Details of the Target
General Information of Target
Target ID | LDTP01056 | |||||
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Target Name | Coiled-coil domain-containing protein 22 (CCDC22) | |||||
Gene Name | CCDC22 | |||||
Gene ID | 28952 | |||||
Synonyms |
CXorf37; Coiled-coil domain-containing protein 22 |
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3D Structure | ||||||
Sequence |
MEEADRILIHSLRQAGTAVPPDVQTLRAFTTELVVEAVVRCLRVINPAVGSGLSPLLPLA
MSARFRLAMSLAQACMDLGYPLELGYQNFLYPSEPDLRDLLLFLAERLPTDASEDADQPA GDSAILLRAIGSQIRDQLALPWVPPHLRTPKLQHLQGSALQKPFHASRLVVPELSSRGEP REFQASPLLLPVPTQVPQPVGRVASLLEHHALQLCQQTGRDRPGDEDWVHRTSRLPPQED TRAQRQRLQKQLTEHLRQSWGLLGAPIQARDLGELLQAWGAGAKTGAPKGSRFTHSEKFT FHLEPQAQATQVSDVPATSRRPEQVTWAAQEQELESLREQLEGVNRSIEEVEADMKTLGV SFVQAESECRHSKLSTAEREQALRLKSRAVELLPDGTANLAKLQLVVENSAQRVIHLAGQ WEKHRVPLLAEYRHLRKLQDCRELESSRRLAEIQELHQSVRAAAEEARRKEEVYKQLMSE LETLPRDVSRLAYTQRILEIVGNIRKQKEEITKILSDTKELQKEINSLSGKLDRTFAVTD ELVFKDAKKDDAVRKAYKYLAALHENCSQLIQTIEDTGTIMREVRDLEEQIETELGKKTL SNLEKIREDYRALRQENAGLLGRVREA |
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Target Bioclass |
Transporter and channel
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Family |
CCDC22 family
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Subcellular location |
Endosome
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Function |
Involved in regulation of NF-kappa-B signaling. Promotes ubiquitination of I-kappa-B-kinase subunit IKBKB and its subsequent proteasomal degradation leading to NF-kappa-B activation; the function may involve association with COMMD8 and a CUL1-dependent E3 ubiquitin ligase complex. May down-regulate NF-kappa-B activity via association with COMMD1 and involving a CUL2-dependent E3 ubiquitin ligase complex. Regulates the cellular localization of COMM domain-containing proteins, such as COMMD1 and COMMD10. Component of the CCC complex, which is involved in the regulation of endosomal recycling of surface proteins, including integrins, signaling receptor and channels. The CCC complex associates with SNX17, retriever and WASH complexes to prevent lysosomal degradation and promote cell surface recycling of numerous cargos such as integrins ITGA5:ITGB1. Plays a role in copper ion homeostasis. Involved in copper-dependent ATP7A trafficking between the trans-Golgi network and vesicles in the cell periphery; the function is proposed to depend on its association within the CCC complex and cooperation with the WASH complex on early endosomes.; (Microbial infection) The CCC complex, in collaboration with the heterotrimeric retriever complex, mediates the exit of human papillomavirus to the cell surface.
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Uniprot ID | ||||||
Ensemble ID | ||||||
HGNC ID |
Probe(s) Labeling This Target
ABPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
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m-APA Probe Info |
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15.00 | LDD0402 | [2] | |
BTD Probe Info |
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C441(0.66) | LDD2094 | [3] | |
DBIA Probe Info |
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C369(1.08) | LDD0531 | [4] | |
1d-yne Probe Info |
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N.A. | LDD0358 | [5] | |
4-Iodoacetamidophenylacetylene Probe Info |
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C369(0.00); C567(0.00) | LDD0038 | [6] | |
IA-alkyne Probe Info |
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C215(0.00); C567(0.00) | LDD0032 | [7] | |
Lodoacetamide azide Probe Info |
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C369(0.00); C567(0.00) | LDD0037 | [6] | |
ENE Probe Info |
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N.A. | LDD0006 | [8] | |
IPM Probe Info |
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N.A. | LDD0005 | [8] | |
STPyne Probe Info |
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N.A. | LDD0009 | [8] | |
TFBX Probe Info |
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C441(0.00); C369(0.00) | LDD0148 | [9] | |
1c-yne Probe Info |
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N.A. | LDD0228 | [5] | |
Acrolein Probe Info |
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C369(0.00); C215(0.00) | LDD0217 | [10] | |
Crotonaldehyde Probe Info |
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N.A. | LDD0219 | [10] | |
Methacrolein Probe Info |
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N.A. | LDD0218 | [10] | |
AOyne Probe Info |
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12.00 | LDD0443 | [11] | |
NAIA_5 Probe Info |
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N.A. | LDD2223 | [12] |
PAL-AfBPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
---|---|---|---|---|---|
C055 Probe Info |
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13.55 | LDD1752 | [13] | |
C158 Probe Info |
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10.63 | LDD1838 | [13] | |
C278 Probe Info |
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50.91 | LDD1948 | [13] | |
C391 Probe Info |
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18.00 | LDD2050 | [13] | |
FFF probe13 Probe Info |
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20.00 | LDD0475 | [14] | |
FFF probe3 Probe Info |
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20.00 | LDD0465 | [14] |
Competitor(s) Related to This Target
Competitor ID | Name | Cell line | Binding Site(Ratio) | Interaction ID | Ref |
---|---|---|---|---|---|
LDCM0214 | AC1 | HCT 116 | C369(1.08) | LDD0531 | [4] |
LDCM0215 | AC10 | HCT 116 | C369(1.09) | LDD0532 | [4] |
LDCM0216 | AC100 | HEK-293T | C369(1.08) | LDD0814 | [4] |
LDCM0217 | AC101 | HEK-293T | C369(1.15) | LDD0815 | [4] |
LDCM0218 | AC102 | HEK-293T | C369(1.13) | LDD0816 | [4] |
LDCM0219 | AC103 | HEK-293T | C369(1.14) | LDD0817 | [4] |
LDCM0220 | AC104 | HEK-293T | C369(1.11) | LDD0818 | [4] |
LDCM0221 | AC105 | HEK-293T | C369(0.99) | LDD0819 | [4] |
LDCM0222 | AC106 | HEK-293T | C369(1.03) | LDD0820 | [4] |
LDCM0223 | AC107 | HEK-293T | C369(1.07) | LDD0821 | [4] |
LDCM0224 | AC108 | HEK-293T | C369(0.97) | LDD0822 | [4] |
LDCM0225 | AC109 | HEK-293T | C369(1.05) | LDD0823 | [4] |
LDCM0226 | AC11 | HCT 116 | C369(0.91) | LDD0543 | [4] |
LDCM0227 | AC110 | HEK-293T | C369(1.21) | LDD0825 | [4] |
LDCM0228 | AC111 | HEK-293T | C369(1.29) | LDD0826 | [4] |
LDCM0229 | AC112 | HEK-293T | C369(1.15) | LDD0827 | [4] |
LDCM0230 | AC113 | HCT 116 | C369(1.09) | LDD0547 | [4] |
LDCM0231 | AC114 | HCT 116 | C369(0.90) | LDD0548 | [4] |
LDCM0232 | AC115 | HCT 116 | C369(0.86) | LDD0549 | [4] |
LDCM0233 | AC116 | HCT 116 | C369(0.84) | LDD0550 | [4] |
LDCM0234 | AC117 | HCT 116 | C369(0.91) | LDD0551 | [4] |
LDCM0235 | AC118 | HCT 116 | C369(1.08) | LDD0552 | [4] |
LDCM0236 | AC119 | HCT 116 | C369(0.87) | LDD0553 | [4] |
LDCM0237 | AC12 | HCT 116 | C369(0.95) | LDD0554 | [4] |
LDCM0238 | AC120 | HCT 116 | C369(0.78) | LDD0555 | [4] |
LDCM0239 | AC121 | HCT 116 | C369(0.93) | LDD0556 | [4] |
LDCM0240 | AC122 | HCT 116 | C369(0.91) | LDD0557 | [4] |
LDCM0241 | AC123 | HCT 116 | C369(1.01) | LDD0558 | [4] |
LDCM0242 | AC124 | HCT 116 | C369(0.96) | LDD0559 | [4] |
LDCM0243 | AC125 | HCT 116 | C369(0.92) | LDD0560 | [4] |
LDCM0244 | AC126 | HCT 116 | C369(1.02) | LDD0561 | [4] |
LDCM0245 | AC127 | HCT 116 | C369(0.84) | LDD0562 | [4] |
LDCM0246 | AC128 | HEK-293T | C369(1.10) | LDD0844 | [4] |
LDCM0247 | AC129 | HEK-293T | C369(1.17) | LDD0845 | [4] |
LDCM0249 | AC130 | HEK-293T | C369(0.99) | LDD0847 | [4] |
LDCM0250 | AC131 | HEK-293T | C369(0.97) | LDD0848 | [4] |
LDCM0251 | AC132 | HEK-293T | C369(1.09) | LDD0849 | [4] |
LDCM0252 | AC133 | HEK-293T | C369(1.06) | LDD0850 | [4] |
LDCM0253 | AC134 | HEK-293T | C369(1.06) | LDD0851 | [4] |
LDCM0254 | AC135 | HEK-293T | C369(1.02) | LDD0852 | [4] |
LDCM0255 | AC136 | HEK-293T | C369(1.15) | LDD0853 | [4] |
LDCM0256 | AC137 | HEK-293T | C369(1.17) | LDD0854 | [4] |
LDCM0257 | AC138 | HEK-293T | C369(1.10) | LDD0855 | [4] |
LDCM0258 | AC139 | HEK-293T | C369(1.14) | LDD0856 | [4] |
LDCM0259 | AC14 | HCT 116 | C369(1.02) | LDD0576 | [4] |
LDCM0260 | AC140 | HEK-293T | C369(1.08) | LDD0858 | [4] |
LDCM0261 | AC141 | HEK-293T | C369(1.28) | LDD0859 | [4] |
LDCM0262 | AC142 | HEK-293T | C369(1.17) | LDD0860 | [4] |
LDCM0263 | AC143 | HCT 116 | C369(0.99) | LDD0580 | [4] |
LDCM0264 | AC144 | HCT 116 | C369(0.62) | LDD0581 | [4] |
LDCM0265 | AC145 | HCT 116 | C369(0.60) | LDD0582 | [4] |
LDCM0266 | AC146 | HCT 116 | C369(0.64) | LDD0583 | [4] |
LDCM0267 | AC147 | HCT 116 | C369(0.91) | LDD0584 | [4] |
LDCM0268 | AC148 | HCT 116 | C369(0.57) | LDD0585 | [4] |
LDCM0269 | AC149 | HCT 116 | C369(0.64) | LDD0586 | [4] |
LDCM0270 | AC15 | HCT 116 | C369(1.02) | LDD0587 | [4] |
LDCM0271 | AC150 | HCT 116 | C369(0.65) | LDD0588 | [4] |
LDCM0272 | AC151 | HCT 116 | C369(0.80) | LDD0589 | [4] |
LDCM0273 | AC152 | HCT 116 | C369(0.61) | LDD0590 | [4] |
LDCM0274 | AC153 | HCT 116 | C369(0.64) | LDD0591 | [4] |
LDCM0621 | AC154 | HCT 116 | C369(0.62) | LDD2158 | [4] |
LDCM0622 | AC155 | HCT 116 | C369(0.64) | LDD2159 | [4] |
LDCM0623 | AC156 | HCT 116 | C369(0.77) | LDD2160 | [4] |
LDCM0624 | AC157 | HCT 116 | C369(0.61) | LDD2161 | [4] |
LDCM0276 | AC17 | HEK-293T | C369(1.13) | LDD0874 | [4] |
LDCM0277 | AC18 | HEK-293T | C369(0.95) | LDD0875 | [4] |
LDCM0278 | AC19 | HEK-293T | C369(0.99) | LDD0876 | [4] |
LDCM0279 | AC2 | HCT 116 | C369(1.19) | LDD0596 | [4] |
LDCM0280 | AC20 | HEK-293T | C369(1.09) | LDD0878 | [4] |
LDCM0281 | AC21 | HEK-293T | C369(0.98) | LDD0879 | [4] |
LDCM0282 | AC22 | HEK-293T | C369(1.12) | LDD0880 | [4] |
LDCM0283 | AC23 | HEK-293T | C369(1.12) | LDD0881 | [4] |
LDCM0284 | AC24 | HEK-293T | C369(1.12) | LDD0882 | [4] |
LDCM0285 | AC25 | HCT 116 | C369(0.79) | LDD0602 | [4] |
LDCM0286 | AC26 | HCT 116 | C369(1.04) | LDD0603 | [4] |
LDCM0287 | AC27 | HCT 116 | C369(0.96) | LDD0604 | [4] |
LDCM0288 | AC28 | HCT 116 | C369(0.94) | LDD0605 | [4] |
LDCM0289 | AC29 | HCT 116 | C369(0.88) | LDD0606 | [4] |
LDCM0290 | AC3 | HCT 116 | C369(1.19) | LDD0607 | [4] |
LDCM0291 | AC30 | HCT 116 | C369(0.84) | LDD0608 | [4] |
LDCM0292 | AC31 | HCT 116 | C369(0.94) | LDD0609 | [4] |
LDCM0293 | AC32 | HCT 116 | C369(0.93) | LDD0610 | [4] |
LDCM0294 | AC33 | HCT 116 | C369(0.81) | LDD0611 | [4] |
LDCM0295 | AC34 | HCT 116 | C369(0.89) | LDD0612 | [4] |
LDCM0296 | AC35 | HCT 116 | C369(0.85) | LDD0613 | [4] |
LDCM0297 | AC36 | HCT 116 | C369(1.55) | LDD0614 | [4] |
LDCM0298 | AC37 | HCT 116 | C369(0.88) | LDD0615 | [4] |
LDCM0299 | AC38 | HCT 116 | C369(0.83) | LDD0616 | [4] |
LDCM0300 | AC39 | HCT 116 | C369(0.81) | LDD0617 | [4] |
LDCM0301 | AC4 | HCT 116 | C369(1.21) | LDD0618 | [4] |
LDCM0302 | AC40 | HCT 116 | C369(0.86) | LDD0619 | [4] |
LDCM0303 | AC41 | HCT 116 | C369(0.85) | LDD0620 | [4] |
LDCM0304 | AC42 | HCT 116 | C369(0.90) | LDD0621 | [4] |
LDCM0305 | AC43 | HCT 116 | C369(1.03) | LDD0622 | [4] |
LDCM0306 | AC44 | HCT 116 | C369(1.12) | LDD0623 | [4] |
LDCM0307 | AC45 | HCT 116 | C369(0.85) | LDD0624 | [4] |
LDCM0308 | AC46 | HEK-293T | C369(0.98) | LDD0906 | [4] |
LDCM0309 | AC47 | HEK-293T | C369(0.77) | LDD0907 | [4] |
LDCM0310 | AC48 | HEK-293T | C369(0.85) | LDD0908 | [4] |
LDCM0311 | AC49 | HEK-293T | C369(0.92) | LDD0909 | [4] |
LDCM0312 | AC5 | HCT 116 | C369(1.05) | LDD0629 | [4] |
LDCM0313 | AC50 | HEK-293T | C369(0.97) | LDD0911 | [4] |
LDCM0314 | AC51 | HEK-293T | C369(0.89) | LDD0912 | [4] |
LDCM0315 | AC52 | HEK-293T | C369(0.89) | LDD0913 | [4] |
LDCM0316 | AC53 | HEK-293T | C369(0.85) | LDD0914 | [4] |
LDCM0317 | AC54 | HEK-293T | C369(0.92) | LDD0915 | [4] |
LDCM0318 | AC55 | HEK-293T | C369(0.84) | LDD0916 | [4] |
LDCM0319 | AC56 | HEK-293T | C369(0.93) | LDD0917 | [4] |
LDCM0320 | AC57 | HEK-293T | C369(0.90) | LDD0918 | [4] |
LDCM0321 | AC58 | HEK-293T | C369(0.81) | LDD0919 | [4] |
LDCM0322 | AC59 | HEK-293T | C369(1.13) | LDD0920 | [4] |
LDCM0323 | AC6 | HCT 116 | C369(1.03) | LDD0640 | [4] |
LDCM0324 | AC60 | HEK-293T | C369(0.70) | LDD0922 | [4] |
LDCM0325 | AC61 | HEK-293T | C369(0.98) | LDD0923 | [4] |
LDCM0326 | AC62 | HEK-293T | C369(0.83) | LDD0924 | [4] |
LDCM0327 | AC63 | HEK-293T | C369(0.93) | LDD0925 | [4] |
LDCM0328 | AC64 | HEK-293T | C369(0.80) | LDD0926 | [4] |
LDCM0329 | AC65 | HEK-293T | C369(0.81) | LDD0927 | [4] |
LDCM0330 | AC66 | HEK-293T | C369(0.74) | LDD0928 | [4] |
LDCM0331 | AC67 | HEK-293T | C369(1.10) | LDD0929 | [4] |
LDCM0332 | AC68 | HCT 116 | C369(0.98) | LDD0649 | [4] |
LDCM0333 | AC69 | HCT 116 | C369(0.95) | LDD0650 | [4] |
LDCM0334 | AC7 | HCT 116 | C369(1.09) | LDD0651 | [4] |
LDCM0335 | AC70 | HCT 116 | C369(1.05) | LDD0652 | [4] |
LDCM0336 | AC71 | HCT 116 | C369(0.92) | LDD0653 | [4] |
LDCM0337 | AC72 | HCT 116 | C369(1.00) | LDD0654 | [4] |
LDCM0338 | AC73 | HCT 116 | C369(1.28) | LDD0655 | [4] |
LDCM0339 | AC74 | HCT 116 | C369(1.07) | LDD0656 | [4] |
LDCM0340 | AC75 | HCT 116 | C369(1.07) | LDD0657 | [4] |
LDCM0341 | AC76 | HCT 116 | C369(1.04) | LDD0658 | [4] |
LDCM0342 | AC77 | HCT 116 | C369(0.87) | LDD0659 | [4] |
LDCM0343 | AC78 | HCT 116 | C369(0.81) | LDD0660 | [4] |
LDCM0344 | AC79 | HCT 116 | C369(0.93) | LDD0661 | [4] |
LDCM0345 | AC8 | HCT 116 | C369(0.97) | LDD0662 | [4] |
LDCM0346 | AC80 | HCT 116 | C369(0.99) | LDD0663 | [4] |
LDCM0347 | AC81 | HCT 116 | C369(1.02) | LDD0664 | [4] |
LDCM0348 | AC82 | HCT 116 | C369(0.93) | LDD0665 | [4] |
LDCM0349 | AC83 | HCT 116 | C369(0.96) | LDD0666 | [4] |
LDCM0350 | AC84 | HCT 116 | C369(0.99) | LDD0667 | [4] |
LDCM0351 | AC85 | HCT 116 | C369(0.88) | LDD0668 | [4] |
LDCM0352 | AC86 | HCT 116 | C369(1.00) | LDD0669 | [4] |
LDCM0353 | AC87 | HCT 116 | C369(1.05) | LDD0670 | [4] |
LDCM0354 | AC88 | HCT 116 | C369(0.96) | LDD0671 | [4] |
LDCM0355 | AC89 | HCT 116 | C369(0.99) | LDD0672 | [4] |
LDCM0357 | AC90 | HCT 116 | C369(1.05) | LDD0674 | [4] |
LDCM0358 | AC91 | HCT 116 | C369(0.99) | LDD0675 | [4] |
LDCM0359 | AC92 | HCT 116 | C369(0.97) | LDD0676 | [4] |
LDCM0360 | AC93 | HCT 116 | C369(0.96) | LDD0677 | [4] |
LDCM0361 | AC94 | HCT 116 | C369(1.08) | LDD0678 | [4] |
LDCM0362 | AC95 | HCT 116 | C369(1.01) | LDD0679 | [4] |
LDCM0363 | AC96 | HCT 116 | C369(1.05) | LDD0680 | [4] |
LDCM0364 | AC97 | HCT 116 | C369(1.00) | LDD0681 | [4] |
LDCM0365 | AC98 | HEK-293T | C369(0.97) | LDD0963 | [4] |
LDCM0366 | AC99 | HEK-293T | C369(1.00) | LDD0964 | [4] |
LDCM0248 | AKOS034007472 | HCT 116 | C369(1.03) | LDD0565 | [4] |
LDCM0356 | AKOS034007680 | HCT 116 | C369(1.01) | LDD0673 | [4] |
LDCM0275 | AKOS034007705 | HCT 116 | C369(1.07) | LDD0592 | [4] |
LDCM0108 | Chloroacetamide | HeLa | N.A. | LDD0222 | [10] |
LDCM0367 | CL1 | HCT 116 | C369(1.04) | LDD0684 | [4] |
LDCM0368 | CL10 | HCT 116 | C369(1.10) | LDD0685 | [4] |
LDCM0369 | CL100 | HCT 116 | C369(1.12) | LDD0686 | [4] |
LDCM0370 | CL101 | HCT 116 | C369(1.13) | LDD0687 | [4] |
LDCM0371 | CL102 | HCT 116 | C369(1.02) | LDD0688 | [4] |
LDCM0372 | CL103 | HCT 116 | C369(1.04) | LDD0689 | [4] |
LDCM0373 | CL104 | HCT 116 | C369(1.05) | LDD0690 | [4] |
LDCM0374 | CL105 | HEK-293T | C369(1.07) | LDD0972 | [4] |
LDCM0375 | CL106 | HEK-293T | C369(1.03) | LDD0973 | [4] |
LDCM0376 | CL107 | HEK-293T | C369(1.00) | LDD0974 | [4] |
LDCM0377 | CL108 | HEK-293T | C369(1.02) | LDD0975 | [4] |
LDCM0378 | CL109 | HEK-293T | C369(1.06) | LDD0976 | [4] |
LDCM0379 | CL11 | HCT 116 | C369(1.09) | LDD0696 | [4] |
LDCM0380 | CL110 | HEK-293T | C369(1.05) | LDD0978 | [4] |
LDCM0381 | CL111 | HEK-293T | C369(1.03) | LDD0979 | [4] |
LDCM0382 | CL112 | HCT 116 | C369(0.79) | LDD0699 | [4] |
LDCM0383 | CL113 | HCT 116 | C369(0.92) | LDD0700 | [4] |
LDCM0384 | CL114 | HCT 116 | C369(0.85) | LDD0701 | [4] |
LDCM0385 | CL115 | HCT 116 | C369(0.87) | LDD0702 | [4] |
LDCM0386 | CL116 | HCT 116 | C369(0.98) | LDD0703 | [4] |
LDCM0387 | CL117 | HCT 116 | C369(1.07) | LDD0704 | [4] |
LDCM0388 | CL118 | HCT 116 | C369(0.91) | LDD0705 | [4] |
LDCM0389 | CL119 | HCT 116 | C369(0.90) | LDD0706 | [4] |
LDCM0390 | CL12 | HCT 116 | C369(1.13) | LDD0707 | [4] |
LDCM0391 | CL120 | HCT 116 | C369(0.98) | LDD0708 | [4] |
LDCM0392 | CL121 | HEK-293T | C369(0.84) | LDD0990 | [4] |
LDCM0393 | CL122 | HEK-293T | C369(0.96) | LDD0991 | [4] |
LDCM0394 | CL123 | HEK-293T | C369(0.93) | LDD0992 | [4] |
LDCM0395 | CL124 | HEK-293T | C369(0.77) | LDD0993 | [4] |
LDCM0396 | CL125 | HEK-293T | C369(0.86) | LDD0994 | [4] |
LDCM0397 | CL126 | HEK-293T | C369(0.81) | LDD0995 | [4] |
LDCM0398 | CL127 | HEK-293T | C369(0.82) | LDD0996 | [4] |
LDCM0399 | CL128 | HEK-293T | C369(0.82) | LDD0997 | [4] |
LDCM0400 | CL13 | HCT 116 | C369(1.15) | LDD0717 | [4] |
LDCM0401 | CL14 | HCT 116 | C369(1.32) | LDD0718 | [4] |
LDCM0402 | CL15 | HCT 116 | C369(1.08) | LDD0719 | [4] |
LDCM0403 | CL16 | HCT 116 | C369(1.07) | LDD0720 | [4] |
LDCM0404 | CL17 | HCT 116 | C369(0.90) | LDD0721 | [4] |
LDCM0405 | CL18 | HCT 116 | C369(0.93) | LDD0722 | [4] |
LDCM0406 | CL19 | HCT 116 | C369(1.05) | LDD0723 | [4] |
LDCM0407 | CL2 | HCT 116 | C369(1.13) | LDD0724 | [4] |
LDCM0408 | CL20 | HCT 116 | C369(1.06) | LDD0725 | [4] |
LDCM0409 | CL21 | HCT 116 | C369(0.94) | LDD0726 | [4] |
LDCM0410 | CL22 | HCT 116 | C369(0.91) | LDD0727 | [4] |
LDCM0411 | CL23 | HCT 116 | C369(1.13) | LDD0728 | [4] |
LDCM0412 | CL24 | HCT 116 | C369(1.08) | LDD0729 | [4] |
LDCM0413 | CL25 | HCT 116 | C369(1.08) | LDD0730 | [4] |
LDCM0414 | CL26 | HCT 116 | C369(1.14) | LDD0731 | [4] |
LDCM0415 | CL27 | HCT 116 | C369(1.03) | LDD0732 | [4] |
LDCM0416 | CL28 | HCT 116 | C369(1.14) | LDD0733 | [4] |
LDCM0417 | CL29 | HCT 116 | C369(1.02) | LDD0734 | [4] |
LDCM0418 | CL3 | HCT 116 | C369(0.97) | LDD0735 | [4] |
LDCM0419 | CL30 | HCT 116 | C369(1.05) | LDD0736 | [4] |
LDCM0420 | CL31 | HCT 116 | C369(0.93) | LDD0737 | [4] |
LDCM0421 | CL32 | HCT 116 | C369(1.02) | LDD0738 | [4] |
LDCM0422 | CL33 | HCT 116 | C369(1.18) | LDD0739 | [4] |
LDCM0423 | CL34 | HCT 116 | C369(1.03) | LDD0740 | [4] |
LDCM0424 | CL35 | HCT 116 | C369(0.79) | LDD0741 | [4] |
LDCM0425 | CL36 | HCT 116 | C369(0.76) | LDD0742 | [4] |
LDCM0426 | CL37 | HCT 116 | C369(0.74) | LDD0743 | [4] |
LDCM0428 | CL39 | HCT 116 | C369(0.62) | LDD0745 | [4] |
LDCM0429 | CL4 | HCT 116 | C369(1.19) | LDD0746 | [4] |
LDCM0430 | CL40 | HCT 116 | C369(0.63) | LDD0747 | [4] |
LDCM0431 | CL41 | HCT 116 | C369(0.51) | LDD0748 | [4] |
LDCM0432 | CL42 | HCT 116 | C369(0.51) | LDD0749 | [4] |
LDCM0433 | CL43 | HCT 116 | C369(0.82) | LDD0750 | [4] |
LDCM0434 | CL44 | HCT 116 | C369(0.96) | LDD0751 | [4] |
LDCM0435 | CL45 | HCT 116 | C369(1.11) | LDD0752 | [4] |
LDCM0436 | CL46 | HCT 116 | C369(0.95) | LDD0753 | [4] |
LDCM0437 | CL47 | HCT 116 | C369(0.79) | LDD0754 | [4] |
LDCM0438 | CL48 | HCT 116 | C369(0.96) | LDD0755 | [4] |
LDCM0439 | CL49 | HCT 116 | C369(0.98) | LDD0756 | [4] |
LDCM0440 | CL5 | HCT 116 | C369(1.01) | LDD0757 | [4] |
LDCM0441 | CL50 | HCT 116 | C369(0.89) | LDD0758 | [4] |
LDCM0442 | CL51 | HCT 116 | C369(0.98) | LDD0759 | [4] |
LDCM0443 | CL52 | HCT 116 | C369(0.87) | LDD0760 | [4] |
LDCM0444 | CL53 | HCT 116 | C369(0.92) | LDD0761 | [4] |
LDCM0445 | CL54 | HCT 116 | C369(0.94) | LDD0762 | [4] |
LDCM0446 | CL55 | HCT 116 | C369(0.86) | LDD0763 | [4] |
LDCM0447 | CL56 | HCT 116 | C369(0.97) | LDD0764 | [4] |
LDCM0448 | CL57 | HCT 116 | C369(0.78) | LDD0765 | [4] |
LDCM0449 | CL58 | HCT 116 | C369(0.87) | LDD0766 | [4] |
LDCM0450 | CL59 | HCT 116 | C369(0.90) | LDD0767 | [4] |
LDCM0451 | CL6 | HCT 116 | C369(1.21) | LDD0768 | [4] |
LDCM0452 | CL60 | HCT 116 | C369(0.88) | LDD0769 | [4] |
LDCM0453 | CL61 | HCT 116 | C369(0.75) | LDD0770 | [4] |
LDCM0454 | CL62 | HCT 116 | C369(0.97) | LDD0771 | [4] |
LDCM0455 | CL63 | HCT 116 | C369(0.70) | LDD0772 | [4] |
LDCM0456 | CL64 | HCT 116 | C369(0.65) | LDD0773 | [4] |
LDCM0457 | CL65 | HCT 116 | C369(0.78) | LDD0774 | [4] |
LDCM0458 | CL66 | HCT 116 | C369(0.68) | LDD0775 | [4] |
LDCM0459 | CL67 | HCT 116 | C369(0.59) | LDD0776 | [4] |
LDCM0460 | CL68 | HCT 116 | C369(0.44) | LDD0777 | [4] |
LDCM0461 | CL69 | HCT 116 | C369(0.58) | LDD0778 | [4] |
LDCM0462 | CL7 | HCT 116 | C369(1.18) | LDD0779 | [4] |
LDCM0463 | CL70 | HCT 116 | C369(0.75) | LDD0780 | [4] |
LDCM0464 | CL71 | HCT 116 | C369(0.76) | LDD0781 | [4] |
LDCM0465 | CL72 | HCT 116 | C369(0.89) | LDD0782 | [4] |
LDCM0466 | CL73 | HCT 116 | C369(0.89) | LDD0783 | [4] |
LDCM0467 | CL74 | HCT 116 | C369(0.86) | LDD0784 | [4] |
LDCM0469 | CL76 | HCT 116 | C369(0.66) | LDD0786 | [4] |
LDCM0470 | CL77 | HCT 116 | C369(0.41) | LDD0787 | [4] |
LDCM0471 | CL78 | HCT 116 | C369(0.41) | LDD0788 | [4] |
LDCM0472 | CL79 | HCT 116 | C369(0.73) | LDD0789 | [4] |
LDCM0473 | CL8 | HCT 116 | C369(1.11) | LDD0790 | [4] |
LDCM0474 | CL80 | HCT 116 | C369(1.01) | LDD0791 | [4] |
LDCM0475 | CL81 | HCT 116 | C369(0.50) | LDD0792 | [4] |
LDCM0476 | CL82 | HCT 116 | C369(0.52) | LDD0793 | [4] |
LDCM0477 | CL83 | HCT 116 | C369(0.52) | LDD0794 | [4] |
LDCM0478 | CL84 | HCT 116 | C369(0.70) | LDD0795 | [4] |
LDCM0479 | CL85 | HCT 116 | C369(0.66) | LDD0796 | [4] |
LDCM0480 | CL86 | HCT 116 | C369(0.38) | LDD0797 | [4] |
LDCM0481 | CL87 | HCT 116 | C369(0.50) | LDD0798 | [4] |
LDCM0482 | CL88 | HCT 116 | C369(0.43) | LDD0799 | [4] |
LDCM0483 | CL89 | HCT 116 | C369(0.75) | LDD0800 | [4] |
LDCM0484 | CL9 | HCT 116 | C369(1.34) | LDD0801 | [4] |
LDCM0485 | CL90 | HCT 116 | C369(0.60) | LDD0802 | [4] |
LDCM0486 | CL91 | HCT 116 | C369(0.86) | LDD0803 | [4] |
LDCM0487 | CL92 | HCT 116 | C369(0.90) | LDD0804 | [4] |
LDCM0488 | CL93 | HCT 116 | C369(0.94) | LDD0805 | [4] |
LDCM0489 | CL94 | HCT 116 | C369(1.04) | LDD0806 | [4] |
LDCM0490 | CL95 | HCT 116 | C369(1.06) | LDD0807 | [4] |
LDCM0491 | CL96 | HCT 116 | C369(0.97) | LDD0808 | [4] |
LDCM0492 | CL97 | HCT 116 | C369(1.05) | LDD0809 | [4] |
LDCM0493 | CL98 | HCT 116 | C369(0.97) | LDD0810 | [4] |
LDCM0494 | CL99 | HCT 116 | C369(0.93) | LDD0811 | [4] |
LDCM0495 | E2913 | HEK-293T | C215(0.95); C369(1.00) | LDD1698 | [15] |
LDCM0468 | Fragment33 | HCT 116 | C369(0.72) | LDD0785 | [4] |
LDCM0427 | Fragment51 | HCT 116 | C369(0.08) | LDD0744 | [4] |
LDCM0022 | KB02 | HEK-293T | C215(0.94); C369(0.94); C567(1.14) | LDD1492 | [15] |
LDCM0023 | KB03 | HEK-293T | C215(1.00); C369(1.04); C567(1.21) | LDD1497 | [15] |
LDCM0024 | KB05 | HMCB | C369(2.34) | LDD3312 | [16] |
LDCM0501 | Nucleophilic fragment 13b | MDA-MB-231 | C441(0.66) | LDD2094 | [3] |
The Interaction Atlas With This Target
The Protein(s) Related To This Target
Enzyme
Transporter and channel
Protein name | Family | Uniprot ID | |||
---|---|---|---|---|---|
Coiled-coil domain-containing protein 93 (CCDC93) | CCDC93 family | Q567U6 | |||
WASH complex subunit 2A (WASHC2A) | FAM21 family | Q641Q2 |
Other
References