVLEGHDRGVNWAAFHPTMPLIVSGADDRQVKIWRMNESKAW
EVDTCRGHYNNVSCAVFHPRQELILSNSEDKSIRVWDMSKRTGVQTFRRDHDRFWVLAAH
PNLNLFAAGHDGGMIVFKLERERPAYAVHGNMLHYVKDRFLRQLDFNSSKDVAVMQLRSG
SKFPVFNMSYNPAENAVLLCTRASNLENSTYDLYTIPKDADSQNPDAPEGKRSSGLTAVW
VARNRFAVLDRMHSLLIKNLKNEITKKVQVPNCDEIFYAGTGNLLLRDADSITLFDVQQK
RTLASVKISKVKYVIWSADMSHVALLAKHAIVICNRKLDALCNIHENIRVKSGAWDESGV
FIYTTSNHIKYAVTTGDHGIIRTLDLPIYVTRVKGNNVYCLDRECRPRVLTIDPTEFKFK
LALINRKYDEVLHMVRNAKLVGQSIIAYLQKKGYPEVALHFVKDEKTRFSLALECGNIEI
ALEAAKALDDKNCWEKLGEVALLQGNHQIVEMCYQRTKNFDKLSFLYLITGNLEKLRKMM
KIAEIRKDMSGHYQNALYLGDVSERVRILKNCGQKSLAYLTAATHGLDEEAESLKETFDP
EKETIPDIDPNAKLLQPPAPIMPLDTNWPLLTVSKGFFEGTIASKGKGGALAADIDIDTV
GTEGWGEDAELQLDEDGFVEATEGLGDDALGKGQEEGGGWDVEEDLELPPELDISPGAAG
GAEDGFFVPPTKGTSPTQIWCNNSQLPVDHILAGSFETAMRLLHDQVGVIQFGPYKQLFL
QTYARGRTTYQALPCLPSMYGYPNRNWKDAGLKNGVPAVGLKLNDLIQRLQLCYQLTTVG
KFEEAVEKFRSILLSVPLLVVDNKQEIAEAQQLITICREYIVGLSVETERKKLPKETLEQ
QKRICEMAAYFTHSNLQPVHMILVLRTALNLFFKLKNFKTAATFARRLLELGPKPEVAQQ
TRKILSACEKNPTDAYQLNYDMHNPFDICAASYRPIYRGKPVEKCPLSGACYSPEFKGQI
CRVTTVTEIGKDVIGLRISPLQFR
Target Bioclass
Other
Subcellular location
Cytoplasm; Secreted
Function
The coatomer is a cytosolic protein complex that binds to dilysine motifs and reversibly associates with Golgi non-clathrin-coated vesicles, which further mediate biosynthetic protein transport from the ER, via the Golgi up to the trans Golgi network. Coatomer complex is required for budding from Golgi membranes, and is essential for the retrograde Golgi-to-ER transport of dilysine-tagged proteins. In mammals, the coatomer can only be recruited by membranes associated to ADP-ribosylation factors (ARFs), which are small GTP-binding proteins; the complex also influences the Golgi structural integrity, as well as the processing, activity, and endocytic recycling of LDL receptors.; Xenin stimulates exocrine pancreatic secretion. It inhibits pentagastrin-stimulated secretion of acid, to induce exocrine pancreatic secretion and to affect small and large intestinal motility. In the gut, xenin interacts with the neurotensin receptor.
Uniprot ID
P53621
Ensemble ID
ENST00000241704.8
HGNC ID
HGNC:2230

Target Site Mutations in Different Cell Lines

Cell line Mutation details Probe for labeling this protein in this cell
A431 SNV: p.T784I DBIA    Probe Info 
CHL1 SNV: p.H502R DBIA    Probe Info 
DANG SNV: p.F541I DBIA    Probe Info 
DOTC24510 SNV: p.D430H DBIA    Probe Info 
GB1 SNV: p.G247S DBIA    Probe Info 
HT115 SNV: p.V200A DBIA    Probe Info 
KPNYN SNV: p.Q1199R DBIA    Probe Info 
KYSE510 SNV: p.R293C DBIA    Probe Info 
MEWO SNV: p.T1055I DBIA    Probe Info 
NCIH1155 SNV: p.A376T DBIA    Probe Info 
NCIH1793 SNV: p.Y458S DBIA    Probe Info 
OCUG1 SNV: p.Q1199R DBIA    Probe Info 
OSRC2 SNV: p.R717L DBIA    Probe Info 
OVK18 SNV: p.R55Ter DBIA    Probe Info 
RL952 SNV: p.D277Y DBIA    Probe Info 
SNGM SNV: p.R55Ter; p.A998D DBIA    Probe Info 
SUPT1 SNV: p.D113N DBIA    Probe Info 

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 47 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
A-EBA
 Probe Info  		3.22  LDD0215  [1]
CY4
 Probe Info  		100.00  LDD0244  [2]
N1
 Probe Info  		100.00  LDD0242  [2]
W1
 Probe Info  		11.56  LDD0235  [3]
TH211
 Probe Info  		Y1160(20.00); Y1177(20.00); Y326(20.00); Y628(20.00)  LDD0257  [4]
TH214
 Probe Info  		Y249(20.00); Y628(19.92)  LDD0258  [4]
TH216
 Probe Info  		Y1156(20.00); Y249(20.00); Y628(20.00); Y733(20.00)  LDD0259  [4]
YN-4
 Probe Info  		100.00  LDD0445  [5]
ONAyne
 Probe Info  		N.A.  LDD0273  [6]
OPA-S-S-alkyne
 Probe Info  		K607(1.94); K1134(2.49); K480(4.64)  LDD3494  [7]
Probe 1
 Probe Info  		Y73(167.26); Y394(9.93); Y579(19.54)  LDD3495  [8]
BTD
 Probe Info  		C673(2.87); C1148(1.43)  LDD1700  [9]
Johansson_61
 Probe Info  		_(20.00)  LDD1490  [10]
AHL-Pu-1
 Probe Info  		C1169(20.00)  LDD0168  [11]
HHS-482
 Probe Info  		Y249(0.84)  LDD0285  [12]
HHS-475
 Probe Info  		Y634(0.05); Y579(0.74); Y608(0.91); Y249(1.00)  LDD0264  [13]
HHS-465
 Probe Info  		Y249(6.42); Y458(1.58); Y579(6.89); Y634(7.34)  LDD2237  [14]
DBIA
 Probe Info  		C245(0.96)  LDD0078  [15]
AMP probe
 Probe Info  		K1134(0.00); K4(0.00)  LDD0200  [16]
ATP probe
 Probe Info  		K1134(0.00); K4(0.00); K531(0.00); K1143(0.00)  LDD0199  [16]
4-Iodoacetamidophenylacetylene
 Probe Info  		C673(0.00); C245(0.00); C85(0.00); C380(0.00)  LDD0038  [17]
IA-alkyne
 Probe Info  		C580(0.00); C975(0.00); C380(0.00); C1185(0.00)  LDD0032  [18]
IPIAA_H
 Probe Info  		N.A.  LDD0030  [19]
IPIAA_L
 Probe Info  		C380(0.00); C522(0.00); C254(0.00); C673(0.00)  LDD0031  [19]
Lodoacetamide azide
 Probe Info  		C673(0.00); C245(0.00); C85(0.00); C380(0.00)  LDD0037  [17]
ATP probe
 Probe Info  		N.A.  LDD0035  [20]
JW-RF-010
 Probe Info  		N.A.  LDD0026  [21]
NAIA_4
 Probe Info  		C41(0.00); C380(0.00); C453(0.00); C522(0.00)  LDD2226  [22]
WYneO
 Probe Info  		N.A.  LDD0022  [23]
1d-yne
 Probe Info  		N.A.  LDD0356  [24]
Compound 10
 Probe Info  		C1185(0.00); C245(0.00)  LDD2216  [25]
IPM
 Probe Info  		C254(0.00); C380(0.00); C975(0.00); C453(0.00)  LDD0147  [21]
NHS
 Probe Info  		K1028(0.00); K825(0.00); K480(0.00)  LDD0010  [23]
PF-06672131
 Probe Info  		N.A.  LDD0017  [26]
SF
 Probe Info  		K631(0.00); Y249(0.00)  LDD0028  [27]
STPyne
 Probe Info  		K1028(0.00); K480(0.00)  LDD0009  [23]
TFBX
 Probe Info  		C453(0.00); C380(0.00); C254(0.00); C1148(0.00)  LDD0148  [21]
VSF
 Probe Info  		N.A.  LDD0007  [23]
Phosphinate-6
 Probe Info  		N.A.  LDD0018  [28]
Ox-W18
 Probe Info  		W295(0.00); W808(0.00)  LDD2175  [29]
1c-yne
 Probe Info  		K607(0.00); K727(0.00); K350(0.00); K619(0.00)  LDD0228  [24]
Acrolein
 Probe Info  		H944(0.00); C1057(0.00); C522(0.00); H558(0.00)  LDD0217  [30]
Cinnamaldehyde
 Probe Info  		N.A.  LDD0220  [30]
Crotonaldehyde
 Probe Info  		N.A.  LDD0219  [30]
Methacrolein
 Probe Info  		C673(0.00); C514(0.00); C245(0.00); C254(0.00)  LDD0218  [30]
m-APA
 Probe Info  		N.A.  LDD0405  [31]
NAIA_5
 Probe Info  		C673(0.00); C245(0.00); C85(0.00); C380(0.00)  LDD2223  [22]
PAL-AfBPP Probe
Click To Hide/Show 4 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
STS-1
 Probe Info  		N.A.  LDD0136  [32]
STS-2
 Probe Info  		N.A.  LDD0138  [32]
Alk-rapa
 Probe Info  		3.48  LDD0213  [33]
DA-2
 Probe Info  		N.A.  LDD0071  [34]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0548  1-(4-(Benzo[d][1,3]dioxol-5-ylmethyl)piperazin-1-yl)-2-nitroethan-1-one MDA-MB-231 C522(0.75); C673(0.53)  LDD2142  [9]
 LDCM0519  1-(6-methoxy-3,4-dihydroquinolin-1(2H)-yl)-2-nitroethan-1-one MDA-MB-231 C673(0.92)  LDD2112  [9]
 LDCM0502  1-(Cyanoacetyl)piperidine MDA-MB-231 C514(0.84); C1148(0.51)  LDD2095  [9]
 LDCM0537  2-Cyano-N,N-dimethylacetamide MDA-MB-231 C522(0.78)  LDD2130  [9]
 LDCM0524  2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide MDA-MB-231 C514(0.97); C1148(0.98); C41(1.52); C673(1.24)  LDD2117  [9]
 LDCM0558  2-Cyano-N-phenylacetamide MDA-MB-231 C1148(1.34); C41(1.93); C522(1.28); C673(1.75)  LDD2152  [9]
 LDCM0510  3-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-3-oxopropanenitrile MDA-MB-231 C1148(0.77); C522(0.92); C1185(0.72)  LDD2103  [9]
 LDCM0539  3-(4-Isopropylpiperazin-1-yl)-3-oxopropanenitrile MDA-MB-231 C673(0.55)  LDD2132  [9]
 LDCM0538  4-(Cyanoacetyl)morpholine MDA-MB-231 C1148(0.63); C41(0.63)  LDD2131  [9]
 LDCM0025  4SU-RNA HEK-293T C1169(20.00)  LDD0168  [11]
 LDCM0026  4SU-RNA+native RNA HEK-293T C1169(4.92)  LDD0169  [11]
 LDCM0214  AC1 HCT 116 C514(1.23)  LDD0531  [15]
 LDCM0215  AC10 HCT 116 C514(1.08)  LDD0532  [15]
 LDCM0216  AC100 HCT 116 C514(1.16)  LDD0533  [15]
 LDCM0217  AC101 HCT 116 C514(1.19)  LDD0534  [15]
 LDCM0218  AC102 HCT 116 C514(1.06)  LDD0535  [15]
 LDCM0219  AC103 HCT 116 C514(1.17)  LDD0536  [15]
 LDCM0220  AC104 HCT 116 C514(1.08)  LDD0537  [15]
 LDCM0221  AC105 HCT 116 C514(0.83)  LDD0538  [15]
 LDCM0222  AC106 HCT 116 C514(0.87)  LDD0539  [15]
 LDCM0223  AC107 HCT 116 C514(0.91)  LDD0540  [15]
 LDCM0224  AC108 HCT 116 C514(0.73)  LDD0541  [15]
 LDCM0225  AC109 HCT 116 C514(0.80)  LDD0542  [15]
 LDCM0226  AC11 HCT 116 C514(1.12)  LDD0543  [15]
 LDCM0227  AC110 HCT 116 C514(0.79)  LDD0544  [15]
 LDCM0228  AC111 HCT 116 C514(1.21)  LDD0545  [15]
 LDCM0229  AC112 HCT 116 C514(0.75)  LDD0546  [15]
 LDCM0230  AC113 HCT 116 C514(1.20)  LDD0547  [15]
 LDCM0231  AC114 HCT 116 C514(1.06)  LDD0548  [15]
 LDCM0232  AC115 HCT 116 C514(1.03)  LDD0549  [15]
 LDCM0233  AC116 HCT 116 C514(1.06)  LDD0550  [15]
 LDCM0234  AC117 HCT 116 C514(1.02)  LDD0551  [15]
 LDCM0235  AC118 HCT 116 C514(1.11)  LDD0552  [15]
 LDCM0236  AC119 HCT 116 C514(1.17)  LDD0553  [15]
 LDCM0237  AC12 HCT 116 C514(0.97)  LDD0554  [15]
 LDCM0238  AC120 HCT 116 C514(1.14)  LDD0555  [15]
 LDCM0239  AC121 HCT 116 C514(1.10)  LDD0556  [15]
 LDCM0240  AC122 HCT 116 C514(1.09)  LDD0557  [15]
 LDCM0241  AC123 HCT 116 C514(1.14)  LDD0558  [15]
 LDCM0242  AC124 HCT 116 C514(1.08)  LDD0559  [15]
 LDCM0243  AC125 HCT 116 C514(1.07)  LDD0560  [15]
 LDCM0244  AC126 HCT 116 C514(1.14)  LDD0561  [15]
 LDCM0245  AC127 HCT 116 C514(1.10)  LDD0562  [15]
 LDCM0246  AC128 HCT 116 C514(1.16)  LDD0563  [15]
 LDCM0247  AC129 HCT 116 C514(1.37)  LDD0564  [15]
 LDCM0249  AC130 HCT 116 C514(1.15)  LDD0566  [15]
 LDCM0250  AC131 HCT 116 C514(1.28)  LDD0567  [15]
 LDCM0251  AC132 HCT 116 C514(1.54)  LDD0568  [15]
 LDCM0252  AC133 HCT 116 C514(1.72)  LDD0569  [15]
 LDCM0253  AC134 HCT 116 C514(1.03)  LDD0570  [15]
 LDCM0254  AC135 HCT 116 C514(1.29)  LDD0571  [15]
 LDCM0255  AC136 HCT 116 C514(1.41)  LDD0572  [15]
 LDCM0256  AC137 HCT 116 C514(1.48)  LDD0573  [15]
 LDCM0257  AC138 HCT 116 C514(0.97)  LDD0574  [15]
 LDCM0258  AC139 HCT 116 C514(1.34)  LDD0575  [15]
 LDCM0259  AC14 HCT 116 C514(1.06)  LDD0576  [15]
 LDCM0260  AC140 HCT 116 C514(1.02)  LDD0577  [15]
 LDCM0261  AC141 HCT 116 C514(1.14)  LDD0578  [15]
 LDCM0262  AC142 HCT 116 C514(1.17)  LDD0579  [15]
 LDCM0263  AC143 HCT 116 C514(1.00)  LDD0580  [15]
 LDCM0264  AC144 HCT 116 C514(0.99)  LDD0581  [15]
 LDCM0265  AC145 HCT 116 C514(0.88)  LDD0582  [15]
 LDCM0266  AC146 HCT 116 C514(1.00)  LDD0583  [15]
 LDCM0267  AC147 HCT 116 C514(0.97)  LDD0584  [15]
 LDCM0268  AC148 HCT 116 C514(1.03)  LDD0585  [15]
 LDCM0269  AC149 HCT 116 C514(0.87)  LDD0586  [15]
 LDCM0270  AC15 HCT 116 C514(1.09)  LDD0587  [15]
 LDCM0271  AC150 HCT 116 C514(0.99)  LDD0588  [15]
 LDCM0272  AC151 HCT 116 C514(1.07)  LDD0589  [15]
 LDCM0273  AC152 HCT 116 C514(0.92)  LDD0590  [15]
 LDCM0274  AC153 HCT 116 C514(0.78)  LDD0591  [15]
 LDCM0621  AC154 HCT 116 C514(0.85)  LDD2158  [15]
 LDCM0622  AC155 HCT 116 C514(0.93)  LDD2159  [15]
 LDCM0623  AC156 HCT 116 C514(0.90)  LDD2160  [15]
 LDCM0624  AC157 HCT 116 C514(0.79)  LDD2161  [15]
 LDCM0276  AC17 HCT 116 C514(1.07)  LDD0593  [15]
 LDCM0277  AC18 HCT 116 C514(1.18)  LDD0594  [15]
 LDCM0278  AC19 HCT 116 C514(1.22)  LDD0595  [15]
 LDCM0279  AC2 HCT 116 C514(1.42)  LDD0596  [15]
 LDCM0280  AC20 HCT 116 C514(1.04)  LDD0597  [15]
 LDCM0281  AC21 HCT 116 C514(1.22)  LDD0598  [15]
 LDCM0282  AC22 HCT 116 C514(1.19)  LDD0599  [15]
 LDCM0283  AC23 HCT 116 C514(1.05)  LDD0600  [15]
 LDCM0284  AC24 HCT 116 C514(1.06)  LDD0601  [15]
 LDCM0285  AC25 HCT 116 C514(1.02)  LDD0602  [15]
 LDCM0286  AC26 HCT 116 C514(1.01)  LDD0603  [15]
 LDCM0287  AC27 HCT 116 C514(1.07)  LDD0604  [15]
 LDCM0288  AC28 HCT 116 C514(1.20)  LDD0605  [15]
 LDCM0289  AC29 HCT 116 C514(1.10)  LDD0606  [15]
 LDCM0290  AC3 HCT 116 C514(1.40)  LDD0607  [15]
 LDCM0291  AC30 HCT 116 C514(0.97)  LDD0608  [15]
 LDCM0292  AC31 HCT 116 C514(1.19)  LDD0609  [15]
 LDCM0293  AC32 HCT 116 C514(0.89)  LDD0610  [15]
 LDCM0294  AC33 HCT 116 C514(0.90)  LDD0611  [15]
 LDCM0295  AC34 HCT 116 C514(0.91)  LDD0612  [15]
 LDCM0296  AC35 HCT 116 C514(1.11)  LDD0613  [15]
 LDCM0297  AC36 HCT 116 C514(1.16)  LDD0614  [15]
 LDCM0298  AC37 HCT 116 C514(1.29)  LDD0615  [15]
 LDCM0299  AC38 HCT 116 C514(1.06)  LDD0616  [15]
 LDCM0300  AC39 HCT 116 C514(1.12)  LDD0617  [15]
 LDCM0301  AC4 HCT 116 C514(1.30)  LDD0618  [15]
 LDCM0302  AC40 HCT 116 C514(1.13)  LDD0619  [15]
 LDCM0303  AC41 HCT 116 C514(1.44)  LDD0620  [15]
 LDCM0304  AC42 HCT 116 C514(1.23)  LDD0621  [15]
 LDCM0305  AC43 HCT 116 C514(1.26)  LDD0622  [15]
 LDCM0306  AC44 HCT 116 C514(1.32)  LDD0623  [15]
 LDCM0307  AC45 HCT 116 C514(1.29)  LDD0624  [15]
 LDCM0308  AC46 HCT 116 C514(1.04)  LDD0625  [15]
 LDCM0309  AC47 HCT 116 C514(0.90)  LDD0626  [15]
 LDCM0310  AC48 HCT 116 C514(0.97)  LDD0627  [15]
 LDCM0311  AC49 HCT 116 C514(0.85)  LDD0628  [15]
 LDCM0312  AC5 HCT 116 C514(1.26)  LDD0629  [15]
 LDCM0313  AC50 HCT 116 C514(0.92)  LDD0630  [15]
 LDCM0314  AC51 HCT 116 C514(0.82)  LDD0631  [15]
 LDCM0315  AC52 HCT 116 C514(0.87)  LDD0632  [15]
 LDCM0316  AC53 HCT 116 C514(1.04)  LDD0633  [15]
 LDCM0317  AC54 HCT 116 C514(0.85)  LDD0634  [15]
 LDCM0318  AC55 HCT 116 C514(1.00)  LDD0635  [15]
 LDCM0319  AC56 HCT 116 C514(0.88)  LDD0636  [15]
 LDCM0320  AC57 HCT 116 C514(1.11)  LDD0637  [15]
 LDCM0321  AC58 HCT 116 C514(0.86)  LDD0638  [15]
 LDCM0322  AC59 HCT 116 C514(1.06)  LDD0639  [15]
 LDCM0323  AC6 HCT 116 C514(1.02)  LDD0640  [15]
 LDCM0324  AC60 HCT 116 C514(1.05)  LDD0641  [15]
 LDCM0325  AC61 HCT 116 C514(1.03)  LDD0642  [15]
 LDCM0326  AC62 HCT 116 C514(1.09)  LDD0643  [15]
 LDCM0327  AC63 HCT 116 C514(1.22)  LDD0644  [15]
 LDCM0328  AC64 HCT 116 C514(1.21)  LDD0645  [15]
 LDCM0329  AC65 HCT 116 C514(1.01)  LDD0646  [15]
 LDCM0330  AC66 HCT 116 C514(1.11)  LDD0647  [15]
 LDCM0331  AC67 HCT 116 C514(1.14)  LDD0648  [15]
 LDCM0332  AC68 HCT 116 C514(0.90)  LDD0649  [15]
 LDCM0333  AC69 HCT 116 C514(0.82)  LDD0650  [15]
 LDCM0334  AC7 HCT 116 C514(1.02)  LDD0651  [15]
 LDCM0335  AC70 HCT 116 C514(0.88)  LDD0652  [15]
 LDCM0336  AC71 HCT 116 C514(0.96)  LDD0653  [15]
 LDCM0337  AC72 HCT 116 C514(0.91)  LDD0654  [15]
 LDCM0338  AC73 HCT 116 C514(0.81)  LDD0655  [15]
 LDCM0339  AC74 HCT 116 C514(0.97)  LDD0656  [15]
 LDCM0340  AC75 HCT 116 C514(0.91)  LDD0657  [15]
 LDCM0341  AC76 HCT 116 C514(1.00)  LDD0658  [15]
 LDCM0342  AC77 HCT 116 C514(0.77)  LDD0659  [15]
 LDCM0343  AC78 HCT 116 C514(0.82)  LDD0660  [15]
 LDCM0344  AC79 HCT 116 C514(0.82)  LDD0661  [15]
 LDCM0345  AC8 HCT 116 C514(1.02)  LDD0662  [15]
 LDCM0346  AC80 HCT 116 C514(0.87)  LDD0663  [15]
 LDCM0347  AC81 HCT 116 C514(0.94)  LDD0664  [15]
 LDCM0348  AC82 HCT 116 C514(0.94)  LDD0665  [15]
 LDCM0349  AC83 HCT 116 C514(0.89)  LDD0666  [15]
 LDCM0350  AC84 HCT 116 C514(0.84)  LDD0667  [15]
 LDCM0351  AC85 HCT 116 C514(0.88)  LDD0668  [15]
 LDCM0352  AC86 HCT 116 C514(0.80)  LDD0669  [15]
 LDCM0353  AC87 HCT 116 C514(1.03)  LDD0670  [15]
 LDCM0354  AC88 HCT 116 C514(0.81)  LDD0671  [15]
 LDCM0355  AC89 HCT 116 C514(0.88)  LDD0672  [15]
 LDCM0357  AC90 HCT 116 C514(1.01)  LDD0674  [15]
 LDCM0358  AC91 HCT 116 C514(0.92)  LDD0675  [15]
 LDCM0359  AC92 HCT 116 C514(0.87)  LDD0676  [15]
 LDCM0360  AC93 HCT 116 C514(0.91)  LDD0677  [15]
 LDCM0361  AC94 HCT 116 C514(1.02)  LDD0678  [15]
 LDCM0362  AC95 HCT 116 C514(1.06)  LDD0679  [15]
 LDCM0363  AC96 HCT 116 C514(0.94)  LDD0680  [15]
 LDCM0364  AC97 HCT 116 C514(0.85)  LDD0681  [15]
 LDCM0365  AC98 HCT 116 C514(1.00)  LDD0682  [15]
 LDCM0366  AC99 HCT 116 C514(0.97)  LDD0683  [15]
 LDCM0545  Acetamide MDA-MB-231 C514(0.42); C1148(0.37); C673(0.65)  LDD2138  [9]
 LDCM0520  AKOS000195272 MDA-MB-231 C41(0.95)  LDD2113  [9]
 LDCM0248  AKOS034007472 HCT 116 C514(1.02)  LDD0565  [15]
 LDCM0356  AKOS034007680 HCT 116 C514(1.11)  LDD0673  [15]
 LDCM0275  AKOS034007705 HCT 116 C514(1.10)  LDD0592  [15]
 LDCM0156  Aniline NCI-H1299 N.A.  LDD0405  [31]
 LDCM0020  ARS-1620 HCC44 C245(0.96)  LDD0078  [15]
 LDCM0498  BS-3668 MDA-MB-231 C514(0.45); C1148(0.55); C752(0.77)  LDD2091  [9]
 LDCM0108  Chloroacetamide HeLa C453(0.00); C254(0.00); H944(0.00); C522(0.00)  LDD0222  [30]
 LDCM0632  CL-Sc Hep-G2 C921(2.21); C453(1.07); C41(0.86); C693(0.84)  LDD2227  [22]
 LDCM0367  CL1 HCT 116 C514(1.00)  LDD0684  [15]
 LDCM0368  CL10 HCT 116 C514(1.12)  LDD0685  [15]
 LDCM0369  CL100 HCT 116 C514(1.08)  LDD0686  [15]
 LDCM0370  CL101 HCT 116 C514(1.04)  LDD0687  [15]
 LDCM0371  CL102 HCT 116 C514(1.10)  LDD0688  [15]
 LDCM0372  CL103 HCT 116 C514(0.99)  LDD0689  [15]
 LDCM0373  CL104 HCT 116 C514(1.10)  LDD0690  [15]
 LDCM0374  CL105 HCT 116 C514(1.36)  LDD0691  [15]
 LDCM0375  CL106 HCT 116 C514(1.20)  LDD0692  [15]
 LDCM0376  CL107 HCT 116 C514(1.20)  LDD0693  [15]
 LDCM0377  CL108 HCT 116 C514(1.07)  LDD0694  [15]
 LDCM0378  CL109 HCT 116 C514(1.32)  LDD0695  [15]
 LDCM0379  CL11 HCT 116 C514(1.20)  LDD0696  [15]
 LDCM0380  CL110 HCT 116 C514(1.07)  LDD0697  [15]
 LDCM0381  CL111 HCT 116 C514(1.03)  LDD0698  [15]
 LDCM0382  CL112 HCT 116 C514(1.10)  LDD0699  [15]
 LDCM0383  CL113 HCT 116 C514(0.88)  LDD0700  [15]
 LDCM0384  CL114 HCT 116 C514(0.99)  LDD0701  [15]
 LDCM0385  CL115 HCT 116 C514(0.88)  LDD0702  [15]
 LDCM0386  CL116 HCT 116 C514(0.85)  LDD0703  [15]
 LDCM0387  CL117 HCT 116 C514(1.15)  LDD0704  [15]
 LDCM0388  CL118 HCT 116 C514(1.49)  LDD0705  [15]
 LDCM0389  CL119 HCT 116 C514(1.28)  LDD0706  [15]
 LDCM0390  CL12 HCT 116 C514(1.28)  LDD0707  [15]
 LDCM0391  CL120 HCT 116 C514(1.17)  LDD0708  [15]
 LDCM0392  CL121 HCT 116 C514(0.97)  LDD0709  [15]
 LDCM0393  CL122 HCT 116 C514(0.92)  LDD0710  [15]
 LDCM0394  CL123 HCT 116 C514(0.99)  LDD0711  [15]
 LDCM0395  CL124 HCT 116 C514(0.97)  LDD0712  [15]
 LDCM0396  CL125 HCT 116 C514(1.09)  LDD0713  [15]
 LDCM0397  CL126 HCT 116 C514(0.88)  LDD0714  [15]
 LDCM0398  CL127 HCT 116 C514(1.16)  LDD0715  [15]
 LDCM0399  CL128 HCT 116 C514(1.14)  LDD0716  [15]
 LDCM0400  CL13 HCT 116 C514(1.09)  LDD0717  [15]
 LDCM0401  CL14 HCT 116 C514(1.22)  LDD0718  [15]
 LDCM0402  CL15 HCT 116 C514(1.08)  LDD0719  [15]
 LDCM0403  CL16 HCT 116 C514(1.05)  LDD0720  [15]
 LDCM0404  CL17 HCT 116 C514(1.11)  LDD0721  [15]
 LDCM0405  CL18 HCT 116 C514(1.00)  LDD0722  [15]
 LDCM0406  CL19 HCT 116 C514(0.88)  LDD0723  [15]
 LDCM0407  CL2 HCT 116 C514(1.20)  LDD0724  [15]
 LDCM0408  CL20 HCT 116 C514(0.93)  LDD0725  [15]
 LDCM0409  CL21 HCT 116 C514(0.96)  LDD0726  [15]
 LDCM0410  CL22 HCT 116 C514(0.81)  LDD0727  [15]
 LDCM0411  CL23 HCT 116 C514(0.88)  LDD0728  [15]
 LDCM0412  CL24 HCT 116 C514(0.85)  LDD0729  [15]
 LDCM0413  CL25 HCT 116 C514(1.12)  LDD0730  [15]
 LDCM0414  CL26 HCT 116 C514(1.01)  LDD0731  [15]
 LDCM0415  CL27 HCT 116 C514(0.86)  LDD0732  [15]
 LDCM0416  CL28 HCT 116 C514(0.99)  LDD0733  [15]
 LDCM0417  CL29 HCT 116 C514(0.96)  LDD0734  [15]
 LDCM0418  CL3 HCT 116 C514(1.13)  LDD0735  [15]
 LDCM0419  CL30 HCT 116 C514(0.94)  LDD0736  [15]
 LDCM0420  CL31 HCT 116 C514(0.94)  LDD0737  [15]
 LDCM0421  CL32 HCT 116 C514(1.03)  LDD0738  [15]
 LDCM0422  CL33 HCT 116 C514(1.08)  LDD0739  [15]
 LDCM0423  CL34 HCT 116 C514(0.97)  LDD0740  [15]
 LDCM0424  CL35 HCT 116 C514(1.07)  LDD0741  [15]
 LDCM0425  CL36 HCT 116 C514(0.79)  LDD0742  [15]
 LDCM0426  CL37 HCT 116 C514(1.00)  LDD0743  [15]
 LDCM0428  CL39 HCT 116 C514(1.11)  LDD0745  [15]
 LDCM0429  CL4 HCT 116 C514(1.26)  LDD0746  [15]
 LDCM0430  CL40 HCT 116 C514(0.96)  LDD0747  [15]
 LDCM0431  CL41 HCT 116 C514(0.96)  LDD0748  [15]
 LDCM0432  CL42 HCT 116 C514(0.84)  LDD0749  [15]
 LDCM0433  CL43 HCT 116 C514(1.00)  LDD0750  [15]
 LDCM0434  CL44 HCT 116 C514(1.14)  LDD0751  [15]
 LDCM0435  CL45 HCT 116 C514(0.95)  LDD0752  [15]
 LDCM0436  CL46 HCT 116 C514(1.02)  LDD0753  [15]
 LDCM0437  CL47 HCT 116 C514(1.03)  LDD0754  [15]
 LDCM0438  CL48 HCT 116 C514(0.91)  LDD0755  [15]
 LDCM0439  CL49 HCT 116 C514(1.49)  LDD0756  [15]
 LDCM0440  CL5 HCT 116 C514(1.20)  LDD0757  [15]
 LDCM0441  CL50 HCT 116 C514(1.03)  LDD0758  [15]
 LDCM0442  CL51 HCT 116 C514(1.05)  LDD0759  [15]
 LDCM0443  CL52 HCT 116 C514(0.88)  LDD0760  [15]
 LDCM0444  CL53 HCT 116 C514(0.88)  LDD0761  [15]
 LDCM0445  CL54 HCT 116 C514(1.12)  LDD0762  [15]
 LDCM0446  CL55 HCT 116 C514(1.33)  LDD0763  [15]
 LDCM0447  CL56 HCT 116 C514(1.17)  LDD0764  [15]
 LDCM0448  CL57 HCT 116 C514(1.23)  LDD0765  [15]
 LDCM0449  CL58 HCT 116 C514(1.12)  LDD0766  [15]
 LDCM0450  CL59 HCT 116 C514(1.43)  LDD0767  [15]
 LDCM0451  CL6 HCT 116 C514(1.16)  LDD0768  [15]
 LDCM0452  CL60 HCT 116 C514(1.41)  LDD0769  [15]
 LDCM0453  CL61 HCT 116 C514(1.05)  LDD0770  [15]
 LDCM0454  CL62 HCT 116 C514(1.07)  LDD0771  [15]
 LDCM0455  CL63 HCT 116 C514(0.89)  LDD0772  [15]
 LDCM0456  CL64 HCT 116 C514(1.17)  LDD0773  [15]
 LDCM0457  CL65 HCT 116 C514(1.25)  LDD0774  [15]
 LDCM0458  CL66 HCT 116 C514(1.26)  LDD0775  [15]
 LDCM0459  CL67 HCT 116 C514(1.14)  LDD0776  [15]
 LDCM0460  CL68 HCT 116 C514(1.13)  LDD0777  [15]
 LDCM0461  CL69 HCT 116 C514(1.02)  LDD0778  [15]
 LDCM0462  CL7 HCT 116 C514(1.30)  LDD0779  [15]
 LDCM0463  CL70 HCT 116 C514(0.94)  LDD0780  [15]
 LDCM0464  CL71 HCT 116 C514(0.98)  LDD0781  [15]
 LDCM0465  CL72 HCT 116 C514(0.98)  LDD0782  [15]
 LDCM0466  CL73 HCT 116 C514(1.22)  LDD0783  [15]
 LDCM0467  CL74 HCT 116 C514(1.08)  LDD0784  [15]
 LDCM0469  CL76 HCT 116 C514(0.98)  LDD0786  [15]
 LDCM0470  CL77 HCT 116 C514(0.81)  LDD0787  [15]
 LDCM0471  CL78 HCT 116 C514(0.91)  LDD0788  [15]
 LDCM0472  CL79 HCT 116 C514(0.93)  LDD0789  [15]
 LDCM0473  CL8 HCT 116 C514(1.04)  LDD0790  [15]
 LDCM0474  CL80 HCT 116 C514(1.12)  LDD0791  [15]
 LDCM0475  CL81 HCT 116 C514(0.98)  LDD0792  [15]
 LDCM0476  CL82 HCT 116 C514(1.07)  LDD0793  [15]
 LDCM0477  CL83 HCT 116 C514(1.04)  LDD0794  [15]
 LDCM0478  CL84 HCT 116 C514(0.96)  LDD0795  [15]
 LDCM0479  CL85 HCT 116 C514(0.84)  LDD0796  [15]
 LDCM0480  CL86 HCT 116 C514(0.98)  LDD0797  [15]
 LDCM0481  CL87 HCT 116 C514(1.05)  LDD0798  [15]
 LDCM0482  CL88 HCT 116 C514(1.02)  LDD0799  [15]
 LDCM0483  CL89 HCT 116 C514(0.90)  LDD0800  [15]
 LDCM0484  CL9 HCT 116 C514(1.14)  LDD0801  [15]
 LDCM0485  CL90 HCT 116 C514(0.97)  LDD0802  [15]
 LDCM0486  CL91 HCT 116 C514(1.06)  LDD0803  [15]
 LDCM0487  CL92 HCT 116 C514(0.98)  LDD0804  [15]
 LDCM0488  CL93 HCT 116 C514(1.10)  LDD0805  [15]
 LDCM0489  CL94 HCT 116 C514(1.40)  LDD0806  [15]
 LDCM0490  CL95 HCT 116 C514(1.13)  LDD0807  [15]
 LDCM0491  CL96 HCT 116 C514(1.14)  LDD0808  [15]
 LDCM0492  CL97 HCT 116 C514(1.07)  LDD0809  [15]
 LDCM0493  CL98 HCT 116 C514(1.09)  LDD0810  [15]
 LDCM0494  CL99 HCT 116 C514(1.06)  LDD0811  [15]
 LDCM0495  E2913 HEK-293T C514(0.77); C254(0.98); C245(0.90); C41(0.96)  LDD1698  [35]
 LDCM0213  Electrophilic fragment 2 MDA-MB-231 C1185(3.55); C522(2.32); C580(2.09); C453(1.76)  LDD1702  [9]
 LDCM0625  F8 Ramos C41(0.84); C85(0.81)  LDD2187  [36]
 LDCM0572  Fragment10 Ramos C41(0.53); C380(1.13)  LDD2189  [36]
 LDCM0573  Fragment11 Ramos C41(0.21); C85(0.50)  LDD2190  [36]
 LDCM0574  Fragment12 Ramos C41(0.52); C380(1.17)  LDD2191  [36]
 LDCM0575  Fragment13 Ramos C41(0.65)  LDD2192  [36]
 LDCM0576  Fragment14 Ramos C41(0.82); C522(0.90); C85(0.65); C975(1.67)  LDD2193  [36]
 LDCM0579  Fragment20 Ramos C41(0.33); C380(0.63)  LDD2194  [36]
 LDCM0580  Fragment21 Ramos C41(0.68); C380(1.36)  LDD2195  [36]
 LDCM0582  Fragment23 Ramos C41(1.25); C380(0.96)  LDD2196  [36]
 LDCM0578  Fragment27 Ramos C41(0.96)  LDD2197  [36]
 LDCM0586  Fragment28 Ramos C41(0.99); C522(0.47); C85(2.57)  LDD2198  [36]
 LDCM0588  Fragment30 Ramos C41(0.81); C380(1.45)  LDD2199  [36]
 LDCM0589  Fragment31 Ramos C41(0.91)  LDD2200  [36]
 LDCM0590  Fragment32 Ramos C41(0.52); C380(0.99)  LDD2201  [36]
 LDCM0468  Fragment33 HCT 116 C514(1.28)  LDD0785  [15]
 LDCM0596  Fragment38 Ramos C41(0.96)  LDD2203  [36]
 LDCM0566  Fragment4 Ramos C41(0.95); C522(0.75); C85(0.57); C975(2.01)  LDD2184  [36]
 LDCM0427  Fragment51 HCT 116 C514(1.06)  LDD0744  [15]
 LDCM0610  Fragment52 Ramos C41(0.56)  LDD2204  [36]
 LDCM0614  Fragment56 Ramos C41(0.73); C380(1.35)  LDD2205  [36]
 LDCM0617  Fragment63-S Jurkat _(20.00)  LDD1490  [10]
 LDCM0569  Fragment7 Ramos C41(0.52); C522(0.75); C85(0.91); C975(0.64)  LDD2186  [36]
 LDCM0571  Fragment9 Ramos C41(0.35); C380(0.93)  LDD2188  [36]
 LDCM0116  HHS-0101 DM93 Y634(0.05); Y579(0.74); Y608(0.91); Y249(1.00)  LDD0264  [13]
 LDCM0117  HHS-0201 DM93 Y1156(0.58); Y579(0.72); Y249(0.93); Y608(1.01)  LDD0265  [13]
 LDCM0118  HHS-0301 DM93 Y634(0.60); Y579(0.77); Y249(0.79); Y608(0.88)  LDD0266  [13]
 LDCM0119  HHS-0401 DM93 Y579(0.82); Y249(0.88); Y608(1.29); Y628(9.88)  LDD0267  [13]
 LDCM0120  HHS-0701 DM93 Y579(0.68); Y249(1.43); Y608(1.48); Y628(6.58)  LDD0268  [13]
 LDCM0107  IAA HeLa H944(0.00); C1057(0.00); H640(0.00); H558(0.00)  LDD0221  [30]
 LDCM0123  JWB131 DM93 Y249(0.84)  LDD0285  [12]
 LDCM0125  JWB146 DM93 Y249(0.86)  LDD0287  [12]
 LDCM0126  JWB150 DM93 Y249(3.86)  LDD0288  [12]
 LDCM0127  JWB152 DM93 Y249(2.19)  LDD0289  [12]
 LDCM0128  JWB198 DM93 Y249(1.40)  LDD0290  [12]
 LDCM0130  JWB211 DM93 Y249(0.86)  LDD0292  [12]
 LDCM0022  KB02 HCT 116 C1185(14.05); C1191(14.05); C580(2.47); C514(1.97)  LDD0080  [15]
 LDCM0023  KB03 HCT 116 C1185(17.21); C1191(17.21); C580(4.35); C514(2.96)  LDD0081  [15]
 LDCM0024  KB05 HCT 116 C1185(7.81); C1191(7.81); C580(3.13); C514(2.75)  LDD0082  [15]
 LDCM0528  N-(4-bromophenyl)-2-cyano-N-phenylacetamide MDA-MB-231 C514(0.40); C1148(0.59); C673(0.85)  LDD2121  [9]
 LDCM0109  NEM HeLa H944(0.00); C254(0.00); H558(0.00); H433(0.00)  LDD0223  [30]
 LDCM0496  Nucleophilic fragment 11a MDA-MB-231 C1148(0.59); C673(0.97)  LDD2089  [9]
 LDCM0497  Nucleophilic fragment 11b MDA-MB-231 C1148(1.19); C522(1.00); C1185(1.09)  LDD2090  [9]
 LDCM0499  Nucleophilic fragment 12b MDA-MB-231 C1185(0.60)  LDD2092  [9]
 LDCM0500  Nucleophilic fragment 13a MDA-MB-231 C514(0.85); C1148(0.92); C41(1.29); C522(1.17)  LDD2093  [9]
 LDCM0501  Nucleophilic fragment 13b MDA-MB-231 C1185(0.91)  LDD2094  [9]
 LDCM0503  Nucleophilic fragment 14b MDA-MB-231 C752(0.08)  LDD2096  [9]
 LDCM0504  Nucleophilic fragment 15a MDA-MB-231 C514(0.77)  LDD2097  [9]
 LDCM0505  Nucleophilic fragment 15b MDA-MB-231 C1148(0.32); C673(0.84); C1185(1.00)  LDD2098  [9]
 LDCM0506  Nucleophilic fragment 16a MDA-MB-231 C514(1.10); C1148(1.02); C41(1.19); C522(1.85)  LDD2099  [9]
 LDCM0507  Nucleophilic fragment 16b MDA-MB-231 C1148(0.43)  LDD2100  [9]
 LDCM0508  Nucleophilic fragment 17a MDA-MB-231 C41(0.89)  LDD2101  [9]
 LDCM0511  Nucleophilic fragment 18b MDA-MB-231 C1148(0.68)  LDD2104  [9]
 LDCM0512  Nucleophilic fragment 19a MDA-MB-231 C1148(1.24); C522(1.00); C1185(1.02)  LDD2105  [9]
 LDCM0513  Nucleophilic fragment 19b MDA-MB-231 C1148(0.51)  LDD2106  [9]
 LDCM0514  Nucleophilic fragment 20a MDA-MB-231 C514(1.00); C41(1.53); C580(1.24)  LDD2107  [9]
 LDCM0515  Nucleophilic fragment 20b MDA-MB-231 C522(0.88); C673(0.38)  LDD2108  [9]
 LDCM0516  Nucleophilic fragment 21a MDA-MB-231 C514(0.48); C1148(0.67); C673(0.77); C580(0.76)  LDD2109  [9]
 LDCM0517  Nucleophilic fragment 21b MDA-MB-231 C522(0.69)  LDD2110  [9]
 LDCM0518  Nucleophilic fragment 22a MDA-MB-231 C514(1.03); C1148(0.97); C522(0.44)  LDD2111  [9]
 LDCM0521  Nucleophilic fragment 23b MDA-MB-231 C1185(0.54)  LDD2114  [9]
 LDCM0522  Nucleophilic fragment 24a MDA-MB-231 C673(0.54)  LDD2115  [9]
 LDCM0525  Nucleophilic fragment 25b MDA-MB-231 C522(1.18)  LDD2118  [9]
 LDCM0526  Nucleophilic fragment 26a MDA-MB-231 C514(1.88); C1148(2.14); C673(1.97)  LDD2119  [9]
 LDCM0527  Nucleophilic fragment 26b MDA-MB-231 C1148(0.74)  LDD2120  [9]
 LDCM0529  Nucleophilic fragment 27b MDA-MB-231 C522(0.37); C673(0.08); C254(0.45); C1191(0.94)  LDD2122  [9]
 LDCM0530  Nucleophilic fragment 28a MDA-MB-231 C514(0.85); C673(0.99); C1013(0.77); C1057(1.31)  LDD2123  [9]
 LDCM0532  Nucleophilic fragment 29a MDA-MB-231 C1148(0.77); C41(1.19); C673(1.00); C1013(1.08)  LDD2125  [9]
 LDCM0533  Nucleophilic fragment 29b MDA-MB-231 C522(0.40); C673(0.08)  LDD2126  [9]
 LDCM0534  Nucleophilic fragment 30a MDA-MB-231 C514(1.15); C1148(0.98); C522(0.99); C673(1.27)  LDD2127  [9]
 LDCM0535  Nucleophilic fragment 30b MDA-MB-231 C514(0.98); C522(1.17); C673(0.95); C1185(0.76)  LDD2128  [9]
 LDCM0536  Nucleophilic fragment 31 MDA-MB-231 C514(0.98); C1148(0.97); C41(1.72); C522(1.43)  LDD2129  [9]
 LDCM0541  Nucleophilic fragment 36 MDA-MB-231 C41(0.83)  LDD2134  [9]
 LDCM0542  Nucleophilic fragment 37 MDA-MB-231 C514(1.20); C1148(1.15); C673(1.81); C254(1.94)  LDD2135  [9]
 LDCM0543  Nucleophilic fragment 38 MDA-MB-231 C514(0.89); C1148(1.23); C673(1.00); C1013(0.96)  LDD2136  [9]
 LDCM0544  Nucleophilic fragment 39 MDA-MB-231 C514(0.83); C1148(1.02); C673(0.91); C1013(0.94)  LDD2137  [9]
 LDCM0211  Nucleophilic fragment 3b MDA-MB-231 C673(2.87); C1148(1.43)  LDD1700  [9]
 LDCM0546  Nucleophilic fragment 40 MDA-MB-231 C1148(0.73); C41(1.12); C673(1.12)  LDD2140  [9]
 LDCM0547  Nucleophilic fragment 41 MDA-MB-231 C673(0.48)  LDD2141  [9]
 LDCM0549  Nucleophilic fragment 43 MDA-MB-231 C1148(0.98)  LDD2143  [9]
 LDCM0550  Nucleophilic fragment 5a MDA-MB-231 C514(1.37); C1148(2.37); C522(3.01); C673(1.46)  LDD2144  [9]
 LDCM0552  Nucleophilic fragment 6a MDA-MB-231 C514(0.83); C1148(1.19); C580(1.14)  LDD2146  [9]
 LDCM0553  Nucleophilic fragment 6b MDA-MB-231 C1148(2.13); C522(2.25)  LDD2147  [9]
 LDCM0554  Nucleophilic fragment 7a MDA-MB-231 C41(0.51)  LDD2148  [9]
 LDCM0556  Nucleophilic fragment 8a MDA-MB-231 C514(0.45); C673(0.66); C1185(1.04)  LDD2150  [9]
 LDCM0557  Nucleophilic fragment 8b MDA-MB-231 C752(0.15)  LDD2151  [9]
 LDCM0559  Nucleophilic fragment 9b MDA-MB-231 C1148(1.56); C1185(1.62)  LDD2153  [9]
 LDCM0628  OTUB2-COV-1 HEK-293T C752(0.82)  LDD2207  [37]
 LDCM0090  Rapamycin JHH-7 3.48  LDD0213  [33]
 LDCM0021  THZ1 HCT 116 C1057(1.07); C41(1.07); C514(1.13); C522(0.93)  LDD2173  [15]

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Mass spectrometry data entry: PXD037665
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Mass spectrometry data entry: PXD042888
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