Details of the Target
General Information of Target
Target ID | LDTP06479 | |||||
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Target Name | Tubulin-specific chaperone E (TBCE) | |||||
Gene Name | TBCE | |||||
Gene ID | 6905 | |||||
Synonyms |
Tubulin-specific chaperone E; Tubulin-folding cofactor E |
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3D Structure | ||||||
Sequence |
MSDTLTADVIGRRVEVNGEHATVRFAGVVPPVAGPWLGVEWDNPERGKHDGSHEGTVYFK
CRHPTGGSFIRPNKVNFGTDFLTAIKNRYVLEDGPEEDRKEQIVTIGNKPVETIGFDSIM KQQSQLSKLQEVSLRNCAVSCAGEKGGVAEACPNIRKVDLSKNLLSSWDEVIHIADQLRH LEVLNVSENKLKFPSGSVLTGTLSVLKVLVLNQTGITWAEVLRCVAGCPGLEELYLESNN IFISERPTDVLQTVKLLDLSSNQLIDENQLYLIAHLPRLEQLILSDTGISSLHFPDAGIG CKTSMFPSLKYLVVNDNQISQWSFFNELEKLPSLRALSCLRNPLTKEDKEAETARLLIIA SIGQLKTLNKCEILPEERRRAELDYRKAFGNEWKQAGGHKDPEKNRLSEEFLTAHPRYQF LCLKYGAPEDWELKTQQPLMLKNQLLTLKIKYPHQLDQKVLEKQLPGSMTIQKVKGLLSR LLKVPVSDLLLSYESPKKPGREIELENDLKSLQFYSVENGDCLLVRW |
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Target Bioclass |
Other
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Family |
TBCE family
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Subcellular location |
Cytoplasm
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Function |
Tubulin-folding protein; involved in the second step of the tubulin folding pathway and in the regulation of tubulin heterodimer dissociation. Required for correct organization of microtubule cytoskeleton and mitotic splindle, and maintenance of the neuronal microtubule network.
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Uniprot ID | ||||||
Ensemble ID | ||||||
HGNC ID |
Target Site Mutations in Different Cell Lines
Cell line | Mutation details | Probe for labeling this protein in this cell | |||
---|---|---|---|---|---|
SW620 | SNV: p.S290F | DBIA Probe Info | |||
UACC257 | SNV: p.A354T | DBIA Probe Info |
Probe(s) Labeling This Target
ABPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
---|---|---|---|---|---|
m-APA Probe Info |
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15.00 | LDD0402 | [1] | |
TH211 Probe Info |
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Y418(13.15); Y271(5.33) | LDD0257 | [2] | |
ONAyne Probe Info |
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K451(10.00) | LDD0275 | [3] | |
Probe 1 Probe Info |
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Y89(28.11); Y385(6.98) | LDD3495 | [4] | |
BTD Probe Info |
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C371(2.17) | LDD1700 | [5] | |
Johansson_61 Probe Info |
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_(10.32) | LDD1485 | [6] | |
DBIA Probe Info |
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C137(6.72); C141(2.51); C522(1.00) | LDD0080 | [7] | |
ATP probe Probe Info |
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K48(0.00); K424(0.00) | LDD0199 | [8] | |
4-Iodoacetamidophenylacetylene Probe Info |
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C152(0.00); C301(0.00); C522(0.00); C422(0.00) | LDD0038 | [9] | |
IA-alkyne Probe Info |
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C371(0.00); C224(0.00); C228(0.00); C152(0.00) | LDD0036 | [9] | |
IPIAA_H Probe Info |
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N.A. | LDD0030 | [10] | |
IPIAA_L Probe Info |
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N.A. | LDD0031 | [10] | |
Lodoacetamide azide Probe Info |
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C371(0.00); C152(0.00); C301(0.00); C522(0.00) | LDD0037 | [9] | |
NAIA_4 Probe Info |
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N.A. | LDD2226 | [11] | |
WYneN Probe Info |
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C152(0.00); C141(0.00) | LDD0021 | [12] | |
Compound 10 Probe Info |
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C141(0.00); C152(0.00); C301(0.00); C422(0.00) | LDD2216 | [13] | |
Compound 11 Probe Info |
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N.A. | LDD2213 | [13] | |
ENE Probe Info |
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N.A. | LDD0006 | [12] | |
IPM Probe Info |
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C141(0.00); C301(0.00) | LDD0005 | [12] | |
NHS Probe Info |
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N.A. | LDD0010 | [12] | |
STPyne Probe Info |
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N.A. | LDD0009 | [12] | |
TFBX Probe Info |
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C339(0.00); C301(0.00); C422(0.00); C141(0.00) | LDD0148 | [14] | |
VSF Probe Info |
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C141(0.00); C371(0.00) | LDD0007 | [12] | |
Phosphinate-6 Probe Info |
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C137(0.00); C301(0.00); C371(0.00); C141(0.00) | LDD0018 | [15] | |
1c-yne Probe Info |
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K434(0.00); K483(0.00) | LDD0228 | [16] | |
Acrolein Probe Info |
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C422(0.00); C141(0.00) | LDD0217 | [17] | |
Methacrolein Probe Info |
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C152(0.00); C141(0.00) | LDD0218 | [17] | |
W1 Probe Info |
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N.A. | LDD0236 | [18] | |
AOyne Probe Info |
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12.50 | LDD0443 | [19] | |
NAIA_5 Probe Info |
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C339(0.00); C152(0.00); C301(0.00); C371(0.00) | LDD2223 | [11] |
PAL-AfBPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
---|---|---|---|---|---|
C186 Probe Info |
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7.94 | LDD1864 | [20] | |
FFF probe14 Probe Info |
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20.00 | LDD0477 | [21] | |
FFF probe3 Probe Info |
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14.59 | LDD0465 | [21] |
Competitor(s) Related to This Target
Competitor ID | Name | Cell line | Binding Site(Ratio) | Interaction ID | Ref |
---|---|---|---|---|---|
LDCM0537 | 2-Cyano-N,N-dimethylacetamide | MDA-MB-231 | C137(1.30) | LDD2130 | [5] |
LDCM0524 | 2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide | MDA-MB-231 | C371(0.96); C141(0.98); C152(1.40); C422(1.24) | LDD2117 | [5] |
LDCM0558 | 2-Cyano-N-phenylacetamide | MDA-MB-231 | C371(1.10) | LDD2152 | [5] |
LDCM0510 | 3-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-3-oxopropanenitrile | MDA-MB-231 | C371(0.90) | LDD2103 | [5] |
LDCM0214 | AC1 | HCT 116 | C137(0.77); C141(0.65); C152(1.12); C371(1.10) | LDD0531 | [7] |
LDCM0215 | AC10 | HCT 116 | C137(0.89); C141(0.83); C152(0.78); C224(0.73) | LDD0532 | [7] |
LDCM0216 | AC100 | HCT 116 | C137(0.51); C141(1.10); C152(0.96); C371(1.02) | LDD0533 | [7] |
LDCM0217 | AC101 | HCT 116 | C137(0.65); C141(1.31); C152(1.01); C371(1.26) | LDD0534 | [7] |
LDCM0218 | AC102 | HCT 116 | C137(0.65); C141(1.09); C152(1.13); C371(0.98) | LDD0535 | [7] |
LDCM0219 | AC103 | HCT 116 | C137(0.49); C141(1.12); C152(0.96); C371(1.08) | LDD0536 | [7] |
LDCM0220 | AC104 | HCT 116 | C137(0.71); C141(1.03); C152(0.99); C371(1.01) | LDD0537 | [7] |
LDCM0221 | AC105 | HCT 116 | C137(0.52); C141(1.15); C152(1.06); C371(1.26) | LDD0538 | [7] |
LDCM0222 | AC106 | HCT 116 | C137(0.64); C141(1.23); C152(0.99); C371(1.25) | LDD0539 | [7] |
LDCM0223 | AC107 | HCT 116 | C137(0.56); C141(1.16); C152(1.07); C371(0.90) | LDD0540 | [7] |
LDCM0224 | AC108 | HCT 116 | C137(0.60); C141(1.17); C152(1.02); C371(0.93) | LDD0541 | [7] |
LDCM0225 | AC109 | HCT 116 | C137(0.77); C141(0.99); C152(1.01); C371(0.83) | LDD0542 | [7] |
LDCM0226 | AC11 | HCT 116 | C137(0.59); C141(0.63); C152(0.66); C224(0.62) | LDD0543 | [7] |
LDCM0227 | AC110 | HCT 116 | C137(0.63); C141(1.20); C152(0.85); C371(0.96) | LDD0544 | [7] |
LDCM0228 | AC111 | HCT 116 | C137(0.54); C141(1.27); C152(0.88); C371(0.94) | LDD0545 | [7] |
LDCM0229 | AC112 | HCT 116 | C137(0.58); C141(1.43); C152(0.91); C371(1.00) | LDD0546 | [7] |
LDCM0230 | AC113 | HCT 116 | C137(0.98); C141(0.95); C152(1.15); C224(0.79) | LDD0547 | [7] |
LDCM0231 | AC114 | HCT 116 | C137(0.91); C141(1.15); C152(0.93); C224(0.50) | LDD0548 | [7] |
LDCM0232 | AC115 | HCT 116 | C137(0.71); C141(1.21); C152(0.85); C224(0.50) | LDD0549 | [7] |
LDCM0233 | AC116 | HCT 116 | C137(0.67); C141(1.11); C152(0.87); C224(0.48) | LDD0550 | [7] |
LDCM0234 | AC117 | HCT 116 | C137(0.84); C141(1.19); C152(1.24); C224(0.58) | LDD0551 | [7] |
LDCM0235 | AC118 | HCT 116 | C137(0.82); C141(1.06); C152(0.93); C224(0.64) | LDD0552 | [7] |
LDCM0236 | AC119 | HCT 116 | C137(0.79); C141(1.00); C152(0.98); C224(0.67) | LDD0553 | [7] |
LDCM0237 | AC12 | HCT 116 | C137(0.86); C141(0.86); C152(0.82); C224(0.96) | LDD0554 | [7] |
LDCM0238 | AC120 | HCT 116 | C137(0.85); C141(0.91); C152(0.82); C224(0.55) | LDD0555 | [7] |
LDCM0239 | AC121 | HCT 116 | C137(1.04); C141(1.12); C152(0.99); C224(0.62) | LDD0556 | [7] |
LDCM0240 | AC122 | HCT 116 | C137(0.88); C141(0.82); C152(0.83); C224(0.55) | LDD0557 | [7] |
LDCM0241 | AC123 | HCT 116 | C137(1.14); C141(1.21); C152(1.08); C224(0.58) | LDD0558 | [7] |
LDCM0242 | AC124 | HCT 116 | C137(1.22); C141(1.17); C152(0.98); C224(0.67) | LDD0559 | [7] |
LDCM0243 | AC125 | HCT 116 | C137(0.93); C141(1.01); C152(1.03); C224(0.55) | LDD0560 | [7] |
LDCM0244 | AC126 | HCT 116 | C137(0.77); C141(0.94); C152(0.89); C224(0.50) | LDD0561 | [7] |
LDCM0245 | AC127 | HCT 116 | C137(0.84); C141(1.12); C152(0.89); C224(0.55) | LDD0562 | [7] |
LDCM0246 | AC128 | HCT 116 | C137(0.68); C141(0.96); C152(0.77); C371(1.42) | LDD0563 | [7] |
LDCM0247 | AC129 | HCT 116 | C137(1.30); C141(1.38); C152(0.69); C371(1.41) | LDD0564 | [7] |
LDCM0249 | AC130 | HCT 116 | C137(0.77); C141(1.02); C152(0.72); C371(1.54) | LDD0566 | [7] |
LDCM0250 | AC131 | HCT 116 | C137(1.41); C141(1.47); C152(0.78); C371(1.22) | LDD0567 | [7] |
LDCM0251 | AC132 | HCT 116 | C137(1.22); C141(1.34); C152(0.63); C371(1.67) | LDD0568 | [7] |
LDCM0252 | AC133 | HCT 116 | C137(0.75); C141(0.98); C152(0.67); C371(1.55) | LDD0569 | [7] |
LDCM0253 | AC134 | HCT 116 | C137(0.78); C141(1.26); C152(0.65); C371(1.71) | LDD0570 | [7] |
LDCM0254 | AC135 | HCT 116 | C137(0.83); C141(1.20); C152(0.65); C371(1.81) | LDD0571 | [7] |
LDCM0255 | AC136 | HCT 116 | C137(0.74); C141(1.02); C152(0.52); C371(1.26) | LDD0572 | [7] |
LDCM0256 | AC137 | HCT 116 | C137(0.96); C141(1.12); C152(0.39); C371(1.20) | LDD0573 | [7] |
LDCM0257 | AC138 | HCT 116 | C137(0.79); C141(1.35); C152(0.53); C371(1.48) | LDD0574 | [7] |
LDCM0258 | AC139 | HCT 116 | C137(0.81); C141(1.17); C152(0.70); C371(1.59) | LDD0575 | [7] |
LDCM0259 | AC14 | HCT 116 | C137(0.78); C141(0.78); C152(0.65); C224(0.75) | LDD0576 | [7] |
LDCM0260 | AC140 | HCT 116 | C137(0.73); C141(1.27); C152(0.61); C371(1.95) | LDD0577 | [7] |
LDCM0261 | AC141 | HCT 116 | C137(0.81); C141(1.16); C152(0.54); C371(1.63) | LDD0578 | [7] |
LDCM0262 | AC142 | HCT 116 | C137(1.04); C141(1.17); C152(0.65); C371(1.52) | LDD0579 | [7] |
LDCM0263 | AC143 | HCT 116 | C422(0.84); C152(0.88); C141(1.04); C371(1.11) | LDD0580 | [7] |
LDCM0264 | AC144 | HCT 116 | C422(0.79); C152(0.84); C371(1.30); C141(1.32) | LDD0581 | [7] |
LDCM0265 | AC145 | HCT 116 | C422(0.89); C152(0.94); C141(1.09); C371(1.16) | LDD0582 | [7] |
LDCM0266 | AC146 | HCT 116 | C422(0.90); C152(1.07); C141(1.23); C371(1.26) | LDD0583 | [7] |
LDCM0267 | AC147 | HCT 116 | C422(0.73); C152(1.02); C371(1.21); C141(1.27) | LDD0584 | [7] |
LDCM0268 | AC148 | HCT 116 | C152(0.83); C422(1.23); C371(1.47); C141(1.90) | LDD0585 | [7] |
LDCM0269 | AC149 | HCT 116 | C152(0.77); C422(1.03); C371(1.36); C141(1.51) | LDD0586 | [7] |
LDCM0270 | AC15 | HCT 116 | C224(0.62); C228(0.62); C152(0.65); C141(0.70) | LDD0587 | [7] |
LDCM0271 | AC150 | HCT 116 | C422(0.90); C152(1.02); C371(1.08); C141(1.13) | LDD0588 | [7] |
LDCM0272 | AC151 | HCT 116 | C422(0.94); C141(0.97); C152(1.11); C371(1.20) | LDD0589 | [7] |
LDCM0273 | AC152 | HCT 116 | C422(0.84); C152(0.90); C371(1.10); C141(1.26) | LDD0590 | [7] |
LDCM0274 | AC153 | HCT 116 | C152(0.98); C422(1.02); C371(1.63); C141(2.24) | LDD0591 | [7] |
LDCM0621 | AC154 | HCT 116 | C141(1.21); C152(1.01); C371(1.21); C422(0.87) | LDD2158 | [7] |
LDCM0622 | AC155 | HCT 116 | C141(1.00); C152(0.89); C371(1.20); C422(0.91) | LDD2159 | [7] |
LDCM0623 | AC156 | HCT 116 | C141(0.81); C152(1.24); C371(1.19); C422(1.05) | LDD2160 | [7] |
LDCM0624 | AC157 | HCT 116 | C141(1.02); C152(1.26); C371(1.29); C422(0.93) | LDD2161 | [7] |
LDCM0276 | AC17 | HCT 116 | C224(0.77); C228(0.77); C137(0.94); C422(0.99) | LDD0593 | [7] |
LDCM0277 | AC18 | HCT 116 | C137(0.51); C224(0.65); C228(0.65); C422(0.86) | LDD0594 | [7] |
LDCM0278 | AC19 | HCT 116 | C137(0.66); C422(0.88); C224(0.92); C228(0.92) | LDD0595 | [7] |
LDCM0279 | AC2 | HCT 116 | C141(0.85); C137(0.87); C422(0.88); C152(0.97) | LDD0596 | [7] |
LDCM0280 | AC20 | HCT 116 | C224(0.71); C228(0.71); C137(0.88); C152(0.98) | LDD0597 | [7] |
LDCM0281 | AC21 | HCT 116 | C137(0.79); C224(0.89); C228(0.89); C152(0.95) | LDD0598 | [7] |
LDCM0282 | AC22 | HCT 116 | C152(0.91); C371(0.92); C224(1.10); C228(1.10) | LDD0599 | [7] |
LDCM0283 | AC23 | HCT 116 | C224(0.91); C228(0.91); C371(0.96); C152(0.99) | LDD0600 | [7] |
LDCM0284 | AC24 | HCT 116 | C224(1.01); C228(1.01); C422(1.05); C137(1.06) | LDD0601 | [7] |
LDCM0285 | AC25 | HCT 116 | C137(0.76); C422(0.83); C152(0.84); C141(0.98) | LDD0602 | [7] |
LDCM0286 | AC26 | HCT 116 | C152(0.67); C422(0.71); C137(0.72); C371(1.12) | LDD0603 | [7] |
LDCM0287 | AC27 | HCT 116 | C152(0.65); C422(0.70); C137(0.75); C141(0.91) | LDD0604 | [7] |
LDCM0288 | AC28 | HCT 116 | C152(0.64); C422(0.70); C137(0.71); C141(1.04) | LDD0605 | [7] |
LDCM0289 | AC29 | HCT 116 | C137(0.56); C152(0.61); C422(0.68); C141(1.05) | LDD0606 | [7] |
LDCM0290 | AC3 | HCT 116 | C141(0.83); C137(0.89); C422(0.90); C152(1.00) | LDD0607 | [7] |
LDCM0291 | AC30 | HCT 116 | C137(0.49); C152(0.57); C422(0.66); C141(0.99) | LDD0608 | [7] |
LDCM0292 | AC31 | HCT 116 | C152(0.64); C422(0.66); C137(0.71); C141(1.08) | LDD0609 | [7] |
LDCM0293 | AC32 | HCT 116 | C152(0.53); C422(0.57); C137(0.57); C141(1.33) | LDD0610 | [7] |
LDCM0294 | AC33 | HCT 116 | C422(0.62); C152(0.65); C137(0.71); C371(1.05) | LDD0611 | [7] |
LDCM0295 | AC34 | HCT 116 | C422(0.62); C137(0.64); C152(0.70); C371(1.04) | LDD0612 | [7] |
LDCM0296 | AC35 | HCT 116 | C141(0.81); C371(0.89); C152(1.31); C422(1.31) | LDD0613 | [7] |
LDCM0297 | AC36 | HCT 116 | C141(0.98); C371(1.02); C137(1.12); C152(1.17) | LDD0614 | [7] |
LDCM0298 | AC37 | HCT 116 | C141(0.77); C371(1.02); C152(1.03); C422(1.06) | LDD0615 | [7] |
LDCM0299 | AC38 | HCT 116 | C141(0.80); C137(1.02); C422(1.07); C152(1.08) | LDD0616 | [7] |
LDCM0300 | AC39 | HCT 116 | C141(0.92); C152(0.98); C137(1.07); C422(1.10) | LDD0617 | [7] |
LDCM0301 | AC4 | HCT 116 | C141(0.77); C422(0.85); C137(0.90); C152(1.06) | LDD0618 | [7] |
LDCM0302 | AC40 | HCT 116 | C141(0.91); C137(0.96); C422(0.99); C152(1.08) | LDD0619 | [7] |
LDCM0303 | AC41 | HCT 116 | C152(0.96); C137(1.01); C141(1.05); C371(1.10) | LDD0620 | [7] |
LDCM0304 | AC42 | HCT 116 | C371(0.91); C152(0.93); C422(0.98); C141(0.99) | LDD0621 | [7] |
LDCM0305 | AC43 | HCT 116 | C371(0.93); C152(0.95); C141(0.96); C422(1.01) | LDD0622 | [7] |
LDCM0306 | AC44 | HCT 116 | C371(0.91); C152(1.01); C141(1.02); C422(1.03) | LDD0623 | [7] |
LDCM0307 | AC45 | HCT 116 | C152(0.86); C371(0.93); C422(1.00); C141(1.04) | LDD0624 | [7] |
LDCM0308 | AC46 | HCT 116 | C137(0.95); C422(1.01); C141(1.05); C152(1.07) | LDD0625 | [7] |
LDCM0309 | AC47 | HCT 116 | C137(0.91); C141(0.99); C422(0.99); C152(1.00) | LDD0626 | [7] |
LDCM0310 | AC48 | HCT 116 | C141(0.93); C152(1.05); C422(1.05); C137(1.16) | LDD0627 | [7] |
LDCM0311 | AC49 | HCT 116 | C152(0.89); C422(0.95); C137(1.05); C371(1.23) | LDD0628 | [7] |
LDCM0312 | AC5 | HCT 116 | C141(0.69); C137(0.87); C422(0.89); C152(1.13) | LDD0629 | [7] |
LDCM0313 | AC50 | HCT 116 | C422(0.97); C152(0.99); C137(1.15); C371(1.29) | LDD0630 | [7] |
LDCM0314 | AC51 | HCT 116 | C141(0.87); C137(1.00); C371(1.12); C422(1.22) | LDD0631 | [7] |
LDCM0315 | AC52 | HCT 116 | C137(1.00); C141(1.06); C422(1.07); C152(1.17) | LDD0632 | [7] |
LDCM0316 | AC53 | HCT 116 | C422(0.91); C137(0.94); C152(0.98); C371(1.06) | LDD0633 | [7] |
LDCM0317 | AC54 | HCT 116 | C141(1.03); C371(1.09); C422(1.10); C137(1.13) | LDD0634 | [7] |
LDCM0318 | AC55 | HCT 116 | C422(0.87); C137(0.92); C152(1.08); C371(1.17) | LDD0635 | [7] |
LDCM0319 | AC56 | HCT 116 | C137(0.93); C152(1.05); C422(1.12); C141(1.23) | LDD0636 | [7] |
LDCM0320 | AC57 | HCT 116 | C422(0.83); C152(0.84); C137(0.86); C141(1.30) | LDD0637 | [7] |
LDCM0321 | AC58 | HCT 116 | C137(0.77); C152(0.82); C422(0.83); C141(1.15) | LDD0638 | [7] |
LDCM0322 | AC59 | HCT 116 | C152(0.73); C137(0.84); C422(0.84); C141(1.48) | LDD0639 | [7] |
LDCM0323 | AC6 | HCT 116 | C371(0.62); C152(0.71); C137(0.73); C224(0.73) | LDD0640 | [7] |
LDCM0324 | AC60 | HCT 116 | C152(0.70); C422(0.81); C137(0.91); C371(1.29) | LDD0641 | [7] |
LDCM0325 | AC61 | HCT 116 | C152(0.77); C137(0.87); C422(0.88); C371(1.28) | LDD0642 | [7] |
LDCM0326 | AC62 | HCT 116 | C152(0.74); C422(0.81); C137(1.04); C141(1.41) | LDD0643 | [7] |
LDCM0327 | AC63 | HCT 116 | C152(0.72); C422(0.87); C137(1.15); C141(1.37) | LDD0644 | [7] |
LDCM0328 | AC64 | HCT 116 | C152(0.71); C422(0.85); C137(1.15); C371(1.44) | LDD0645 | [7] |
LDCM0329 | AC65 | HCT 116 | C152(0.77); C422(0.79); C137(0.80); C141(1.52) | LDD0646 | [7] |
LDCM0330 | AC66 | HCT 116 | C137(0.76); C152(0.86); C422(0.89); C371(1.46) | LDD0647 | [7] |
LDCM0331 | AC67 | HCT 116 | C152(0.72); C137(0.77); C422(0.82); C141(1.57) | LDD0648 | [7] |
LDCM0332 | AC68 | HCT 116 | C152(0.78); C141(0.90); C137(0.96); C371(1.03) | LDD0649 | [7] |
LDCM0333 | AC69 | HCT 116 | C141(0.73); C152(0.74); C371(0.80); C137(1.04) | LDD0650 | [7] |
LDCM0334 | AC7 | HCT 116 | C371(0.71); C137(0.77); C141(0.79); C224(0.80) | LDD0651 | [7] |
LDCM0335 | AC70 | HCT 116 | C152(0.73); C141(0.80); C137(0.87); C371(1.09) | LDD0652 | [7] |
LDCM0336 | AC71 | HCT 116 | C371(0.74); C141(0.84); C152(0.94); C137(1.10) | LDD0653 | [7] |
LDCM0337 | AC72 | HCT 116 | C141(0.85); C137(0.87); C152(0.88); C371(1.09) | LDD0654 | [7] |
LDCM0338 | AC73 | HCT 116 | C141(0.77); C152(0.80); C137(0.85); C371(1.11) | LDD0655 | [7] |
LDCM0339 | AC74 | HCT 116 | C141(0.70); C371(0.84); C152(0.86); C137(0.96) | LDD0656 | [7] |
LDCM0340 | AC75 | HCT 116 | C141(0.84); C152(0.90); C137(0.93); C422(1.07) | LDD0657 | [7] |
LDCM0341 | AC76 | HCT 116 | C152(0.76); C141(0.78); C371(0.91); C137(1.07) | LDD0658 | [7] |
LDCM0342 | AC77 | HCT 116 | C141(0.83); C371(0.83); C152(0.83); C137(1.02) | LDD0659 | [7] |
LDCM0343 | AC78 | HCT 116 | C141(0.80); C152(0.81); C371(0.93); C137(1.04) | LDD0660 | [7] |
LDCM0344 | AC79 | HCT 116 | C152(0.88); C141(0.90); C137(0.98); C371(0.99) | LDD0661 | [7] |
LDCM0345 | AC8 | HCT 116 | C371(0.63); C137(0.67); C224(0.73); C228(0.73) | LDD0662 | [7] |
LDCM0346 | AC80 | HCT 116 | C141(0.91); C152(0.97); C422(1.01); C371(1.14) | LDD0663 | [7] |
LDCM0347 | AC81 | HCT 116 | C141(0.74); C137(1.02); C152(1.07); C371(1.17) | LDD0664 | [7] |
LDCM0348 | AC82 | HCT 116 | C141(0.85); C137(0.95); C371(0.96); C152(1.01) | LDD0665 | [7] |
LDCM0349 | AC83 | HCT 116 | C137(0.58); C422(0.78); C152(0.91); C141(0.95) | LDD0666 | [7] |
LDCM0350 | AC84 | HCT 116 | C137(0.62); C422(0.77); C141(0.88); C152(0.90) | LDD0667 | [7] |
LDCM0351 | AC85 | HCT 116 | C137(0.56); C422(0.78); C141(0.83); C152(0.89) | LDD0668 | [7] |
LDCM0352 | AC86 | HCT 116 | C152(0.81); C137(0.83); C422(0.83); C141(0.98) | LDD0669 | [7] |
LDCM0353 | AC87 | HCT 116 | C137(0.83); C141(0.87); C152(0.92); C422(0.94) | LDD0670 | [7] |
LDCM0354 | AC88 | HCT 116 | C141(0.89); C422(0.89); C137(0.91); C152(0.97) | LDD0671 | [7] |
LDCM0355 | AC89 | HCT 116 | C422(0.72); C137(0.77); C141(0.79); C152(0.83) | LDD0672 | [7] |
LDCM0357 | AC90 | HCT 116 | C152(0.91); C141(1.10); C371(1.13); C422(1.28) | LDD0674 | [7] |
LDCM0358 | AC91 | HCT 116 | C137(0.70); C422(0.72); C152(0.82); C141(0.94) | LDD0675 | [7] |
LDCM0359 | AC92 | HCT 116 | C137(0.63); C141(0.73); C422(0.74); C152(0.86) | LDD0676 | [7] |
LDCM0360 | AC93 | HCT 116 | C137(0.63); C141(0.68); C152(0.79); C422(0.84) | LDD0677 | [7] |
LDCM0361 | AC94 | HCT 116 | C422(0.77); C137(0.85); C141(0.88); C371(0.97) | LDD0678 | [7] |
LDCM0362 | AC95 | HCT 116 | C137(0.70); C422(0.78); C141(0.87); C152(0.95) | LDD0679 | [7] |
LDCM0363 | AC96 | HCT 116 | C422(0.68); C141(0.82); C137(0.84); C152(0.98) | LDD0680 | [7] |
LDCM0364 | AC97 | HCT 116 | C137(0.64); C422(0.74); C152(0.83); C141(0.90) | LDD0681 | [7] |
LDCM0365 | AC98 | HCT 116 | C422(0.53); C137(0.56); C152(0.98); C371(1.28) | LDD0682 | [7] |
LDCM0366 | AC99 | HCT 116 | C137(0.49); C422(0.71); C371(0.95); C152(1.03) | LDD0683 | [7] |
LDCM0248 | AKOS034007472 | HCT 116 | C137(0.87); C141(0.83); C152(0.77); C224(0.98) | LDD0565 | [7] |
LDCM0356 | AKOS034007680 | HCT 116 | C371(0.65); C224(0.67); C228(0.67); C152(0.68) | LDD0673 | [7] |
LDCM0275 | AKOS034007705 | HCT 116 | C224(0.50); C228(0.50); C137(0.57); C141(0.62) | LDD0592 | [7] |
LDCM0020 | ARS-1620 | HCC44 | C141(1.04); C422(1.02) | LDD2171 | [7] |
LDCM0108 | Chloroacetamide | HeLa | C422(0.00); H415(0.00); H180(0.00) | LDD0222 | [17] |
LDCM0632 | CL-Sc | Hep-G2 | C137(20.00); C371(0.95); C301(0.46) | LDD2227 | [11] |
LDCM0367 | CL1 | HCT 116 | C152(0.79); C371(0.94); C422(1.23); C141(1.25) | LDD0684 | [7] |
LDCM0368 | CL10 | HCT 116 | C224(0.59); C228(0.59); C422(0.82); C152(0.97) | LDD0685 | [7] |
LDCM0369 | CL100 | HCT 116 | C141(0.73); C137(0.74); C422(0.86); C152(1.05) | LDD0686 | [7] |
LDCM0370 | CL101 | HCT 116 | C371(0.63); C224(0.64); C228(0.64); C137(0.71) | LDD0687 | [7] |
LDCM0371 | CL102 | HCT 116 | C371(0.61); C152(0.72); C224(0.88); C228(0.88) | LDD0688 | [7] |
LDCM0372 | CL103 | HCT 116 | C371(0.79); C152(0.82); C141(0.87); C137(0.87) | LDD0689 | [7] |
LDCM0373 | CL104 | HCT 116 | C152(0.70); C371(0.81); C422(0.92); C224(0.92) | LDD0690 | [7] |
LDCM0374 | CL105 | HCT 116 | C224(0.63); C228(0.63); C137(0.78); C422(0.86) | LDD0691 | [7] |
LDCM0375 | CL106 | HCT 116 | C224(0.48); C228(0.48); C137(0.50); C422(0.85) | LDD0692 | [7] |
LDCM0376 | CL107 | HCT 116 | C137(0.46); C224(0.55); C228(0.55); C422(0.82) | LDD0693 | [7] |
LDCM0377 | CL108 | HCT 116 | C137(0.44); C224(0.55); C228(0.55); C422(0.82) | LDD0694 | [7] |
LDCM0378 | CL109 | HCT 116 | C224(0.71); C228(0.71); C137(0.74); C422(0.81) | LDD0695 | [7] |
LDCM0379 | CL11 | HCT 116 | C224(0.62); C228(0.62); C422(0.84); C137(0.95) | LDD0696 | [7] |
LDCM0380 | CL110 | HCT 116 | C137(0.65); C224(0.67); C228(0.67); C422(0.82) | LDD0697 | [7] |
LDCM0381 | CL111 | HCT 116 | C137(0.69); C224(0.82); C228(0.82); C422(0.88) | LDD0698 | [7] |
LDCM0382 | CL112 | HCT 116 | C152(0.81); C137(0.90); C422(0.96); C371(1.00) | LDD0699 | [7] |
LDCM0383 | CL113 | HCT 116 | C152(0.55); C137(0.60); C422(0.66); C371(1.22) | LDD0700 | [7] |
LDCM0384 | CL114 | HCT 116 | C152(0.65); C422(0.75); C137(0.77); C371(1.16) | LDD0701 | [7] |
LDCM0385 | CL115 | HCT 116 | C137(0.62); C152(0.65); C422(0.69); C371(1.06) | LDD0702 | [7] |
LDCM0386 | CL116 | HCT 116 | C137(0.65); C422(0.71); C152(0.79); C371(1.13) | LDD0703 | [7] |
LDCM0387 | CL117 | HCT 116 | C371(1.05); C152(1.08); C422(1.11); C137(1.15) | LDD0704 | [7] |
LDCM0388 | CL118 | HCT 116 | C152(0.94); C371(0.97); C422(1.01); C141(1.11) | LDD0705 | [7] |
LDCM0389 | CL119 | HCT 116 | C152(0.94); C141(0.98); C422(0.98); C137(1.09) | LDD0706 | [7] |
LDCM0390 | CL12 | HCT 116 | C224(0.60); C228(0.60); C422(0.87); C152(1.10) | LDD0707 | [7] |
LDCM0391 | CL120 | HCT 116 | C141(0.88); C137(0.98); C152(0.98); C422(1.05) | LDD0708 | [7] |
LDCM0392 | CL121 | HCT 116 | C152(0.74); C141(0.83); C422(0.89); C137(0.94) | LDD0709 | [7] |
LDCM0393 | CL122 | HCT 116 | C422(0.92); C152(0.98); C137(1.04); C371(1.14) | LDD0710 | [7] |
LDCM0394 | CL123 | HCT 116 | C422(0.97); C152(1.02); C137(1.07); C371(1.11) | LDD0711 | [7] |
LDCM0395 | CL124 | HCT 116 | C422(0.94); C152(0.97); C137(1.12); C371(1.15) | LDD0712 | [7] |
LDCM0396 | CL125 | HCT 116 | C137(0.80); C422(0.91); C152(1.02); C371(1.18) | LDD0713 | [7] |
LDCM0397 | CL126 | HCT 116 | C137(0.79); C152(0.88); C422(0.97); C371(1.17) | LDD0714 | [7] |
LDCM0398 | CL127 | HCT 116 | C137(0.71); C152(0.76); C422(0.86); C371(1.29) | LDD0715 | [7] |
LDCM0399 | CL128 | HCT 116 | C137(0.75); C152(0.80); C422(0.86); C141(1.02) | LDD0716 | [7] |
LDCM0400 | CL13 | HCT 116 | C224(0.72); C228(0.72); C422(0.87); C137(0.95) | LDD0717 | [7] |
LDCM0401 | CL14 | HCT 116 | C224(0.81); C228(0.81); C422(0.89); C152(0.97) | LDD0718 | [7] |
LDCM0402 | CL15 | HCT 116 | C224(0.84); C228(0.84); C422(0.92); C152(1.07) | LDD0719 | [7] |
LDCM0403 | CL16 | HCT 116 | C137(0.69); C371(0.72); C422(0.83); C152(1.09) | LDD0720 | [7] |
LDCM0404 | CL17 | HCT 116 | C422(0.86); C152(1.09); C137(1.47); C141(3.66) | LDD0721 | [7] |
LDCM0405 | CL18 | HCT 116 | C137(0.64); C422(0.75); C152(1.19); C141(1.57) | LDD0722 | [7] |
LDCM0406 | CL19 | HCT 116 | C137(0.75); C422(0.88); C152(1.15); C141(1.58) | LDD0723 | [7] |
LDCM0407 | CL2 | HCT 116 | C152(0.95); C141(1.04); C371(1.06); C224(1.09) | LDD0724 | [7] |
LDCM0408 | CL20 | HCT 116 | C137(0.64); C422(0.78); C152(1.14); C141(1.52) | LDD0725 | [7] |
LDCM0409 | CL21 | HCT 116 | C137(0.82); C422(0.87); C152(1.19); C141(1.60) | LDD0726 | [7] |
LDCM0410 | CL22 | HCT 116 | C137(0.66); C422(0.89); C152(1.55); C141(2.83) | LDD0727 | [7] |
LDCM0411 | CL23 | HCT 116 | C137(0.71); C422(0.84); C152(1.05); C141(1.22) | LDD0728 | [7] |
LDCM0412 | CL24 | HCT 116 | C137(0.65); C141(2.06); C152(1.12); C422(0.80) | LDD0729 | [7] |
LDCM0413 | CL25 | HCT 116 | C137(0.72); C141(1.51); C152(1.12); C422(0.87) | LDD0730 | [7] |
LDCM0414 | CL26 | HCT 116 | C137(0.60); C141(1.17); C152(1.16); C422(0.84) | LDD0731 | [7] |
LDCM0415 | CL27 | HCT 116 | C137(0.80); C141(1.23); C152(1.65); C422(0.82) | LDD0732 | [7] |
LDCM0416 | CL28 | HCT 116 | C137(0.71); C141(1.45); C152(1.21); C422(0.81) | LDD0733 | [7] |
LDCM0417 | CL29 | HCT 116 | C137(0.74); C141(1.37); C152(1.25); C422(0.79) | LDD0734 | [7] |
LDCM0418 | CL3 | HCT 116 | C137(1.47); C141(1.31); C152(1.09); C224(1.37) | LDD0735 | [7] |
LDCM0419 | CL30 | HCT 116 | C137(0.65); C141(1.02); C152(1.17); C422(0.89) | LDD0736 | [7] |
LDCM0420 | CL31 | HCT 116 | C137(0.80); C141(0.76); C152(0.98); C371(0.86) | LDD0737 | [7] |
LDCM0421 | CL32 | HCT 116 | C137(0.59); C141(0.83); C152(0.77); C371(0.95) | LDD0738 | [7] |
LDCM0422 | CL33 | HCT 116 | C137(0.77); C141(1.07); C152(0.59); C371(1.05) | LDD0739 | [7] |
LDCM0423 | CL34 | HCT 116 | C137(0.70); C141(1.36); C152(0.69); C371(0.81) | LDD0740 | [7] |
LDCM0424 | CL35 | HCT 116 | C137(0.52); C141(0.92); C152(0.65); C371(1.09) | LDD0741 | [7] |
LDCM0425 | CL36 | HCT 116 | C137(0.43); C141(0.81); C152(0.73); C371(0.91) | LDD0742 | [7] |
LDCM0426 | CL37 | HCT 116 | C137(0.90); C141(1.07); C152(0.77); C371(0.94) | LDD0743 | [7] |
LDCM0428 | CL39 | HCT 116 | C137(0.48); C141(0.78); C152(0.76); C371(0.97) | LDD0745 | [7] |
LDCM0429 | CL4 | HCT 116 | C137(1.48); C141(1.28); C152(0.80); C224(0.94) | LDD0746 | [7] |
LDCM0430 | CL40 | HCT 116 | C137(0.68); C141(0.99); C152(0.72); C371(0.94) | LDD0747 | [7] |
LDCM0431 | CL41 | HCT 116 | C137(0.58); C141(0.79); C152(0.79); C371(1.01) | LDD0748 | [7] |
LDCM0432 | CL42 | HCT 116 | C137(0.59); C141(0.97); C152(0.70); C371(0.88) | LDD0749 | [7] |
LDCM0433 | CL43 | HCT 116 | C137(0.76); C141(0.97); C152(0.71); C371(0.94) | LDD0750 | [7] |
LDCM0434 | CL44 | HCT 116 | C137(0.53); C141(0.80); C152(0.80); C371(0.93) | LDD0751 | [7] |
LDCM0435 | CL45 | HCT 116 | C137(0.48); C141(0.94); C152(0.75); C371(0.90) | LDD0752 | [7] |
LDCM0436 | CL46 | HCT 116 | C137(2.70); C141(2.73); C152(0.81); C224(1.87) | LDD0753 | [7] |
LDCM0437 | CL47 | HCT 116 | C137(1.84); C141(1.89); C152(0.97); C224(1.22) | LDD0754 | [7] |
LDCM0438 | CL48 | HCT 116 | C137(1.47); C141(1.57); C152(0.84); C224(1.26) | LDD0755 | [7] |
LDCM0439 | CL49 | HCT 116 | C137(1.65); C141(1.59); C152(1.15); C224(1.30) | LDD0756 | [7] |
LDCM0440 | CL5 | HCT 116 | C137(1.09); C141(1.03); C152(1.01); C224(0.84) | LDD0757 | [7] |
LDCM0441 | CL50 | HCT 116 | C137(1.95); C141(1.98); C152(0.82); C224(1.36) | LDD0758 | [7] |
LDCM0442 | CL51 | HCT 116 | C137(1.82); C141(1.76); C152(0.89); C224(1.47) | LDD0759 | [7] |
LDCM0443 | CL52 | HCT 116 | C137(1.96); C141(2.09); C152(0.80); C224(1.62) | LDD0760 | [7] |
LDCM0444 | CL53 | HCT 116 | C137(1.51); C141(1.64); C152(0.79); C224(1.33) | LDD0761 | [7] |
LDCM0445 | CL54 | HCT 116 | C137(2.05); C141(2.09); C152(0.74); C224(2.08) | LDD0762 | [7] |
LDCM0446 | CL55 | HCT 116 | C137(2.03); C141(2.01); C152(0.81); C224(2.56) | LDD0763 | [7] |
LDCM0447 | CL56 | HCT 116 | C137(1.26); C141(1.34); C152(0.88); C224(0.89) | LDD0764 | [7] |
LDCM0448 | CL57 | HCT 116 | C137(1.56); C141(1.58); C152(1.07); C224(1.61) | LDD0765 | [7] |
LDCM0449 | CL58 | HCT 116 | C137(1.47); C141(1.52); C152(0.72); C224(1.34) | LDD0766 | [7] |
LDCM0450 | CL59 | HCT 116 | C137(1.36); C141(1.35); C152(0.92); C224(1.12) | LDD0767 | [7] |
LDCM0451 | CL6 | HCT 116 | C137(0.94); C141(0.95); C152(1.01); C224(0.74) | LDD0768 | [7] |
LDCM0452 | CL60 | HCT 116 | C137(1.38); C141(1.35); C152(0.85); C224(1.32) | LDD0769 | [7] |
LDCM0453 | CL61 | HCT 116 | C137(0.94); C141(1.00); C224(0.93); C228(0.93) | LDD0770 | [7] |
LDCM0454 | CL62 | HCT 116 | C137(0.88); C141(0.95); C224(0.80); C228(0.80) | LDD0771 | [7] |
LDCM0455 | CL63 | HCT 116 | C137(0.97); C141(1.08); C224(0.73); C228(0.73) | LDD0772 | [7] |
LDCM0456 | CL64 | HCT 116 | C137(0.81); C141(0.81); C224(0.63); C228(0.63) | LDD0773 | [7] |
LDCM0457 | CL65 | HCT 116 | C137(0.86); C141(0.89); C224(0.75); C228(0.75) | LDD0774 | [7] |
LDCM0458 | CL66 | HCT 116 | C137(0.78); C141(0.83); C224(0.53); C228(0.53) | LDD0775 | [7] |
LDCM0459 | CL67 | HCT 116 | C137(0.87); C141(0.83); C224(0.55); C228(0.55) | LDD0776 | [7] |
LDCM0460 | CL68 | HCT 116 | C137(0.73); C141(0.76); C224(0.56); C228(0.56) | LDD0777 | [7] |
LDCM0461 | CL69 | HCT 116 | C137(0.95); C141(1.10); C224(0.50); C228(0.50) | LDD0778 | [7] |
LDCM0462 | CL7 | HCT 116 | C137(1.22); C141(1.31); C152(1.20); C224(0.64) | LDD0779 | [7] |
LDCM0463 | CL70 | HCT 116 | C137(0.88); C141(0.93); C224(0.55); C228(0.55) | LDD0780 | [7] |
LDCM0464 | CL71 | HCT 116 | C137(0.83); C141(0.92); C224(0.57); C228(0.57) | LDD0781 | [7] |
LDCM0465 | CL72 | HCT 116 | C137(0.88); C141(0.93); C224(1.04); C228(1.04) | LDD0782 | [7] |
LDCM0466 | CL73 | HCT 116 | C137(1.11); C141(1.23); C224(0.93); C228(0.93) | LDD0783 | [7] |
LDCM0467 | CL74 | HCT 116 | C137(1.02); C141(1.09); C224(0.77); C228(0.77) | LDD0784 | [7] |
LDCM0469 | CL76 | HCT 116 | C137(0.82); C141(0.85); C152(0.98); C371(0.93) | LDD0786 | [7] |
LDCM0470 | CL77 | HCT 116 | C137(0.96); C141(1.02); C152(0.82); C371(0.90) | LDD0787 | [7] |
LDCM0471 | CL78 | HCT 116 | C137(0.89); C141(0.95); C152(0.97); C371(1.01) | LDD0788 | [7] |
LDCM0472 | CL79 | HCT 116 | C137(0.78); C141(0.82); C152(0.97); C371(1.01) | LDD0789 | [7] |
LDCM0473 | CL8 | HCT 116 | C137(1.18); C141(1.67); C152(0.93); C224(0.63) | LDD0790 | [7] |
LDCM0474 | CL80 | HCT 116 | C137(0.79); C141(0.82); C152(0.90); C371(1.06) | LDD0791 | [7] |
LDCM0475 | CL81 | HCT 116 | C137(0.83); C141(0.83); C152(1.20); C371(0.99) | LDD0792 | [7] |
LDCM0476 | CL82 | HCT 116 | C137(0.83); C141(0.82); C152(0.97); C371(1.00) | LDD0793 | [7] |
LDCM0477 | CL83 | HCT 116 | C137(0.88); C141(0.82); C152(0.93); C371(0.93) | LDD0794 | [7] |
LDCM0478 | CL84 | HCT 116 | C137(0.81); C141(0.80); C152(0.79); C371(1.03) | LDD0795 | [7] |
LDCM0479 | CL85 | HCT 116 | C137(0.81); C141(0.81); C152(0.94); C371(1.01) | LDD0796 | [7] |
LDCM0480 | CL86 | HCT 116 | C137(0.81); C141(0.81); C152(1.37); C371(0.91) | LDD0797 | [7] |
LDCM0481 | CL87 | HCT 116 | C137(0.92); C141(0.82); C152(1.05); C371(1.00) | LDD0798 | [7] |
LDCM0482 | CL88 | HCT 116 | C137(0.91); C141(0.81); C152(0.86); C371(1.08) | LDD0799 | [7] |
LDCM0483 | CL89 | HCT 116 | C137(0.83); C141(0.81); C152(1.02); C371(1.06) | LDD0800 | [7] |
LDCM0484 | CL9 | HCT 116 | C137(1.07); C141(1.04); C152(0.94); C224(0.73) | LDD0801 | [7] |
LDCM0485 | CL90 | HCT 116 | C137(1.20); C141(1.20); C152(0.92); C371(0.95) | LDD0802 | [7] |
LDCM0486 | CL91 | HCT 116 | C137(0.96); C141(1.00); C152(0.91); C371(1.10) | LDD0803 | [7] |
LDCM0487 | CL92 | HCT 116 | C137(1.05); C141(1.14); C152(1.20); C371(0.99) | LDD0804 | [7] |
LDCM0488 | CL93 | HCT 116 | C137(0.93); C141(0.84); C152(1.13); C371(1.03) | LDD0805 | [7] |
LDCM0489 | CL94 | HCT 116 | C137(0.92); C141(0.87); C152(0.99); C371(1.05) | LDD0806 | [7] |
LDCM0490 | CL95 | HCT 116 | C137(0.96); C141(1.01); C152(1.28); C371(1.05) | LDD0807 | [7] |
LDCM0491 | CL96 | HCT 116 | C137(0.90); C141(0.99); C152(1.04); C371(1.06) | LDD0808 | [7] |
LDCM0492 | CL97 | HCT 116 | C137(0.88); C141(0.94); C152(0.89); C371(1.07) | LDD0809 | [7] |
LDCM0493 | CL98 | HCT 116 | C137(0.86); C141(0.87); C152(0.88); C371(1.28) | LDD0810 | [7] |
LDCM0494 | CL99 | HCT 116 | C137(0.89); C141(0.78); C152(1.19); C371(1.18) | LDD0811 | [7] |
LDCM0634 | CY-0357 | Hep-G2 | C371(1.45) | LDD2228 | [11] |
LDCM0495 | E2913 | HEK-293T | C371(1.01); C422(0.98); C522(0.99); C301(1.08) | LDD1698 | [22] |
LDCM0213 | Electrophilic fragment 2 | MDA-MB-231 | C301(1.23); C141(0.94) | LDD1702 | [5] |
LDCM0625 | F8 | Ramos | C371(1.73) | LDD2187 | [23] |
LDCM0572 | Fragment10 | Ramos | C371(1.23) | LDD2189 | [23] |
LDCM0573 | Fragment11 | Ramos | C371(0.64) | LDD2190 | [23] |
LDCM0574 | Fragment12 | Ramos | C371(0.75) | LDD2191 | [23] |
LDCM0575 | Fragment13 | Ramos | C371(0.98) | LDD2192 | [23] |
LDCM0576 | Fragment14 | Ramos | C371(0.62) | LDD2193 | [23] |
LDCM0579 | Fragment20 | Ramos | C371(0.62) | LDD2194 | [23] |
LDCM0580 | Fragment21 | Ramos | C371(0.92) | LDD2195 | [23] |
LDCM0582 | Fragment23 | Ramos | C371(0.83) | LDD2196 | [23] |
LDCM0578 | Fragment27 | Ramos | C371(0.97) | LDD2197 | [23] |
LDCM0586 | Fragment28 | Ramos | C371(0.64) | LDD2198 | [23] |
LDCM0588 | Fragment30 | Ramos | C371(1.29) | LDD2199 | [23] |
LDCM0589 | Fragment31 | Ramos | C371(0.90) | LDD2200 | [23] |
LDCM0590 | Fragment32 | Ramos | C371(0.74) | LDD2201 | [23] |
LDCM0468 | Fragment33 | HCT 116 | C137(0.81); C141(0.87); C224(0.58); C228(0.58) | LDD0785 | [7] |
LDCM0596 | Fragment38 | Ramos | C371(0.64) | LDD2203 | [23] |
LDCM0566 | Fragment4 | Ramos | C371(1.03) | LDD2184 | [23] |
LDCM0427 | Fragment51 | HCT 116 | C137(0.58); C141(1.29); C152(0.73); C371(0.78) | LDD0744 | [7] |
LDCM0610 | Fragment52 | Ramos | C371(1.58) | LDD2204 | [23] |
LDCM0614 | Fragment56 | Ramos | C371(1.04) | LDD2205 | [23] |
LDCM0569 | Fragment7 | Jurkat | _(10.32) | LDD1485 | [6] |
LDCM0571 | Fragment9 | Ramos | C371(0.68) | LDD2188 | [23] |
LDCM0107 | IAA | HeLa | N.A. | LDD0221 | [17] |
LDCM0022 | KB02 | HCT 116 | C137(6.72); C141(2.51); C522(1.00) | LDD0080 | [7] |
LDCM0023 | KB03 | HCT 116 | C137(3.84); C141(1.22); C522(0.93) | LDD0081 | [7] |
LDCM0024 | KB05 | HCT 116 | C137(5.67); C141(1.14); C522(1.03) | LDD0082 | [7] |
LDCM0509 | N-(4-bromo-3,5-dimethylphenyl)-2-nitroacetamide | MDA-MB-231 | C371(1.01) | LDD2102 | [5] |
LDCM0109 | NEM | HeLa | H180(0.00); H415(0.00) | LDD0223 | [17] |
LDCM0496 | Nucleophilic fragment 11a | MDA-MB-231 | C371(0.69) | LDD2089 | [5] |
LDCM0497 | Nucleophilic fragment 11b | MDA-MB-231 | C371(1.11); C141(1.19) | LDD2090 | [5] |
LDCM0499 | Nucleophilic fragment 12b | MDA-MB-231 | C141(0.90) | LDD2092 | [5] |
LDCM0500 | Nucleophilic fragment 13a | MDA-MB-231 | C371(0.99) | LDD2093 | [5] |
LDCM0501 | Nucleophilic fragment 13b | MDA-MB-231 | C371(0.92); C141(1.58) | LDD2094 | [5] |
LDCM0505 | Nucleophilic fragment 15b | MDA-MB-231 | C371(0.95); C141(1.07) | LDD2098 | [5] |
LDCM0506 | Nucleophilic fragment 16a | MDA-MB-231 | C371(1.10); C141(1.03); C137(1.75) | LDD2099 | [5] |
LDCM0512 | Nucleophilic fragment 19a | MDA-MB-231 | C371(0.93); C141(1.87) | LDD2105 | [5] |
LDCM0514 | Nucleophilic fragment 20a | MDA-MB-231 | C141(1.09) | LDD2107 | [5] |
LDCM0516 | Nucleophilic fragment 21a | MDA-MB-231 | C371(0.96); C141(1.14) | LDD2109 | [5] |
LDCM0518 | Nucleophilic fragment 22a | MDA-MB-231 | C371(0.97) | LDD2111 | [5] |
LDCM0521 | Nucleophilic fragment 23b | MDA-MB-231 | C371(0.68) | LDD2114 | [5] |
LDCM0526 | Nucleophilic fragment 26a | MDA-MB-231 | C371(2.48) | LDD2119 | [5] |
LDCM0527 | Nucleophilic fragment 26b | MDA-MB-231 | C371(0.52) | LDD2120 | [5] |
LDCM0530 | Nucleophilic fragment 28a | MDA-MB-231 | C371(0.71); C141(0.99) | LDD2123 | [5] |
LDCM0531 | Nucleophilic fragment 28b | MDA-MB-231 | C371(0.26) | LDD2124 | [5] |
LDCM0532 | Nucleophilic fragment 29a | MDA-MB-231 | C371(0.51); C141(0.95) | LDD2125 | [5] |
LDCM0534 | Nucleophilic fragment 30a | MDA-MB-231 | C371(1.15); C141(0.99) | LDD2127 | [5] |
LDCM0536 | Nucleophilic fragment 31 | MDA-MB-231 | C371(1.10); C141(0.64) | LDD2129 | [5] |
LDCM0542 | Nucleophilic fragment 37 | MDA-MB-231 | C371(1.05) | LDD2135 | [5] |
LDCM0543 | Nucleophilic fragment 38 | MDA-MB-231 | C141(1.16); C137(1.24); C422(0.86) | LDD2136 | [5] |
LDCM0544 | Nucleophilic fragment 39 | MDA-MB-231 | C141(0.95); C422(0.99) | LDD2137 | [5] |
LDCM0211 | Nucleophilic fragment 3b | MDA-MB-231 | C371(2.17) | LDD1700 | [5] |
LDCM0546 | Nucleophilic fragment 40 | MDA-MB-231 | C371(0.81); C141(1.19) | LDD2140 | [5] |
LDCM0547 | Nucleophilic fragment 41 | MDA-MB-231 | C141(0.56) | LDD2141 | [5] |
LDCM0552 | Nucleophilic fragment 6a | MDA-MB-231 | C371(1.21); C152(0.95) | LDD2146 | [5] |
LDCM0553 | Nucleophilic fragment 6b | MDA-MB-231 | C371(0.31) | LDD2147 | [5] |
LDCM0559 | Nucleophilic fragment 9b | MDA-MB-231 | C371(0.88); C141(2.35) | LDD2153 | [5] |
LDCM0627 | NUDT7-COV-1 | HEK-293T | C141(1.36); C141(1.29) | LDD2206 | [24] |
LDCM0628 | OTUB2-COV-1 | HEK-293T | C141(0.55) | LDD2207 | [24] |
LDCM0131 | RA190 | MM1.R | C141(1.22) | LDD0304 | [25] |
LDCM0021 | THZ1 | HCT 116 | C141(1.04); C422(1.02) | LDD2173 | [7] |
References