Details of the Target
General Information of Target
Target ID | LDTP08369 | |||||
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Target Name | ATP-dependent RNA helicase DDX42 (DDX42) | |||||
Gene Name | DDX42 | |||||
Gene ID | 11325 | |||||
Synonyms |
ATP-dependent RNA helicase DDX42; EC 3.6.4.13; DEAD box protein 42; RNA helicase-like protein; RHELP; RNA helicase-related protein; RNAHP; SF3b DEAD box protein; Splicing factor 3B-associated 125 kDa protein; SF3b125
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3D Structure | ||||||
Sequence |
MNWNKGGPGTKRGFGFGGFAISAGKKEEPKLPQQSHSAFGATSSSSGFGKSAPPQLPSFY
KIGSKRANFDEENAYFEDEEEDSSNVDLPYIPAENSPTRQQFHSKPVDSDSDDDPLEAFM AEVEDQAARDMKRLEEKDKERKNVKGIRDDIEEEDDQEAYFRYMAENPTAGVVQEEEEDN LEYDSDGNPIAPTKKIIDPLPPIDHSEIDYPPFEKNFYNEHEEITNLTPQQLIDLRHKLN LRVSGAAPPRPGSSFAHFGFDEQLMHQIRKSEYTQPTPIQCQGVPVALSGRDMIGIAKTG SGKTAAFIWPMLIHIMDQKELEPGDGPIAVIVCPTRELCQQIHAECKRFGKAYNLRSVAV YGGGSMWEQAKALQEGAEIVVCTPGRLIDHVKKKATNLQRVSYLVFDEADRMFDMGFEYQ VRSIASHVRPDRQTLLFSATFRKKIEKLARDILIDPIRVVQGDIGEANEDVTQIVEILHS GPSKWNWLTRRLVEFTSSGSVLLFVTKKANAEELANNLKQEGHNLGLLHGDMDQSERNKV ISDFKKKDIPVLVATDVAARGLDIPSIKTVINYDVARDIDTHTHRIGRTGRAGEKGVAYT LLTPKDSNFAGDLVRNLEGANQHVSKELLDLAMQNAWFRKSRFKGGKGKKLNIGGGGLGY RERPGLGSENMDRGNNNVMSNYEAYKPSTGAMGDRLTAMKAAFQSQYKSHFVAASLSNQK AGSSAAGASGWTSAGSLNSVPTNSAQQGHNSPDSPVTSAAKGIPGFGNTGNISGAPVTYP SAGAQGVNNTASGNNSREGTGGSNGKRERYTENRGSSRHSHGETGNRHSDSPRHGDGGRH GDGYRHPESSSRHTDGHRHGENRHGGSAGRHGENRGANDGRNGESRKEAFNRESKMEPKM EPKVDSSKMDKVDSKTDKTADGFAVPEPPKRKKSRWDS |
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Target Bioclass |
Enzyme
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Family |
DEAD box helicase family, DDX42 subfamily
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Subcellular location |
Cytoplasm; Nucleus, Cajal body
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Function |
ATP-dependent RNA helicase that binds to partially double-stranded RNAs (dsRNAs) in order to unwind RNA secondary structures. Unwinding is promoted in the presence of single-strand binding proteins. Mediates also RNA duplex formation thereby displacing the single-strand RNA binding protein. ATP and ADP modulate its activity: ATP binding and hydrolysis by DDX42 triggers RNA strand separation, whereas the ADP-bound form of the protein triggers annealing of complementary RNA strands. Required for assembly of the 17S U2 SnRNP complex of the spliceosome, a large ribonucleoprotein complex that removes introns from transcribed pre-mRNAs: DDX42 associates transiently with the SF3B subcomplex of the 17S U2 SnRNP complex and is released after fulfilling its role in the assembly of 17S U2 SnRNP. Involved in the survival of cells by interacting with TP53BP2 and thereby counteracting the apoptosis-stimulating activity of TP53BP2. Relocalizes TP53BP2 to the cytoplasm.
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Uniprot ID | ||||||
Ensemble ID | ||||||
HGNC ID | ||||||
ChEMBL ID |
Target Site Mutations in Different Cell Lines
Cell line | Mutation details | Probe for labeling this protein in this cell | |||
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CCK81 | SNV: p.R429H | DBIA Probe Info | |||
HCC70 | SNV: p.A372S | DBIA Probe Info | |||
KYSE150 | Substitution: p.N143I | DBIA Probe Info | |||
RL952 | SNV: p.A170V | . | |||
SH4 | SNV: p.D198N | DBIA Probe Info |
Probe(s) Labeling This Target
ABPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
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CY4 Probe Info |
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100.00 | LDD0244 | [1] | |
C-Sul Probe Info |
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3.67 | LDD0066 | [2] | |
Probe 1 Probe Info |
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Y60(12.15); Y160(15.64); Y660(18.44); Y707(91.94) | LDD3495 | [3] | |
BTD Probe Info |
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C346(1.68); C382(1.63) | LDD2099 | [4] | |
HHS-475 Probe Info |
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Y779(0.72); Y707(0.77); Y361(1.74) | LDD0264 | [5] | |
HHS-465 Probe Info |
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Y361(10.00) | LDD2237 | [6] | |
DBIA Probe Info |
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C281(1.02); C333(0.91); C339(0.90); C346(0.87) | LDD0531 | [7] | |
5E-2FA Probe Info |
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N.A. | LDD2235 | [8] | |
ATP probe Probe Info |
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K270(0.00); K347(0.00); K195(0.00) | LDD0199 | [9] | |
m-APA Probe Info |
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N.A. | LDD2231 | [8] | |
4-Iodoacetamidophenylacetylene Probe Info |
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C382(0.00); C333(0.00); C281(0.00) | LDD0038 | [10] | |
IA-alkyne Probe Info |
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C281(0.00); C333(0.00) | LDD0032 | [11] | |
IPIAA_H Probe Info |
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N.A. | LDD0030 | [12] | |
IPIAA_L Probe Info |
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N.A. | LDD0031 | [12] | |
Lodoacetamide azide Probe Info |
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C382(0.00); C333(0.00); C281(0.00) | LDD0037 | [10] | |
TFBX Probe Info |
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C382(0.00); C281(0.00) | LDD0027 | [13] | |
Compound 10 Probe Info |
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N.A. | LDD2216 | [14] | |
IPM Probe Info |
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N.A. | LDD0147 | [13] | |
SF Probe Info |
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Y707(0.00); Y60(0.00) | LDD0028 | [15] | |
STPyne Probe Info |
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N.A. | LDD0009 | [16] | |
1c-yne Probe Info |
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N.A. | LDD0228 | [17] | |
1d-yne Probe Info |
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N.A. | LDD0357 | [17] | |
Acrolein Probe Info |
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C339(0.00); C333(0.00); H623(0.00); C346(0.00) | LDD0217 | [18] | |
Crotonaldehyde Probe Info |
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N.A. | LDD0219 | [18] | |
Methacrolein Probe Info |
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C382(0.00); C339(0.00) | LDD0218 | [18] | |
NAIA_5 Probe Info |
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N.A. | LDD2223 | [19] |
PAL-AfBPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
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FFF probe13 Probe Info |
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8.77 | LDD0475 | [20] | |
FFF probe2 Probe Info |
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9.53 | LDD0463 | [20] | |
VE-P Probe Info |
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N.A. | LDD0396 | [21] |
Competitor(s) Related to This Target
Competitor ID | Name | Cell line | Binding Site(Ratio) | Interaction ID | Ref |
---|---|---|---|---|---|
LDCM0524 | 2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide | MDA-MB-231 | C382(1.27) | LDD2117 | [4] |
LDCM0214 | AC1 | HCT 116 | C281(1.02); C333(0.91); C339(0.90); C346(0.87) | LDD0531 | [7] |
LDCM0215 | AC10 | HCT 116 | C281(0.80); C333(0.84); C339(1.30); C346(1.23) | LDD0532 | [7] |
LDCM0216 | AC100 | HCT 116 | C281(0.70); C333(0.73); C339(0.78); C346(0.91) | LDD0533 | [7] |
LDCM0217 | AC101 | HCT 116 | C281(0.66); C333(0.78); C339(0.69); C346(0.74) | LDD0534 | [7] |
LDCM0218 | AC102 | HCT 116 | C281(0.62); C333(0.83); C339(0.69); C346(0.74) | LDD0535 | [7] |
LDCM0219 | AC103 | HCT 116 | C281(0.54); C333(0.60); C339(0.63); C346(0.62) | LDD0536 | [7] |
LDCM0220 | AC104 | HCT 116 | C281(0.55); C333(0.69); C339(0.65); C346(0.70) | LDD0537 | [7] |
LDCM0221 | AC105 | HCT 116 | C281(0.61); C333(0.71); C339(0.66); C346(0.69) | LDD0538 | [7] |
LDCM0222 | AC106 | HCT 116 | C281(0.68); C333(0.70); C339(0.63); C346(0.65) | LDD0539 | [7] |
LDCM0223 | AC107 | HCT 116 | C281(0.60); C333(0.76); C339(0.82); C346(0.87) | LDD0540 | [7] |
LDCM0224 | AC108 | HCT 116 | C281(0.59); C333(0.78); C339(0.82); C346(0.83) | LDD0541 | [7] |
LDCM0225 | AC109 | HCT 116 | C281(0.61); C333(0.72); C339(0.73); C346(0.82) | LDD0542 | [7] |
LDCM0226 | AC11 | HCT 116 | C281(0.63); C333(0.83); C339(1.33); C346(1.26) | LDD0543 | [7] |
LDCM0227 | AC110 | HCT 116 | C281(0.63); C333(0.76); C339(0.74); C346(0.80) | LDD0544 | [7] |
LDCM0228 | AC111 | HCT 116 | C281(0.58); C333(0.71); C339(0.77); C346(0.74) | LDD0545 | [7] |
LDCM0229 | AC112 | HCT 116 | C281(0.62); C333(0.67); C339(0.72); C346(0.70) | LDD0546 | [7] |
LDCM0230 | AC113 | HCT 116 | C281(1.00); C333(0.90); C339(1.03); C346(1.05) | LDD0547 | [7] |
LDCM0231 | AC114 | HCT 116 | C281(1.08); C333(0.82); C339(0.98); C346(0.97) | LDD0548 | [7] |
LDCM0232 | AC115 | HCT 116 | C281(0.89); C333(1.05); C339(0.88); C346(0.89) | LDD0549 | [7] |
LDCM0233 | AC116 | HCT 116 | C281(0.87); C333(0.98); C339(0.98); C346(0.97) | LDD0550 | [7] |
LDCM0234 | AC117 | HCT 116 | C281(0.88); C333(0.77); C339(0.97); C346(1.02) | LDD0551 | [7] |
LDCM0235 | AC118 | HCT 116 | C281(0.90); C333(0.92); C339(1.00); C346(1.04) | LDD0552 | [7] |
LDCM0236 | AC119 | HCT 116 | C281(0.95); C333(0.90); C339(0.99); C346(0.99) | LDD0553 | [7] |
LDCM0237 | AC12 | HCT 116 | C281(0.77); C333(0.96); C339(1.20); C346(1.19) | LDD0554 | [7] |
LDCM0238 | AC120 | HCT 116 | C281(0.87); C333(0.88); C339(1.02); C346(1.01) | LDD0555 | [7] |
LDCM0239 | AC121 | HCT 116 | C281(1.02); C333(0.84); C339(1.15); C346(1.12) | LDD0556 | [7] |
LDCM0240 | AC122 | HCT 116 | C281(0.92); C333(0.85); C339(1.01); C346(1.03) | LDD0557 | [7] |
LDCM0241 | AC123 | HCT 116 | C281(1.21); C333(0.97); C339(0.97); C346(1.01) | LDD0558 | [7] |
LDCM0242 | AC124 | HCT 116 | C281(1.02); C333(0.79); C339(1.08); C346(1.06) | LDD0559 | [7] |
LDCM0243 | AC125 | HCT 116 | C281(1.16); C333(0.87); C339(0.98); C346(1.02) | LDD0560 | [7] |
LDCM0244 | AC126 | HCT 116 | C281(0.96); C333(1.04); C339(0.96); C346(1.00) | LDD0561 | [7] |
LDCM0245 | AC127 | HCT 116 | C281(1.09); C333(0.95); C339(1.03); C346(1.02) | LDD0562 | [7] |
LDCM0246 | AC128 | HCT 116 | C281(1.04); C333(0.95); C339(1.09); C346(1.03) | LDD0563 | [7] |
LDCM0247 | AC129 | HCT 116 | C281(0.93); C333(1.32); C339(1.07); C346(1.09) | LDD0564 | [7] |
LDCM0249 | AC130 | HCT 116 | C281(0.83); C333(1.20); C339(0.98); C346(0.97) | LDD0566 | [7] |
LDCM0250 | AC131 | HCT 116 | C281(1.03); C333(0.80); C339(1.14); C346(0.96) | LDD0567 | [7] |
LDCM0251 | AC132 | HCT 116 | C281(0.91); C333(0.97); C339(1.12); C346(1.00) | LDD0568 | [7] |
LDCM0252 | AC133 | HCT 116 | C281(0.93); C333(1.12); C339(1.03); C346(0.94) | LDD0569 | [7] |
LDCM0253 | AC134 | HCT 116 | C281(0.79); C333(0.94); C339(1.09); C346(0.88) | LDD0570 | [7] |
LDCM0254 | AC135 | HCT 116 | C281(0.82); C333(0.96); C339(1.02); C346(0.93) | LDD0571 | [7] |
LDCM0255 | AC136 | HCT 116 | C281(0.83); C333(1.43); C339(0.99); C346(0.94) | LDD0572 | [7] |
LDCM0256 | AC137 | HCT 116 | C281(0.75); C333(1.02); C339(1.02); C346(0.96) | LDD0573 | [7] |
LDCM0257 | AC138 | HCT 116 | C281(0.81); C333(1.03); C339(1.09); C346(0.95) | LDD0574 | [7] |
LDCM0258 | AC139 | HCT 116 | C281(0.77); C333(1.11); C339(0.96); C346(0.88) | LDD0575 | [7] |
LDCM0259 | AC14 | HCT 116 | C281(0.72); C333(0.81); C339(1.42); C346(1.28) | LDD0576 | [7] |
LDCM0260 | AC140 | HCT 116 | C281(0.79); C333(0.84); C339(1.05); C346(0.90) | LDD0577 | [7] |
LDCM0261 | AC141 | HCT 116 | C281(0.81); C333(0.83); C339(1.09); C346(0.92) | LDD0578 | [7] |
LDCM0262 | AC142 | HCT 116 | C281(0.84); C333(1.33); C339(1.17); C346(1.05) | LDD0579 | [7] |
LDCM0263 | AC143 | HCT 116 | C281(1.02); C333(0.97); C339(0.74); C346(0.77) | LDD0580 | [7] |
LDCM0264 | AC144 | HCT 116 | C339(0.63); C346(0.74); C333(0.75); C382(0.82) | LDD0581 | [7] |
LDCM0265 | AC145 | HCT 116 | C339(0.72); C346(0.73); C382(0.80); C333(0.81) | LDD0582 | [7] |
LDCM0266 | AC146 | HCT 116 | C339(0.56); C346(0.71); C333(0.76); C281(0.82) | LDD0583 | [7] |
LDCM0267 | AC147 | HCT 116 | C346(0.62); C339(0.72); C333(0.76); C281(0.81) | LDD0584 | [7] |
LDCM0268 | AC148 | HCT 116 | C339(0.56); C346(0.61); C281(0.72); C333(0.82) | LDD0585 | [7] |
LDCM0269 | AC149 | HCT 116 | C339(0.57); C346(0.59); C281(0.64); C333(0.74) | LDD0586 | [7] |
LDCM0270 | AC15 | HCT 116 | C281(0.77); C333(0.79); C382(1.02); C346(1.22) | LDD0587 | [7] |
LDCM0271 | AC150 | HCT 116 | C346(0.66); C339(0.70); C333(0.75); C281(0.82) | LDD0588 | [7] |
LDCM0272 | AC151 | HCT 116 | C346(0.65); C339(0.72); C333(0.86); C281(0.88) | LDD0589 | [7] |
LDCM0273 | AC152 | HCT 116 | C346(0.56); C339(0.60); C281(0.71); C333(0.74) | LDD0590 | [7] |
LDCM0274 | AC153 | HCT 116 | C339(0.56); C346(0.63); C281(0.78); C333(0.82) | LDD0591 | [7] |
LDCM0621 | AC154 | HCT 116 | C281(0.79); C333(0.71); C339(0.59); C346(0.57) | LDD2158 | [7] |
LDCM0622 | AC155 | HCT 116 | C281(0.90); C333(0.73); C339(0.57); C346(0.60) | LDD2159 | [7] |
LDCM0623 | AC156 | HCT 116 | C281(0.86); C333(1.07); C339(0.83); C346(0.74) | LDD2160 | [7] |
LDCM0624 | AC157 | HCT 116 | C281(1.29); C333(1.04); C339(0.66); C346(0.65) | LDD2161 | [7] |
LDCM0276 | AC17 | HCT 116 | C339(0.99); C346(1.03); C333(1.24); C382(1.39) | LDD0593 | [7] |
LDCM0277 | AC18 | HCT 116 | C382(0.81); C339(0.82); C346(0.86); C281(0.97) | LDD0594 | [7] |
LDCM0278 | AC19 | HCT 116 | C382(0.79); C346(0.90); C339(0.91); C333(1.12) | LDD0595 | [7] |
LDCM0279 | AC2 | HCT 116 | C333(0.80); C281(0.88); C339(0.88); C346(0.96) | LDD0596 | [7] |
LDCM0280 | AC20 | HCT 116 | C382(0.83); C339(0.99); C346(0.99); C281(1.57) | LDD0597 | [7] |
LDCM0281 | AC21 | HCT 116 | C382(0.92); C339(0.96); C346(0.97); C281(1.17) | LDD0598 | [7] |
LDCM0282 | AC22 | HCT 116 | C339(1.05); C346(1.08); C333(1.09); C382(1.11) | LDD0599 | [7] |
LDCM0283 | AC23 | HCT 116 | C339(0.97); C333(0.98); C346(1.00); C382(1.00) | LDD0600 | [7] |
LDCM0284 | AC24 | HCT 116 | C382(0.83); C339(1.02); C346(1.04); C333(1.06) | LDD0601 | [7] |
LDCM0285 | AC25 | HCT 116 | C281(0.84); C339(0.88); C382(0.90); C346(0.96) | LDD0602 | [7] |
LDCM0286 | AC26 | HCT 116 | C333(0.70); C339(0.77); C281(0.83); C346(0.84) | LDD0603 | [7] |
LDCM0287 | AC27 | HCT 116 | C339(0.71); C346(0.74); C281(0.81); C382(0.99) | LDD0604 | [7] |
LDCM0288 | AC28 | HCT 116 | C333(0.65); C339(0.77); C281(0.79); C346(0.80) | LDD0605 | [7] |
LDCM0289 | AC29 | HCT 116 | C281(0.76); C346(0.78); C339(0.78); C333(1.04) | LDD0606 | [7] |
LDCM0290 | AC3 | HCT 116 | C333(0.87); C281(0.92); C346(0.95); C339(0.95) | LDD0607 | [7] |
LDCM0291 | AC30 | HCT 116 | C281(0.72); C333(0.73); C339(0.73); C346(0.73) | LDD0608 | [7] |
LDCM0292 | AC31 | HCT 116 | C333(0.68); C339(0.73); C281(0.73); C346(0.74) | LDD0609 | [7] |
LDCM0293 | AC32 | HCT 116 | C281(0.63); C339(0.69); C346(0.72); C382(0.96) | LDD0610 | [7] |
LDCM0294 | AC33 | HCT 116 | C339(0.67); C346(0.69); C281(0.69); C382(0.79) | LDD0611 | [7] |
LDCM0295 | AC34 | HCT 116 | C333(0.61); C281(0.66); C339(0.71); C346(0.76) | LDD0612 | [7] |
LDCM0296 | AC35 | HCT 116 | C382(1.00); C333(1.06); C281(1.14); C346(1.17) | LDD0613 | [7] |
LDCM0297 | AC36 | HCT 116 | C333(0.87); C382(0.98); C339(1.01); C346(1.03) | LDD0614 | [7] |
LDCM0298 | AC37 | HCT 116 | C333(0.79); C346(1.07); C281(1.08); C339(1.13) | LDD0615 | [7] |
LDCM0299 | AC38 | HCT 116 | C346(0.91); C382(0.92); C339(0.95); C333(0.99) | LDD0616 | [7] |
LDCM0300 | AC39 | HCT 116 | C382(0.96); C333(0.98); C339(1.02); C346(1.02) | LDD0617 | [7] |
LDCM0301 | AC4 | HCT 116 | C333(0.88); C281(0.91); C346(0.95); C339(1.02) | LDD0618 | [7] |
LDCM0302 | AC40 | HCT 116 | C382(0.90); C346(0.90); C333(0.92); C339(0.94) | LDD0619 | [7] |
LDCM0303 | AC41 | HCT 116 | C333(0.65); C281(1.01); C339(1.02); C382(1.06) | LDD0620 | [7] |
LDCM0304 | AC42 | HCT 116 | C333(0.81); C346(0.92); C339(0.93); C382(0.98) | LDD0621 | [7] |
LDCM0305 | AC43 | HCT 116 | C333(0.77); C339(0.85); C346(0.89); C281(0.94) | LDD0622 | [7] |
LDCM0306 | AC44 | HCT 116 | C333(0.71); C346(0.96); C339(1.02); C281(1.07) | LDD0623 | [7] |
LDCM0307 | AC45 | HCT 116 | C333(0.74); C346(0.96); C281(0.97); C339(1.03) | LDD0624 | [7] |
LDCM0308 | AC46 | HCT 116 | C382(0.89); C281(0.90); C346(0.98); C339(1.05) | LDD0625 | [7] |
LDCM0309 | AC47 | HCT 116 | C382(0.87); C281(0.89); C339(1.04); C346(1.08) | LDD0626 | [7] |
LDCM0310 | AC48 | HCT 116 | C281(0.89); C346(1.01); C382(1.01); C339(1.02) | LDD0627 | [7] |
LDCM0311 | AC49 | HCT 116 | C281(0.87); C346(0.88); C339(0.91); C382(0.93) | LDD0628 | [7] |
LDCM0312 | AC5 | HCT 116 | C281(0.97); C339(1.00); C346(1.07); C333(1.07) | LDD0629 | [7] |
LDCM0313 | AC50 | HCT 116 | C382(0.78); C346(0.88); C281(0.94); C339(0.94) | LDD0630 | [7] |
LDCM0314 | AC51 | HCT 116 | C281(1.06); C346(1.07); C382(1.08); C339(1.22) | LDD0631 | [7] |
LDCM0315 | AC52 | HCT 116 | C382(0.94); C346(0.97); C281(0.98); C339(0.99) | LDD0632 | [7] |
LDCM0316 | AC53 | HCT 116 | C346(0.87); C281(0.94); C382(0.95); C339(0.96) | LDD0633 | [7] |
LDCM0317 | AC54 | HCT 116 | C281(0.88); C346(0.93); C382(0.93); C339(0.95) | LDD0634 | [7] |
LDCM0318 | AC55 | HCT 116 | C382(0.82); C281(0.92); C346(0.97); C339(1.03) | LDD0635 | [7] |
LDCM0319 | AC56 | HCT 116 | C382(0.92); C346(1.04); C281(1.07); C339(1.14) | LDD0636 | [7] |
LDCM0320 | AC57 | HCT 116 | C382(0.70); C281(0.70); C339(0.81); C346(0.82) | LDD0637 | [7] |
LDCM0321 | AC58 | HCT 116 | C382(0.63); C339(0.73); C346(0.74); C281(0.81) | LDD0638 | [7] |
LDCM0322 | AC59 | HCT 116 | C281(0.68); C382(0.69); C346(0.75); C339(0.75) | LDD0639 | [7] |
LDCM0323 | AC6 | HCT 116 | C333(0.69); C281(0.75); C382(0.92); C346(1.18) | LDD0640 | [7] |
LDCM0324 | AC60 | HCT 116 | C382(0.68); C281(0.68); C333(0.69); C346(0.73) | LDD0641 | [7] |
LDCM0325 | AC61 | HCT 116 | C281(0.71); C346(0.74); C382(0.75); C339(0.79) | LDD0642 | [7] |
LDCM0326 | AC62 | HCT 116 | C382(0.68); C281(0.69); C346(0.73); C339(0.81) | LDD0643 | [7] |
LDCM0327 | AC63 | HCT 116 | C382(0.64); C281(0.73); C333(0.79); C346(0.79) | LDD0644 | [7] |
LDCM0328 | AC64 | HCT 116 | C382(0.73); C281(0.73); C333(0.76); C346(0.82) | LDD0645 | [7] |
LDCM0329 | AC65 | HCT 116 | C281(0.63); C346(0.75); C339(0.81); C382(0.84) | LDD0646 | [7] |
LDCM0330 | AC66 | HCT 116 | C281(0.67); C346(0.74); C339(0.76); C382(0.79) | LDD0647 | [7] |
LDCM0331 | AC67 | HCT 116 | C281(0.59); C346(0.67); C382(0.76); C333(0.76) | LDD0648 | [7] |
LDCM0332 | AC68 | HCT 116 | C281(0.90); C333(0.96); C382(1.01); C346(1.05) | LDD0649 | [7] |
LDCM0333 | AC69 | HCT 116 | C281(0.98); C382(1.00); C346(1.06); C339(1.15) | LDD0650 | [7] |
LDCM0334 | AC7 | HCT 116 | C281(0.84); C382(0.93); C333(1.01); C346(1.20) | LDD0651 | [7] |
LDCM0335 | AC70 | HCT 116 | C382(0.73); C339(0.73); C346(0.84); C333(0.84) | LDD0652 | [7] |
LDCM0336 | AC71 | HCT 116 | C339(1.00); C346(1.03); C281(1.08); C333(1.10) | LDD0653 | [7] |
LDCM0337 | AC72 | HCT 116 | C339(0.67); C346(0.81); C281(1.02); C382(1.14) | LDD0654 | [7] |
LDCM0338 | AC73 | HCT 116 | C333(0.76); C339(0.84); C346(0.96); C281(1.05) | LDD0655 | [7] |
LDCM0339 | AC74 | HCT 116 | C382(1.00); C339(1.07); C281(1.10); C346(1.14) | LDD0656 | [7] |
LDCM0340 | AC75 | HCT 116 | C333(0.91); C339(1.00); C346(1.04); C281(1.13) | LDD0657 | [7] |
LDCM0341 | AC76 | HCT 116 | C382(0.87); C333(0.94); C346(0.95); C339(0.97) | LDD0658 | [7] |
LDCM0342 | AC77 | HCT 116 | C382(0.90); C281(0.91); C346(0.94); C339(1.03) | LDD0659 | [7] |
LDCM0343 | AC78 | HCT 116 | C281(0.97); C333(1.01); C382(1.08); C346(1.09) | LDD0660 | [7] |
LDCM0344 | AC79 | HCT 116 | C339(0.92); C346(0.98); C281(1.02); C382(1.04) | LDD0661 | [7] |
LDCM0345 | AC8 | HCT 116 | C281(0.76); C333(0.89); C382(0.98); C346(1.17) | LDD0662 | [7] |
LDCM0346 | AC80 | HCT 116 | C333(0.90); C339(0.97); C346(0.98); C382(1.01) | LDD0663 | [7] |
LDCM0347 | AC81 | HCT 116 | C333(0.99); C339(1.01); C382(1.05); C281(1.09) | LDD0664 | [7] |
LDCM0348 | AC82 | HCT 116 | C339(1.07); C333(1.15); C281(1.16); C346(1.16) | LDD0665 | [7] |
LDCM0349 | AC83 | HCT 116 | C281(0.68); C382(0.77); C339(0.78); C333(0.79) | LDD0666 | [7] |
LDCM0350 | AC84 | HCT 116 | C333(0.68); C281(0.69); C382(0.81); C346(0.85) | LDD0667 | [7] |
LDCM0351 | AC85 | HCT 116 | C281(0.70); C333(0.71); C339(0.81); C346(0.82) | LDD0668 | [7] |
LDCM0352 | AC86 | HCT 116 | C281(0.71); C346(0.78); C382(0.79); C339(0.80) | LDD0669 | [7] |
LDCM0353 | AC87 | HCT 116 | C382(0.65); C333(0.85); C346(0.91); C281(0.92) | LDD0670 | [7] |
LDCM0354 | AC88 | HCT 116 | C281(0.80); C382(0.82); C333(0.83); C346(0.86) | LDD0671 | [7] |
LDCM0355 | AC89 | HCT 116 | C281(0.71); C346(0.74); C333(0.77); C339(0.81) | LDD0672 | [7] |
LDCM0357 | AC90 | HCT 116 | C382(0.73); C333(0.93); C281(0.94); C346(1.04) | LDD0674 | [7] |
LDCM0358 | AC91 | HCT 116 | C382(0.71); C281(0.71); C333(0.73); C346(0.74) | LDD0675 | [7] |
LDCM0359 | AC92 | HCT 116 | C333(0.65); C281(0.70); C346(0.71); C339(0.73) | LDD0676 | [7] |
LDCM0360 | AC93 | HCT 116 | C333(0.72); C346(0.77); C382(0.79); C281(0.84) | LDD0677 | [7] |
LDCM0361 | AC94 | HCT 116 | C382(0.59); C333(0.79); C281(0.89); C346(0.95) | LDD0678 | [7] |
LDCM0362 | AC95 | HCT 116 | C382(0.77); C333(0.79); C339(0.80); C346(0.82) | LDD0679 | [7] |
LDCM0363 | AC96 | HCT 116 | C281(0.75); C382(0.76); C333(0.82); C346(0.88) | LDD0680 | [7] |
LDCM0364 | AC97 | HCT 116 | C382(0.67); C346(0.67); C333(0.70); C339(0.70) | LDD0681 | [7] |
LDCM0365 | AC98 | HCT 116 | C281(0.51); C382(0.57); C339(0.61); C346(0.61) | LDD0682 | [7] |
LDCM0366 | AC99 | HCT 116 | C382(0.49); C281(0.64); C339(0.75); C333(0.81) | LDD0683 | [7] |
LDCM0520 | AKOS000195272 | MDA-MB-231 | C346(0.76) | LDD2113 | [4] |
LDCM0248 | AKOS034007472 | HCT 116 | C281(0.78); C333(0.87); C339(1.29); C346(1.22) | LDD0565 | [7] |
LDCM0356 | AKOS034007680 | HCT 116 | C333(0.74); C281(0.92); C382(1.07); C346(1.13) | LDD0673 | [7] |
LDCM0275 | AKOS034007705 | HCT 116 | C333(0.65); C281(0.71); C382(0.95); C346(1.10) | LDD0592 | [7] |
LDCM0108 | Chloroacetamide | HeLa | C382(0.00); H710(0.00); H584(0.00); H840(0.00) | LDD0222 | [18] |
LDCM0632 | CL-Sc | Hep-G2 | C382(3.64) | LDD2227 | [19] |
LDCM0367 | CL1 | HCT 116 | C382(0.66); C281(0.87); C333(0.96); C339(1.07) | LDD0684 | [7] |
LDCM0368 | CL10 | HCT 116 | C382(0.68); C346(0.72); C281(0.78); C339(0.79) | LDD0685 | [7] |
LDCM0369 | CL100 | HCT 116 | C333(0.73); C339(0.91); C346(0.94); C281(0.98) | LDD0686 | [7] |
LDCM0370 | CL101 | HCT 116 | C281(0.76); C333(0.76); C382(1.04); C346(1.19) | LDD0687 | [7] |
LDCM0371 | CL102 | HCT 116 | C333(0.84); C281(0.88); C382(1.09); C346(1.18) | LDD0688 | [7] |
LDCM0372 | CL103 | HCT 116 | C281(0.96); C382(1.12); C346(1.20); C333(1.31) | LDD0689 | [7] |
LDCM0373 | CL104 | HCT 116 | C333(0.74); C281(0.87); C382(1.02); C346(1.25) | LDD0690 | [7] |
LDCM0374 | CL105 | HCT 116 | C339(0.89); C346(0.92); C281(1.05); C382(1.12) | LDD0691 | [7] |
LDCM0375 | CL106 | HCT 116 | C382(0.60); C346(0.95); C339(0.97); C281(1.06) | LDD0692 | [7] |
LDCM0376 | CL107 | HCT 116 | C382(0.71); C339(0.93); C346(0.97); C281(1.03) | LDD0693 | [7] |
LDCM0377 | CL108 | HCT 116 | C339(0.86); C346(0.92); C281(0.99); C382(1.13) | LDD0694 | [7] |
LDCM0378 | CL109 | HCT 116 | C382(0.71); C339(0.84); C346(0.85); C281(1.15) | LDD0695 | [7] |
LDCM0379 | CL11 | HCT 116 | C346(0.79); C339(0.87); C281(0.92); C333(0.93) | LDD0696 | [7] |
LDCM0380 | CL110 | HCT 116 | C382(0.71); C339(0.87); C346(0.87); C281(0.93) | LDD0697 | [7] |
LDCM0381 | CL111 | HCT 116 | C382(0.82); C339(0.87); C346(0.88); C333(1.15) | LDD0698 | [7] |
LDCM0382 | CL112 | HCT 116 | C333(0.85); C281(0.85); C346(0.92); C339(0.97) | LDD0699 | [7] |
LDCM0383 | CL113 | HCT 116 | C281(0.64); C339(0.78); C346(0.80); C333(0.82) | LDD0700 | [7] |
LDCM0384 | CL114 | HCT 116 | C333(0.66); C281(0.67); C346(0.78); C339(0.80) | LDD0701 | [7] |
LDCM0385 | CL115 | HCT 116 | C333(0.67); C339(0.71); C346(0.75); C281(0.78) | LDD0702 | [7] |
LDCM0386 | CL116 | HCT 116 | C339(0.72); C281(0.74); C346(0.78); C333(0.90) | LDD0703 | [7] |
LDCM0387 | CL117 | HCT 116 | C346(0.94); C339(1.00); C382(1.05); C281(1.05) | LDD0704 | [7] |
LDCM0388 | CL118 | HCT 116 | C346(1.01); C281(1.01); C382(1.01); C339(1.02) | LDD0705 | [7] |
LDCM0389 | CL119 | HCT 116 | C333(0.88); C346(0.91); C339(0.92); C281(0.95) | LDD0706 | [7] |
LDCM0390 | CL12 | HCT 116 | C346(0.74); C339(0.75); C281(0.96); C333(0.99) | LDD0707 | [7] |
LDCM0391 | CL120 | HCT 116 | C333(0.82); C281(1.02); C346(1.03); C339(1.04) | LDD0708 | [7] |
LDCM0392 | CL121 | HCT 116 | C281(0.67); C382(0.89); C346(1.15); C339(1.48) | LDD0709 | [7] |
LDCM0393 | CL122 | HCT 116 | C281(0.86); C382(0.86); C339(0.91); C346(0.93) | LDD0710 | [7] |
LDCM0394 | CL123 | HCT 116 | C281(0.81); C346(0.84); C382(0.85); C339(0.88) | LDD0711 | [7] |
LDCM0395 | CL124 | HCT 116 | C339(0.84); C346(0.87); C382(0.87); C281(0.87) | LDD0712 | [7] |
LDCM0396 | CL125 | HCT 116 | C333(0.86); C346(0.89); C382(0.91); C339(0.93) | LDD0713 | [7] |
LDCM0397 | CL126 | HCT 116 | C346(0.75); C339(0.80); C382(0.92); C333(1.02) | LDD0714 | [7] |
LDCM0398 | CL127 | HCT 116 | C382(0.68); C281(0.74); C346(0.75); C333(0.77) | LDD0715 | [7] |
LDCM0399 | CL128 | HCT 116 | C382(0.63); C339(0.76); C281(0.76); C346(0.77) | LDD0716 | [7] |
LDCM0400 | CL13 | HCT 116 | C382(0.71); C339(0.71); C346(0.77); C333(0.88) | LDD0717 | [7] |
LDCM0401 | CL14 | HCT 116 | C382(0.77); C339(0.78); C346(0.81); C333(0.94) | LDD0718 | [7] |
LDCM0402 | CL15 | HCT 116 | C382(0.69); C346(0.77); C339(0.79); C333(0.92) | LDD0719 | [7] |
LDCM0403 | CL16 | HCT 116 | C346(0.78); C281(0.81); C339(0.82); C333(1.18) | LDD0720 | [7] |
LDCM0404 | CL17 | HCT 116 | C339(0.73); C346(0.78); C281(0.93); C333(1.06) | LDD0721 | [7] |
LDCM0405 | CL18 | HCT 116 | C339(0.67); C281(0.72); C346(0.73); C333(1.02) | LDD0722 | [7] |
LDCM0406 | CL19 | HCT 116 | C339(0.79); C281(0.80); C346(0.82); C333(1.16) | LDD0723 | [7] |
LDCM0407 | CL2 | HCT 116 | C382(0.59); C281(0.97); C346(1.00); C339(1.05) | LDD0724 | [7] |
LDCM0408 | CL20 | HCT 116 | C339(0.67); C346(0.71); C281(0.78); C333(1.01) | LDD0725 | [7] |
LDCM0409 | CL21 | HCT 116 | C339(0.69); C346(0.73); C281(0.77); C333(1.01) | LDD0726 | [7] |
LDCM0410 | CL22 | HCT 116 | C281(0.88); C346(0.91); C339(0.91); C333(1.41) | LDD0727 | [7] |
LDCM0411 | CL23 | HCT 116 | C339(0.74); C346(0.75); C281(0.78); C333(1.12) | LDD0728 | [7] |
LDCM0412 | CL24 | HCT 116 | C281(0.70); C346(0.71); C339(0.73); C333(1.04) | LDD0729 | [7] |
LDCM0413 | CL25 | HCT 116 | C281(0.76); C333(1.15); C339(0.84); C346(0.76) | LDD0730 | [7] |
LDCM0414 | CL26 | HCT 116 | C281(0.75); C333(1.05); C339(0.73); C346(0.74) | LDD0731 | [7] |
LDCM0415 | CL27 | HCT 116 | C281(0.91); C333(1.23); C339(0.73); C346(0.75) | LDD0732 | [7] |
LDCM0416 | CL28 | HCT 116 | C281(0.72); C333(0.99); C339(0.72); C346(0.72) | LDD0733 | [7] |
LDCM0417 | CL29 | HCT 116 | C281(0.81); C333(0.98); C339(0.62); C346(0.70) | LDD0734 | [7] |
LDCM0418 | CL3 | HCT 116 | C281(1.10); C333(1.08); C339(1.17); C346(1.02) | LDD0735 | [7] |
LDCM0419 | CL30 | HCT 116 | C281(0.87); C333(1.29); C339(0.85); C346(0.79) | LDD0736 | [7] |
LDCM0420 | CL31 | HCT 116 | C281(0.92); C333(1.12); C339(0.89); C346(0.88) | LDD0737 | [7] |
LDCM0421 | CL32 | HCT 116 | C281(0.64); C333(0.81); C339(0.80); C346(0.80) | LDD0738 | [7] |
LDCM0422 | CL33 | HCT 116 | C281(0.67); C333(0.77); C339(0.79); C346(0.82) | LDD0739 | [7] |
LDCM0423 | CL34 | HCT 116 | C281(0.65); C333(0.88); C339(0.79); C346(0.73) | LDD0740 | [7] |
LDCM0424 | CL35 | HCT 116 | C281(0.66); C333(0.92); C339(0.71); C346(0.68) | LDD0741 | [7] |
LDCM0425 | CL36 | HCT 116 | C281(0.76); C333(0.92); C339(0.80); C346(0.76) | LDD0742 | [7] |
LDCM0426 | CL37 | HCT 116 | C281(0.76); C333(1.07); C339(0.71); C346(0.67) | LDD0743 | [7] |
LDCM0428 | CL39 | HCT 116 | C281(0.82); C333(0.85); C339(0.74); C346(0.72) | LDD0745 | [7] |
LDCM0429 | CL4 | HCT 116 | C281(0.86); C333(1.09); C339(0.91); C346(0.89) | LDD0746 | [7] |
LDCM0430 | CL40 | HCT 116 | C281(0.74); C333(0.82); C339(0.66); C346(0.64) | LDD0747 | [7] |
LDCM0431 | CL41 | HCT 116 | C281(0.86); C333(1.00); C339(0.67); C346(0.63) | LDD0748 | [7] |
LDCM0432 | CL42 | HCT 116 | C281(0.95); C333(0.89); C339(0.77); C346(0.77) | LDD0749 | [7] |
LDCM0433 | CL43 | HCT 116 | C281(0.85); C333(0.89); C339(0.71); C346(0.63) | LDD0750 | [7] |
LDCM0434 | CL44 | HCT 116 | C281(0.75); C333(1.09); C339(0.68); C346(0.63) | LDD0751 | [7] |
LDCM0435 | CL45 | HCT 116 | C281(0.69); C333(1.02); C339(0.72); C346(0.67) | LDD0752 | [7] |
LDCM0436 | CL46 | HCT 116 | C281(1.42); C333(0.66); C339(1.10); C346(1.05) | LDD0753 | [7] |
LDCM0437 | CL47 | HCT 116 | C281(1.21); C333(0.79); C339(1.13); C346(1.09) | LDD0754 | [7] |
LDCM0438 | CL48 | HCT 116 | C281(1.21); C333(0.76); C339(1.05); C346(0.97) | LDD0755 | [7] |
LDCM0439 | CL49 | HCT 116 | C281(1.25); C333(1.35); C339(1.00); C346(0.97) | LDD0756 | [7] |
LDCM0440 | CL5 | HCT 116 | C281(1.09); C333(1.23); C339(0.99); C346(0.94) | LDD0757 | [7] |
LDCM0441 | CL50 | HCT 116 | C281(1.40); C333(0.63); C339(1.02); C346(1.00) | LDD0758 | [7] |
LDCM0442 | CL51 | HCT 116 | C281(1.34); C333(0.85); C339(1.08); C346(1.06) | LDD0759 | [7] |
LDCM0443 | CL52 | HCT 116 | C281(1.25); C333(0.82); C339(0.91); C346(1.01) | LDD0760 | [7] |
LDCM0444 | CL53 | HCT 116 | C281(1.38); C333(0.72); C339(1.00); C346(0.97) | LDD0761 | [7] |
LDCM0445 | CL54 | HCT 116 | C281(1.32); C333(1.22); C339(1.06); C346(0.93) | LDD0762 | [7] |
LDCM0446 | CL55 | HCT 116 | C281(1.37); C333(0.82); C339(1.17); C346(1.08) | LDD0763 | [7] |
LDCM0447 | CL56 | HCT 116 | C281(1.11); C333(0.78); C339(0.99); C346(0.99) | LDD0764 | [7] |
LDCM0448 | CL57 | HCT 116 | C281(1.26); C333(0.92); C339(1.08); C346(1.06) | LDD0765 | [7] |
LDCM0449 | CL58 | HCT 116 | C281(1.48); C333(0.72); C339(0.93); C346(1.00) | LDD0766 | [7] |
LDCM0450 | CL59 | HCT 116 | C281(1.16); C333(1.03); C339(0.95); C346(1.00) | LDD0767 | [7] |
LDCM0451 | CL6 | HCT 116 | C281(0.83); C333(0.82); C339(0.82); C346(0.71) | LDD0768 | [7] |
LDCM0452 | CL60 | HCT 116 | C281(1.12); C333(0.81); C339(0.96); C346(1.00) | LDD0769 | [7] |
LDCM0453 | CL61 | HCT 116 | C281(0.88); C333(0.93); C339(0.96); C346(1.01) | LDD0770 | [7] |
LDCM0454 | CL62 | HCT 116 | C281(0.78); C333(0.88); C339(0.89); C346(0.94) | LDD0771 | [7] |
LDCM0455 | CL63 | HCT 116 | C281(0.87); C333(0.85); C339(0.84); C346(0.88) | LDD0772 | [7] |
LDCM0456 | CL64 | HCT 116 | C281(1.07); C333(0.81); C339(0.87); C346(0.86) | LDD0773 | [7] |
LDCM0457 | CL65 | HCT 116 | C281(0.94); C333(0.89); C339(0.92); C346(0.98) | LDD0774 | [7] |
LDCM0458 | CL66 | HCT 116 | C281(0.92); C333(0.74); C339(0.87); C346(0.90) | LDD0775 | [7] |
LDCM0459 | CL67 | HCT 116 | C281(1.49); C333(0.86); C339(0.90); C346(0.93) | LDD0776 | [7] |
LDCM0460 | CL68 | HCT 116 | C281(2.03); C333(0.69); C339(1.01); C346(1.03) | LDD0777 | [7] |
LDCM0461 | CL69 | HCT 116 | C281(0.81); C333(0.75); C339(0.77); C346(0.80) | LDD0778 | [7] |
LDCM0462 | CL7 | HCT 116 | C281(1.00); C333(1.01); C339(0.81); C346(0.80) | LDD0779 | [7] |
LDCM0463 | CL70 | HCT 116 | C281(0.86); C333(0.80); C339(0.83); C346(0.88) | LDD0780 | [7] |
LDCM0464 | CL71 | HCT 116 | C281(0.77); C333(0.81); C339(0.92); C346(0.91) | LDD0781 | [7] |
LDCM0465 | CL72 | HCT 116 | C281(0.99); C333(0.85); C339(0.95); C346(1.01) | LDD0782 | [7] |
LDCM0466 | CL73 | HCT 116 | C281(1.39); C333(0.76); C339(0.89); C346(0.96) | LDD0783 | [7] |
LDCM0467 | CL74 | HCT 116 | C281(1.13); C333(0.86); C339(0.82); C346(0.82) | LDD0784 | [7] |
LDCM0469 | CL76 | HCT 116 | C281(1.38); C339(1.02); C346(1.01) | LDD0786 | [7] |
LDCM0470 | CL77 | HCT 116 | C281(1.35); C339(1.04); C346(1.02) | LDD0787 | [7] |
LDCM0471 | CL78 | HCT 116 | C281(0.98); C339(0.95); C346(1.04) | LDD0788 | [7] |
LDCM0472 | CL79 | HCT 116 | C281(1.52); C339(0.99); C346(1.01) | LDD0789 | [7] |
LDCM0473 | CL8 | HCT 116 | C281(0.90); C333(0.81); C339(0.77); C346(0.70) | LDD0790 | [7] |
LDCM0474 | CL80 | HCT 116 | C281(0.99); C339(0.98); C346(0.98) | LDD0791 | [7] |
LDCM0475 | CL81 | HCT 116 | C281(1.94); C339(1.01); C346(1.07) | LDD0792 | [7] |
LDCM0476 | CL82 | HCT 116 | C281(1.91); C339(0.96); C346(1.06) | LDD0793 | [7] |
LDCM0477 | CL83 | HCT 116 | C281(1.39); C339(1.14); C346(1.02) | LDD0794 | [7] |
LDCM0478 | CL84 | HCT 116 | C281(1.27); C339(1.12); C346(1.09) | LDD0795 | [7] |
LDCM0479 | CL85 | HCT 116 | C281(1.46); C339(1.04); C346(0.95) | LDD0796 | [7] |
LDCM0480 | CL86 | HCT 116 | C281(1.30); C339(1.11); C346(1.12) | LDD0797 | [7] |
LDCM0481 | CL87 | HCT 116 | C281(2.10); C339(0.96); C346(1.02) | LDD0798 | [7] |
LDCM0482 | CL88 | HCT 116 | C281(2.23); C339(0.99); C346(0.99) | LDD0799 | [7] |
LDCM0483 | CL89 | HCT 116 | C281(1.16); C339(1.18); C346(1.16) | LDD0800 | [7] |
LDCM0484 | CL9 | HCT 116 | C281(0.84); C333(0.95); C339(0.84); C346(0.83) | LDD0801 | [7] |
LDCM0485 | CL90 | HCT 116 | C281(1.49); C339(1.15); C346(1.15) | LDD0802 | [7] |
LDCM0486 | CL91 | HCT 116 | C281(0.98); C333(0.88); C339(0.95); C346(1.09) | LDD0803 | [7] |
LDCM0487 | CL92 | HCT 116 | C281(0.98); C333(0.85); C339(1.03); C346(1.25) | LDD0804 | [7] |
LDCM0488 | CL93 | HCT 116 | C281(1.05); C333(0.95); C339(1.11); C346(1.05) | LDD0805 | [7] |
LDCM0489 | CL94 | HCT 116 | C281(1.06); C333(0.83); C339(0.97); C346(0.96) | LDD0806 | [7] |
LDCM0490 | CL95 | HCT 116 | C281(0.85); C333(0.75); C339(0.92); C346(0.99) | LDD0807 | [7] |
LDCM0491 | CL96 | HCT 116 | C281(0.80); C333(1.10); C339(0.96); C346(0.96) | LDD0808 | [7] |
LDCM0492 | CL97 | HCT 116 | C281(0.78); C333(0.83); C339(0.83); C346(0.84) | LDD0809 | [7] |
LDCM0493 | CL98 | HCT 116 | C281(0.76); C333(0.88); C339(0.89); C346(0.89) | LDD0810 | [7] |
LDCM0494 | CL99 | HCT 116 | C281(0.87); C333(0.95); C339(0.89); C346(0.91) | LDD0811 | [7] |
LDCM0495 | E2913 | HEK-293T | C281(1.13); C382(1.03); C333(0.82); C346(1.12) | LDD1698 | [22] |
LDCM0468 | Fragment33 | HCT 116 | C281(1.04); C333(0.82); C339(0.97); C346(0.98) | LDD0785 | [7] |
LDCM0427 | Fragment51 | HCT 116 | C281(0.86); C333(0.98); C339(0.78); C346(0.76) | LDD0744 | [7] |
LDCM0116 | HHS-0101 | DM93 | Y779(0.72); Y707(0.77); Y361(1.74) | LDD0264 | [5] |
LDCM0117 | HHS-0201 | DM93 | Y707(0.68); Y779(0.78); Y361(3.71); Y685(9.39) | LDD0265 | [5] |
LDCM0118 | HHS-0301 | DM93 | Y707(0.46); Y779(1.90); Y361(3.74) | LDD0266 | [5] |
LDCM0119 | HHS-0401 | DM93 | Y707(0.41); Y779(0.75) | LDD0267 | [5] |
LDCM0120 | HHS-0701 | DM93 | Y779(0.79); Y707(1.07); Y685(3.01); Y361(4.27) | LDD0268 | [5] |
LDCM0107 | IAA | HeLa | H710(0.00); C339(0.00); C333(0.00) | LDD0221 | [18] |
LDCM0022 | KB02 | HEK-293T | C346(0.84); C281(1.05); C382(0.99); C333(1.05) | LDD1492 | [22] |
LDCM0023 | KB03 | HEK-293T | C346(0.85); C281(1.00); C382(1.01); C333(1.07) | LDD1497 | [22] |
LDCM0024 | KB05 | HMCB | C382(2.16); C333(1.30); C281(2.26) | LDD3312 | [23] |
LDCM0109 | NEM | HeLa | H710(0.00); H582(0.00); H479(0.00); H205(0.00) | LDD0223 | [18] |
LDCM0506 | Nucleophilic fragment 16a | MDA-MB-231 | C346(1.68); C382(1.63) | LDD2099 | [4] |
LDCM0507 | Nucleophilic fragment 16b | MDA-MB-231 | C382(0.63) | LDD2100 | [4] |
LDCM0508 | Nucleophilic fragment 17a | MDA-MB-231 | C382(0.81) | LDD2101 | [4] |
LDCM0516 | Nucleophilic fragment 21a | MDA-MB-231 | C382(0.91) | LDD2109 | [4] |
LDCM0518 | Nucleophilic fragment 22a | MDA-MB-231 | C346(0.97) | LDD2111 | [4] |
LDCM0526 | Nucleophilic fragment 26a | MDA-MB-231 | C346(1.83) | LDD2119 | [4] |
LDCM0530 | Nucleophilic fragment 28a | MDA-MB-231 | C382(0.96) | LDD2123 | [4] |
LDCM0534 | Nucleophilic fragment 30a | MDA-MB-231 | C346(1.13); C382(1.23) | LDD2127 | [4] |
LDCM0541 | Nucleophilic fragment 36 | MDA-MB-231 | C346(0.60); C382(0.60) | LDD2134 | [4] |
LDCM0542 | Nucleophilic fragment 37 | MDA-MB-231 | C346(1.83); C339(1.06) | LDD2135 | [4] |
LDCM0543 | Nucleophilic fragment 38 | MDA-MB-231 | C346(1.90); C382(1.50) | LDD2136 | [4] |
LDCM0544 | Nucleophilic fragment 39 | MDA-MB-231 | C382(1.00) | LDD2137 | [4] |
LDCM0546 | Nucleophilic fragment 40 | MDA-MB-231 | C346(1.32) | LDD2140 | [4] |
LDCM0550 | Nucleophilic fragment 5a | MDA-MB-231 | C346(3.27) | LDD2144 | [4] |
LDCM0551 | Nucleophilic fragment 5b | MDA-MB-231 | C382(0.22) | LDD2145 | [4] |
LDCM0554 | Nucleophilic fragment 7a | MDA-MB-231 | C382(0.64) | LDD2148 | [4] |
LDCM0556 | Nucleophilic fragment 8a | MDA-MB-231 | C333(0.72) | LDD2150 | [4] |
References