Details of the Target

General Information of Target

Target ID LDTP12826
Target Name Bcl-2-associated transcription factor 1 (BCLAF1)
Gene Name BCLAF1
Gene ID 9774
Synonyms
BTF; KIAA0164; Bcl-2-associated transcription factor 1; Btf; BCLAF1 and THRAP3 family member 1
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MKPSPAGTAKELEPPAPARGEQRTAEPEGRWREKGEADTERQRTRERQEATLAGLAELEY
LRQRQELLVRGALRGAGGAGAAAPRAGELLGEAAQRSRLEEKFLEENILLLRKQLNCLRR
RDAGLLNQLQELDKQISDLRLDVEKTSEEHLETDSRPSSGFYELSDGASGSLSNSSNSVF
SECLSSCHSSTCFCSPLEATLSLSDGCPKSADLIGLLEYKEGHCEDQASGAVCRSLSTPQ
FNSLDVIADVNPKYQCDLVSKNGNDVYRYPSPLHAVAVQSPMFLLCLTGNPLREEDRLGN
HASDICGGSELDAVKTDSSLPSPSSLWSASHPSSSKKMDGYILSLVQKKTHPVRTNKPRT
SVNADPTKGLLRNGSVCVRAPGGVSQGNSVNLKNSKQACLPSGGIPSLNNGTFSPPKQWS
KESKAEQAESKRVPLPEGCPSGAASDLQSKHLPKTAKPASQEHARCSAIGTGESPKESAQ
LSGASPKESPSRGPAPPQENKVVQPLKKMSQKNSLQGVPPATPPLLSTAFPVEERPALDF
KSEGSSQSLEEAHLVKAQFIPGQQPSVRLHRGHRNMGVVKNSSLKHRGPALQGLENGLPT
VREKTRAGSKKCRFPDDLDTNKKLKKASSKGRKSGGGPEAGVPGRPAGGGHRAGSRAHGH
GREAVVAKPKHKRTDYRRWKSSAEISYEEALRRARRGRRENVGLYPAPVPLPYASPYAYV
ASDSEYSAECESLFHSTVVDTSEDEQSNYTTNCFGDSESSVSEGEFVGESTTTSDSEESG
GLIWSQFVQTLPIQTVTAPDLHNHPAKTFVKIKASHNLKKKILRFRSGSLKLMTTV
Target Bioclass
Other
Family
BCLAF1/THRAP3 family
Subcellular location
Cytoplasm
Function Death-promoting transcriptional repressor. May be involved in cyclin-D1/CCND1 mRNA stability through the SNARP complex which associates with both the 3'end of the CCND1 gene and its mRNA.
Uniprot ID
Q9NYF8
Ensemble ID
ENST00000353331.8
HGNC ID
HGNC:16863

Target Site Mutations in Different Cell Lines

Cell line Mutation details Probe for labeling this protein in this cell
CAL51 SNV: p.R915H .
HT115 SNV: p.R654I; p.R801Q DBIA    Probe Info 
HUH28 SNV: p.R704T .
MFE319 SNV: p.K919N DBIA    Probe Info 
SHP77 SNV: p.R667L .

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 40 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
m-APA
 Probe Info  		15.00  LDD0402  [2]
P1
 Probe Info  		2.69  LDD0448  [3]
P2
 Probe Info  		4.20  LDD0449  [3]
P3
 Probe Info  		4.01  LDD0450  [3]
CY-1
 Probe Info  		100.00  LDD0243  [4]
FBP2
 Probe Info  		2.12  LDD0323  [5]
ONAyne
 Probe Info  		K712(1.79)  LDD0274  [6]
Probe 1
 Probe Info  		Y408(28.84); Y466(41.95); Y839(31.93)  LDD3495  [7]
BTD
 Probe Info  		C688(0.78)  LDD1700  [8]
AHL-Pu-1
 Probe Info  		C688(2.14)  LDD0169  [9]
HHS-475
 Probe Info  		Y438(0.91); Y322(18.42)  LDD0264  [10]
DBIA
 Probe Info  		C688(0.82)  LDD0531  [11]
5E-2FA
 Probe Info  		N.A.  LDD2235  [12]
AMP probe
 Probe Info  		N.A.  LDD0200  [13]
ATP probe
 Probe Info  		K593(0.00); K462(0.00); K421(0.00); K831(0.00)  LDD0199  [13]
4-Iodoacetamidophenylacetylene
 Probe Info  		C688(0.00); C242(0.00)  LDD0038  [14]
IA-alkyne
 Probe Info  		C688(0.00); C242(0.00)  LDD0036  [14]
IPIAA_L
 Probe Info  		N.A.  LDD0031  [15]
Lodoacetamide azide
 Probe Info  		C688(0.00); C242(0.00)  LDD0037  [14]
NAIA_4
 Probe Info  		N.A.  LDD2226  [16]
NAIA_5
 Probe Info  		C688(0.00); C242(0.00)  LDD2224  [16]
TFBX
 Probe Info  		N.A.  LDD0027  [17]
Compound 10
 Probe Info  		N.A.  LDD2216  [18]
Compound 11
 Probe Info  		N.A.  LDD2213  [18]
IPM
 Probe Info  		N.A.  LDD0005  [19]
NHS
 Probe Info  		K506(0.00); K517(0.00); K421(0.00); K332(0.00)  LDD0010  [19]
SF
 Probe Info  		Y511(0.00); Y466(0.00); Y322(0.00); K725(0.00)  LDD0028  [20]
STPyne
 Probe Info  		K550(0.00); K567(0.00)  LDD0009  [19]
VSF
 Probe Info  		C688(0.00); C242(0.00)  LDD0007  [19]
Phosphinate-6
 Probe Info  		C242(0.00); C688(0.00)  LDD0018  [21]
Ox-W18
 Probe Info  		N.A.  LDD2175  [22]
1c-yne
 Probe Info  		K462(0.00); K204(0.00); K550(0.00)  LDD0228  [23]
1d-yne
 Probe Info  		N.A.  LDD0357  [23]
Acrolein
 Probe Info  		C688(0.00); H608(0.00); H577(0.00); H615(0.00)  LDD0217  [24]
Crotonaldehyde
 Probe Info  		H591(0.00); H642(0.00)  LDD0219  [24]
W1
 Probe Info  		E603(0.00); S600(0.00)  LDD0236  [25]
AOyne
 Probe Info  		6.30  LDD0443  [26]
MPP-AC
 Probe Info  		N.A.  LDD0428  [27]
HHS-465
 Probe Info  		N.A.  LDD2240  [28]
HHS-482
 Probe Info  		Y892(0.80)  LDD2239  [29]
PAL-AfBPP Probe
Click To Hide/Show 5 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
C187
 Probe Info  		15.56  LDD1865  [30]
C191
 Probe Info  		13.45  LDD1868  [30]
C193
 Probe Info  		5.98  LDD1869  [30]
FFF probe13
 Probe Info  		5.85  LDD0475  [31]
IMP2070
 Probe Info  		1.48  LDD0370  [32]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0548  1-(4-(Benzo[d][1,3]dioxol-5-ylmethyl)piperazin-1-yl)-2-nitroethan-1-one MDA-MB-231 C242(1.17); C688(0.66)  LDD2142  [8]
 LDCM0519  1-(6-methoxy-3,4-dihydroquinolin-1(2H)-yl)-2-nitroethan-1-one MDA-MB-231 C242(1.12)  LDD2112  [8]
 LDCM0502  1-(Cyanoacetyl)piperidine MDA-MB-231 C242(0.64); C688(0.57)  LDD2095  [8]
 LDCM0537  2-Cyano-N,N-dimethylacetamide MDA-MB-231 C688(1.04)  LDD2130  [8]
 LDCM0524  2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide MDA-MB-231 C688(0.95)  LDD2117  [8]
 LDCM0558  2-Cyano-N-phenylacetamide MDA-MB-231 C688(1.06)  LDD2152  [8]
 LDCM0510  3-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-3-oxopropanenitrile MDA-MB-231 C688(0.98)  LDD2103  [8]
 LDCM0539  3-(4-Isopropylpiperazin-1-yl)-3-oxopropanenitrile MDA-MB-231 C242(0.72)  LDD2132  [8]
 LDCM0026  4SU-RNA+native RNA HEK-293T C688(2.14)  LDD0169  [9]
 LDCM0214  AC1 HCT 116 C688(0.82)  LDD0531  [11]
 LDCM0215  AC10 HCT 116 C688(1.07)  LDD0532  [11]
 LDCM0216  AC100 HCT 116 C688(1.47)  LDD0533  [11]
 LDCM0217  AC101 HCT 116 C688(1.35)  LDD0534  [11]
 LDCM0218  AC102 HCT 116 C688(0.98)  LDD0535  [11]
 LDCM0219  AC103 HCT 116 C688(1.25)  LDD0536  [11]
 LDCM0220  AC104 HCT 116 C688(0.98)  LDD0537  [11]
 LDCM0221  AC105 HCT 116 C688(1.74)  LDD0538  [11]
 LDCM0222  AC106 HCT 116 C688(2.05)  LDD0539  [11]
 LDCM0223  AC107 HCT 116 C688(1.37)  LDD0540  [11]
 LDCM0224  AC108 HCT 116 C688(1.65)  LDD0541  [11]
 LDCM0225  AC109 HCT 116 C688(0.97)  LDD0542  [11]
 LDCM0226  AC11 HCT 116 C688(1.15)  LDD0543  [11]
 LDCM0227  AC110 HCT 116 C688(1.38)  LDD0544  [11]
 LDCM0228  AC111 HCT 116 C688(1.42)  LDD0545  [11]
 LDCM0229  AC112 HCT 116 C688(1.42)  LDD0546  [11]
 LDCM0230  AC113 HCT 116 C688(0.90)  LDD0547  [11]
 LDCM0231  AC114 HCT 116 C688(1.20)  LDD0548  [11]
 LDCM0232  AC115 HCT 116 C688(1.35)  LDD0549  [11]
 LDCM0233  AC116 HCT 116 C688(1.23)  LDD0550  [11]
 LDCM0234  AC117 HCT 116 C688(1.27)  LDD0551  [11]
 LDCM0235  AC118 HCT 116 C688(1.03)  LDD0552  [11]
 LDCM0236  AC119 HCT 116 C688(1.06)  LDD0553  [11]
 LDCM0237  AC12 HCT 116 C688(0.94)  LDD0554  [11]
 LDCM0238  AC120 HCT 116 C688(0.72)  LDD0555  [11]
 LDCM0239  AC121 HCT 116 C688(1.11)  LDD0556  [11]
 LDCM0240  AC122 HCT 116 C688(1.16)  LDD0557  [11]
 LDCM0241  AC123 HCT 116 C688(0.97)  LDD0558  [11]
 LDCM0242  AC124 HCT 116 C688(1.02)  LDD0559  [11]
 LDCM0243  AC125 HCT 116 C688(1.21)  LDD0560  [11]
 LDCM0244  AC126 HCT 116 C688(1.33)  LDD0561  [11]
 LDCM0245  AC127 HCT 116 C688(1.41)  LDD0562  [11]
 LDCM0246  AC128 HCT 116 C688(0.09)  LDD0563  [11]
 LDCM0247  AC129 HCT 116 C688(0.11)  LDD0564  [11]
 LDCM0249  AC130 HCT 116 C688(0.11)  LDD0566  [11]
 LDCM0250  AC131 HCT 116 C688(0.10)  LDD0567  [11]
 LDCM0251  AC132 HCT 116 C688(0.12)  LDD0568  [11]
 LDCM0252  AC133 HCT 116 C688(0.11)  LDD0569  [11]
 LDCM0253  AC134 HCT 116 C688(0.15)  LDD0570  [11]
 LDCM0254  AC135 HCT 116 C688(0.13)  LDD0571  [11]
 LDCM0255  AC136 HCT 116 C688(0.17)  LDD0572  [11]
 LDCM0256  AC137 HCT 116 C688(0.12)  LDD0573  [11]
 LDCM0257  AC138 HCT 116 C688(0.14)  LDD0574  [11]
 LDCM0258  AC139 HCT 116 C688(0.14)  LDD0575  [11]
 LDCM0259  AC14 HCT 116 C688(0.91)  LDD0576  [11]
 LDCM0260  AC140 HCT 116 C688(0.16)  LDD0577  [11]
 LDCM0261  AC141 HCT 116 C688(0.16)  LDD0578  [11]
 LDCM0262  AC142 HCT 116 C688(0.11)  LDD0579  [11]
 LDCM0263  AC143 HCT 116 C688(1.20)  LDD0580  [11]
 LDCM0264  AC144 HCT 116 C688(1.85)  LDD0581  [11]
 LDCM0265  AC145 HCT 116 C688(1.27)  LDD0582  [11]
 LDCM0266  AC146 HCT 116 C688(1.44)  LDD0583  [11]
 LDCM0267  AC147 HCT 116 C688(1.67)  LDD0584  [11]
 LDCM0268  AC148 HCT 116 C688(2.10)  LDD0585  [11]
 LDCM0269  AC149 HCT 116 C688(1.87)  LDD0586  [11]
 LDCM0270  AC15 HCT 116 C688(1.06)  LDD0587  [11]
 LDCM0271  AC150 HCT 116 C688(1.12)  LDD0588  [11]
 LDCM0272  AC151 HCT 116 C688(1.28)  LDD0589  [11]
 LDCM0273  AC152 HCT 116 C688(1.29)  LDD0590  [11]
 LDCM0274  AC153 HCT 116 C688(3.28)  LDD0591  [11]
 LDCM0621  AC154 HCT 116 C688(1.89)  LDD2158  [11]
 LDCM0622  AC155 HCT 116 C688(1.36)  LDD2159  [11]
 LDCM0623  AC156 HCT 116 C688(1.13)  LDD2160  [11]
 LDCM0624  AC157 HCT 116 C688(1.36)  LDD2161  [11]
 LDCM0276  AC17 HCT 116 C688(0.35)  LDD0593  [11]
 LDCM0277  AC18 HCT 116 C688(0.42)  LDD0594  [11]
 LDCM0278  AC19 HCT 116 C688(0.34)  LDD0595  [11]
 LDCM0279  AC2 HCT 116 C688(1.14)  LDD0596  [11]
 LDCM0280  AC20 HCT 116 C688(0.38)  LDD0597  [11]
 LDCM0281  AC21 HCT 116 C688(0.37)  LDD0598  [11]
 LDCM0282  AC22 HCT 116 C688(0.37)  LDD0599  [11]
 LDCM0283  AC23 HCT 116 C688(0.31)  LDD0600  [11]
 LDCM0284  AC24 HCT 116 C688(0.28)  LDD0601  [11]
 LDCM0285  AC25 HCT 116 C688(7.92)  LDD0602  [11]
 LDCM0286  AC26 HCT 116 C688(6.79)  LDD0603  [11]
 LDCM0287  AC27 HCT 116 C688(6.76)  LDD0604  [11]
 LDCM0288  AC28 HCT 116 C688(6.88)  LDD0605  [11]
 LDCM0289  AC29 HCT 116 C688(7.10)  LDD0606  [11]
 LDCM0290  AC3 HCT 116 C688(1.00)  LDD0607  [11]
 LDCM0291  AC30 HCT 116 C688(5.80)  LDD0608  [11]
 LDCM0292  AC31 HCT 116 C688(5.88)  LDD0609  [11]
 LDCM0293  AC32 HCT 116 C688(6.17)  LDD0610  [11]
 LDCM0294  AC33 HCT 116 C688(6.35)  LDD0611  [11]
 LDCM0295  AC34 HCT 116 C688(7.11)  LDD0612  [11]
 LDCM0296  AC35 HEK-293T C688(0.96)  LDD0894  [11]
 LDCM0297  AC36 HEK-293T C688(0.54)  LDD0895  [11]
 LDCM0298  AC37 HEK-293T C688(1.22)  LDD0896  [11]
 LDCM0299  AC38 HEK-293T C688(1.03)  LDD0897  [11]
 LDCM0300  AC39 HEK-293T C688(1.66)  LDD0898  [11]
 LDCM0301  AC4 HCT 116 C688(0.92)  LDD0618  [11]
 LDCM0302  AC40 HEK-293T C688(0.84)  LDD0900  [11]
 LDCM0303  AC41 HEK-293T C688(0.99)  LDD0901  [11]
 LDCM0304  AC42 HEK-293T C688(0.97)  LDD0902  [11]
 LDCM0305  AC43 HEK-293T C688(1.00)  LDD0903  [11]
 LDCM0306  AC44 HEK-293T C688(0.93)  LDD0904  [11]
 LDCM0307  AC45 HEK-293T C688(1.19)  LDD0905  [11]
 LDCM0308  AC46 HCT 116 C688(1.12)  LDD0625  [11]
 LDCM0309  AC47 HCT 116 C688(1.19)  LDD0626  [11]
 LDCM0310  AC48 HCT 116 C688(1.30)  LDD0627  [11]
 LDCM0311  AC49 HCT 116 C688(1.65)  LDD0628  [11]
 LDCM0312  AC5 HCT 116 C688(0.96)  LDD0629  [11]
 LDCM0313  AC50 HCT 116 C688(2.16)  LDD0630  [11]
 LDCM0314  AC51 HCT 116 C688(1.12)  LDD0631  [11]
 LDCM0315  AC52 HCT 116 C688(1.48)  LDD0632  [11]
 LDCM0316  AC53 HCT 116 C688(1.67)  LDD0633  [11]
 LDCM0317  AC54 HCT 116 C688(1.42)  LDD0634  [11]
 LDCM0318  AC55 HCT 116 C688(2.18)  LDD0635  [11]
 LDCM0319  AC56 HCT 116 C688(3.26)  LDD0636  [11]
 LDCM0320  AC57 HCT 116 C688(0.99)  LDD0637  [11]
 LDCM0321  AC58 HCT 116 C688(0.92)  LDD0638  [11]
 LDCM0322  AC59 HCT 116 C688(1.09)  LDD0639  [11]
 LDCM0323  AC6 HCT 116 C688(0.96)  LDD0640  [11]
 LDCM0324  AC60 HCT 116 C688(1.18)  LDD0641  [11]
 LDCM0325  AC61 HCT 116 C688(0.90)  LDD0642  [11]
 LDCM0326  AC62 HCT 116 C688(1.09)  LDD0643  [11]
 LDCM0327  AC63 HCT 116 C688(1.13)  LDD0644  [11]
 LDCM0328  AC64 HCT 116 C688(1.24)  LDD0645  [11]
 LDCM0329  AC65 HCT 116 C688(1.16)  LDD0646  [11]
 LDCM0330  AC66 HCT 116 C688(1.05)  LDD0647  [11]
 LDCM0331  AC67 HCT 116 C688(1.31)  LDD0648  [11]
 LDCM0332  AC68 HCT 116 C688(1.89)  LDD0649  [11]
 LDCM0333  AC69 HCT 116 C688(2.08)  LDD0650  [11]
 LDCM0334  AC7 HCT 116 C688(1.10)  LDD0651  [11]
 LDCM0335  AC70 HCT 116 C688(2.06)  LDD0652  [11]
 LDCM0336  AC71 HCT 116 C688(1.43)  LDD0653  [11]
 LDCM0337  AC72 HCT 116 C688(2.01)  LDD0654  [11]
 LDCM0338  AC73 HCT 116 C688(2.59)  LDD0655  [11]
 LDCM0339  AC74 HCT 116 C688(1.94)  LDD0656  [11]
 LDCM0340  AC75 HCT 116 C688(3.14)  LDD0657  [11]
 LDCM0341  AC76 HCT 116 C688(2.16)  LDD0658  [11]
 LDCM0342  AC77 HCT 116 C688(2.03)  LDD0659  [11]
 LDCM0343  AC78 HCT 116 C688(1.73)  LDD0660  [11]
 LDCM0344  AC79 HCT 116 C688(1.87)  LDD0661  [11]
 LDCM0345  AC8 HCT 116 C688(1.20)  LDD0662  [11]
 LDCM0346  AC80 HCT 116 C688(1.89)  LDD0663  [11]
 LDCM0347  AC81 HCT 116 C688(1.56)  LDD0664  [11]
 LDCM0348  AC82 HCT 116 C688(2.35)  LDD0665  [11]
 LDCM0349  AC83 HCT 116 C688(1.89)  LDD0666  [11]
 LDCM0350  AC84 HCT 116 C688(1.39)  LDD0667  [11]
 LDCM0351  AC85 HCT 116 C688(0.96)  LDD0668  [11]
 LDCM0352  AC86 HCT 116 C688(1.42)  LDD0669  [11]
 LDCM0353  AC87 HCT 116 C688(1.16)  LDD0670  [11]
 LDCM0354  AC88 HCT 116 C688(1.24)  LDD0671  [11]
 LDCM0355  AC89 HCT 116 C688(1.92)  LDD0672  [11]
 LDCM0357  AC90 HCT 116 C688(0.89)  LDD0674  [11]
 LDCM0358  AC91 HCT 116 C688(2.82)  LDD0675  [11]
 LDCM0359  AC92 HCT 116 C688(2.80)  LDD0676  [11]
 LDCM0360  AC93 HCT 116 C688(1.10)  LDD0677  [11]
 LDCM0361  AC94 HCT 116 C688(0.82)  LDD0678  [11]
 LDCM0362  AC95 HCT 116 C688(1.61)  LDD0679  [11]
 LDCM0363  AC96 HCT 116 C688(2.03)  LDD0680  [11]
 LDCM0364  AC97 HCT 116 C688(1.66)  LDD0681  [11]
 LDCM0365  AC98 HCT 116 C688(1.25)  LDD0682  [11]
 LDCM0366  AC99 HCT 116 C688(1.38)  LDD0683  [11]
 LDCM0545  Acetamide MDA-MB-231 C242(0.55); C688(0.32)  LDD2138  [8]
 LDCM0248  AKOS034007472 HCT 116 C688(1.11)  LDD0565  [11]
 LDCM0356  AKOS034007680 HCT 116 C688(1.25)  LDD0673  [11]
 LDCM0275  AKOS034007705 HCT 116 C688(1.00)  LDD0592  [11]
 LDCM0156  Aniline NCI-H1299 11.43  LDD0403  [2]
 LDCM0498  BS-3668 MDA-MB-231 C242(0.42); C688(0.42)  LDD2091  [8]
 LDCM0108  Chloroacetamide HeLa H608(0.00); H614(0.00); H615(0.00); H543(0.00)  LDD0222  [24]
 LDCM0632  CL-Sc Hep-G2 C688(20.00); C688(0.94); C688(0.63)  LDD2227  [16]
 LDCM0367  CL1 HCT 116 C688(1.22)  LDD0684  [11]
 LDCM0368  CL10 HCT 116 C688(1.35)  LDD0685  [11]
 LDCM0369  CL100 HCT 116 C688(1.08)  LDD0686  [11]
 LDCM0370  CL101 HCT 116 C688(0.77)  LDD0687  [11]
 LDCM0371  CL102 HCT 116 C688(0.86)  LDD0688  [11]
 LDCM0372  CL103 HCT 116 C688(0.96)  LDD0689  [11]
 LDCM0373  CL104 HCT 116 C688(0.97)  LDD0690  [11]
 LDCM0374  CL105 HCT 116 C688(0.33)  LDD0691  [11]
 LDCM0375  CL106 HCT 116 C688(0.33)  LDD0692  [11]
 LDCM0376  CL107 HCT 116 C688(0.51)  LDD0693  [11]
 LDCM0377  CL108 HCT 116 C688(0.34)  LDD0694  [11]
 LDCM0378  CL109 HCT 116 C688(0.45)  LDD0695  [11]
 LDCM0379  CL11 HCT 116 C688(0.98)  LDD0696  [11]
 LDCM0380  CL110 HCT 116 C688(0.38)  LDD0697  [11]
 LDCM0381  CL111 HCT 116 C688(0.34)  LDD0698  [11]
 LDCM0382  CL112 HCT 116 C688(4.05)  LDD0699  [11]
 LDCM0383  CL113 HCT 116 C688(5.82)  LDD0700  [11]
 LDCM0384  CL114 HCT 116 C688(7.14)  LDD0701  [11]
 LDCM0385  CL115 HCT 116 C688(7.35)  LDD0702  [11]
 LDCM0386  CL116 HCT 116 C688(7.63)  LDD0703  [11]
 LDCM0387  CL117 HEK-293T C688(1.12)  LDD0985  [11]
 LDCM0388  CL118 HEK-293T C688(0.71)  LDD0986  [11]
 LDCM0389  CL119 HEK-293T C688(1.00)  LDD0987  [11]
 LDCM0390  CL12 HCT 116 C688(1.33)  LDD0707  [11]
 LDCM0391  CL120 HEK-293T C688(1.09)  LDD0989  [11]
 LDCM0392  CL121 HCT 116 C688(1.53)  LDD0709  [11]
 LDCM0393  CL122 HCT 116 C688(1.14)  LDD0710  [11]
 LDCM0394  CL123 HCT 116 C688(1.38)  LDD0711  [11]
 LDCM0395  CL124 HCT 116 C688(1.62)  LDD0712  [11]
 LDCM0396  CL125 HCT 116 C688(0.99)  LDD0713  [11]
 LDCM0397  CL126 HCT 116 C688(0.87)  LDD0714  [11]
 LDCM0398  CL127 HCT 116 C688(1.10)  LDD0715  [11]
 LDCM0399  CL128 HCT 116 C688(0.95)  LDD0716  [11]
 LDCM0400  CL13 HCT 116 C688(1.21)  LDD0717  [11]
 LDCM0401  CL14 HCT 116 C688(1.30)  LDD0718  [11]
 LDCM0402  CL15 HCT 116 C688(1.06)  LDD0719  [11]
 LDCM0403  CL16 HCT 116 C688(1.07)  LDD0720  [11]
 LDCM0404  CL17 HCT 116 C688(0.65)  LDD0721  [11]
 LDCM0405  CL18 HCT 116 C688(0.96)  LDD0722  [11]
 LDCM0406  CL19 HCT 116 C688(0.88)  LDD0723  [11]
 LDCM0407  CL2 HCT 116 C688(1.19)  LDD0724  [11]
 LDCM0408  CL20 HCT 116 C688(1.06)  LDD0725  [11]
 LDCM0409  CL21 HCT 116 C688(0.89)  LDD0726  [11]
 LDCM0410  CL22 HCT 116 C688(0.80)  LDD0727  [11]
 LDCM0411  CL23 HCT 116 C688(1.02)  LDD0728  [11]
 LDCM0412  CL24 HCT 116 C688(1.02)  LDD0729  [11]
 LDCM0413  CL25 HCT 116 C688(0.95)  LDD0730  [11]
 LDCM0414  CL26 HCT 116 C688(1.23)  LDD0731  [11]
 LDCM0415  CL27 HCT 116 C688(0.99)  LDD0732  [11]
 LDCM0416  CL28 HCT 116 C688(1.25)  LDD0733  [11]
 LDCM0417  CL29 HCT 116 C688(1.11)  LDD0734  [11]
 LDCM0418  CL3 HCT 116 C688(1.47)  LDD0735  [11]
 LDCM0419  CL30 HCT 116 C688(1.11)  LDD0736  [11]
 LDCM0420  CL31 HEK-293T C688(1.22)  LDD1018  [11]
 LDCM0421  CL32 HCT 116 C688(1.08)  LDD0738  [11]
 LDCM0422  CL33 HCT 116 C688(0.91)  LDD0739  [11]
 LDCM0423  CL34 HCT 116 C688(0.91)  LDD0740  [11]
 LDCM0424  CL35 HCT 116 C688(1.04)  LDD0741  [11]
 LDCM0425  CL36 HCT 116 C688(0.80)  LDD0742  [11]
 LDCM0426  CL37 HCT 116 C688(1.05)  LDD0743  [11]
 LDCM0428  CL39 HCT 116 C688(1.15)  LDD0745  [11]
 LDCM0429  CL4 HCT 116 C688(1.01)  LDD0746  [11]
 LDCM0430  CL40 HCT 116 C688(0.89)  LDD0747  [11]
 LDCM0431  CL41 HCT 116 C688(0.95)  LDD0748  [11]
 LDCM0432  CL42 HCT 116 C688(0.71)  LDD0749  [11]
 LDCM0433  CL43 HCT 116 C688(0.98)  LDD0750  [11]
 LDCM0434  CL44 HCT 116 C688(1.13)  LDD0751  [11]
 LDCM0435  CL45 HCT 116 C688(1.01)  LDD0752  [11]
 LDCM0436  CL46 HCT 116 C688(0.82)  LDD0753  [11]
 LDCM0437  CL47 HCT 116 C688(0.87)  LDD0754  [11]
 LDCM0438  CL48 HCT 116 C688(1.08)  LDD0755  [11]
 LDCM0439  CL49 HCT 116 C688(0.77)  LDD0756  [11]
 LDCM0440  CL5 HCT 116 C688(1.16)  LDD0757  [11]
 LDCM0441  CL50 HCT 116 C688(0.93)  LDD0758  [11]
 LDCM0442  CL51 HCT 116 C688(1.02)  LDD0759  [11]
 LDCM0443  CL52 HCT 116 C688(1.04)  LDD0760  [11]
 LDCM0444  CL53 HCT 116 C688(0.95)  LDD0761  [11]
 LDCM0445  CL54 HCT 116 C688(0.93)  LDD0762  [11]
 LDCM0446  CL55 HCT 116 C688(0.94)  LDD0763  [11]
 LDCM0447  CL56 HCT 116 C688(0.87)  LDD0764  [11]
 LDCM0448  CL57 HCT 116 C688(0.81)  LDD0765  [11]
 LDCM0449  CL58 HCT 116 C688(1.03)  LDD0766  [11]
 LDCM0450  CL59 HCT 116 C688(1.03)  LDD0767  [11]
 LDCM0451  CL6 HCT 116 C688(1.30)  LDD0768  [11]
 LDCM0452  CL60 HCT 116 C688(0.86)  LDD0769  [11]
 LDCM0453  CL61 HEK-293T C242(0.85); C688(0.94)  LDD1656  [33]
 LDCM0454  CL62 HEK-293T C242(1.05); C688(1.13)  LDD1657  [33]
 LDCM0455  CL63 HEK-293T C242(0.86); C688(1.08)  LDD1658  [33]
 LDCM0456  CL64 HEK-293T C242(0.95); C688(1.11)  LDD1659  [33]
 LDCM0457  CL65 HEK-293T C242(1.18); C688(1.12)  LDD1660  [33]
 LDCM0458  CL66 HEK-293T C688(1.16)  LDD1661  [33]
 LDCM0459  CL67 HEK-293T C242(0.85); C688(1.14)  LDD1662  [33]
 LDCM0460  CL68 HEK-293T C242(0.69); C688(1.16)  LDD1663  [33]
 LDCM0461  CL69 HEK-293T C242(0.88); C688(1.14)  LDD1664  [33]
 LDCM0462  CL7 HCT 116 C688(1.14)  LDD0779  [11]
 LDCM0463  CL70 HEK-293T C242(1.08); C688(1.15)  LDD1666  [33]
 LDCM0464  CL71 HEK-293T C242(0.86); C688(1.21)  LDD1667  [33]
 LDCM0465  CL72 HEK-293T C242(0.95); C688(1.10)  LDD1668  [33]
 LDCM0466  CL73 HEK-293T C242(0.81); C688(0.99)  LDD1669  [33]
 LDCM0467  CL74 HEK-293T C242(0.94); C688(1.08)  LDD1670  [33]
 LDCM0469  CL76 HEK-293T C688(1.18)  LDD1067  [11]
 LDCM0470  CL77 HEK-293T C688(1.06)  LDD1068  [11]
 LDCM0471  CL78 HEK-293T C688(0.90)  LDD1069  [11]
 LDCM0472  CL79 HEK-293T C688(0.86)  LDD1070  [11]
 LDCM0473  CL8 HCT 116 C688(1.05)  LDD0790  [11]
 LDCM0474  CL80 HEK-293T C688(1.06)  LDD1072  [11]
 LDCM0475  CL81 HEK-293T C688(0.85)  LDD1073  [11]
 LDCM0476  CL82 HEK-293T C688(0.78)  LDD1074  [11]
 LDCM0477  CL83 HEK-293T C688(0.78)  LDD1075  [11]
 LDCM0478  CL84 HEK-293T C688(1.05)  LDD1076  [11]
 LDCM0479  CL85 HEK-293T C688(1.03)  LDD1077  [11]
 LDCM0480  CL86 HEK-293T C688(0.98)  LDD1078  [11]
 LDCM0481  CL87 HEK-293T C688(1.20)  LDD1079  [11]
 LDCM0482  CL88 HEK-293T C688(1.35)  LDD1080  [11]
 LDCM0483  CL89 HEK-293T C688(0.98)  LDD1081  [11]
 LDCM0484  CL9 HCT 116 C688(1.31)  LDD0801  [11]
 LDCM0485  CL90 HEK-293T C688(1.29)  LDD1083  [11]
 LDCM0486  CL91 HCT 116 C688(0.77)  LDD0803  [11]
 LDCM0487  CL92 HCT 116 C688(0.76)  LDD0804  [11]
 LDCM0488  CL93 HCT 116 C688(0.81)  LDD0805  [11]
 LDCM0489  CL94 HCT 116 C688(0.89)  LDD0806  [11]
 LDCM0490  CL95 HCT 116 C688(0.81)  LDD0807  [11]
 LDCM0491  CL96 HCT 116 C688(0.86)  LDD0808  [11]
 LDCM0492  CL97 HCT 116 C688(0.93)  LDD0809  [11]
 LDCM0493  CL98 HCT 116 C688(0.96)  LDD0810  [11]
 LDCM0494  CL99 HCT 116 C688(0.96)  LDD0811  [11]
 LDCM0495  E2913 HEK-293T C242(1.05); C688(1.19)  LDD1698  [33]
 LDCM0213  Electrophilic fragment 2 MDA-MB-231 C242(1.03)  LDD1702  [8]
 LDCM0625  F8 Ramos C688(1.02); C242(1.43)  LDD2187  [34]
 LDCM0572  Fragment10 Ramos C688(0.67); C242(1.09)  LDD2189  [34]
 LDCM0573  Fragment11 Ramos C688(0.34); C242(0.50)  LDD2190  [34]
 LDCM0574  Fragment12 Ramos C688(0.56); C242(0.92)  LDD2191  [34]
 LDCM0575  Fragment13 Ramos C688(0.72); C242(1.09)  LDD2192  [34]
 LDCM0576  Fragment14 Ramos C688(0.71); C242(0.76)  LDD2193  [34]
 LDCM0579  Fragment20 Ramos C688(0.61); C242(0.62)  LDD2194  [34]
 LDCM0580  Fragment21 Ramos C688(0.88); C242(0.86)  LDD2195  [34]
 LDCM0582  Fragment23 Ramos C688(0.85); C242(1.20)  LDD2196  [34]
 LDCM0578  Fragment27 Ramos C688(0.86); C242(0.94)  LDD2197  [34]
 LDCM0586  Fragment28 Ramos C688(0.60); C242(0.81)  LDD2198  [34]
 LDCM0588  Fragment30 Ramos C688(0.74); C242(1.33)  LDD2199  [34]
 LDCM0589  Fragment31 Ramos C688(0.79); C242(0.95)  LDD2200  [34]
 LDCM0590  Fragment32 Ramos C688(0.70); C242(1.05)  LDD2201  [34]
 LDCM0468  Fragment33 HEK-293T C242(0.82); C688(1.17)  LDD1671  [33]
 LDCM0596  Fragment38 Ramos C688(1.30); C242(0.96)  LDD2203  [34]
 LDCM0566  Fragment4 Ramos C688(0.69); C242(0.79)  LDD2184  [34]
 LDCM0427  Fragment51 HCT 116 C688(0.89)  LDD0744  [11]
 LDCM0610  Fragment52 Ramos C688(0.75); C242(1.32)  LDD2204  [34]
 LDCM0614  Fragment56 Ramos C688(0.73); C242(1.28)  LDD2205  [34]
 LDCM0569  Fragment7 Ramos C688(0.79); C242(0.90)  LDD2186  [34]
 LDCM0571  Fragment9 Ramos C688(0.50); C242(0.82)  LDD2188  [34]
 LDCM0116  HHS-0101 DM93 Y438(0.91); Y322(18.42)  LDD0264  [10]
 LDCM0117  HHS-0201 DM93 Y438(0.87); Y322(7.88)  LDD0265  [10]
 LDCM0118  HHS-0301 DM93 Y438(0.94); Y322(9.71)  LDD0266  [10]
 LDCM0119  HHS-0401 DM93 Y892(0.45); Y438(0.73); Y322(7.62)  LDD0267  [10]
 LDCM0120  HHS-0701 DM93 Y438(0.50)  LDD0268  [10]
 LDCM0107  IAA HeLa H577(0.00); H614(0.00); H428(0.00); H591(0.00)  LDD0221  [24]
 LDCM0022  KB02 HEK-293T C688(0.93); C242(1.01)  LDD1492  [33]
 LDCM0023  KB03 HEK-293T C688(1.00); C242(0.99)  LDD1497  [33]
 LDCM0024  KB05 G361 C688(2.05)  LDD3311  [35]
 LDCM0145  MCC950 THP-1 1.48  LDD0370  [32]
 LDCM0509  N-(4-bromo-3,5-dimethylphenyl)-2-nitroacetamide MDA-MB-231 C688(1.02)  LDD2102  [8]
 LDCM0528  N-(4-bromophenyl)-2-cyano-N-phenylacetamide MDA-MB-231 C688(0.74)  LDD2121  [8]
 LDCM0109  NEM HeLa H543(0.00); H428(0.00); H577(0.00); H608(0.00)  LDD0223  [24]
 LDCM0499  Nucleophilic fragment 12b MDA-MB-231 C242(1.02); C688(1.13)  LDD2092  [8]
 LDCM0500  Nucleophilic fragment 13a MDA-MB-231 C688(0.91)  LDD2093  [8]
 LDCM0501  Nucleophilic fragment 13b MDA-MB-231 C242(1.31); C688(1.62)  LDD2094  [8]
 LDCM0503  Nucleophilic fragment 14b MDA-MB-231 C242(1.02); C688(0.17)  LDD2096  [8]
 LDCM0505  Nucleophilic fragment 15b MDA-MB-231 C242(0.90); C688(0.80)  LDD2098  [8]
 LDCM0506  Nucleophilic fragment 16a MDA-MB-231 C688(0.65)  LDD2099  [8]
 LDCM0507  Nucleophilic fragment 16b MDA-MB-231 C242(0.90); C688(0.56)  LDD2100  [8]
 LDCM0511  Nucleophilic fragment 18b MDA-MB-231 C242(1.12); C688(0.80)  LDD2104  [8]
 LDCM0512  Nucleophilic fragment 19a MDA-MB-231 C688(1.31)  LDD2105  [8]
 LDCM0513  Nucleophilic fragment 19b MDA-MB-231 C242(0.65)  LDD2106  [8]
 LDCM0514  Nucleophilic fragment 20a MDA-MB-231 C688(0.98)  LDD2107  [8]
 LDCM0515  Nucleophilic fragment 20b MDA-MB-231 C688(0.43)  LDD2108  [8]
 LDCM0516  Nucleophilic fragment 21a MDA-MB-231 C688(1.05)  LDD2109  [8]
 LDCM0517  Nucleophilic fragment 21b MDA-MB-231 C242(0.98)  LDD2110  [8]
 LDCM0518  Nucleophilic fragment 22a MDA-MB-231 C688(0.75)  LDD2111  [8]
 LDCM0521  Nucleophilic fragment 23b MDA-MB-231 C242(0.75); C688(1.83)  LDD2114  [8]
 LDCM0522  Nucleophilic fragment 24a MDA-MB-231 C688(0.63)  LDD2115  [8]
 LDCM0523  Nucleophilic fragment 24b MDA-MB-231 C242(1.08); C688(0.28)  LDD2116  [8]
 LDCM0525  Nucleophilic fragment 25b MDA-MB-231 C242(1.23); C688(0.31)  LDD2118  [8]
 LDCM0526  Nucleophilic fragment 26a MDA-MB-231 C688(1.73)  LDD2119  [8]
 LDCM0527  Nucleophilic fragment 26b MDA-MB-231 C688(0.86)  LDD2120  [8]
 LDCM0529  Nucleophilic fragment 27b MDA-MB-231 C242(1.41); C688(0.26)  LDD2122  [8]
 LDCM0530  Nucleophilic fragment 28a MDA-MB-231 C688(0.82)  LDD2123  [8]
 LDCM0531  Nucleophilic fragment 28b MDA-MB-231 C242(1.29); C688(0.23)  LDD2124  [8]
 LDCM0532  Nucleophilic fragment 29a MDA-MB-231 C688(0.62)  LDD2125  [8]
 LDCM0533  Nucleophilic fragment 29b MDA-MB-231 C242(1.05); C688(0.16)  LDD2126  [8]
 LDCM0534  Nucleophilic fragment 30a MDA-MB-231 C688(0.77)  LDD2127  [8]
 LDCM0535  Nucleophilic fragment 30b MDA-MB-231 C688(1.04)  LDD2128  [8]
 LDCM0536  Nucleophilic fragment 31 MDA-MB-231 C688(0.88)  LDD2129  [8]
 LDCM0543  Nucleophilic fragment 38 MDA-MB-231 C688(1.14)  LDD2136  [8]
 LDCM0544  Nucleophilic fragment 39 MDA-MB-231 C688(1.00)  LDD2137  [8]
 LDCM0211  Nucleophilic fragment 3b MDA-MB-231 C688(0.78)  LDD1700  [8]
 LDCM0547  Nucleophilic fragment 41 MDA-MB-231 C242(0.89); C688(0.50)  LDD2141  [8]
 LDCM0549  Nucleophilic fragment 43 MDA-MB-231 C688(1.08)  LDD2143  [8]
 LDCM0550  Nucleophilic fragment 5a MDA-MB-231 C688(2.66)  LDD2144  [8]
 LDCM0552  Nucleophilic fragment 6a MDA-MB-231 C688(0.87)  LDD2146  [8]
 LDCM0553  Nucleophilic fragment 6b MDA-MB-231 C688(3.13)  LDD2147  [8]
 LDCM0555  Nucleophilic fragment 7b MDA-MB-231 C242(1.27); C688(0.23)  LDD2149  [8]
 LDCM0556  Nucleophilic fragment 8a MDA-MB-231 C242(0.39); C688(0.40)  LDD2150  [8]
 LDCM0557  Nucleophilic fragment 8b MDA-MB-231 C242(1.04); C688(0.38)  LDD2151  [8]
 LDCM0628  OTUB2-COV-1 HEK-293T C688(0.62)  LDD2207  [36]

The Interaction Atlas With This Target

The Protein(s) Related To This Target

Transporter and channel
Click To Hide/Show 1 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Apoptosis regulator Bcl-2 (BCL2) Bcl-2 family P10415
Other
Click To Hide/Show 1 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Emerin (EMD) . P50402

References

1 Labeling Preferences of Diazirines with Protein Biomolecules. J Am Chem Soc. 2021 May 5;143(17):6691-6700. doi: 10.1021/jacs.1c02509. Epub 2021 Apr 20.
Mass spectrometry data entry: PXD025140
2 Quantitative and Site-Specific Chemoproteomic Profiling of Targets of Acrolein. Chem Res Toxicol. 2019 Mar 18;32(3):467-473. doi: 10.1021/acs.chemrestox.8b00343. Epub 2019 Jan 15.
3 Comparison of Different Competitive Proteome Profiling Approaches in Target Identification of Covalent Inhibitors. Chembiochem. 2022 Dec 16;23(24):e202200389. doi: 10.1002/cbic.202200389. Epub 2022 Nov 22.
4 Cyclopropenone, Cyclopropeniminium Ion, and Cyclopropenethione as Novel Electrophilic Warheads for Potential Target Discovery of Triple-Negative Breast Cancer. J Med Chem. 2023 Feb 23;66(4):2851-2864. doi: 10.1021/acs.jmedchem.2c01889. Epub 2023 Feb 10.
5 Tranylcypromine specificity for monoamine oxidase is limited by promiscuous protein labelling and lysosomal trapping. RSC Chem Biol. 2020 Aug 12;1(4):209-213. doi: 10.1039/d0cb00048e. eCollection 2020 Oct 1.
Mass spectrometry data entry: PXD018580
6 A Paal-Knorr agent for chemoproteomic profiling of targets of isoketals in cells. Chem Sci. 2021 Oct 15;12(43):14557-14563. doi: 10.1039/d1sc02230j. eCollection 2021 Nov 10.
Mass spectrometry data entry: PXD028270
7 An Azo Coupling-Based Chemoproteomic Approach to Systematically Profile the Tyrosine Reactivity in the Human Proteome. Anal Chem. 2021 Jul 27;93(29):10334-10342. doi: 10.1021/acs.analchem.1c01935. Epub 2021 Jul 12.
8 Nucleophilic covalent ligand discovery for the cysteine redoxome. Nat Chem Biol. 2023 Nov;19(11):1309-1319. doi: 10.1038/s41589-023-01330-5. Epub 2023 May 29.
Mass spectrometry data entry: PXD039908 , PXD029761
9 Chemoproteomic capture of RNA binding activity in living cells. Nat Commun. 2023 Oct 7;14(1):6282. doi: 10.1038/s41467-023-41844-z.
Mass spectrometry data entry: PXD044625
10 Discovery of a Cell-Active SuTEx Ligand of Prostaglandin Reductase 2. Chembiochem. 2021 Jun 15;22(12):2134-2139. doi: 10.1002/cbic.202000879. Epub 2021 Apr 29.
11 Reimagining high-throughput profiling of reactive cysteines for cell-based screening of large electrophile libraries. Nat Biotechnol. 2021 May;39(5):630-641. doi: 10.1038/s41587-020-00778-3. Epub 2021 Jan 4.
12 Global profiling of functional histidines in live cells using small-molecule photosensitizer and chemical probe relay labelling. Nat Chem. 2024 Jun 4. doi: 10.1038/s41557-024-01545-6. Online ahead of print.
Mass spectrometry data entry: PXD042377
13 Targeted Proteomic Approaches for Proteome-Wide Characterizations of the AMP-Binding Capacities of Kinases. J Proteome Res. 2022 Aug 5;21(8):2063-2070. doi: 10.1021/acs.jproteome.2c00225. Epub 2022 Jul 12.
14 Enhancing Cysteine Chemoproteomic Coverage through Systematic Assessment of Click Chemistry Product Fragmentation. Anal Chem. 2022 Mar 8;94(9):3800-3810. doi: 10.1021/acs.analchem.1c04402. Epub 2022 Feb 23.
Mass spectrometry data entry: PXD028853
15 SP3-Enabled Rapid and High Coverage Chemoproteomic Identification of Cell-State-Dependent Redox-Sensitive Cysteines. Mol Cell Proteomics. 2022 Apr;21(4):100218. doi: 10.1016/j.mcpro.2022.100218. Epub 2022 Feb 25.
Mass spectrometry data entry: PXD029500 , PXD031647
16 N-Acryloylindole-alkyne (NAIA) enables imaging and profiling new ligandable cysteines and oxidized thiols by chemoproteomics. Nat Commun. 2023 Jun 15;14(1):3564. doi: 10.1038/s41467-023-39268-w.
Mass spectrometry data entry: PXD041264
17 Chemoproteomic Profiling by Cysteine Fluoroalkylation Reveals Myrocin G as an Inhibitor of the Nonhomologous End Joining DNA Repair Pathway. J Am Chem Soc. 2021 Dec 8;143(48):20332-20342. doi: 10.1021/jacs.1c09724. Epub 2021 Nov 24.
Mass spectrometry data entry: PXD029255
18 Multiplexed CuAAC Suzuki-Miyaura Labeling for Tandem Activity-Based Chemoproteomic Profiling. Anal Chem. 2021 Feb 2;93(4):2610-2618. doi: 10.1021/acs.analchem.0c04726. Epub 2021 Jan 20.
Mass spectrometry data entry: PXD022279
19 A modification-centric assessment tool for the performance of chemoproteomic probes. Nat Chem Biol. 2022 Aug;18(8):904-912. doi: 10.1038/s41589-022-01074-8. Epub 2022 Jul 21.
Mass spectrometry data entry: PXD027758 , PXD027755 , PXD027760 , PXD027762 , PXD027756 , PXD027591 , PXD007149 , PXD030064 , PXD032392 , PXD027789 , PXD027767 , PXD027764
20 Solid Phase Synthesis of Fluorosulfate Containing Macrocycles for Chemoproteomic Workflows. bioRxiv [Preprint]. 2023 Feb 18:2023.02.17.529022. doi: 10.1101/2023.02.17.529022.
Mass spectrometry data entry: PXD039931
21 DFT-Guided Discovery of Ethynyl-Triazolyl-Phosphinates as Modular Electrophiles for Chemoselective Cysteine Bioconjugation and Profiling. Angew Chem Int Ed Engl. 2022 Oct 10;61(41):e202205348. doi: 10.1002/anie.202205348. Epub 2022 Aug 22.
Mass spectrometry data entry: PXD033004
22 Oxidative cyclization reagents reveal tryptophan cation- interactions. Nature. 2024 Mar;627(8004):680-687. doi: 10.1038/s41586-024-07140-6. Epub 2024 Mar 6.
Mass spectrometry data entry: PXD001377 , PXD005252
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Mass spectrometry data entry: PXD038010
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Mass spectrometry data entry: PXD041587
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Mass spectrometry data entry: PXD024915 , PXD024913
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Mass spectrometry data entry: PXD044402
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Mass spectrometry data entry: PXD027578
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Mass spectrometry data entry: PXD047840
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