Details of the Target
General Information of Target
Target ID | LDTP01556 | |||||
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Target Name | Vesicle-associated membrane protein-associated protein B/C (VAPB) | |||||
Gene Name | VAPB | |||||
Gene ID | 9217 | |||||
Synonyms |
Vesicle-associated membrane protein-associated protein B/C; VAMP-B/VAMP-C; VAMP-associated protein B/C; VAP-B/VAP-C |
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3D Structure | ||||||
Sequence |
MAKVEQVLSLEPQHELKFRGPFTDVVTTNLKLGNPTDRNVCFKVKTTAPRRYCVRPNSGI
IDAGASINVSVMLQPFDYDPNEKSKHKFMVQSMFAPTDTSDMEAVWKEAKPEDLMDSKLR CVFELPAENDKPHDVEINKIISTTASKTETPIVSKSLSSSLDDTEVKKVMEECKRLQGEV QRLREENKQFKEEDGLRMRKTVQSNSPISALAPTGKEEGLSTRLLALVVLFFIVGVIIGK IAL |
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Target Bioclass |
Transporter and channel
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Family |
VAMP-associated protein (VAP) (TC 9.B.17) family
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Subcellular location |
Endoplasmic reticulum membrane
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Function |
Endoplasmic reticulum (ER)-anchored protein that mediates the formation of contact sites between the ER and endosomes via interaction with FFAT motif-containing proteins such as STARD3 or WDR44. Interacts with STARD3 in a FFAT motif phosphorylation dependent manner. Via interaction with WDR44 participates in neosynthesized protein export. Participates in the endoplasmic reticulum unfolded protein response (UPR) by inducing ERN1/IRE1 activity. Involved in cellular calcium homeostasis regulation.
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Uniprot ID | ||||||
Ensemble ID | ||||||
HGNC ID |
Probe(s) Labeling This Target
ABPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
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m-APA Probe Info |
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15.00 | LDD0402 | [1] | |
YN-1 Probe Info |
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100.00 | LDD0444 | [2] | |
ONAyne Probe Info |
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K118(1.01) | LDD0274 | [3] | |
STPyne Probe Info |
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K118(6.13) | LDD0277 | [3] | |
OPA-S-S-alkyne Probe Info |
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K174(1.61); K45(4.46) | LDD3494 | [4] | |
BTD Probe Info |
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C173(1.38) | LDD2090 | [5] | |
DA-P3 Probe Info |
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4.85 | LDD0181 | [6] | |
AHL-Pu-1 Probe Info |
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C173(2.72) | LDD0171 | [7] | |
Alkyne-RA190 Probe Info |
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3.33 | LDD0300 | [8] | |
DBIA Probe Info |
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C121(0.60) | LDD0533 | [9] | |
5E-2FA Probe Info |
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N.A. | LDD2235 | [10] | |
ATP probe Probe Info |
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N.A. | LDD0199 | [11] | |
IA-alkyne Probe Info |
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N.A. | LDD0032 | [12] | |
Lodoacetamide azide Probe Info |
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C121(0.00); C173(0.00) | LDD0037 | [13] | |
JW-RF-010 Probe Info |
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N.A. | LDD0026 | [14] | |
TFBX Probe Info |
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N.A. | LDD0027 | [14] | |
IPM Probe Info |
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N.A. | LDD0005 | [15] | |
NHS Probe Info |
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K3(0.00); K167(0.00); K168(0.00); K118(0.00) | LDD0010 | [15] | |
Phosphinate-6 Probe Info |
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C53(0.00); C173(0.00) | LDD0018 | [16] | |
1c-yne Probe Info |
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N.A. | LDD0228 | [17] | |
Acrolein Probe Info |
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H14(0.00); C173(0.00); C121(0.00) | LDD0217 | [18] | |
Crotonaldehyde Probe Info |
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N.A. | LDD0219 | [18] | |
Methacrolein Probe Info |
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N.A. | LDD0218 | [18] | |
W1 Probe Info |
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N.A. | LDD0236 | [19] | |
AOyne Probe Info |
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14.80 | LDD0443 | [20] | |
NAIA_5 Probe Info |
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C121(0.00); C173(0.00); C41(0.00) | LDD2223 | [21] | |
TPP-AC Probe Info |
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N.A. | LDD0427 | [22] |
PAL-AfBPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
---|---|---|---|---|---|
FFF probe13 Probe Info |
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20.00 | LDD0475 | [23] | |
FFF probe14 Probe Info |
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20.00 | LDD0477 | [23] | |
FFF probe2 Probe Info |
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15.03 | LDD0463 | [23] | |
FFF probe3 Probe Info |
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20.00 | LDD0464 | [23] | |
OEA-DA Probe Info |
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4.57 | LDD0046 | [24] | |
STS-1 Probe Info |
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N.A. | LDD0068 | [25] |
Competitor(s) Related to This Target
Competitor ID | Name | Cell line | Binding Site(Ratio) | Interaction ID | Ref |
---|---|---|---|---|---|
LDCM0548 | 1-(4-(Benzo[d][1,3]dioxol-5-ylmethyl)piperazin-1-yl)-2-nitroethan-1-one | MDA-MB-231 | C173(0.71); C121(0.84) | LDD2142 | [5] |
LDCM0519 | 1-(6-methoxy-3,4-dihydroquinolin-1(2H)-yl)-2-nitroethan-1-one | MDA-MB-231 | C173(0.87) | LDD2112 | [5] |
LDCM0524 | 2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide | MDA-MB-231 | C173(1.55); C121(1.48) | LDD2117 | [5] |
LDCM0510 | 3-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-3-oxopropanenitrile | MDA-MB-231 | C173(1.33) | LDD2103 | [5] |
LDCM0539 | 3-(4-Isopropylpiperazin-1-yl)-3-oxopropanenitrile | MDA-MB-231 | C121(0.91) | LDD2132 | [5] |
LDCM0025 | 4SU-RNA | HEK-293T | C53(2.16) | LDD0371 | [7] |
LDCM0026 | 4SU-RNA+native RNA | DM93 | C173(2.72) | LDD0171 | [7] |
LDCM0214 | AC1 | PaTu 8988t | C121(0.57) | LDD1093 | [9] |
LDCM0215 | AC10 | PaTu 8988t | C121(0.41) | LDD1094 | [9] |
LDCM0216 | AC100 | HCT 116 | C121(0.60) | LDD0533 | [9] |
LDCM0217 | AC101 | HCT 116 | C121(0.61) | LDD0534 | [9] |
LDCM0218 | AC102 | HCT 116 | C121(0.65) | LDD0535 | [9] |
LDCM0219 | AC103 | HCT 116 | C121(0.53) | LDD0536 | [9] |
LDCM0220 | AC104 | HCT 116 | C121(0.82) | LDD0537 | [9] |
LDCM0221 | AC105 | HCT 116 | C121(0.69) | LDD0538 | [9] |
LDCM0222 | AC106 | HCT 116 | C121(0.60) | LDD0539 | [9] |
LDCM0223 | AC107 | HCT 116 | C121(0.63) | LDD0540 | [9] |
LDCM0224 | AC108 | HCT 116 | C121(0.56) | LDD0541 | [9] |
LDCM0225 | AC109 | HCT 116 | C121(0.84) | LDD0542 | [9] |
LDCM0226 | AC11 | PaTu 8988t | C121(0.79) | LDD1105 | [9] |
LDCM0227 | AC110 | HCT 116 | C121(0.50) | LDD0544 | [9] |
LDCM0228 | AC111 | HCT 116 | C121(0.50) | LDD0545 | [9] |
LDCM0229 | AC112 | HCT 116 | C121(0.52) | LDD0546 | [9] |
LDCM0230 | AC113 | HCT 116 | C121(0.36) | LDD0547 | [9] |
LDCM0231 | AC114 | HCT 116 | C121(0.35) | LDD0548 | [9] |
LDCM0232 | AC115 | HCT 116 | C121(0.41) | LDD0549 | [9] |
LDCM0233 | AC116 | HCT 116 | C121(0.47) | LDD0550 | [9] |
LDCM0234 | AC117 | HCT 116 | C121(0.48) | LDD0551 | [9] |
LDCM0235 | AC118 | HCT 116 | C121(0.40) | LDD0552 | [9] |
LDCM0236 | AC119 | HCT 116 | C121(0.35) | LDD0553 | [9] |
LDCM0237 | AC12 | PaTu 8988t | C121(0.66) | LDD1116 | [9] |
LDCM0238 | AC120 | HCT 116 | C121(0.48) | LDD0555 | [9] |
LDCM0239 | AC121 | HCT 116 | C121(0.30) | LDD0556 | [9] |
LDCM0240 | AC122 | HCT 116 | C121(0.34) | LDD0557 | [9] |
LDCM0241 | AC123 | HCT 116 | C121(0.32) | LDD0558 | [9] |
LDCM0242 | AC124 | HCT 116 | C121(0.32) | LDD0559 | [9] |
LDCM0243 | AC125 | HCT 116 | C121(0.47) | LDD0560 | [9] |
LDCM0244 | AC126 | HCT 116 | C121(0.44) | LDD0561 | [9] |
LDCM0245 | AC127 | HCT 116 | C121(0.33) | LDD0562 | [9] |
LDCM0246 | AC128 | HCT 116 | C121(0.65) | LDD0563 | [9] |
LDCM0247 | AC129 | HCT 116 | C121(0.68) | LDD0564 | [9] |
LDCM0249 | AC130 | HCT 116 | C121(0.52) | LDD0566 | [9] |
LDCM0250 | AC131 | HCT 116 | C121(0.53) | LDD0567 | [9] |
LDCM0251 | AC132 | HCT 116 | C121(0.80) | LDD0568 | [9] |
LDCM0252 | AC133 | HCT 116 | C121(0.57) | LDD0569 | [9] |
LDCM0253 | AC134 | HCT 116 | C121(0.55) | LDD0570 | [9] |
LDCM0254 | AC135 | HCT 116 | C121(0.57) | LDD0571 | [9] |
LDCM0255 | AC136 | HCT 116 | C121(0.57) | LDD0572 | [9] |
LDCM0256 | AC137 | HCT 116 | C121(0.55) | LDD0573 | [9] |
LDCM0257 | AC138 | HCT 116 | C121(0.46) | LDD0574 | [9] |
LDCM0258 | AC139 | HCT 116 | C121(0.54) | LDD0575 | [9] |
LDCM0259 | AC14 | PaTu 8988t | C121(0.70) | LDD1138 | [9] |
LDCM0260 | AC140 | HCT 116 | C121(0.49) | LDD0577 | [9] |
LDCM0261 | AC141 | HCT 116 | C121(0.55) | LDD0578 | [9] |
LDCM0262 | AC142 | HCT 116 | C121(0.56) | LDD0579 | [9] |
LDCM0263 | AC143 | HCT 116 | C121(0.87) | LDD0580 | [9] |
LDCM0264 | AC144 | HCT 116 | C121(0.76) | LDD0581 | [9] |
LDCM0265 | AC145 | HCT 116 | C121(0.87) | LDD0582 | [9] |
LDCM0266 | AC146 | HCT 116 | C121(0.63) | LDD0583 | [9] |
LDCM0267 | AC147 | HCT 116 | C121(0.86) | LDD0584 | [9] |
LDCM0268 | AC148 | HCT 116 | C121(0.55) | LDD0585 | [9] |
LDCM0269 | AC149 | HCT 116 | C121(0.68) | LDD0586 | [9] |
LDCM0270 | AC15 | PaTu 8988t | C121(0.46) | LDD1149 | [9] |
LDCM0271 | AC150 | HCT 116 | C121(1.00) | LDD0588 | [9] |
LDCM0272 | AC151 | HCT 116 | C121(0.76) | LDD0589 | [9] |
LDCM0273 | AC152 | HCT 116 | C121(0.72) | LDD0590 | [9] |
LDCM0274 | AC153 | HCT 116 | C121(0.55) | LDD0591 | [9] |
LDCM0621 | AC154 | HCT 116 | C121(0.81) | LDD2158 | [9] |
LDCM0622 | AC155 | HCT 116 | C121(0.71) | LDD2159 | [9] |
LDCM0623 | AC156 | HCT 116 | C121(0.89) | LDD2160 | [9] |
LDCM0624 | AC157 | HCT 116 | C121(0.89) | LDD2161 | [9] |
LDCM0276 | AC17 | PaTu 8988t | C121(1.23) | LDD1155 | [9] |
LDCM0277 | AC18 | PaTu 8988t | C121(0.87) | LDD1156 | [9] |
LDCM0278 | AC19 | PaTu 8988t | C121(0.96) | LDD1157 | [9] |
LDCM0279 | AC2 | PaTu 8988t | C121(0.81) | LDD1158 | [9] |
LDCM0280 | AC20 | PaTu 8988t | C121(0.97) | LDD1159 | [9] |
LDCM0281 | AC21 | PaTu 8988t | C121(1.15) | LDD1160 | [9] |
LDCM0282 | AC22 | PaTu 8988t | C121(0.96) | LDD1161 | [9] |
LDCM0283 | AC23 | PaTu 8988t | C121(0.88) | LDD1162 | [9] |
LDCM0284 | AC24 | PaTu 8988t | C121(0.90) | LDD1163 | [9] |
LDCM0285 | AC25 | HEK-293T | C173(1.33); C121(0.98); C53(1.06) | LDD1524 | [26] |
LDCM0286 | AC26 | HEK-293T | C173(1.42); C121(1.02); C53(0.98) | LDD1525 | [26] |
LDCM0287 | AC27 | HEK-293T | C173(1.16); C121(1.14); C53(0.96) | LDD1526 | [26] |
LDCM0288 | AC28 | HEK-293T | C173(1.52); C121(1.10); C53(1.13) | LDD1527 | [26] |
LDCM0289 | AC29 | HEK-293T | C173(1.15); C121(1.02); C53(0.89) | LDD1528 | [26] |
LDCM0290 | AC3 | PaTu 8988t | C121(0.79) | LDD1169 | [9] |
LDCM0291 | AC30 | HEK-293T | C173(1.28); C121(1.25); C53(1.14) | LDD1530 | [26] |
LDCM0292 | AC31 | HEK-293T | C173(1.10); C121(1.08); C53(1.02) | LDD1531 | [26] |
LDCM0293 | AC32 | HEK-293T | C173(1.04); C121(1.03); C53(1.11) | LDD1532 | [26] |
LDCM0294 | AC33 | HEK-293T | C173(1.29); C121(1.02); C53(1.13) | LDD1533 | [26] |
LDCM0295 | AC34 | HEK-293T | C173(1.35); C121(1.02); C53(1.09) | LDD1534 | [26] |
LDCM0296 | AC35 | PaTu 8988t | C121(0.59) | LDD1175 | [9] |
LDCM0297 | AC36 | PaTu 8988t | C121(0.46) | LDD1176 | [9] |
LDCM0298 | AC37 | PaTu 8988t | C121(0.83) | LDD1177 | [9] |
LDCM0299 | AC38 | PaTu 8988t | C121(0.55) | LDD1178 | [9] |
LDCM0300 | AC39 | PaTu 8988t | C121(0.54) | LDD1179 | [9] |
LDCM0301 | AC4 | PaTu 8988t | C121(0.71) | LDD1180 | [9] |
LDCM0302 | AC40 | PaTu 8988t | C121(0.54) | LDD1181 | [9] |
LDCM0303 | AC41 | PaTu 8988t | C121(0.98) | LDD1182 | [9] |
LDCM0304 | AC42 | PaTu 8988t | C121(0.95) | LDD1183 | [9] |
LDCM0305 | AC43 | PaTu 8988t | C121(1.00) | LDD1184 | [9] |
LDCM0306 | AC44 | PaTu 8988t | C121(0.93) | LDD1185 | [9] |
LDCM0307 | AC45 | PaTu 8988t | C121(0.84) | LDD1186 | [9] |
LDCM0308 | AC46 | PaTu 8988t | C121(0.52) | LDD1187 | [9] |
LDCM0309 | AC47 | PaTu 8988t | C121(0.67) | LDD1188 | [9] |
LDCM0310 | AC48 | PaTu 8988t | C121(0.65) | LDD1189 | [9] |
LDCM0311 | AC49 | PaTu 8988t | C121(0.54) | LDD1190 | [9] |
LDCM0312 | AC5 | PaTu 8988t | C121(0.76) | LDD1191 | [9] |
LDCM0313 | AC50 | PaTu 8988t | C121(0.56) | LDD1192 | [9] |
LDCM0314 | AC51 | PaTu 8988t | C121(0.17) | LDD1193 | [9] |
LDCM0315 | AC52 | PaTu 8988t | C121(0.67) | LDD1194 | [9] |
LDCM0316 | AC53 | PaTu 8988t | C121(0.54) | LDD1195 | [9] |
LDCM0317 | AC54 | PaTu 8988t | C121(0.59) | LDD1196 | [9] |
LDCM0318 | AC55 | PaTu 8988t | C121(0.39) | LDD1197 | [9] |
LDCM0319 | AC56 | PaTu 8988t | C121(0.30) | LDD1198 | [9] |
LDCM0320 | AC57 | HCT 116 | C121(0.71) | LDD0637 | [9] |
LDCM0321 | AC58 | HCT 116 | C121(1.17) | LDD0638 | [9] |
LDCM0322 | AC59 | HCT 116 | C121(0.66) | LDD0639 | [9] |
LDCM0323 | AC6 | PaTu 8988t | C121(0.82) | LDD1202 | [9] |
LDCM0324 | AC60 | HCT 116 | C121(0.64) | LDD0641 | [9] |
LDCM0325 | AC61 | HCT 116 | C121(0.56) | LDD0642 | [9] |
LDCM0326 | AC62 | HCT 116 | C121(0.68) | LDD0643 | [9] |
LDCM0327 | AC63 | HCT 116 | C121(0.78) | LDD0644 | [9] |
LDCM0328 | AC64 | HCT 116 | C121(0.66) | LDD0645 | [9] |
LDCM0329 | AC65 | HCT 116 | C121(0.35) | LDD0646 | [9] |
LDCM0330 | AC66 | HCT 116 | C121(0.31) | LDD0647 | [9] |
LDCM0331 | AC67 | HCT 116 | C121(0.18) | LDD0648 | [9] |
LDCM0332 | AC68 | HCT 116 | C121(0.79) | LDD0649 | [9] |
LDCM0333 | AC69 | HCT 116 | C121(0.63) | LDD0650 | [9] |
LDCM0334 | AC7 | PaTu 8988t | C121(1.37) | LDD1213 | [9] |
LDCM0335 | AC70 | HCT 116 | C121(0.43) | LDD0652 | [9] |
LDCM0336 | AC71 | HCT 116 | C121(0.76) | LDD0653 | [9] |
LDCM0337 | AC72 | HCT 116 | C121(1.02) | LDD0654 | [9] |
LDCM0338 | AC73 | HCT 116 | C121(0.55) | LDD0655 | [9] |
LDCM0339 | AC74 | HCT 116 | C121(0.50) | LDD0656 | [9] |
LDCM0340 | AC75 | HCT 116 | C121(0.46) | LDD0657 | [9] |
LDCM0341 | AC76 | HCT 116 | C121(0.95) | LDD0658 | [9] |
LDCM0342 | AC77 | HCT 116 | C121(0.63) | LDD0659 | [9] |
LDCM0343 | AC78 | HCT 116 | C121(0.62) | LDD0660 | [9] |
LDCM0344 | AC79 | HCT 116 | C121(1.16) | LDD0661 | [9] |
LDCM0345 | AC8 | PaTu 8988t | C121(0.69) | LDD1224 | [9] |
LDCM0346 | AC80 | HCT 116 | C121(0.90) | LDD0663 | [9] |
LDCM0347 | AC81 | HCT 116 | C121(0.80) | LDD0664 | [9] |
LDCM0348 | AC82 | HCT 116 | C121(0.28) | LDD0665 | [9] |
LDCM0349 | AC83 | HCT 116 | C121(0.75) | LDD0666 | [9] |
LDCM0350 | AC84 | HCT 116 | C121(0.76) | LDD0667 | [9] |
LDCM0351 | AC85 | HCT 116 | C121(0.68) | LDD0668 | [9] |
LDCM0352 | AC86 | HCT 116 | C121(0.67) | LDD0669 | [9] |
LDCM0353 | AC87 | HCT 116 | C121(0.65) | LDD0670 | [9] |
LDCM0354 | AC88 | HCT 116 | C121(0.73) | LDD0671 | [9] |
LDCM0355 | AC89 | HCT 116 | C121(0.63) | LDD0672 | [9] |
LDCM0357 | AC90 | HCT 116 | C121(0.75) | LDD0674 | [9] |
LDCM0358 | AC91 | HCT 116 | C121(0.75) | LDD0675 | [9] |
LDCM0359 | AC92 | HCT 116 | C121(0.73) | LDD0676 | [9] |
LDCM0360 | AC93 | HCT 116 | C121(0.70) | LDD0677 | [9] |
LDCM0361 | AC94 | HCT 116 | C121(1.10) | LDD0678 | [9] |
LDCM0362 | AC95 | HCT 116 | C121(0.56) | LDD0679 | [9] |
LDCM0363 | AC96 | HCT 116 | C121(0.87) | LDD0680 | [9] |
LDCM0364 | AC97 | HCT 116 | C121(0.62) | LDD0681 | [9] |
LDCM0365 | AC98 | HCT 116 | C121(0.59) | LDD0682 | [9] |
LDCM0366 | AC99 | HCT 116 | C121(0.66) | LDD0683 | [9] |
LDCM0545 | Acetamide | MDA-MB-231 | C173(0.63) | LDD2138 | [5] |
LDCM0520 | AKOS000195272 | MDA-MB-231 | C173(0.67); C121(0.63) | LDD2113 | [5] |
LDCM0248 | AKOS034007472 | PaTu 8988t | C121(0.50) | LDD1127 | [9] |
LDCM0356 | AKOS034007680 | PaTu 8988t | C121(0.63) | LDD1235 | [9] |
LDCM0275 | AKOS034007705 | PaTu 8988t | C121(0.47) | LDD1154 | [9] |
LDCM0156 | Aniline | NCI-H1299 | 12.14 | LDD0403 | [1] |
LDCM0498 | BS-3668 | MDA-MB-231 | C173(1.14) | LDD2091 | [5] |
LDCM0108 | Chloroacetamide | HeLa | C173(0.00); H14(0.00) | LDD0222 | [18] |
LDCM0632 | CL-Sc | Hep-G2 | C173(1.95); C121(0.90); C173(0.23) | LDD2227 | [21] |
LDCM0367 | CL1 | HCT 116 | C121(0.83) | LDD0684 | [9] |
LDCM0368 | CL10 | HCT 116 | C121(0.95) | LDD0685 | [9] |
LDCM0369 | CL100 | PaTu 8988t | C121(0.82) | LDD1248 | [9] |
LDCM0370 | CL101 | PaTu 8988t | C121(0.82) | LDD1249 | [9] |
LDCM0371 | CL102 | PaTu 8988t | C121(0.95) | LDD1250 | [9] |
LDCM0372 | CL103 | PaTu 8988t | C121(0.62) | LDD1251 | [9] |
LDCM0373 | CL104 | PaTu 8988t | C121(0.81) | LDD1252 | [9] |
LDCM0374 | CL105 | PaTu 8988t | C121(1.13) | LDD1253 | [9] |
LDCM0375 | CL106 | PaTu 8988t | C121(0.99) | LDD1254 | [9] |
LDCM0376 | CL107 | PaTu 8988t | C121(1.00) | LDD1255 | [9] |
LDCM0377 | CL108 | PaTu 8988t | C121(1.08) | LDD1256 | [9] |
LDCM0378 | CL109 | PaTu 8988t | C121(1.08) | LDD1257 | [9] |
LDCM0379 | CL11 | HCT 116 | C121(1.05) | LDD0696 | [9] |
LDCM0380 | CL110 | PaTu 8988t | C121(0.71) | LDD1259 | [9] |
LDCM0381 | CL111 | PaTu 8988t | C121(0.65) | LDD1260 | [9] |
LDCM0382 | CL112 | HEK-293T | C173(1.21); C121(1.01); C53(1.14) | LDD1586 | [26] |
LDCM0383 | CL113 | HEK-293T | C173(1.46); C121(1.03); C53(1.08) | LDD1587 | [26] |
LDCM0384 | CL114 | HEK-293T | C173(1.07); C121(1.23); C53(1.08) | LDD1588 | [26] |
LDCM0385 | CL115 | HEK-293T | C173(1.34); C121(1.15); C53(1.26) | LDD1589 | [26] |
LDCM0386 | CL116 | HEK-293T | C173(1.29); C121(1.03); C53(1.10) | LDD1590 | [26] |
LDCM0387 | CL117 | PaTu 8988t | C121(0.92) | LDD1266 | [9] |
LDCM0388 | CL118 | PaTu 8988t | C121(1.01) | LDD1267 | [9] |
LDCM0389 | CL119 | PaTu 8988t | C121(0.98) | LDD1268 | [9] |
LDCM0390 | CL12 | HCT 116 | C121(1.09) | LDD0707 | [9] |
LDCM0391 | CL120 | PaTu 8988t | C121(0.61) | LDD1270 | [9] |
LDCM0392 | CL121 | PaTu 8988t | C121(0.74) | LDD1271 | [9] |
LDCM0393 | CL122 | PaTu 8988t | C121(0.68) | LDD1272 | [9] |
LDCM0394 | CL123 | PaTu 8988t | C121(0.51) | LDD1273 | [9] |
LDCM0395 | CL124 | PaTu 8988t | C121(0.37) | LDD1274 | [9] |
LDCM0396 | CL125 | HCT 116 | C121(1.26) | LDD0713 | [9] |
LDCM0397 | CL126 | HCT 116 | C121(0.73) | LDD0714 | [9] |
LDCM0398 | CL127 | HCT 116 | C121(0.95) | LDD0715 | [9] |
LDCM0399 | CL128 | HCT 116 | C121(1.28) | LDD0716 | [9] |
LDCM0400 | CL13 | HCT 116 | C121(1.40) | LDD0717 | [9] |
LDCM0401 | CL14 | HCT 116 | C121(0.85) | LDD0718 | [9] |
LDCM0402 | CL15 | HCT 116 | C121(1.12) | LDD0719 | [9] |
LDCM0403 | CL16 | PaTu 8988t | C121(0.85) | LDD1282 | [9] |
LDCM0404 | CL17 | PaTu 8988t | C121(0.93) | LDD1283 | [9] |
LDCM0405 | CL18 | PaTu 8988t | C121(0.74) | LDD1284 | [9] |
LDCM0406 | CL19 | PaTu 8988t | C121(0.83) | LDD1285 | [9] |
LDCM0407 | CL2 | HCT 116 | C121(0.81) | LDD0724 | [9] |
LDCM0408 | CL20 | PaTu 8988t | C121(0.79) | LDD1287 | [9] |
LDCM0409 | CL21 | PaTu 8988t | C121(0.58) | LDD1288 | [9] |
LDCM0410 | CL22 | PaTu 8988t | C121(0.72) | LDD1289 | [9] |
LDCM0411 | CL23 | PaTu 8988t | C121(0.50) | LDD1290 | [9] |
LDCM0412 | CL24 | PaTu 8988t | C121(0.56) | LDD1291 | [9] |
LDCM0413 | CL25 | PaTu 8988t | C121(0.47) | LDD1292 | [9] |
LDCM0414 | CL26 | PaTu 8988t | C121(0.57) | LDD1293 | [9] |
LDCM0415 | CL27 | PaTu 8988t | C121(0.59) | LDD1294 | [9] |
LDCM0416 | CL28 | PaTu 8988t | C121(0.55) | LDD1295 | [9] |
LDCM0417 | CL29 | PaTu 8988t | C121(0.40) | LDD1296 | [9] |
LDCM0418 | CL3 | HCT 116 | C121(0.83) | LDD0735 | [9] |
LDCM0419 | CL30 | PaTu 8988t | C121(0.48) | LDD1298 | [9] |
LDCM0420 | CL31 | PaTu 8988t | C121(0.81) | LDD1299 | [9] |
LDCM0421 | CL32 | PaTu 8988t | C121(0.87) | LDD1300 | [9] |
LDCM0422 | CL33 | PaTu 8988t | C121(0.51) | LDD1301 | [9] |
LDCM0423 | CL34 | PaTu 8988t | C121(0.55) | LDD1302 | [9] |
LDCM0424 | CL35 | PaTu 8988t | C121(0.52) | LDD1303 | [9] |
LDCM0425 | CL36 | PaTu 8988t | C121(0.36) | LDD1304 | [9] |
LDCM0426 | CL37 | PaTu 8988t | C121(0.47) | LDD1305 | [9] |
LDCM0428 | CL39 | PaTu 8988t | C121(0.54) | LDD1307 | [9] |
LDCM0429 | CL4 | HCT 116 | C121(0.89) | LDD0746 | [9] |
LDCM0430 | CL40 | PaTu 8988t | C121(0.87) | LDD1309 | [9] |
LDCM0431 | CL41 | PaTu 8988t | C121(0.65) | LDD1310 | [9] |
LDCM0432 | CL42 | PaTu 8988t | C121(0.72) | LDD1311 | [9] |
LDCM0433 | CL43 | PaTu 8988t | C121(0.62) | LDD1312 | [9] |
LDCM0434 | CL44 | PaTu 8988t | C121(0.71) | LDD1313 | [9] |
LDCM0435 | CL45 | PaTu 8988t | C121(0.62) | LDD1314 | [9] |
LDCM0436 | CL46 | PaTu 8988t | C121(0.93) | LDD1315 | [9] |
LDCM0437 | CL47 | PaTu 8988t | C121(0.78) | LDD1316 | [9] |
LDCM0438 | CL48 | PaTu 8988t | C121(0.88) | LDD1317 | [9] |
LDCM0439 | CL49 | PaTu 8988t | C121(1.03) | LDD1318 | [9] |
LDCM0440 | CL5 | HCT 116 | C121(0.98) | LDD0757 | [9] |
LDCM0441 | CL50 | PaTu 8988t | C121(0.93) | LDD1320 | [9] |
LDCM0442 | CL51 | PaTu 8988t | C121(0.85) | LDD1321 | [9] |
LDCM0443 | CL52 | PaTu 8988t | C121(0.97) | LDD1322 | [9] |
LDCM0444 | CL53 | PaTu 8988t | C121(0.63) | LDD1323 | [9] |
LDCM0445 | CL54 | PaTu 8988t | C121(0.52) | LDD1324 | [9] |
LDCM0446 | CL55 | PaTu 8988t | C121(0.71) | LDD1325 | [9] |
LDCM0447 | CL56 | PaTu 8988t | C121(0.16) | LDD1326 | [9] |
LDCM0448 | CL57 | PaTu 8988t | C121(0.61) | LDD1327 | [9] |
LDCM0449 | CL58 | PaTu 8988t | C121(0.65) | LDD1328 | [9] |
LDCM0450 | CL59 | PaTu 8988t | C121(0.44) | LDD1329 | [9] |
LDCM0451 | CL6 | HCT 116 | C121(0.79) | LDD0768 | [9] |
LDCM0452 | CL60 | PaTu 8988t | C121(0.68) | LDD1331 | [9] |
LDCM0453 | CL61 | PaTu 8988t | C121(0.86) | LDD1332 | [9] |
LDCM0454 | CL62 | PaTu 8988t | C121(1.06) | LDD1333 | [9] |
LDCM0455 | CL63 | PaTu 8988t | C121(1.03) | LDD1334 | [9] |
LDCM0456 | CL64 | PaTu 8988t | C121(1.29) | LDD1335 | [9] |
LDCM0457 | CL65 | PaTu 8988t | C121(1.14) | LDD1336 | [9] |
LDCM0458 | CL66 | PaTu 8988t | C121(1.12) | LDD1337 | [9] |
LDCM0459 | CL67 | PaTu 8988t | C121(1.19) | LDD1338 | [9] |
LDCM0460 | CL68 | PaTu 8988t | C121(1.07) | LDD1339 | [9] |
LDCM0461 | CL69 | PaTu 8988t | C121(1.03) | LDD1340 | [9] |
LDCM0462 | CL7 | HCT 116 | C121(1.12) | LDD0779 | [9] |
LDCM0463 | CL70 | PaTu 8988t | C121(0.92) | LDD1342 | [9] |
LDCM0464 | CL71 | PaTu 8988t | C121(1.11) | LDD1343 | [9] |
LDCM0465 | CL72 | PaTu 8988t | C121(1.13) | LDD1344 | [9] |
LDCM0466 | CL73 | PaTu 8988t | C121(1.05) | LDD1345 | [9] |
LDCM0467 | CL74 | PaTu 8988t | C121(1.00) | LDD1346 | [9] |
LDCM0469 | CL76 | PaTu 8988t | C121(0.62) | LDD1348 | [9] |
LDCM0470 | CL77 | PaTu 8988t | C121(0.79) | LDD1349 | [9] |
LDCM0471 | CL78 | PaTu 8988t | C121(0.72) | LDD1350 | [9] |
LDCM0472 | CL79 | PaTu 8988t | C121(1.08) | LDD1351 | [9] |
LDCM0473 | CL8 | HCT 116 | C121(0.69) | LDD0790 | [9] |
LDCM0474 | CL80 | PaTu 8988t | C121(0.76) | LDD1353 | [9] |
LDCM0475 | CL81 | PaTu 8988t | C121(0.66) | LDD1354 | [9] |
LDCM0476 | CL82 | PaTu 8988t | C121(0.66) | LDD1355 | [9] |
LDCM0477 | CL83 | PaTu 8988t | C121(0.63) | LDD1356 | [9] |
LDCM0478 | CL84 | PaTu 8988t | C121(0.72) | LDD1357 | [9] |
LDCM0479 | CL85 | PaTu 8988t | C121(1.04) | LDD1358 | [9] |
LDCM0480 | CL86 | PaTu 8988t | C121(0.81) | LDD1359 | [9] |
LDCM0481 | CL87 | PaTu 8988t | C121(0.57) | LDD1360 | [9] |
LDCM0482 | CL88 | PaTu 8988t | C121(0.65) | LDD1361 | [9] |
LDCM0483 | CL89 | PaTu 8988t | C121(0.78) | LDD1362 | [9] |
LDCM0484 | CL9 | HCT 116 | C121(0.97) | LDD0801 | [9] |
LDCM0485 | CL90 | PaTu 8988t | C121(0.99) | LDD1364 | [9] |
LDCM0486 | CL91 | PaTu 8988t | C121(0.70) | LDD1365 | [9] |
LDCM0487 | CL92 | PaTu 8988t | C121(0.71) | LDD1366 | [9] |
LDCM0488 | CL93 | PaTu 8988t | C121(0.65) | LDD1367 | [9] |
LDCM0489 | CL94 | PaTu 8988t | C121(0.54) | LDD1368 | [9] |
LDCM0490 | CL95 | PaTu 8988t | C121(0.45) | LDD1369 | [9] |
LDCM0491 | CL96 | PaTu 8988t | C121(0.66) | LDD1370 | [9] |
LDCM0492 | CL97 | PaTu 8988t | C121(0.74) | LDD1371 | [9] |
LDCM0493 | CL98 | PaTu 8988t | C121(0.64) | LDD1372 | [9] |
LDCM0494 | CL99 | PaTu 8988t | C121(0.78) | LDD1373 | [9] |
LDCM0495 | E2913 | HEK-293T | C173(1.34); C121(1.07); C53(1.12) | LDD1698 | [26] |
LDCM0213 | Electrophilic fragment 2 | MDA-MB-231 | C121(0.99); C173(0.83) | LDD1702 | [5] |
LDCM0625 | F8 | Ramos | C173(1.31); C121(0.53) | LDD2187 | [27] |
LDCM0572 | Fragment10 | Ramos | C173(1.12); C121(0.79) | LDD2189 | [27] |
LDCM0573 | Fragment11 | Ramos | C173(0.25); C121(1.75) | LDD2190 | [27] |
LDCM0574 | Fragment12 | Ramos | C173(0.78); C121(0.74) | LDD2191 | [27] |
LDCM0575 | Fragment13 | Ramos | C173(0.94); C121(0.60) | LDD2192 | [27] |
LDCM0576 | Fragment14 | Ramos | C173(0.55); C121(0.60) | LDD2193 | [27] |
LDCM0579 | Fragment20 | Ramos | C173(0.97); C121(0.83) | LDD2194 | [27] |
LDCM0580 | Fragment21 | Ramos | C173(0.81); C121(0.83) | LDD2195 | [27] |
LDCM0582 | Fragment23 | Ramos | C173(0.91); C121(0.72) | LDD2196 | [27] |
LDCM0578 | Fragment27 | Ramos | C173(0.89); C121(0.85) | LDD2197 | [27] |
LDCM0586 | Fragment28 | Ramos | C173(0.73); C121(0.48) | LDD2198 | [27] |
LDCM0588 | Fragment30 | Ramos | C173(1.27); C121(1.55) | LDD2199 | [27] |
LDCM0589 | Fragment31 | Ramos | C173(0.73); C121(0.78) | LDD2200 | [27] |
LDCM0590 | Fragment32 | Ramos | C173(1.39); C121(0.52) | LDD2201 | [27] |
LDCM0468 | Fragment33 | PaTu 8988t | C121(1.14) | LDD1347 | [9] |
LDCM0596 | Fragment38 | Ramos | C173(0.81); C121(1.01) | LDD2203 | [27] |
LDCM0566 | Fragment4 | Ramos | C173(0.82); C121(0.84) | LDD2184 | [27] |
LDCM0427 | Fragment51 | PaTu 8988t | C121(0.46) | LDD1306 | [9] |
LDCM0610 | Fragment52 | Ramos | C173(1.09) | LDD2204 | [27] |
LDCM0614 | Fragment56 | Ramos | C173(1.47); C121(1.56) | LDD2205 | [27] |
LDCM0569 | Fragment7 | Ramos | C173(0.88); C121(0.71) | LDD2186 | [27] |
LDCM0571 | Fragment9 | Ramos | C173(0.89); C121(0.65) | LDD2188 | [27] |
LDCM0107 | IAA | HeLa | N.A. | LDD0221 | [18] |
LDCM0022 | KB02 | HEK-293T | C173(1.17); C121(0.99) | LDD1492 | [26] |
LDCM0023 | KB03 | HEK-293T | C173(1.01); C121(0.92) | LDD1497 | [26] |
LDCM0024 | KB05 | HMCB | C121(2.16) | LDD3312 | [28] |
LDCM0509 | N-(4-bromo-3,5-dimethylphenyl)-2-nitroacetamide | MDA-MB-231 | C173(0.78) | LDD2102 | [5] |
LDCM0528 | N-(4-bromophenyl)-2-cyano-N-phenylacetamide | MDA-MB-231 | C173(0.44) | LDD2121 | [5] |
LDCM0109 | NEM | HeLa | H14(0.00); K3(0.00) | LDD0223 | [18] |
LDCM0497 | Nucleophilic fragment 11b | MDA-MB-231 | C173(1.38) | LDD2090 | [5] |
LDCM0500 | Nucleophilic fragment 13a | MDA-MB-231 | C173(0.87) | LDD2093 | [5] |
LDCM0501 | Nucleophilic fragment 13b | MDA-MB-231 | C173(1.15); C121(1.33) | LDD2094 | [5] |
LDCM0503 | Nucleophilic fragment 14b | MDA-MB-231 | C121(0.91) | LDD2096 | [5] |
LDCM0504 | Nucleophilic fragment 15a | MDA-MB-231 | C173(0.79) | LDD2097 | [5] |
LDCM0505 | Nucleophilic fragment 15b | MDA-MB-231 | C173(0.56); C121(0.91) | LDD2098 | [5] |
LDCM0506 | Nucleophilic fragment 16a | MDA-MB-231 | C173(1.46) | LDD2099 | [5] |
LDCM0507 | Nucleophilic fragment 16b | MDA-MB-231 | C173(0.96); C121(0.46) | LDD2100 | [5] |
LDCM0508 | Nucleophilic fragment 17a | MDA-MB-231 | C173(0.74) | LDD2101 | [5] |
LDCM0511 | Nucleophilic fragment 18b | MDA-MB-231 | C173(0.66); C121(0.38) | LDD2104 | [5] |
LDCM0513 | Nucleophilic fragment 19b | MDA-MB-231 | C173(0.78) | LDD2106 | [5] |
LDCM0514 | Nucleophilic fragment 20a | MDA-MB-231 | C173(1.10) | LDD2107 | [5] |
LDCM0515 | Nucleophilic fragment 20b | MDA-MB-231 | C173(0.71); C121(0.58) | LDD2108 | [5] |
LDCM0516 | Nucleophilic fragment 21a | MDA-MB-231 | C173(1.10); C121(0.85) | LDD2109 | [5] |
LDCM0517 | Nucleophilic fragment 21b | MDA-MB-231 | C173(2.08) | LDD2110 | [5] |
LDCM0518 | Nucleophilic fragment 22a | MDA-MB-231 | C173(1.49) | LDD2111 | [5] |
LDCM0521 | Nucleophilic fragment 23b | MDA-MB-231 | C173(0.59) | LDD2114 | [5] |
LDCM0522 | Nucleophilic fragment 24a | MDA-MB-231 | C173(0.47) | LDD2115 | [5] |
LDCM0526 | Nucleophilic fragment 26a | MDA-MB-231 | C121(1.49) | LDD2119 | [5] |
LDCM0527 | Nucleophilic fragment 26b | MDA-MB-231 | C121(1.31) | LDD2120 | [5] |
LDCM0530 | Nucleophilic fragment 28a | MDA-MB-231 | C173(1.10) | LDD2123 | [5] |
LDCM0532 | Nucleophilic fragment 29a | MDA-MB-231 | C173(1.13); C121(1.10) | LDD2125 | [5] |
LDCM0534 | Nucleophilic fragment 30a | MDA-MB-231 | C173(1.41); C121(0.76) | LDD2127 | [5] |
LDCM0536 | Nucleophilic fragment 31 | MDA-MB-231 | C173(1.06) | LDD2129 | [5] |
LDCM0540 | Nucleophilic fragment 35 | MDA-MB-231 | C173(0.30) | LDD2133 | [5] |
LDCM0541 | Nucleophilic fragment 36 | MDA-MB-231 | C173(0.34); C121(0.73) | LDD2134 | [5] |
LDCM0542 | Nucleophilic fragment 37 | MDA-MB-231 | C173(1.04); C121(1.07) | LDD2135 | [5] |
LDCM0543 | Nucleophilic fragment 38 | MDA-MB-231 | C173(1.68) | LDD2136 | [5] |
LDCM0544 | Nucleophilic fragment 39 | MDA-MB-231 | C173(1.48); C121(1.26) | LDD2137 | [5] |
LDCM0546 | Nucleophilic fragment 40 | MDA-MB-231 | C173(0.92) | LDD2140 | [5] |
LDCM0547 | Nucleophilic fragment 41 | MDA-MB-231 | C173(0.75) | LDD2141 | [5] |
LDCM0550 | Nucleophilic fragment 5a | MDA-MB-231 | C173(3.06); C121(2.41) | LDD2144 | [5] |
LDCM0551 | Nucleophilic fragment 5b | MDA-MB-231 | C173(4.97) | LDD2145 | [5] |
LDCM0552 | Nucleophilic fragment 6a | MDA-MB-231 | C173(1.37) | LDD2146 | [5] |
LDCM0553 | Nucleophilic fragment 6b | MDA-MB-231 | C121(1.77) | LDD2147 | [5] |
LDCM0554 | Nucleophilic fragment 7a | MDA-MB-231 | C173(0.38); C121(0.48) | LDD2148 | [5] |
LDCM0556 | Nucleophilic fragment 8a | MDA-MB-231 | C173(0.45) | LDD2150 | [5] |
LDCM0559 | Nucleophilic fragment 9b | MDA-MB-231 | C173(0.99) | LDD2153 | [5] |
LDCM0628 | OTUB2-COV-1 | HEK-293T | C173(0.85) | LDD2207 | [29] |
LDCM0029 | Quercetin | HEK-293T | 4.85 | LDD0181 | [6] |
LDCM0131 | RA190 | MM1.R | 3.33 | LDD0300 | [8] |
The Interaction Atlas With This Target
The Protein(s) Related To This Target
Enzyme
Transporter and channel
Transcription factor
Protein name | Family | Uniprot ID | |||
---|---|---|---|---|---|
Zinc finger and BTB domain-containing protein 22 (ZBTB22) | Krueppel C2H2-type zinc-finger protein family | O15209 |
GPCR
Protein name | Family | Uniprot ID | |||
---|---|---|---|---|---|
Probable G-protein coupled receptor 25 (GPR25) | G-protein coupled receptor 1 family | O00155 |
Immunoglobulin
Protein name | Family | Uniprot ID | |||
---|---|---|---|---|---|
B-cell antigen receptor complex-associated protein alpha chain (CD79A) | . | P11912 |
Other
References