Details of the Target
General Information of Target
Target ID | LDTP11833 | |||||
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Target Name | Rab3 GTPase-activating protein non-catalytic subunit (RAB3GAP2) | |||||
Gene Name | RAB3GAP2 | |||||
Gene ID | 25782 | |||||
Synonyms |
KIAA0839; Rab3 GTPase-activating protein non-catalytic subunit; RGAP-iso; Rab3 GTPase-activating protein 150 kDa subunit; Rab3-GAP p150; Rab3-GAP150; Rab3-GAP regulatory subunit |
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3D Structure | ||||||
Sequence |
MAPAGRPGAKKGILERLESGEVVIGDGSFLITLEKRGYVKAGLWTPEAVIEHPDAVRQLH
MEFLRAGSNVMQTFTFSASEDNMESKWEDVNAAACDLAREVAGKGDALVAGGICQTSIYK YQKDEARIKKLFRQQLEVFAWKNVDFLIAEYFEHVEEAVWAVEVLKESDRPVAVTMCIGP EGDMHDITPGECAVRLVKAGASIVGVNCRFGPDTSLKTMELMKEGLEWAGLKAHLMVQPL GFHAPDCGKEGFVDLPEYPFGLESRVATRWDIQKYAREAYNLGVRYIGGCCGFEPYHIRA IAEELAPERGFLPPASEKHGSWGSGLDMHTKPWIRARARREYWENLLPASGRPFCPSLSK |
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Target Bioclass |
Other
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Family |
Rab3-GAP regulatory subunit family
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Subcellular location |
Cytoplasm
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Function |
Regulatory subunit of the Rab3 GTPase-activating (Rab3GAP) complex composed of RAB3GAP1 and RAB3GAP2, which has GTPase-activating protein (GAP) activity towards various Rab3 subfamily members (RAB3A, RAB3B, RAB3C and RAB3D), RAB5A and RAB43, and guanine nucleotide exchange factor (GEF) activity towards RAB18. As part of the Rab3GAP complex, acts as a GAP for Rab3 proteins by converting active RAB3-GTP to the inactive form RAB3-GDP. Rab3 proteins are involved in regulated exocytosis of neurotransmitters and hormones. The Rab3GAP complex, acts as a GEF for RAB18 by promoting the conversion of inactive RAB18-GDP to the active form RAB18-GTP. Required for recruiting and activating RAB18 at the endoplasmic reticulum (ER) membrane where it maintains proper ER structure. Required for normal eye and brain development. May participate in neurodevelopmental processes such as proliferation, migration and differentiation before synapse formation, and non-synaptic vesicular release of neurotransmitters.
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Uniprot ID | ||||||
Ensemble ID | ||||||
HGNC ID |
Target Site Mutations in Different Cell Lines
Cell line | Mutation details | Probe for labeling this protein in this cell | |||
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A431 | SNV: p.Q815Ter | DBIA Probe Info | |||
HCT15 | SNV: p.D448N | . | |||
HT | SNV: p.F1171V | DBIA Probe Info | |||
HT115 | SNV: p.S107N; p.P500L | . | |||
Ishikawa (Heraklio) 02 ER | Deletion: p.F1034LfsTer5 | DBIA Probe Info | |||
KYSE410 | SNV: p.T372I | DBIA Probe Info | |||
MV411 | SNV: p.Q1214K | DBIA Probe Info | |||
RKO | SNV: p.P1207L | DBIA Probe Info |
Probe(s) Labeling This Target
ABPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
---|---|---|---|---|---|
m-APA Probe Info |
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14.25 | LDD0402 | [1] | |
CY-1 Probe Info |
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100.00 | LDD0243 | [2] | |
STPyne Probe Info |
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K103(3.45); K1075(10.00); K1363(1.22); K558(1.41) | LDD0277 | [3] | |
BTD Probe Info |
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C608(1.12) | LDD2090 | [4] | |
AHL-Pu-1 Probe Info |
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C896(7.03) | LDD0170 | [5] | |
Acrolein Probe Info |
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H1314(0.00); H440(0.00) | LDD0225 | [6] | |
DBIA Probe Info |
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C1336(1.40); C67(1.50) | LDD0080 | [7] | |
ATP probe Probe Info |
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K1075(0.00); K1078(0.00) | LDD0199 | [8] | |
4-Iodoacetamidophenylacetylene Probe Info |
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C78(0.00); C896(0.00) | LDD0038 | [9] | |
IA-alkyne Probe Info |
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C608(0.00); C896(0.00) | LDD0036 | [9] | |
IPIAA_L Probe Info |
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N.A. | LDD0031 | [10] | |
Lodoacetamide azide Probe Info |
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C896(0.00); C78(0.00) | LDD0037 | [9] | |
WYneN Probe Info |
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N.A. | LDD0021 | [11] | |
WYneO Probe Info |
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N.A. | LDD0022 | [11] | |
IPM Probe Info |
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N.A. | LDD0147 | [12] | |
TFBX Probe Info |
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N.A. | LDD0148 | [12] | |
1c-yne Probe Info |
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N.A. | LDD0228 | [13] | |
W1 Probe Info |
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N.A. | LDD0236 | [14] | |
AOyne Probe Info |
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12.00 | LDD0443 | [15] | |
NAIA_5 Probe Info |
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C1336(0.00); C636(0.00); C155(0.00); C828(0.00) | LDD2223 | [16] |
PAL-AfBPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
---|---|---|---|---|---|
FFF probe11 Probe Info |
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5.40 | LDD0472 | [17] | |
FFF probe14 Probe Info |
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20.00 | LDD0477 | [17] |
Competitor(s) Related to This Target
Competitor ID | Name | Cell line | Binding Site(Ratio) | Interaction ID | Ref |
---|---|---|---|---|---|
LDCM0519 | 1-(6-methoxy-3,4-dihydroquinolin-1(2H)-yl)-2-nitroethan-1-one | MDA-MB-231 | C608(0.92) | LDD2112 | [4] |
LDCM0524 | 2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide | MDA-MB-231 | C608(1.15) | LDD2117 | [4] |
LDCM0510 | 3-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-3-oxopropanenitrile | MDA-MB-231 | C608(1.03) | LDD2103 | [4] |
LDCM0025 | 4SU-RNA | DM93 | C896(7.03) | LDD0170 | [5] |
LDCM0026 | 4SU-RNA+native RNA | HEK-293T | C608(2.11) | LDD0372 | [5] |
LDCM0214 | AC1 | HCT 116 | C1336(0.93); C391(1.15); C395(1.15); C608(1.11) | LDD0531 | [7] |
LDCM0215 | AC10 | HCT 116 | C1336(1.05); C391(0.95); C395(0.95); C608(0.93) | LDD0532 | [7] |
LDCM0216 | AC100 | HCT 116 | C1336(0.71); C391(0.82); C395(0.82) | LDD0533 | [7] |
LDCM0217 | AC101 | HCT 116 | C1336(0.75); C391(0.88); C395(0.88) | LDD0534 | [7] |
LDCM0218 | AC102 | HCT 116 | C1336(0.77); C391(0.76); C395(0.76) | LDD0535 | [7] |
LDCM0219 | AC103 | HCT 116 | C1336(0.83); C391(0.83); C395(0.83) | LDD0536 | [7] |
LDCM0220 | AC104 | HCT 116 | C1336(0.83); C391(0.69); C395(0.69) | LDD0537 | [7] |
LDCM0221 | AC105 | HCT 116 | C1336(0.83); C391(0.75); C395(0.75) | LDD0538 | [7] |
LDCM0222 | AC106 | HCT 116 | C1336(0.88); C391(0.70); C395(0.70) | LDD0539 | [7] |
LDCM0223 | AC107 | HCT 116 | C1336(0.90); C391(0.81); C395(0.81) | LDD0540 | [7] |
LDCM0224 | AC108 | HCT 116 | C1336(0.73); C391(0.76); C395(0.76) | LDD0541 | [7] |
LDCM0225 | AC109 | HCT 116 | C1336(0.74); C391(1.06); C395(1.06) | LDD0542 | [7] |
LDCM0226 | AC11 | HCT 116 | C1336(1.05); C391(1.24); C395(1.24); C608(0.83) | LDD0543 | [7] |
LDCM0227 | AC110 | HCT 116 | C1336(0.71); C391(0.81); C395(0.81) | LDD0544 | [7] |
LDCM0228 | AC111 | HCT 116 | C1336(0.74); C391(0.73); C395(0.73) | LDD0545 | [7] |
LDCM0229 | AC112 | HCT 116 | C1336(0.78); C391(0.69); C395(0.69) | LDD0546 | [7] |
LDCM0230 | AC113 | HCT 116 | C1336(0.95); C391(0.79); C395(0.79); C608(1.23) | LDD0547 | [7] |
LDCM0231 | AC114 | HCT 116 | C1336(0.97); C391(1.05); C395(0.95); C608(1.08) | LDD0548 | [7] |
LDCM0232 | AC115 | HCT 116 | C1336(1.06); C391(1.00); C395(1.08); C608(1.05) | LDD0549 | [7] |
LDCM0233 | AC116 | HCT 116 | C1336(1.07); C391(1.26); C395(1.11); C608(1.18) | LDD0550 | [7] |
LDCM0234 | AC117 | HCT 116 | C1336(0.96); C391(1.12); C395(1.11); C608(1.25) | LDD0551 | [7] |
LDCM0235 | AC118 | HCT 116 | C1336(0.94); C391(1.08); C395(1.06); C608(1.13) | LDD0552 | [7] |
LDCM0236 | AC119 | HCT 116 | C1336(1.01); C391(0.94); C395(0.93); C608(1.22) | LDD0553 | [7] |
LDCM0237 | AC12 | HCT 116 | C1336(0.97); C391(1.17); C395(1.17); C608(0.90) | LDD0554 | [7] |
LDCM0238 | AC120 | HCT 116 | C1336(1.08); C391(0.98); C395(1.00); C608(1.08) | LDD0555 | [7] |
LDCM0239 | AC121 | HCT 116 | C1336(1.01); C391(1.10); C395(1.17); C608(1.28) | LDD0556 | [7] |
LDCM0240 | AC122 | HCT 116 | C1336(1.00); C391(0.98); C395(1.04); C608(1.05) | LDD0557 | [7] |
LDCM0241 | AC123 | HCT 116 | C1336(0.96); C391(1.19); C395(1.17); C608(1.17) | LDD0558 | [7] |
LDCM0242 | AC124 | HCT 116 | C1336(0.89); C391(1.29); C395(1.11); C608(1.28) | LDD0559 | [7] |
LDCM0243 | AC125 | HCT 116 | C1336(0.94); C391(1.32); C395(1.32); C608(1.21) | LDD0560 | [7] |
LDCM0244 | AC126 | HCT 116 | C1336(1.07); C391(1.12); C395(1.20); C608(1.05) | LDD0561 | [7] |
LDCM0245 | AC127 | HCT 116 | C1336(1.05); C391(1.14); C395(1.27); C608(1.27) | LDD0562 | [7] |
LDCM0246 | AC128 | HCT 116 | C1336(1.41); C391(1.53); C395(1.53); C608(1.53) | LDD0563 | [7] |
LDCM0247 | AC129 | HCT 116 | C1336(1.01); C391(1.30); C395(1.30); C608(1.30) | LDD0564 | [7] |
LDCM0249 | AC130 | HCT 116 | C1336(1.09); C391(1.40); C395(1.40); C608(1.25) | LDD0566 | [7] |
LDCM0250 | AC131 | HCT 116 | C1336(0.88); C391(1.42); C395(1.42); C608(1.31) | LDD0567 | [7] |
LDCM0251 | AC132 | HCT 116 | C1336(1.04); C391(1.34); C395(1.34); C608(1.08) | LDD0568 | [7] |
LDCM0252 | AC133 | HCT 116 | C1336(1.10); C391(1.69); C395(1.69); C608(1.23) | LDD0569 | [7] |
LDCM0253 | AC134 | HCT 116 | C1336(1.14); C391(1.20); C395(1.20); C608(1.06) | LDD0570 | [7] |
LDCM0254 | AC135 | HCT 116 | C1336(1.09); C391(1.29); C395(1.29); C608(1.14) | LDD0571 | [7] |
LDCM0255 | AC136 | HCT 116 | C1336(1.17); C391(1.19); C395(1.19); C608(1.17) | LDD0572 | [7] |
LDCM0256 | AC137 | HCT 116 | C1336(1.04); C391(1.12); C395(1.12); C608(1.15) | LDD0573 | [7] |
LDCM0257 | AC138 | HCT 116 | C1336(1.12); C391(1.70); C395(1.70); C608(1.09) | LDD0574 | [7] |
LDCM0258 | AC139 | HCT 116 | C1336(1.12); C391(1.21); C395(1.21); C608(1.06) | LDD0575 | [7] |
LDCM0259 | AC14 | HCT 116 | C1336(1.05); C391(1.40); C395(1.40); C608(1.01) | LDD0576 | [7] |
LDCM0260 | AC140 | HCT 116 | C1336(1.10); C391(1.39); C395(1.39); C608(0.95) | LDD0577 | [7] |
LDCM0261 | AC141 | HCT 116 | C1336(1.06); C391(1.00); C395(1.00); C608(0.94) | LDD0578 | [7] |
LDCM0262 | AC142 | HCT 116 | C1336(1.00); C391(1.36); C395(1.36); C608(1.17) | LDD0579 | [7] |
LDCM0263 | AC143 | HCT 116 | C391(0.74); C395(0.74); C1336(1.01) | LDD0580 | [7] |
LDCM0264 | AC144 | HCT 116 | C395(0.93); C391(1.00); C1336(1.07) | LDD0581 | [7] |
LDCM0265 | AC145 | HCT 116 | C395(0.97); C1336(1.00); C391(1.00) | LDD0582 | [7] |
LDCM0266 | AC146 | HCT 116 | C1336(1.06); C395(1.24); C391(1.33) | LDD0583 | [7] |
LDCM0267 | AC147 | HCT 116 | C1336(1.12); C395(1.17); C391(1.24) | LDD0584 | [7] |
LDCM0268 | AC148 | HCT 116 | C391(1.17); C395(1.34); C1336(1.49) | LDD0585 | [7] |
LDCM0269 | AC149 | HCT 116 | C391(1.02); C1336(1.16); C395(1.42) | LDD0586 | [7] |
LDCM0270 | AC15 | HCT 116 | C608(0.97); C391(1.07); C395(1.07); C1336(1.08) | LDD0587 | [7] |
LDCM0271 | AC150 | HCT 116 | C391(1.04); C1336(1.07); C395(1.24) | LDD0588 | [7] |
LDCM0272 | AC151 | HCT 116 | C1336(0.96); C391(1.16); C395(1.21) | LDD0589 | [7] |
LDCM0273 | AC152 | HCT 116 | C391(1.02); C1336(1.23); C395(1.24) | LDD0590 | [7] |
LDCM0274 | AC153 | HCT 116 | C391(1.26); C395(1.57); C1336(1.71) | LDD0591 | [7] |
LDCM0621 | AC154 | HCT 116 | C1336(1.08); C391(1.23); C395(1.40) | LDD2158 | [7] |
LDCM0622 | AC155 | HCT 116 | C1336(0.99); C391(1.27); C395(1.30) | LDD2159 | [7] |
LDCM0623 | AC156 | HCT 116 | C1336(0.97); C391(1.25); C395(1.31) | LDD2160 | [7] |
LDCM0624 | AC157 | HCT 116 | C1336(0.86); C391(1.19); C395(1.29) | LDD2161 | [7] |
LDCM0276 | AC17 | HCT 116 | C391(0.83); C395(0.83); C1336(0.98) | LDD0593 | [7] |
LDCM0277 | AC18 | HCT 116 | C391(0.91); C395(0.91); C1336(1.29) | LDD0594 | [7] |
LDCM0278 | AC19 | HCT 116 | C1336(0.96); C391(1.02); C395(1.02) | LDD0595 | [7] |
LDCM0279 | AC2 | HCT 116 | C391(0.97); C395(0.97); C608(0.97); C1336(0.98) | LDD0596 | [7] |
LDCM0280 | AC20 | HCT 116 | C391(0.81); C395(0.81); C1336(1.01) | LDD0597 | [7] |
LDCM0281 | AC21 | HCT 116 | C391(0.95); C395(0.95); C1336(0.99) | LDD0598 | [7] |
LDCM0282 | AC22 | HCT 116 | C391(0.94); C395(0.94); C1336(0.99) | LDD0599 | [7] |
LDCM0283 | AC23 | HCT 116 | C391(0.68); C395(0.68); C1336(1.12) | LDD0600 | [7] |
LDCM0284 | AC24 | HCT 116 | C391(0.87); C395(0.87); C1336(0.98) | LDD0601 | [7] |
LDCM0285 | AC25 | HCT 116 | C391(0.92); C395(0.92); C608(0.96); C1336(1.05) | LDD0602 | [7] |
LDCM0286 | AC26 | HCT 116 | C391(0.77); C395(0.77); C608(0.81); C1336(1.08) | LDD0603 | [7] |
LDCM0287 | AC27 | HCT 116 | C608(0.85); C391(0.89); C395(0.89); C1336(1.09) | LDD0604 | [7] |
LDCM0288 | AC28 | HCT 116 | C608(0.88); C391(0.92); C395(0.92); C1336(1.10) | LDD0605 | [7] |
LDCM0289 | AC29 | HCT 116 | C391(0.71); C395(0.71); C608(0.87); C1336(1.03) | LDD0606 | [7] |
LDCM0290 | AC3 | HCT 116 | C1336(0.91); C608(0.97); C391(1.18); C395(1.18) | LDD0607 | [7] |
LDCM0291 | AC30 | HCT 116 | C608(0.75); C391(0.75); C395(0.75); C1336(1.09) | LDD0608 | [7] |
LDCM0292 | AC31 | HCT 116 | C608(0.96); C391(0.98); C395(0.98); C1336(1.12) | LDD0609 | [7] |
LDCM0293 | AC32 | HCT 116 | C608(0.68); C391(0.69); C395(0.69); C1336(1.24) | LDD0610 | [7] |
LDCM0294 | AC33 | HCT 116 | C608(0.80); C391(0.99); C395(0.99); C1336(1.14) | LDD0611 | [7] |
LDCM0295 | AC34 | HCT 116 | C608(0.91); C391(0.95); C395(0.95); C1336(1.28) | LDD0612 | [7] |
LDCM0296 | AC35 | HCT 116 | C1336(0.89); C608(0.97) | LDD0613 | [7] |
LDCM0297 | AC36 | HCT 116 | C608(0.89); C1336(0.91) | LDD0614 | [7] |
LDCM0298 | AC37 | HCT 116 | C1336(0.89); C608(0.96) | LDD0615 | [7] |
LDCM0299 | AC38 | HCT 116 | C1336(0.92); C608(0.93) | LDD0616 | [7] |
LDCM0300 | AC39 | HCT 116 | C608(0.96); C1336(1.05) | LDD0617 | [7] |
LDCM0301 | AC4 | HCT 116 | C391(0.92); C395(0.92); C1336(0.94); C608(1.01) | LDD0618 | [7] |
LDCM0302 | AC40 | HCT 116 | C608(1.04); C1336(1.11) | LDD0619 | [7] |
LDCM0303 | AC41 | HCT 116 | C608(0.93); C1336(1.01) | LDD0620 | [7] |
LDCM0304 | AC42 | HCT 116 | C1336(1.02); C608(1.05) | LDD0621 | [7] |
LDCM0305 | AC43 | HCT 116 | C608(0.86); C1336(1.03) | LDD0622 | [7] |
LDCM0306 | AC44 | HCT 116 | C608(0.96); C1336(1.06) | LDD0623 | [7] |
LDCM0307 | AC45 | HCT 116 | C608(1.01); C1336(1.15) | LDD0624 | [7] |
LDCM0308 | AC46 | HCT 116 | C608(0.88); C636(0.93); C1336(0.99); C391(1.23) | LDD0625 | [7] |
LDCM0309 | AC47 | HCT 116 | C608(0.84); C391(1.08); C395(1.08); C1336(1.08) | LDD0626 | [7] |
LDCM0310 | AC48 | HCT 116 | C608(0.93); C1336(1.11); C391(1.13); C395(1.13) | LDD0627 | [7] |
LDCM0311 | AC49 | HCT 116 | C608(0.76); C391(0.97); C395(0.97); C636(1.14) | LDD0628 | [7] |
LDCM0312 | AC5 | HCT 116 | C1336(0.99); C608(1.00); C391(1.19); C395(1.19) | LDD0629 | [7] |
LDCM0313 | AC50 | HCT 116 | C608(0.86); C636(0.98); C391(1.03); C395(1.03) | LDD0630 | [7] |
LDCM0314 | AC51 | HCT 116 | C1336(0.92); C608(0.96); C391(1.05); C395(1.05) | LDD0631 | [7] |
LDCM0315 | AC52 | HCT 116 | C608(0.87); C636(0.92); C1336(1.01); C391(1.23) | LDD0632 | [7] |
LDCM0316 | AC53 | HCT 116 | C608(0.81); C391(1.06); C395(1.06); C1336(1.14) | LDD0633 | [7] |
LDCM0317 | AC54 | HCT 116 | C391(0.89); C395(0.89); C636(1.01); C608(1.05) | LDD0634 | [7] |
LDCM0318 | AC55 | HCT 116 | C608(0.81); C636(0.97); C391(1.18); C395(1.18) | LDD0635 | [7] |
LDCM0319 | AC56 | HCT 116 | C608(0.96); C636(0.98); C391(1.02); C395(1.02) | LDD0636 | [7] |
LDCM0320 | AC57 | HCT 116 | C1336(1.07); C391(1.30); C395(1.30) | LDD0637 | [7] |
LDCM0321 | AC58 | HCT 116 | C391(1.06); C395(1.06); C1336(1.13) | LDD0638 | [7] |
LDCM0322 | AC59 | HCT 116 | C1336(1.16); C391(1.21); C395(1.21) | LDD0639 | [7] |
LDCM0323 | AC6 | HCT 116 | C608(0.92); C391(0.96); C395(0.96); C1336(1.06) | LDD0640 | [7] |
LDCM0324 | AC60 | HCT 116 | C1336(1.06); C391(1.16); C395(1.16) | LDD0641 | [7] |
LDCM0325 | AC61 | HCT 116 | C1336(1.06); C391(1.38); C395(1.38) | LDD0642 | [7] |
LDCM0326 | AC62 | HCT 116 | C1336(1.13); C391(2.18); C395(2.18) | LDD0643 | [7] |
LDCM0327 | AC63 | HCT 116 | C1336(1.06); C391(1.20); C395(1.20) | LDD0644 | [7] |
LDCM0328 | AC64 | HCT 116 | C1336(1.22); C391(1.77); C395(1.77) | LDD0645 | [7] |
LDCM0329 | AC65 | HCT 116 | C1336(1.22); C391(1.36); C395(1.36) | LDD0646 | [7] |
LDCM0330 | AC66 | HCT 116 | C1336(1.20); C391(1.46); C395(1.46) | LDD0647 | [7] |
LDCM0331 | AC67 | HCT 116 | C391(1.16); C395(1.16); C1336(1.29) | LDD0648 | [7] |
LDCM0332 | AC68 | HCT 116 | C391(0.96); C395(0.96); C1336(1.12) | LDD0649 | [7] |
LDCM0333 | AC69 | HCT 116 | C391(0.86); C395(0.86); C1336(1.19) | LDD0650 | [7] |
LDCM0334 | AC7 | HCT 116 | C608(0.99); C1336(1.10); C391(1.19); C395(1.19) | LDD0651 | [7] |
LDCM0335 | AC70 | HCT 116 | C391(0.91); C395(0.91); C1336(1.14) | LDD0652 | [7] |
LDCM0336 | AC71 | HCT 116 | C391(1.07); C395(1.07); C1336(1.14) | LDD0653 | [7] |
LDCM0337 | AC72 | HCT 116 | C391(0.86); C395(0.86); C1336(1.13) | LDD0654 | [7] |
LDCM0338 | AC73 | HCT 116 | C391(1.01); C395(1.01); C1336(1.45) | LDD0655 | [7] |
LDCM0339 | AC74 | HCT 116 | C391(1.07); C395(1.07); C1336(1.44) | LDD0656 | [7] |
LDCM0340 | AC75 | HCT 116 | C391(0.98); C395(0.98); C1336(1.57) | LDD0657 | [7] |
LDCM0341 | AC76 | HCT 116 | C391(0.97); C395(0.97); C1336(1.14) | LDD0658 | [7] |
LDCM0342 | AC77 | HCT 116 | C391(0.95); C395(0.95); C1336(1.19) | LDD0659 | [7] |
LDCM0343 | AC78 | HCT 116 | C391(1.04); C395(1.04); C1336(1.11) | LDD0660 | [7] |
LDCM0344 | AC79 | HCT 116 | C391(1.01); C395(1.01); C1336(1.16) | LDD0661 | [7] |
LDCM0345 | AC8 | HCT 116 | C391(0.81); C395(0.81); C608(0.84); C1336(1.11) | LDD0662 | [7] |
LDCM0346 | AC80 | HCT 116 | C391(0.92); C395(0.92); C1336(1.14) | LDD0663 | [7] |
LDCM0347 | AC81 | HCT 116 | C391(0.88); C395(0.88); C1336(1.07) | LDD0664 | [7] |
LDCM0348 | AC82 | HCT 116 | C391(0.95); C395(0.95); C1336(1.64) | LDD0665 | [7] |
LDCM0349 | AC83 | HCT 116 | C636(0.72); C608(0.73); C1336(1.43) | LDD0666 | [7] |
LDCM0350 | AC84 | HCT 116 | C608(0.78); C636(0.86); C1336(1.29) | LDD0667 | [7] |
LDCM0351 | AC85 | HCT 116 | C608(0.81); C636(0.92); C1336(1.17) | LDD0668 | [7] |
LDCM0352 | AC86 | HCT 116 | C608(0.82); C636(0.96); C1336(1.11) | LDD0669 | [7] |
LDCM0353 | AC87 | HCT 116 | C608(0.75); C1336(1.05); C636(1.42) | LDD0670 | [7] |
LDCM0354 | AC88 | HCT 116 | C608(0.75); C636(0.97); C1336(1.01) | LDD0671 | [7] |
LDCM0355 | AC89 | HCT 116 | C608(0.68); C636(0.78); C1336(1.15) | LDD0672 | [7] |
LDCM0357 | AC90 | HCT 116 | C608(0.65); C1336(1.12); C636(1.24) | LDD0674 | [7] |
LDCM0358 | AC91 | HCT 116 | C636(0.79); C608(0.97); C1336(1.34) | LDD0675 | [7] |
LDCM0359 | AC92 | HCT 116 | C608(0.83); C636(0.83); C1336(1.22) | LDD0676 | [7] |
LDCM0360 | AC93 | HCT 116 | C608(0.70); C636(0.82); C1336(1.03) | LDD0677 | [7] |
LDCM0361 | AC94 | HCT 116 | C636(0.92); C1336(1.11); C608(1.24) | LDD0678 | [7] |
LDCM0362 | AC95 | HCT 116 | C608(0.76); C1336(0.95); C636(1.12) | LDD0679 | [7] |
LDCM0363 | AC96 | HCT 116 | C636(0.83); C608(1.08); C1336(1.09) | LDD0680 | [7] |
LDCM0364 | AC97 | HCT 116 | C608(0.71); C636(0.77); C1336(1.17) | LDD0681 | [7] |
LDCM0365 | AC98 | HCT 116 | C391(0.76); C395(0.76); C1336(1.15) | LDD0682 | [7] |
LDCM0366 | AC99 | HCT 116 | C391(0.64); C395(0.64); C1336(0.75) | LDD0683 | [7] |
LDCM0248 | AKOS034007472 | HCT 116 | C1336(1.02); C391(1.27); C395(1.27); C608(1.04) | LDD0565 | [7] |
LDCM0356 | AKOS034007680 | HCT 116 | C608(0.96); C1336(1.05); C391(1.48); C395(1.48) | LDD0673 | [7] |
LDCM0275 | AKOS034007705 | HCT 116 | C608(0.88); C391(0.97); C395(0.97); C1336(1.45) | LDD0592 | [7] |
LDCM0156 | Aniline | NCI-H1299 | 11.35 | LDD0403 | [1] |
LDCM0632 | CL-Sc | Hep-G2 | C1336(20.00) | LDD2227 | [16] |
LDCM0367 | CL1 | HCT 116 | C608(0.86); C1336(0.93); C391(1.21); C395(1.21) | LDD0684 | [7] |
LDCM0368 | CL10 | HCT 116 | C608(0.79); C1336(1.07); C391(1.12); C395(1.12) | LDD0685 | [7] |
LDCM0369 | CL100 | HCT 116 | C1336(0.91); C608(1.01); C391(1.11); C395(1.11) | LDD0686 | [7] |
LDCM0370 | CL101 | HCT 116 | C608(0.85); C1336(1.12); C391(1.20); C395(1.20) | LDD0687 | [7] |
LDCM0371 | CL102 | HCT 116 | C608(0.89); C391(1.02); C395(1.02); C1336(1.05) | LDD0688 | [7] |
LDCM0372 | CL103 | HCT 116 | C608(0.97); C1336(1.05); C391(1.26); C395(1.26) | LDD0689 | [7] |
LDCM0373 | CL104 | HCT 116 | C608(0.93); C1336(1.01); C391(1.14); C395(1.14) | LDD0690 | [7] |
LDCM0374 | CL105 | HCT 116 | C391(1.07); C395(1.07); C1336(1.08) | LDD0691 | [7] |
LDCM0375 | CL106 | HCT 116 | C391(1.02); C395(1.02); C1336(1.27) | LDD0692 | [7] |
LDCM0376 | CL107 | HCT 116 | C391(1.09); C395(1.09); C1336(1.20) | LDD0693 | [7] |
LDCM0377 | CL108 | HCT 116 | C391(0.97); C395(0.97); C1336(1.20) | LDD0694 | [7] |
LDCM0378 | CL109 | HCT 116 | C391(0.92); C395(0.92); C1336(1.01) | LDD0695 | [7] |
LDCM0379 | CL11 | HCT 116 | C608(0.68); C1336(1.11); C391(1.17); C395(1.17) | LDD0696 | [7] |
LDCM0380 | CL110 | HCT 116 | C391(0.91); C395(0.91); C1336(1.11) | LDD0697 | [7] |
LDCM0381 | CL111 | HCT 116 | C391(0.96); C395(0.96); C1336(1.00) | LDD0698 | [7] |
LDCM0382 | CL112 | HCT 116 | C391(0.91); C395(0.91); C1336(0.98); C608(1.01) | LDD0699 | [7] |
LDCM0383 | CL113 | HCT 116 | C391(0.67); C395(0.67); C608(0.85); C1336(1.17) | LDD0700 | [7] |
LDCM0384 | CL114 | HCT 116 | C391(0.67); C395(0.67); C608(0.78); C1336(1.09) | LDD0701 | [7] |
LDCM0385 | CL115 | HCT 116 | C391(0.75); C395(0.75); C608(0.80); C1336(1.08) | LDD0702 | [7] |
LDCM0386 | CL116 | HCT 116 | C608(0.88); C391(0.93); C395(0.93); C1336(1.12) | LDD0703 | [7] |
LDCM0387 | CL117 | HCT 116 | C608(1.02); C1336(1.38) | LDD0704 | [7] |
LDCM0388 | CL118 | HCT 116 | C608(0.87); C1336(1.01) | LDD0705 | [7] |
LDCM0389 | CL119 | HCT 116 | C608(0.83); C1336(1.06) | LDD0706 | [7] |
LDCM0390 | CL12 | HCT 116 | C608(0.96); C1336(1.17); C391(1.41); C395(1.41) | LDD0707 | [7] |
LDCM0391 | CL120 | HCT 116 | C608(0.98); C1336(1.05) | LDD0708 | [7] |
LDCM0392 | CL121 | HCT 116 | C636(0.78); C1336(0.79); C608(0.85); C391(1.24) | LDD0709 | [7] |
LDCM0393 | CL122 | HCT 116 | C608(0.92); C391(1.14); C395(1.14); C1336(1.14) | LDD0710 | [7] |
LDCM0394 | CL123 | HCT 116 | C608(0.58); C391(0.95); C395(0.95); C636(0.96) | LDD0711 | [7] |
LDCM0395 | CL124 | HCT 116 | C608(0.84); C391(0.97); C395(0.97); C636(1.05) | LDD0712 | [7] |
LDCM0396 | CL125 | HCT 116 | C391(1.03); C395(1.03); C1336(1.04) | LDD0713 | [7] |
LDCM0397 | CL126 | HCT 116 | C1336(1.09); C391(1.11); C395(1.11) | LDD0714 | [7] |
LDCM0398 | CL127 | HCT 116 | C1336(1.07); C391(1.35); C395(1.35) | LDD0715 | [7] |
LDCM0399 | CL128 | HCT 116 | C1336(1.15); C391(1.29); C395(1.29) | LDD0716 | [7] |
LDCM0400 | CL13 | HCT 116 | C1336(1.02); C608(1.05); C391(1.09); C395(1.09) | LDD0717 | [7] |
LDCM0401 | CL14 | HCT 116 | C608(0.85); C1336(0.92); C391(1.45); C395(1.45) | LDD0718 | [7] |
LDCM0402 | CL15 | HCT 116 | C1336(0.96); C608(0.97); C391(1.40); C395(1.40) | LDD0719 | [7] |
LDCM0403 | CL16 | HCT 116 | C608(0.86); C636(0.95); C1336(0.96); C391(1.09) | LDD0720 | [7] |
LDCM0404 | CL17 | HCT 116 | C608(0.90); C636(0.95); C1336(0.98); C391(1.01) | LDD0721 | [7] |
LDCM0405 | CL18 | HCT 116 | C608(0.85); C1336(0.92); C636(1.09); C391(1.20) | LDD0722 | [7] |
LDCM0406 | CL19 | HCT 116 | C636(0.78); C608(1.00); C1336(1.03); C391(1.11) | LDD0723 | [7] |
LDCM0407 | CL2 | HCT 116 | C391(0.94); C395(0.94); C1336(0.95); C608(1.04) | LDD0724 | [7] |
LDCM0408 | CL20 | HCT 116 | C636(0.84); C608(0.87); C1336(1.05); C391(1.20) | LDD0725 | [7] |
LDCM0409 | CL21 | HCT 116 | C636(0.80); C608(1.05); C391(1.16); C395(1.16) | LDD0726 | [7] |
LDCM0410 | CL22 | HCT 116 | C636(0.82); C391(1.08); C395(1.08); C608(1.10) | LDD0727 | [7] |
LDCM0411 | CL23 | HCT 116 | C636(0.84); C608(0.85); C1336(0.97); C391(1.00) | LDD0728 | [7] |
LDCM0412 | CL24 | HCT 116 | C1336(1.20); C391(1.14); C395(1.14); C608(0.85) | LDD0729 | [7] |
LDCM0413 | CL25 | HCT 116 | C1336(1.06); C391(1.05); C395(1.05); C608(0.78) | LDD0730 | [7] |
LDCM0414 | CL26 | HCT 116 | C1336(0.93); C391(1.05); C395(1.05); C608(0.78) | LDD0731 | [7] |
LDCM0415 | CL27 | HCT 116 | C1336(0.99); C391(1.25); C395(1.25); C608(0.81) | LDD0732 | [7] |
LDCM0416 | CL28 | HCT 116 | C1336(1.05); C391(1.26); C395(1.26); C608(0.74) | LDD0733 | [7] |
LDCM0417 | CL29 | HCT 116 | C1336(1.08); C391(1.23); C395(1.23); C608(0.74) | LDD0734 | [7] |
LDCM0418 | CL3 | HCT 116 | C1336(0.93); C391(1.08); C395(1.08); C608(0.73) | LDD0735 | [7] |
LDCM0419 | CL30 | HCT 116 | C1336(0.95); C391(1.17); C395(1.17); C608(0.73) | LDD0736 | [7] |
LDCM0420 | CL31 | HCT 116 | C1336(1.10); C391(0.89); C395(0.89); C608(1.14) | LDD0737 | [7] |
LDCM0421 | CL32 | HCT 116 | C1336(1.04); C391(0.88); C395(0.88); C608(1.02) | LDD0738 | [7] |
LDCM0422 | CL33 | HCT 116 | C1336(0.96); C391(0.91); C395(0.91); C608(0.98) | LDD0739 | [7] |
LDCM0423 | CL34 | HCT 116 | C1336(1.23); C391(1.04); C395(1.04); C608(1.07) | LDD0740 | [7] |
LDCM0424 | CL35 | HCT 116 | C1336(1.15); C391(0.81); C395(0.81); C608(0.90) | LDD0741 | [7] |
LDCM0425 | CL36 | HCT 116 | C1336(1.16); C391(1.07); C395(1.07); C608(0.96) | LDD0742 | [7] |
LDCM0426 | CL37 | HCT 116 | C1336(1.21); C391(1.22); C395(1.22); C608(1.13) | LDD0743 | [7] |
LDCM0428 | CL39 | HCT 116 | C1336(1.20); C391(0.85); C395(0.85); C608(0.94) | LDD0745 | [7] |
LDCM0429 | CL4 | HCT 116 | C1336(0.95); C391(0.75); C395(0.75); C608(0.84) | LDD0746 | [7] |
LDCM0430 | CL40 | HCT 116 | C1336(1.03); C391(1.06); C395(1.06); C608(1.27) | LDD0747 | [7] |
LDCM0431 | CL41 | HCT 116 | C1336(1.08); C391(1.11); C395(1.11); C608(0.99) | LDD0748 | [7] |
LDCM0432 | CL42 | HCT 116 | C1336(1.46); C391(1.04); C395(1.04); C608(1.05) | LDD0749 | [7] |
LDCM0433 | CL43 | HCT 116 | C1336(1.25); C391(0.97); C395(0.97); C608(1.00) | LDD0750 | [7] |
LDCM0434 | CL44 | HCT 116 | C1336(1.16); C391(0.80); C395(0.80); C608(1.07) | LDD0751 | [7] |
LDCM0435 | CL45 | HCT 116 | C1336(1.23); C391(0.79); C395(0.79); C608(1.02) | LDD0752 | [7] |
LDCM0436 | CL46 | HCT 116 | C1336(0.94); C391(1.11); C395(1.11); C608(0.86) | LDD0753 | [7] |
LDCM0437 | CL47 | HCT 116 | C1336(0.93); C391(1.12); C395(1.12); C608(0.96) | LDD0754 | [7] |
LDCM0438 | CL48 | HCT 116 | C1336(0.91); C391(0.97); C395(0.97); C608(0.96) | LDD0755 | [7] |
LDCM0439 | CL49 | HCT 116 | C1336(1.00); C391(1.33); C395(1.33); C608(0.95) | LDD0756 | [7] |
LDCM0440 | CL5 | HCT 116 | C1336(0.94); C391(1.12); C395(1.12); C608(0.97) | LDD0757 | [7] |
LDCM0441 | CL50 | HCT 116 | C1336(1.02); C391(1.22); C395(1.22); C608(0.93) | LDD0758 | [7] |
LDCM0442 | CL51 | HCT 116 | C1336(0.84); C391(1.03); C395(1.03); C608(0.87) | LDD0759 | [7] |
LDCM0443 | CL52 | HCT 116 | C1336(0.90); C391(1.03); C395(1.03); C608(0.72) | LDD0760 | [7] |
LDCM0444 | CL53 | HCT 116 | C1336(0.85); C391(1.01); C395(1.01); C608(1.34) | LDD0761 | [7] |
LDCM0445 | CL54 | HCT 116 | C1336(1.04); C391(1.38); C395(1.38); C608(0.96) | LDD0762 | [7] |
LDCM0446 | CL55 | HCT 116 | C1336(0.91); C391(1.13); C395(1.13); C608(1.03) | LDD0763 | [7] |
LDCM0447 | CL56 | HCT 116 | C1336(1.03); C391(0.89); C395(0.89); C608(1.16) | LDD0764 | [7] |
LDCM0448 | CL57 | HCT 116 | C1336(0.86); C391(0.88); C395(0.88); C608(1.09) | LDD0765 | [7] |
LDCM0449 | CL58 | HCT 116 | C1336(0.99); C391(1.01); C395(1.01); C608(0.97) | LDD0766 | [7] |
LDCM0450 | CL59 | HCT 116 | C1336(1.14); C391(0.98); C395(0.98); C608(0.97) | LDD0767 | [7] |
LDCM0451 | CL6 | HCT 116 | C1336(1.06); C391(1.52); C395(1.52); C608(0.86) | LDD0768 | [7] |
LDCM0452 | CL60 | HCT 116 | C1336(1.06); C391(1.07); C395(1.07); C608(1.01) | LDD0769 | [7] |
LDCM0453 | CL61 | HCT 116 | C1336(1.02); C391(1.04); C395(1.04); C636(0.93) | LDD0770 | [7] |
LDCM0454 | CL62 | HCT 116 | C1336(1.20); C391(0.89); C395(0.89); C636(0.74) | LDD0771 | [7] |
LDCM0455 | CL63 | HCT 116 | C1336(1.07); C391(0.86); C395(0.86); C636(0.87) | LDD0772 | [7] |
LDCM0456 | CL64 | HCT 116 | C1336(1.23); C391(0.93); C395(0.93); C636(0.67) | LDD0773 | [7] |
LDCM0457 | CL65 | HCT 116 | C1336(1.14); C391(0.90); C395(0.90); C636(0.80) | LDD0774 | [7] |
LDCM0458 | CL66 | HCT 116 | C1336(1.46); C391(0.80); C395(0.80); C636(0.77) | LDD0775 | [7] |
LDCM0459 | CL67 | HCT 116 | C1336(1.28); C391(0.86); C395(0.86); C636(0.74) | LDD0776 | [7] |
LDCM0460 | CL68 | HCT 116 | C1336(1.13); C391(0.82); C395(0.82); C636(0.95) | LDD0777 | [7] |
LDCM0461 | CL69 | HCT 116 | C1336(1.00); C391(0.96); C395(0.96); C636(1.11) | LDD0778 | [7] |
LDCM0462 | CL7 | HCT 116 | C1336(1.08); C391(1.24); C395(1.24); C608(0.83) | LDD0779 | [7] |
LDCM0463 | CL70 | HCT 116 | C1336(1.16); C391(0.75); C395(0.75); C636(0.80) | LDD0780 | [7] |
LDCM0464 | CL71 | HCT 116 | C1336(1.15); C391(0.78); C395(0.78); C636(0.79) | LDD0781 | [7] |
LDCM0465 | CL72 | HCT 116 | C1336(1.09); C391(0.94); C395(0.94); C636(0.80) | LDD0782 | [7] |
LDCM0466 | CL73 | HCT 116 | C1336(1.14); C391(0.88); C395(0.88); C636(0.72) | LDD0783 | [7] |
LDCM0467 | CL74 | HCT 116 | C1336(1.10); C391(0.89); C395(0.89); C636(0.63) | LDD0784 | [7] |
LDCM0469 | CL76 | HCT 116 | C1336(0.93); C391(1.08); C395(1.08); C608(1.06) | LDD0786 | [7] |
LDCM0470 | CL77 | HCT 116 | C1336(0.95); C391(0.89); C395(0.89); C608(1.00) | LDD0787 | [7] |
LDCM0471 | CL78 | HCT 116 | C1336(0.92); C391(0.95); C395(0.95); C608(1.01) | LDD0788 | [7] |
LDCM0472 | CL79 | HCT 116 | C1336(1.07); C391(0.92); C395(0.92); C608(1.04) | LDD0789 | [7] |
LDCM0473 | CL8 | HCT 116 | C1336(1.35); C391(1.00); C395(1.00); C608(0.81) | LDD0790 | [7] |
LDCM0474 | CL80 | HCT 116 | C1336(0.95); C391(1.02); C395(1.02); C608(1.21) | LDD0791 | [7] |
LDCM0475 | CL81 | HCT 116 | C1336(1.01); C391(0.90); C395(0.90); C608(1.04) | LDD0792 | [7] |
LDCM0476 | CL82 | HCT 116 | C1336(1.37); C391(1.04); C395(1.04); C608(1.01) | LDD0793 | [7] |
LDCM0477 | CL83 | HCT 116 | C1336(1.32); C391(1.04); C395(1.04); C608(1.11) | LDD0794 | [7] |
LDCM0478 | CL84 | HCT 116 | C1336(1.62); C391(1.06); C395(1.06); C608(1.10) | LDD0795 | [7] |
LDCM0479 | CL85 | HCT 116 | C1336(1.12); C391(0.82); C395(0.82); C608(1.11) | LDD0796 | [7] |
LDCM0480 | CL86 | HCT 116 | C1336(0.99); C391(0.80); C395(0.80); C608(1.12) | LDD0797 | [7] |
LDCM0481 | CL87 | HCT 116 | C1336(1.13); C391(0.97); C395(0.97); C608(1.01) | LDD0798 | [7] |
LDCM0482 | CL88 | HCT 116 | C1336(1.21); C391(0.94); C395(0.94); C608(1.04) | LDD0799 | [7] |
LDCM0483 | CL89 | HCT 116 | C1336(1.66); C391(0.93); C395(0.93); C608(1.09) | LDD0800 | [7] |
LDCM0484 | CL9 | HCT 116 | C1336(1.00); C391(0.85); C395(0.85); C608(1.11) | LDD0801 | [7] |
LDCM0485 | CL90 | HCT 116 | C1336(1.00); C391(0.97); C395(0.97); C608(1.11) | LDD0802 | [7] |
LDCM0486 | CL91 | HCT 116 | C1336(0.99); C391(0.93); C395(0.93); C608(1.03) | LDD0803 | [7] |
LDCM0487 | CL92 | HCT 116 | C1336(0.96); C391(1.07); C395(1.07); C608(1.08) | LDD0804 | [7] |
LDCM0488 | CL93 | HCT 116 | C1336(0.94); C391(1.11); C395(1.11); C608(1.02) | LDD0805 | [7] |
LDCM0489 | CL94 | HCT 116 | C1336(1.05); C391(1.04); C395(1.04); C608(0.95) | LDD0806 | [7] |
LDCM0490 | CL95 | HCT 116 | C1336(1.12); C391(0.97); C395(0.97); C608(0.93) | LDD0807 | [7] |
LDCM0491 | CL96 | HCT 116 | C1336(0.95); C391(1.04); C395(1.04); C608(1.01) | LDD0808 | [7] |
LDCM0492 | CL97 | HCT 116 | C1336(0.95); C391(1.01); C395(1.01); C608(0.90) | LDD0809 | [7] |
LDCM0493 | CL98 | HCT 116 | C1336(0.98); C391(0.99); C395(0.99); C608(0.96) | LDD0810 | [7] |
LDCM0494 | CL99 | HCT 116 | C1336(0.96); C391(0.96); C395(0.96); C608(0.97) | LDD0811 | [7] |
LDCM0495 | E2913 | HEK-293T | C608(0.90); C636(0.95); C1336(0.94); C896(0.98) | LDD1698 | [18] |
LDCM0213 | Electrophilic fragment 2 | MDA-MB-231 | C608(21.70); C896(14.65) | LDD1702 | [4] |
LDCM0625 | F8 | Ramos | C1336(0.96) | LDD2187 | [19] |
LDCM0572 | Fragment10 | Ramos | C1336(1.13) | LDD2189 | [19] |
LDCM0573 | Fragment11 | Ramos | C1336(0.13); C608(0.21) | LDD2190 | [19] |
LDCM0574 | Fragment12 | Ramos | C1336(0.84) | LDD2191 | [19] |
LDCM0575 | Fragment13 | Ramos | C1336(0.65) | LDD2192 | [19] |
LDCM0576 | Fragment14 | Ramos | C1336(1.65); C608(1.90) | LDD2193 | [19] |
LDCM0579 | Fragment20 | Ramos | C1336(1.18) | LDD2194 | [19] |
LDCM0580 | Fragment21 | Ramos | C1336(0.61) | LDD2195 | [19] |
LDCM0582 | Fragment23 | Ramos | C1336(0.59) | LDD2196 | [19] |
LDCM0578 | Fragment27 | Ramos | C1336(0.59) | LDD2197 | [19] |
LDCM0586 | Fragment28 | Ramos | C1336(0.61); C608(8.39) | LDD2198 | [19] |
LDCM0588 | Fragment30 | Ramos | C1336(0.77) | LDD2199 | [19] |
LDCM0589 | Fragment31 | Ramos | C1336(0.68) | LDD2200 | [19] |
LDCM0590 | Fragment32 | Ramos | C1336(0.70) | LDD2201 | [19] |
LDCM0468 | Fragment33 | HCT 116 | C1336(1.09); C391(0.82); C395(0.82); C636(0.72) | LDD0785 | [7] |
LDCM0596 | Fragment38 | Ramos | C1336(0.62) | LDD2203 | [19] |
LDCM0566 | Fragment4 | Ramos | C1336(0.82); C608(2.00) | LDD2184 | [19] |
LDCM0427 | Fragment51 | HCT 116 | C1336(1.53); C391(0.87); C395(0.87); C608(1.35) | LDD0744 | [7] |
LDCM0610 | Fragment52 | Ramos | C1336(1.14) | LDD2204 | [19] |
LDCM0614 | Fragment56 | Ramos | C1336(0.66) | LDD2205 | [19] |
LDCM0569 | Fragment7 | Ramos | C1336(0.95); C608(1.19) | LDD2186 | [19] |
LDCM0571 | Fragment9 | Ramos | C1336(2.11) | LDD2188 | [19] |
LDCM0015 | HNE | MDA-MB-231 | C1336(1.05) | LDD0346 | [19] |
LDCM0022 | KB02 | HCT 116 | C1336(1.40); C67(1.50) | LDD0080 | [7] |
LDCM0023 | KB03 | HCT 116 | C1336(1.45); C67(1.00) | LDD0081 | [7] |
LDCM0024 | KB05 | HCT 116 | C1336(8.63); C67(1.42) | LDD0082 | [7] |
LDCM0509 | N-(4-bromo-3,5-dimethylphenyl)-2-nitroacetamide | MDA-MB-231 | C608(0.95) | LDD2102 | [4] |
LDCM0109 | NEM | HeLa | H1314(0.00); H440(0.00) | LDD0225 | [6] |
LDCM0497 | Nucleophilic fragment 11b | MDA-MB-231 | C608(1.12) | LDD2090 | [4] |
LDCM0499 | Nucleophilic fragment 12b | MDA-MB-231 | C608(0.84) | LDD2092 | [4] |
LDCM0505 | Nucleophilic fragment 15b | MDA-MB-231 | C608(0.82) | LDD2098 | [4] |
LDCM0506 | Nucleophilic fragment 16a | MDA-MB-231 | C608(1.07) | LDD2099 | [4] |
LDCM0512 | Nucleophilic fragment 19a | MDA-MB-231 | C608(0.96) | LDD2105 | [4] |
LDCM0515 | Nucleophilic fragment 20b | MDA-MB-231 | C608(0.70) | LDD2108 | [4] |
LDCM0530 | Nucleophilic fragment 28a | MDA-MB-231 | C608(1.42) | LDD2123 | [4] |
LDCM0534 | Nucleophilic fragment 30a | MDA-MB-231 | C608(1.31) | LDD2127 | [4] |
LDCM0541 | Nucleophilic fragment 36 | MDA-MB-231 | C608(0.53) | LDD2134 | [4] |
LDCM0542 | Nucleophilic fragment 37 | MDA-MB-231 | C608(1.56) | LDD2135 | [4] |
LDCM0543 | Nucleophilic fragment 38 | MDA-MB-231 | C608(1.29) | LDD2136 | [4] |
LDCM0544 | Nucleophilic fragment 39 | MDA-MB-231 | C608(1.09) | LDD2137 | [4] |
LDCM0546 | Nucleophilic fragment 40 | MDA-MB-231 | C608(0.75) | LDD2140 | [4] |
LDCM0552 | Nucleophilic fragment 6a | MDA-MB-231 | C608(1.07) | LDD2146 | [4] |
LDCM0554 | Nucleophilic fragment 7a | MDA-MB-231 | C608(0.64) | LDD2148 | [4] |
LDCM0556 | Nucleophilic fragment 8a | MDA-MB-231 | C608(0.68) | LDD2150 | [4] |
LDCM0559 | Nucleophilic fragment 9b | MDA-MB-231 | C608(2.22) | LDD2153 | [4] |
LDCM0131 | RA190 | MM1.R | C67(1.24) | LDD0304 | [20] |
References