Details of the Target

General Information of Target

Target ID LDTP10374
Target Name Unconventional myosin-XIX (MYO19)
Gene Name MYO19
Gene ID 80179
Synonyms
MYOHD1; Unconventional myosin-XIX; Myosin head domain-containing protein 1
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MDETVAEFIKRTILKIPMNELTTILKAWDFLSENQLQTVNFRQRKESVVQHLIHLCEEKR
ASISDAALLDIIYMQFHQHQKVWEVFQMSKGPGEDVDLFDMKQFKNSFKKILQRALKNVT
VSFRETEENAVWIRIAWGTQYTKPNQYKPTYVVYYSQTPYAFTSSSMLRRNTPLLGQALT
IASKHHQIVKMDLRSRYLDSLKAIVFKQYNQTFETHNSTTPLQERSLGLDINMDSRIIHE
NIVEKERVQRITQETFGDYPQPQLEFAQYKLETKFKSGLNGSILAEREEPLRCLIKFSSP
HLLEALKSLAPAGIADAPLSPLLTCIPNKRMNYFKIRDK
Target Bioclass
Enzyme
Family
TRAFAC class myosin-kinesin ATPase superfamily, Myosin family
Subcellular location
Mitochondrion outer membrane
Function
Actin-based motor molecule with ATPase activity that localizes to the mitochondrion outer membrane. Motor protein that moves towards the plus-end of actin filaments. Required for mitochondrial inheritance during mitosis. May be involved in mitochondrial transport or positioning.
Uniprot ID
Q96H55
Ensemble ID
ENST00000610930.4
HGNC ID
HGNC:26234

Target Site Mutations in Different Cell Lines

Cell line Mutation details Probe for labeling this protein in this cell
CAKI1 SNV: p.P572S DBIA    Probe Info 
CAL72 SNV: p.Y687F DBIA    Probe Info 
CASKI SNV: p.E634D DBIA    Probe Info 
CCK81 SNV: p.W263C DBIA    Probe Info 
HCC1806 SNV: p.K103M DBIA    Probe Info 
HUCCT1 SNV: p.A786G DBIA    Probe Info 
Ishikawa (Heraklio) 02 ER SNV: p.L204P DBIA    Probe Info 
KMCH1 SNV: p.D316Y DBIA    Probe Info 
KURAMOCHI SNV: p.W772L DBIA    Probe Info 
OCILY3 SNV: p.D326G .
SKNAS Insertion: p.Y93SfsTer11 DBIA    Probe Info 
SW480 SNV: p.T41S .
SW837 Substitution: p.C321P DBIA    Probe Info 

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 13 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
BTD
 Probe Info  		C227(0.99)  LDD2109  [1]
AHL-Pu-1
 Probe Info  		C755(2.03)  LDD0168  [2]
DBIA
 Probe Info  		C275(1.19); C242(1.04); C186(0.98)  LDD0078  [3]
IA-alkyne
 Probe Info  		C937(0.00); C764(0.00); C755(0.00); C515(0.00)  LDD0162  [4]
NAIA_4
 Probe Info  		C186(0.00); C515(0.00); C678(0.00); C937(0.00)  LDD2226  [5]
NAIA_5
 Probe Info  		C515(0.00); C186(0.00); C755(0.00)  LDD2224  [5]
TFBX
 Probe Info  		C678(0.00); C764(0.00)  LDD0027  [6]
WYneN
 Probe Info  		C227(0.00); C678(0.00)  LDD0021  [7]
IPM
 Probe Info  		C515(0.00); C845(0.00)  LDD0005  [7]
Acrolein
 Probe Info  		N.A.  LDD0217  [8]
Crotonaldehyde
 Probe Info  		N.A.  LDD0219  [8]
Methacrolein
 Probe Info  		C275(0.00); C515(0.00)  LDD0218  [8]
AOyne
 Probe Info  		14.30  LDD0443  [9]
PAL-AfBPP Probe
Click To Hide/Show 3 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
FFF probe11
 Probe Info  		20.00  LDD0472  [10]
FFF probe3
 Probe Info  		20.00  LDD0465  [10]
STS-2
 Probe Info  		N.A.  LDD0139  [11]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0524  2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide MDA-MB-231 C227(0.90)  LDD2117  [1]
 LDCM0025  4SU-RNA HEK-293T C755(2.03)  LDD0168  [2]
 LDCM0026  4SU-RNA+native RNA DM93 C845(2.78); C755(3.37)  LDD0171  [2]
 LDCM0214  AC1 HCT 116 C186(0.81); C227(0.66); C275(1.42); C755(1.11)  LDD0531  [3]
 LDCM0215  AC10 HCT 116 C186(0.95); C242(0.79); C275(1.28); C767(1.07)  LDD0532  [3]
 LDCM0216  AC100 HCT 116 C186(1.45); C275(1.15); C678(0.78); C764(0.85)  LDD0533  [3]
 LDCM0217  AC101 HCT 116 C186(1.29); C275(1.26); C678(0.80); C764(0.95)  LDD0534  [3]
 LDCM0218  AC102 HCT 116 C186(1.00); C275(1.45); C678(0.81); C764(0.91)  LDD0535  [3]
 LDCM0219  AC103 HCT 116 C186(1.08); C275(1.89); C678(0.90); C764(1.08)  LDD0536  [3]
 LDCM0220  AC104 HCT 116 C186(1.35); C275(1.62); C678(0.95); C764(0.91)  LDD0537  [3]
 LDCM0221  AC105 HCT 116 C186(1.55); C275(1.62); C678(0.89); C764(0.90)  LDD0538  [3]
 LDCM0222  AC106 HCT 116 C186(1.16); C275(1.52); C678(0.82); C764(0.96)  LDD0539  [3]
 LDCM0223  AC107 HCT 116 C186(1.08); C275(1.91); C678(0.77); C764(1.06)  LDD0540  [3]
 LDCM0224  AC108 HCT 116 C186(1.16); C275(1.07); C678(0.89); C764(0.82)  LDD0541  [3]
 LDCM0225  AC109 HCT 116 C186(1.29); C275(1.05); C678(0.80); C764(0.71)  LDD0542  [3]
 LDCM0226  AC11 HCT 116 C186(1.06); C242(0.75); C275(1.23); C767(1.06)  LDD0543  [3]
 LDCM0227  AC110 HCT 116 C186(1.29); C275(1.12); C678(0.81); C764(0.91)  LDD0544  [3]
 LDCM0228  AC111 HCT 116 C186(1.04); C275(1.26); C678(0.72); C764(0.83)  LDD0545  [3]
 LDCM0229  AC112 HCT 116 C186(1.13); C275(1.43); C678(0.83); C764(1.15)  LDD0546  [3]
 LDCM0230  AC113 HCT 116 C186(0.98); C227(0.68); C242(0.79); C275(1.09)  LDD0547  [3]
 LDCM0231  AC114 HCT 116 C186(0.97); C227(0.99); C242(0.75); C275(1.45)  LDD0548  [3]
 LDCM0232  AC115 HCT 116 C186(0.98); C227(0.89); C242(0.69); C275(1.31)  LDD0549  [3]
 LDCM0233  AC116 HCT 116 C186(0.89); C227(1.14); C242(0.74); C275(1.41)  LDD0550  [3]
 LDCM0234  AC117 HCT 116 C186(0.99); C227(0.72); C242(0.83); C275(1.06)  LDD0551  [3]
 LDCM0235  AC118 HCT 116 C186(1.00); C227(0.78); C242(0.77); C275(1.16)  LDD0552  [3]
 LDCM0236  AC119 HCT 116 C186(0.89); C227(0.92); C242(0.68); C275(1.31)  LDD0553  [3]
 LDCM0237  AC12 HCT 116 C186(0.98); C242(0.84); C275(1.24); C767(1.29)  LDD0554  [3]
 LDCM0238  AC120 HCT 116 C186(0.84); C227(0.94); C242(0.62); C275(1.25)  LDD0555  [3]
 LDCM0239  AC121 HCT 116 C186(0.92); C227(0.58); C242(0.68); C275(1.10)  LDD0556  [3]
 LDCM0240  AC122 HCT 116 C186(0.99); C227(1.09); C242(0.79); C275(1.23)  LDD0557  [3]
 LDCM0241  AC123 HCT 116 C186(0.83); C227(0.61); C242(0.82); C275(1.08)  LDD0558  [3]
 LDCM0242  AC124 HCT 116 C186(1.14); C227(0.94); C242(0.74); C275(1.01)  LDD0559  [3]
 LDCM0243  AC125 HCT 116 C186(0.94); C227(1.33); C242(1.07); C275(1.38)  LDD0560  [3]
 LDCM0244  AC126 HCT 116 C186(0.90); C227(0.88); C242(0.82); C275(1.55)  LDD0561  [3]
 LDCM0245  AC127 HCT 116 C186(0.89); C227(0.85); C242(0.80); C275(1.32)  LDD0562  [3]
 LDCM0246  AC128 HCT 116 C242(0.73); C275(0.96); C755(1.76)  LDD0563  [3]
 LDCM0247  AC129 HCT 116 C242(0.94); C275(1.04); C755(1.03)  LDD0564  [3]
 LDCM0249  AC130 HCT 116 C242(0.84); C275(1.24); C755(1.53)  LDD0566  [3]
 LDCM0250  AC131 HCT 116 C242(1.21); C275(1.25); C755(1.21)  LDD0567  [3]
 LDCM0251  AC132 HCT 116 C242(1.05); C275(1.73); C755(1.33)  LDD0568  [3]
 LDCM0252  AC133 HCT 116 C242(0.94); C275(1.61); C755(1.46)  LDD0569  [3]
 LDCM0253  AC134 HCT 116 C242(0.78); C275(1.33); C755(1.48)  LDD0570  [3]
 LDCM0254  AC135 HCT 116 C242(0.95); C275(1.25); C755(1.74)  LDD0571  [3]
 LDCM0255  AC136 HCT 116 C242(0.80); C275(1.53); C755(1.29)  LDD0572  [3]
 LDCM0256  AC137 HCT 116 C242(0.88); C275(1.45); C755(1.54)  LDD0573  [3]
 LDCM0257  AC138 HCT 116 C242(0.91); C275(1.38); C755(1.53)  LDD0574  [3]
 LDCM0258  AC139 HCT 116 C242(0.93); C275(2.19); C755(1.33)  LDD0575  [3]
 LDCM0259  AC14 HCT 116 C186(0.92); C242(0.95); C275(0.87); C767(0.98)  LDD0576  [3]
 LDCM0260  AC140 HCT 116 C242(0.83); C275(2.65); C755(1.79)  LDD0577  [3]
 LDCM0261  AC141 HCT 116 C242(0.87); C275(1.91); C755(1.41)  LDD0578  [3]
 LDCM0262  AC142 HCT 116 C242(1.00); C275(1.14); C755(1.06)  LDD0579  [3]
 LDCM0263  AC143 HCT 116 C227(0.67); C242(0.84); C764(0.90); C767(1.13)  LDD0580  [3]
 LDCM0264  AC144 HCT 116 C227(0.74); C764(0.92); C242(0.92); C767(1.13)  LDD0581  [3]
 LDCM0265  AC145 HCT 116 C242(0.81); C764(0.89); C767(1.04); C678(1.11)  LDD0582  [3]
 LDCM0266  AC146 HCT 116 C242(0.71); C764(0.77); C767(0.98); C678(1.04)  LDD0583  [3]
 LDCM0267  AC147 HCT 116 C242(0.93); C767(1.20); C764(1.24); C678(1.26)  LDD0584  [3]
 LDCM0268  AC148 HCT 116 C764(0.61); C242(0.83); C227(0.84); C767(1.00)  LDD0585  [3]
 LDCM0269  AC149 HCT 116 C764(0.65); C242(0.84); C767(0.98); C678(1.04)  LDD0586  [3]
 LDCM0270  AC15 HCT 116 C275(0.90); C186(0.90); C767(1.02); C242(1.21)  LDD0587  [3]
 LDCM0271  AC150 HCT 116 C242(0.85); C764(0.87); C767(0.91); C678(1.04)  LDD0588  [3]
 LDCM0272  AC151 HCT 116 C764(0.74); C242(0.91); C275(1.20); C678(1.22)  LDD0589  [3]
 LDCM0273  AC152 HCT 116 C764(0.65); C767(0.89); C242(0.92); C227(1.06)  LDD0590  [3]
 LDCM0274  AC153 HCT 116 C764(0.44); C242(0.97); C227(1.00); C767(1.02)  LDD0591  [3]
 LDCM0621  AC154 HCT 116 C227(1.10); C242(0.85); C275(1.69); C678(1.07)  LDD2158  [3]
 LDCM0622  AC155 HCT 116 C227(1.05); C242(0.77); C275(1.79); C678(1.13)  LDD2159  [3]
 LDCM0623  AC156 HCT 116 C227(2.17); C242(0.81); C275(1.23); C678(1.02)  LDD2160  [3]
 LDCM0624  AC157 HCT 116 C227(0.95); C242(0.87); C275(1.26); C678(0.94)  LDD2161  [3]
 LDCM0276  AC17 HCT 116 C764(0.96); C767(1.08); C826(1.09); C275(1.21)  LDD0593  [3]
 LDCM0277  AC18 HCT 116 C275(0.87); C767(0.87); C764(0.89); C242(1.07)  LDD0594  [3]
 LDCM0278  AC19 HCT 116 C767(0.92); C764(1.14); C826(1.19); C275(1.20)  LDD0595  [3]
 LDCM0279  AC2 HCT 116 C227(0.67); C186(0.94); C767(1.11); C764(1.17)  LDD0596  [3]
 LDCM0280  AC20 HCT 116 C275(0.80); C764(0.97); C767(0.99); C826(1.15)  LDD0597  [3]
 LDCM0281  AC21 HCT 116 C767(0.73); C275(0.82); C764(0.91); C826(1.07)  LDD0598  [3]
 LDCM0282  AC22 HCT 116 C764(0.97); C767(0.99); C275(1.13); C826(1.14)  LDD0599  [3]
 LDCM0283  AC23 HCT 116 C767(0.84); C275(0.89); C764(0.92); C242(1.13)  LDD0600  [3]
 LDCM0284  AC24 HCT 116 C764(0.86); C767(0.87); C826(0.87); C275(0.90)  LDD0601  [3]
 LDCM0285  AC25 HCT 116 C242(0.82); C826(0.95); C275(0.96); C227(1.03)  LDD0602  [3]
 LDCM0286  AC26 HCT 116 C242(0.76); C227(0.91); C275(1.05); C826(1.08)  LDD0603  [3]
 LDCM0287  AC27 HCT 116 C242(0.81); C227(0.84); C275(1.06); C767(1.31)  LDD0604  [3]
 LDCM0288  AC28 HCT 116 C242(0.75); C227(1.05); C275(1.05); C767(1.15)  LDD0605  [3]
 LDCM0289  AC29 HCT 116 C242(1.15); C227(1.24); C275(1.29); C767(1.42)  LDD0606  [3]
 LDCM0290  AC3 HCT 116 C186(0.90); C767(0.92); C764(0.96); C227(1.10)  LDD0607  [3]
 LDCM0291  AC30 HCT 116 C242(0.88); C767(1.15); C275(1.35); C826(1.39)  LDD0608  [3]
 LDCM0292  AC31 HCT 116 C242(0.83); C275(1.07); C826(1.22); C767(1.23)  LDD0609  [3]
 LDCM0293  AC32 HCT 116 C242(0.79); C275(1.22); C826(1.43); C767(1.45)  LDD0610  [3]
 LDCM0294  AC33 HCT 116 C242(0.91); C275(0.95); C227(0.97); C826(1.05)  LDD0611  [3]
 LDCM0295  AC34 HCT 116 C227(0.80); C275(0.96); C242(1.04); C767(1.09)  LDD0612  [3]
 LDCM0296  AC35 HCT 116 C227(0.69); C275(0.75); C826(0.79); C767(0.89)  LDD0613  [3]
 LDCM0297  AC36 HCT 116 C227(0.72); C275(0.79); C826(0.79); C767(0.91)  LDD0614  [3]
 LDCM0298  AC37 HCT 116 C227(0.66); C678(0.69); C275(0.75); C826(0.82)  LDD0615  [3]
 LDCM0299  AC38 HCT 116 C275(0.87); C767(0.92); C227(1.07); C826(1.19)  LDD0616  [3]
 LDCM0300  AC39 HCT 116 C275(0.92); C767(0.93); C826(0.97); C678(1.05)  LDD0617  [3]
 LDCM0301  AC4 HCT 116 C227(0.88); C186(0.92); C767(1.12); C764(1.15)  LDD0618  [3]
 LDCM0302  AC40 HCT 116 C275(0.78); C227(0.78); C767(0.81); C678(0.88)  LDD0619  [3]
 LDCM0303  AC41 HCT 116 C227(0.68); C826(0.77); C767(0.91); C275(0.91)  LDD0620  [3]
 LDCM0304  AC42 HCT 116 C275(0.89); C767(0.99); C678(1.03); C227(1.04)  LDD0621  [3]
 LDCM0305  AC43 HCT 116 C227(0.84); C826(0.94); C275(0.95); C767(0.98)  LDD0622  [3]
 LDCM0306  AC44 HCT 116 C227(0.48); C826(0.69); C275(0.71); C767(0.90)  LDD0623  [3]
 LDCM0307  AC45 HCT 116 C227(0.51); C826(0.71); C275(0.72); C767(0.92)  LDD0624  [3]
 LDCM0308  AC46 HCT 116 C767(1.10); C826(1.22); C227(1.35); C275(1.35)  LDD0625  [3]
 LDCM0309  AC47 HCT 116 C826(1.05); C275(1.25); C227(1.29); C767(1.29)  LDD0626  [3]
 LDCM0310  AC48 HCT 116 C227(0.99); C767(1.19); C826(1.34); C275(1.35)  LDD0627  [3]
 LDCM0311  AC49 HCT 116 C826(1.00); C767(1.00); C275(1.03); C227(1.31)  LDD0628  [3]
 LDCM0312  AC5 HCT 116 C227(0.85); C186(0.94); C764(1.24); C767(1.40)  LDD0629  [3]
 LDCM0313  AC50 HCT 116 C826(1.04); C767(1.12); C227(1.34); C275(1.37)  LDD0630  [3]
 LDCM0314  AC51 HCT 116 C275(0.71); C826(0.81); C227(1.05); C767(1.26)  LDD0631  [3]
 LDCM0315  AC52 HCT 116 C826(0.86); C275(0.91); C227(1.18); C767(1.21)  LDD0632  [3]
 LDCM0316  AC53 HCT 116 C826(0.78); C275(0.97); C767(1.03); C227(1.05)  LDD0633  [3]
 LDCM0317  AC54 HCT 116 C826(0.71); C227(0.98); C275(1.21); C767(1.46)  LDD0634  [3]
 LDCM0318  AC55 HCT 116 C826(0.91); C227(1.13); C767(1.37); C275(1.44)  LDD0635  [3]
 LDCM0319  AC56 HCT 116 C826(1.01); C227(1.16); C767(1.22); C275(1.61)  LDD0636  [3]
 LDCM0320  AC57 HCT 116 C242(0.83); C764(1.03); C678(1.05); C767(1.06)  LDD0637  [3]
 LDCM0321  AC58 HCT 116 C227(0.79); C678(0.93); C764(1.05); C242(1.08)  LDD0638  [3]
 LDCM0322  AC59 HCT 116 C242(0.95); C678(0.95); C764(1.09); C767(1.15)  LDD0639  [3]
 LDCM0323  AC6 HCT 116 C186(0.99); C242(1.08); C767(1.10); C275(1.23)  LDD0640  [3]
 LDCM0324  AC60 HCT 116 C678(0.91); C242(0.94); C764(1.10); C767(1.16)  LDD0641  [3]
 LDCM0325  AC61 HCT 116 C678(0.85); C242(0.92); C764(0.98); C227(1.01)  LDD0642  [3]
 LDCM0326  AC62 HCT 116 C678(0.88); C242(1.00); C227(1.03); C767(1.06)  LDD0643  [3]
 LDCM0327  AC63 HCT 116 C227(0.82); C242(0.90); C767(0.95); C678(1.09)  LDD0644  [3]
 LDCM0328  AC64 HCT 116 C242(0.97); C767(1.04); C678(1.12); C764(1.16)  LDD0645  [3]
 LDCM0329  AC65 HCT 116 C678(0.92); C242(0.96); C767(1.09); C764(1.18)  LDD0646  [3]
 LDCM0330  AC66 HCT 116 C227(0.93); C242(0.98); C767(0.99); C678(1.01)  LDD0647  [3]
 LDCM0331  AC67 HCT 116 C242(0.91); C678(0.99); C767(1.14); C227(1.16)  LDD0648  [3]
 LDCM0332  AC68 HCT 116 C275(0.86); C767(0.90); C764(0.90); C242(0.91)  LDD0649  [3]
 LDCM0333  AC69 HCT 116 C275(0.79); C764(0.87); C242(1.01); C755(1.31)  LDD0650  [3]
 LDCM0334  AC7 HCT 116 C242(1.02); C186(1.05); C275(1.14); C767(1.23)  LDD0651  [3]
 LDCM0335  AC70 HCT 116 C764(0.99); C275(1.26); C767(1.38); C242(1.40)  LDD0652  [3]
 LDCM0336  AC71 HCT 116 C764(0.72); C275(0.89); C767(0.94); C242(1.06)  LDD0653  [3]
 LDCM0337  AC72 HCT 116 C242(0.99); C767(1.06); C275(1.08); C764(1.14)  LDD0654  [3]
 LDCM0338  AC73 HCT 116 C764(1.07); C767(1.09); C242(1.25); C275(1.28)  LDD0655  [3]
 LDCM0339  AC74 HCT 116 C764(0.86); C767(1.10); C275(1.29); C242(1.31)  LDD0656  [3]
 LDCM0340  AC75 HCT 116 C764(0.87); C242(1.23); C767(1.23); C755(2.07)  LDD0657  [3]
 LDCM0341  AC76 HCT 116 C275(0.99); C764(1.05); C242(1.10); C767(1.10)  LDD0658  [3]
 LDCM0342  AC77 HCT 116 C764(0.61); C275(1.00); C242(1.08); C767(1.42)  LDD0659  [3]
 LDCM0343  AC78 HCT 116 C764(0.65); C275(0.92); C242(1.00); C767(1.05)  LDD0660  [3]
 LDCM0344  AC79 HCT 116 C764(0.88); C275(1.03); C242(1.05); C767(1.23)  LDD0661  [3]
 LDCM0345  AC8 HCT 116 C242(0.91); C186(0.99); C275(1.01); C767(1.27)  LDD0662  [3]
 LDCM0346  AC80 HCT 116 C764(0.91); C275(1.04); C242(1.07); C767(1.11)  LDD0663  [3]
 LDCM0347  AC81 HCT 116 C755(0.67); C764(0.76); C275(0.87); C242(0.95)  LDD0664  [3]
 LDCM0348  AC82 HCT 116 C764(0.79); C767(0.95); C242(1.26); C275(1.63)  LDD0665  [3]
 LDCM0349  AC83 HCT 116 C242(0.84); C678(1.20); C764(1.32); C826(1.36)  LDD0666  [3]
 LDCM0350  AC84 HCT 116 C826(0.79); C242(0.81); C678(0.95); C764(1.37)  LDD0667  [3]
 LDCM0351  AC85 HCT 116 C242(0.75); C678(0.98); C826(1.00); C764(1.18)  LDD0668  [3]
 LDCM0352  AC86 HCT 116 C242(0.77); C678(1.14); C764(1.16); C767(1.16)  LDD0669  [3]
 LDCM0353  AC87 HCT 116 C242(0.86); C767(0.98); C275(1.04); C678(1.09)  LDD0670  [3]
 LDCM0354  AC88 HCT 116 C242(0.85); C678(0.92); C764(1.12); C275(1.21)  LDD0671  [3]
 LDCM0355  AC89 HCT 116 C242(0.85); C678(1.11); C764(1.18); C767(1.26)  LDD0672  [3]
 LDCM0357  AC90 HCT 116 C242(0.94); C275(1.04); C764(1.04); C767(1.21)  LDD0674  [3]
 LDCM0358  AC91 HCT 116 C242(0.82); C678(1.05); C826(1.28); C764(1.33)  LDD0675  [3]
 LDCM0359  AC92 HCT 116 C242(0.77); C678(0.99); C826(1.39); C764(1.48)  LDD0676  [3]
 LDCM0360  AC93 HCT 116 C242(0.78); C826(0.79); C678(1.01); C767(1.06)  LDD0677  [3]
 LDCM0361  AC94 HCT 116 C826(0.72); C242(0.84); C275(1.00); C764(1.25)  LDD0678  [3]
 LDCM0362  AC95 HCT 116 C242(0.83); C275(1.08); C678(1.15); C764(1.18)  LDD0679  [3]
 LDCM0363  AC96 HCT 116 C826(0.55); C242(0.79); C275(1.10); C764(1.35)  LDD0680  [3]
 LDCM0364  AC97 HCT 116 C242(0.79); C678(1.22); C764(1.30); C767(1.50)  LDD0681  [3]
 LDCM0365  AC98 HCT 116 C764(0.97); C678(1.13); C186(1.33); C767(1.35)  LDD0682  [3]
 LDCM0366  AC99 HCT 116 C764(0.91); C678(0.94); C275(1.24); C767(1.32)  LDD0683  [3]
 LDCM0248  AKOS034007472 HCT 116 C186(1.04); C242(0.81); C275(1.24); C767(1.02)  LDD0565  [3]
 LDCM0356  AKOS034007680 HCT 116 C242(0.84); C186(1.00); C275(1.13); C767(1.26)  LDD0673  [3]
 LDCM0275  AKOS034007705 HCT 116 C242(1.01); C275(1.04); C186(1.08); C767(1.11)  LDD0592  [3]
 LDCM0020  ARS-1620 HCC44 C275(1.19); C242(1.04); C186(0.98)  LDD0078  [3]
 LDCM0630  CCW28-3 231MFP C845(1.21)  LDD2214  [12]
 LDCM0108  Chloroacetamide HeLa N.A.  LDD0222  [8]
 LDCM0632  CL-Sc Hep-G2 C515(20.00); C186(2.41)  LDD2227  [5]
 LDCM0367  CL1 HCT 116 C227(0.78); C767(1.07); C764(1.07); C826(1.08)  LDD0684  [3]
 LDCM0368  CL10 HCT 116 C227(0.89); C275(1.02); C826(1.06); C764(1.12)  LDD0685  [3]
 LDCM0369  CL100 HCT 116 C227(0.83); C186(0.94); C767(0.97); C764(1.14)  LDD0686  [3]
 LDCM0370  CL101 HCT 116 C186(0.95); C242(0.96); C767(1.02); C275(1.09)  LDD0687  [3]
 LDCM0371  CL102 HCT 116 C242(0.79); C186(0.89); C767(1.14); C275(1.36)  LDD0688  [3]
 LDCM0372  CL103 HCT 116 C242(0.84); C186(0.88); C275(1.15); C767(1.18)  LDD0689  [3]
 LDCM0373  CL104 HCT 116 C242(0.86); C186(1.04); C767(1.07); C275(1.16)  LDD0690  [3]
 LDCM0374  CL105 HCT 116 C764(0.95); C767(0.97); C242(1.08); C275(1.35)  LDD0691  [3]
 LDCM0375  CL106 HCT 116 C764(1.00); C767(1.05); C242(1.25); C826(1.33)  LDD0692  [3]
 LDCM0376  CL107 HCT 116 C767(0.92); C242(1.03); C275(1.40); C764(1.42)  LDD0693  [3]
 LDCM0377  CL108 HCT 116 C764(1.02); C767(1.17); C275(1.34); C242(1.48)  LDD0694  [3]
 LDCM0378  CL109 HCT 116 C767(0.89); C242(1.04); C764(1.04); C275(1.39)  LDD0695  [3]
 LDCM0379  CL11 HCT 116 C227(0.98); C826(1.13); C767(1.32); C764(1.38)  LDD0696  [3]
 LDCM0380  CL110 HCT 116 C764(0.80); C767(0.85); C242(1.07); C826(1.46)  LDD0697  [3]
 LDCM0381  CL111 HCT 116 C764(0.95); C767(0.98); C242(1.17); C275(1.37)  LDD0698  [3]
 LDCM0382  CL112 HCT 116 C242(0.73); C275(0.94); C826(1.01); C227(1.12)  LDD0699  [3]
 LDCM0383  CL113 HCT 116 C227(0.84); C242(0.85); C275(1.15); C826(1.27)  LDD0700  [3]
 LDCM0384  CL114 HCT 116 C242(0.89); C227(1.18); C275(1.37); C826(1.42)  LDD0701  [3]
 LDCM0385  CL115 HCT 116 C242(0.74); C227(1.10); C767(1.16); C275(1.19)  LDD0702  [3]
 LDCM0386  CL116 HCT 116 C242(0.69); C227(0.91); C275(1.05); C826(1.18)  LDD0703  [3]
 LDCM0387  CL117 HCT 116 C227(0.83); C275(0.84); C767(0.89); C755(1.14)  LDD0704  [3]
 LDCM0388  CL118 HCT 116 C227(0.84); C767(0.95); C275(0.99); C826(1.15)  LDD0705  [3]
 LDCM0389  CL119 HCT 116 C826(0.88); C767(0.91); C227(0.97); C275(1.00)  LDD0706  [3]
 LDCM0390  CL12 HCT 116 C275(0.98); C826(0.98); C764(1.03); C767(1.39)  LDD0707  [3]
 LDCM0391  CL120 HCT 116 C227(0.77); C767(0.96); C826(1.05); C678(1.06)  LDD0708  [3]
 LDCM0392  CL121 HCT 116 C826(0.71); C767(1.00); C227(1.08); C275(1.42)  LDD0709  [3]
 LDCM0393  CL122 HCT 116 C227(0.90); C275(0.96); C767(1.15); C826(1.51)  LDD0710  [3]
 LDCM0394  CL123 HCT 116 C767(1.08); C826(1.11); C275(1.64); C227(1.74)  LDD0711  [3]
 LDCM0395  CL124 HCT 116 C826(0.88); C227(0.96); C767(1.25); C275(1.51)  LDD0712  [3]
 LDCM0396  CL125 HCT 116 C242(0.79); C678(0.96); C764(1.04); C227(1.10)  LDD0713  [3]
 LDCM0397  CL126 HCT 116 C764(0.96); C227(1.01); C242(1.02); C678(1.04)  LDD0714  [3]
 LDCM0398  CL127 HCT 116 C764(0.91); C242(0.95); C678(0.99); C767(1.10)  LDD0715  [3]
 LDCM0399  CL128 HCT 116 C242(0.96); C678(0.97); C227(1.00); C764(1.10)  LDD0716  [3]
 LDCM0400  CL13 HCT 116 C275(0.96); C227(0.97); C826(0.98); C764(1.03)  LDD0717  [3]
 LDCM0401  CL14 HCT 116 C227(0.89); C826(1.06); C275(1.23); C764(1.25)  LDD0718  [3]
 LDCM0402  CL15 HCT 116 C227(0.85); C764(1.11); C826(1.16); C275(1.25)  LDD0719  [3]
 LDCM0403  CL16 HCT 116 C186(0.88); C275(1.12); C767(1.16); C764(1.62)  LDD0720  [3]
 LDCM0404  CL17 HCT 116 C186(0.84); C242(0.87); C767(0.90); C275(1.29)  LDD0721  [3]
 LDCM0405  CL18 HCT 116 C186(0.80); C242(0.85); C678(1.00); C764(1.10)  LDD0722  [3]
 LDCM0406  CL19 HCT 116 C186(0.80); C764(0.91); C242(1.00); C767(1.04)  LDD0723  [3]
 LDCM0407  CL2 HCT 116 C826(0.93); C764(0.98); C767(1.05); C227(1.18)  LDD0724  [3]
 LDCM0408  CL20 HCT 116 C242(0.93); C186(0.93); C764(1.04); C678(1.17)  LDD0725  [3]
 LDCM0409  CL21 HCT 116 C242(0.86); C764(0.89); C186(0.91); C767(1.29)  LDD0726  [3]
 LDCM0410  CL22 HCT 116 C764(0.82); C678(0.92); C186(1.00); C242(1.38)  LDD0727  [3]
 LDCM0411  CL23 HCT 116 C186(0.73); C678(1.04); C764(1.10); C242(1.14)  LDD0728  [3]
 LDCM0412  CL24 HCT 116 C186(0.70); C678(0.90); C242(0.93); C767(1.08)  LDD0729  [3]
 LDCM0413  CL25 HCT 116 C186(0.78); C242(0.82); C275(1.54); C678(1.06)  LDD0730  [3]
 LDCM0414  CL26 HCT 116 C186(0.71); C242(0.97); C275(1.25); C678(1.01)  LDD0731  [3]
 LDCM0415  CL27 HCT 116 C186(0.75); C242(0.86); C275(1.32); C678(0.91)  LDD0732  [3]
 LDCM0416  CL28 HCT 116 C186(0.83); C242(0.87); C275(1.23); C678(1.11)  LDD0733  [3]
 LDCM0417  CL29 HCT 116 C186(0.90); C242(1.31); C275(1.14); C678(0.99)  LDD0734  [3]
 LDCM0418  CL3 HCT 116 C227(0.90); C275(0.83); C764(0.96); C767(1.10)  LDD0735  [3]
 LDCM0419  CL30 HCT 116 C186(0.76); C242(1.14); C275(0.97); C678(1.16)  LDD0736  [3]
 LDCM0420  CL31 HCT 116 C186(0.92); C227(1.02); C242(0.99); C275(1.00)  LDD0737  [3]
 LDCM0421  CL32 HCT 116 C186(0.95); C227(0.82); C242(1.16); C275(0.91)  LDD0738  [3]
 LDCM0422  CL33 HCT 116 C186(0.98); C227(0.95); C242(1.64); C275(0.95)  LDD0739  [3]
 LDCM0423  CL34 HCT 116 C186(1.07); C227(1.29); C242(1.46); C275(0.98)  LDD0740  [3]
 LDCM0424  CL35 HCT 116 C186(1.05); C227(1.14); C242(1.53); C275(1.18)  LDD0741  [3]
 LDCM0425  CL36 HCT 116 C186(1.01); C227(1.01); C242(1.26); C275(0.75)  LDD0742  [3]
 LDCM0426  CL37 HCT 116 C186(1.09); C227(1.03); C242(1.47); C275(1.04)  LDD0743  [3]
 LDCM0428  CL39 HCT 116 C186(1.01); C227(1.19); C242(1.44); C275(0.93)  LDD0745  [3]
 LDCM0429  CL4 HCT 116 C227(0.95); C275(1.04); C764(1.09); C767(1.22)  LDD0746  [3]
 LDCM0430  CL40 HCT 116 C186(1.24); C227(1.21); C242(1.13); C275(1.03)  LDD0747  [3]
 LDCM0431  CL41 HCT 116 C186(1.01); C227(1.02); C242(1.12); C275(0.68)  LDD0748  [3]
 LDCM0432  CL42 HCT 116 C186(0.96); C227(1.28); C242(1.84); C275(0.78)  LDD0749  [3]
 LDCM0433  CL43 HCT 116 C186(1.04); C227(1.09); C242(1.71); C275(0.92)  LDD0750  [3]
 LDCM0434  CL44 HCT 116 C186(1.12); C227(1.23); C242(1.51); C275(1.14)  LDD0751  [3]
 LDCM0435  CL45 HCT 116 C186(1.15); C227(1.17); C242(1.59); C275(1.00)  LDD0752  [3]
 LDCM0436  CL46 HCT 116 C242(0.68); C275(1.22); C678(0.79); C764(0.96)  LDD0753  [3]
 LDCM0437  CL47 HCT 116 C242(0.91); C275(0.95); C678(0.87); C764(0.99)  LDD0754  [3]
 LDCM0438  CL48 HCT 116 C242(0.74); C275(0.97); C678(0.86); C764(0.78)  LDD0755  [3]
 LDCM0439  CL49 HCT 116 C242(0.79); C275(1.22); C678(0.90); C764(1.14)  LDD0756  [3]
 LDCM0440  CL5 HCT 116 C227(0.95); C275(1.07); C764(1.16); C767(1.23)  LDD0757  [3]
 LDCM0441  CL50 HCT 116 C242(0.73); C275(1.07); C678(0.86); C764(0.87)  LDD0758  [3]
 LDCM0442  CL51 HCT 116 C242(0.73); C275(1.24); C678(0.83); C764(0.88)  LDD0759  [3]
 LDCM0443  CL52 HCT 116 C242(0.82); C275(1.29); C678(0.85); C764(0.93)  LDD0760  [3]
 LDCM0444  CL53 HCT 116 C242(1.41); C275(0.74); C678(0.95); C764(1.03)  LDD0761  [3]
 LDCM0445  CL54 HCT 116 C242(0.87); C275(1.08); C678(0.96); C764(0.92)  LDD0762  [3]
 LDCM0446  CL55 HCT 116 C242(0.94); C275(0.85); C678(0.79); C764(1.02)  LDD0763  [3]
 LDCM0447  CL56 HCT 116 C242(1.21); C275(0.94); C678(0.93); C764(0.96)  LDD0764  [3]
 LDCM0448  CL57 HCT 116 C242(1.19); C275(0.91); C678(0.95); C764(0.99)  LDD0765  [3]
 LDCM0449  CL58 HCT 116 C242(0.97); C275(0.95); C678(0.76); C764(0.88)  LDD0766  [3]
 LDCM0450  CL59 HCT 116 C242(1.06); C275(0.99); C678(0.93); C764(1.01)  LDD0767  [3]
 LDCM0451  CL6 HCT 116 C227(0.75); C275(1.10); C764(1.13); C767(1.29)  LDD0768  [3]
 LDCM0452  CL60 HCT 116 C242(0.72); C275(1.22); C678(0.93); C764(0.95)  LDD0769  [3]
 LDCM0453  CL61 HCT 116 C242(0.97); C275(0.99); C755(1.01); C764(1.03)  LDD0770  [3]
 LDCM0454  CL62 HCT 116 C242(0.82); C275(1.37); C755(1.22); C764(1.41)  LDD0771  [3]
 LDCM0455  CL63 HCT 116 C242(0.95); C275(1.63); C755(1.24); C764(1.10)  LDD0772  [3]
 LDCM0456  CL64 HCT 116 C242(0.90); C275(1.29); C755(1.55); C764(1.22)  LDD0773  [3]
 LDCM0457  CL65 HCT 116 C242(1.04); C275(1.60); C755(1.15); C764(1.11)  LDD0774  [3]
 LDCM0458  CL66 HCT 116 C242(0.96); C275(1.32); C755(1.85); C764(1.51)  LDD0775  [3]
 LDCM0459  CL67 HCT 116 C242(1.50); C275(1.23); C755(1.43); C764(1.42)  LDD0776  [3]
 LDCM0460  CL68 HCT 116 C242(1.53); C275(1.30); C755(1.32); C764(1.04)  LDD0777  [3]
 LDCM0461  CL69 HCT 116 C242(1.04); C275(1.08); C755(1.31); C764(1.03)  LDD0778  [3]
 LDCM0462  CL7 HCT 116 C227(1.13); C275(1.13); C764(1.13); C767(1.42)  LDD0779  [3]
 LDCM0463  CL70 HCT 116 C242(1.02); C275(1.04); C755(1.10); C764(0.84)  LDD0780  [3]
 LDCM0464  CL71 HCT 116 C242(1.22); C275(1.48); C755(1.35); C764(1.50)  LDD0781  [3]
 LDCM0465  CL72 HCT 116 C242(1.21); C275(0.99); C755(1.12); C764(1.03)  LDD0782  [3]
 LDCM0466  CL73 HCT 116 C242(1.20); C275(1.39); C755(1.52); C764(1.33)  LDD0783  [3]
 LDCM0467  CL74 HCT 116 C242(1.38); C275(1.22); C755(1.52); C764(1.01)  LDD0784  [3]
 LDCM0469  CL76 HCT 116 C275(0.96); C764(1.25); C767(0.92); C826(1.03)  LDD0786  [3]
 LDCM0470  CL77 HCT 116 C275(0.95); C764(1.21); C767(0.89); C826(0.85)  LDD0787  [3]
 LDCM0471  CL78 HCT 116 C275(0.87); C764(1.09); C767(1.17); C826(0.86)  LDD0788  [3]
 LDCM0472  CL79 HCT 116 C275(1.19); C764(1.14); C767(0.93); C826(1.07)  LDD0789  [3]
 LDCM0473  CL8 HCT 116 C227(0.83); C275(1.94); C764(1.01); C767(1.51)  LDD0790  [3]
 LDCM0474  CL80 HCT 116 C275(1.15); C764(1.03); C767(0.91); C826(1.13)  LDD0791  [3]
 LDCM0475  CL81 HCT 116 C275(1.29); C764(1.16); C767(0.94); C826(0.83)  LDD0792  [3]
 LDCM0476  CL82 HCT 116 C275(1.13); C764(1.65); C767(0.84); C826(0.94)  LDD0793  [3]
 LDCM0477  CL83 HCT 116 C275(1.14); C764(1.21); C767(0.80); C826(0.91)  LDD0794  [3]
 LDCM0478  CL84 HCT 116 C275(1.22); C764(1.51); C767(0.97); C826(0.82)  LDD0795  [3]
 LDCM0479  CL85 HCT 116 C275(1.12); C764(1.01); C767(1.08); C826(0.87)  LDD0796  [3]
 LDCM0480  CL86 HCT 116 C275(0.84); C764(1.09); C767(0.90); C826(0.98)  LDD0797  [3]
 LDCM0481  CL87 HCT 116 C275(1.09); C764(1.12); C767(0.91); C826(0.94)  LDD0798  [3]
 LDCM0482  CL88 HCT 116 C275(0.81); C764(1.75); C767(0.92); C826(0.81)  LDD0799  [3]
 LDCM0483  CL89 HCT 116 C275(0.85); C764(1.60); C767(1.04); C826(1.02)  LDD0800  [3]
 LDCM0484  CL9 HCT 116 C227(1.02); C275(1.32); C764(0.93); C767(1.21)  LDD0801  [3]
 LDCM0485  CL90 HCT 116 C275(1.01); C764(0.83); C767(0.94); C826(1.07)  LDD0802  [3]
 LDCM0486  CL91 HCT 116 C186(0.77); C227(0.78); C275(1.04); C755(1.12)  LDD0803  [3]
 LDCM0487  CL92 HCT 116 C186(0.93); C227(0.62); C275(1.13); C755(1.55)  LDD0804  [3]
 LDCM0488  CL93 HCT 116 C186(0.82); C227(0.86); C275(1.14); C755(1.26)  LDD0805  [3]
 LDCM0489  CL94 HCT 116 C186(0.89); C227(1.02); C275(1.44); C755(1.78)  LDD0806  [3]
 LDCM0490  CL95 HCT 116 C186(0.95); C227(0.61); C275(1.69); C755(1.60)  LDD0807  [3]
 LDCM0491  CL96 HCT 116 C186(0.77); C227(0.82); C275(1.38); C755(1.49)  LDD0808  [3]
 LDCM0492  CL97 HCT 116 C186(0.99); C227(0.95); C275(1.39); C755(1.19)  LDD0809  [3]
 LDCM0493  CL98 HCT 116 C186(0.94); C227(1.84); C275(1.37); C755(1.34)  LDD0810  [3]
 LDCM0494  CL99 HCT 116 C186(0.87); C227(1.05); C275(1.21); C755(1.32)  LDD0811  [3]
 LDCM0495  E2913 HEK-293T C678(0.95); C275(1.04); C242(0.98); C227(0.98)  LDD1698  [13]
 LDCM0213  Electrophilic fragment 2 MDA-MB-231 C227(2.35)  LDD1702  [1]
 LDCM0625  F8 Ramos C227(1.42)  LDD2187  [14]
 LDCM0572  Fragment10 Ramos C227(1.72)  LDD2189  [14]
 LDCM0575  Fragment13 Ramos C227(1.04)  LDD2192  [14]
 LDCM0576  Fragment14 Ramos C227(7.84)  LDD2193  [14]
 LDCM0579  Fragment20 Ramos C227(1.82)  LDD2194  [14]
 LDCM0580  Fragment21 Ramos C227(1.07)  LDD2195  [14]
 LDCM0582  Fragment23 Ramos C227(0.70)  LDD2196  [14]
 LDCM0578  Fragment27 Ramos C227(1.08)  LDD2197  [14]
 LDCM0586  Fragment28 Ramos C227(0.83)  LDD2198  [14]
 LDCM0588  Fragment30 Ramos C227(1.14)  LDD2199  [14]
 LDCM0589  Fragment31 Ramos C227(0.91)  LDD2200  [14]
 LDCM0590  Fragment32 Ramos C227(1.72)  LDD2201  [14]
 LDCM0468  Fragment33 HCT 116 C242(0.93); C275(1.32); C755(1.43); C764(1.35)  LDD0785  [3]
 LDCM0596  Fragment38 Ramos C227(0.97)  LDD2203  [14]
 LDCM0427  Fragment51 HCT 116 C186(0.97); C227(1.28); C242(1.62); C275(0.97)  LDD0744  [3]
 LDCM0610  Fragment52 Ramos C227(1.47)  LDD2204  [14]
 LDCM0614  Fragment56 Ramos C227(0.93)  LDD2205  [14]
 LDCM0107  IAA HeLa N.A.  LDD0221  [8]
 LDCM0022  KB02 HEK-293T C227(0.91); C678(1.04); C275(0.84)  LDD1492  [13]
 LDCM0023  KB03 HEK-293T C227(0.98); C678(0.94); C275(0.96)  LDD1497  [13]
 LDCM0024  KB05 G361 C767(2.53); C227(2.96); C764(1.69)  LDD3311  [15]
 LDCM0109  NEM HeLa H94(0.00); H539(0.00)  LDD0224  [8]
 LDCM0516  Nucleophilic fragment 21a MDA-MB-231 C227(0.99)  LDD2109  [1]
 LDCM0021  THZ1 HCT 116 C767(1.08); C275(0.94)  LDD2173  [3]

References

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Mass spectrometry data entry: PXD039908 , PXD029761
2 Chemoproteomic capture of RNA binding activity in living cells. Nat Commun. 2023 Oct 7;14(1):6282. doi: 10.1038/s41467-023-41844-z.
Mass spectrometry data entry: PXD044625
3 Reimagining high-throughput profiling of reactive cysteines for cell-based screening of large electrophile libraries. Nat Biotechnol. 2021 May;39(5):630-641. doi: 10.1038/s41587-020-00778-3. Epub 2021 Jan 4.
4 SP3-FAIMS Chemoproteomics for High-Coverage Profiling of the Human Cysteinome*. Chembiochem. 2021 May 14;22(10):1841-1851. doi: 10.1002/cbic.202000870. Epub 2021 Feb 18.
Mass spectrometry data entry: PXD023056 , PXD023059 , PXD023058 , PXD023057 , PXD023060
5 N-Acryloylindole-alkyne (NAIA) enables imaging and profiling new ligandable cysteines and oxidized thiols by chemoproteomics. Nat Commun. 2023 Jun 15;14(1):3564. doi: 10.1038/s41467-023-39268-w.
Mass spectrometry data entry: PXD041264
6 Chemoproteomic Profiling by Cysteine Fluoroalkylation Reveals Myrocin G as an Inhibitor of the Nonhomologous End Joining DNA Repair Pathway. J Am Chem Soc. 2021 Dec 8;143(48):20332-20342. doi: 10.1021/jacs.1c09724. Epub 2021 Nov 24.
Mass spectrometry data entry: PXD029255
7 A modification-centric assessment tool for the performance of chemoproteomic probes. Nat Chem Biol. 2022 Aug;18(8):904-912. doi: 10.1038/s41589-022-01074-8. Epub 2022 Jul 21.
Mass spectrometry data entry: PXD027758 , PXD027755 , PXD027760 , PXD027762 , PXD027756 , PXD027591 , PXD007149 , PXD030064 , PXD032392 , PXD027789 , PXD027767 , PXD027764
8 ACR-Based Probe for the Quantitative Profiling of Histidine Reactivity in the Human Proteome. J Am Chem Soc. 2023 Mar 8;145(9):5252-5260. doi: 10.1021/jacs.2c12653. Epub 2023 Feb 27.
9 Chemoproteomic profiling of targets of lipid-derived electrophiles by bioorthogonal aminooxy probe. Redox Biol. 2017 Aug;12:712-718. doi: 10.1016/j.redox.2017.04.001. Epub 2017 Apr 5.
10 Ligand and Target Discovery by Fragment-Based Screening in Human Cells. Cell. 2017 Jan 26;168(3):527-541.e29. doi: 10.1016/j.cell.2016.12.029. Epub 2017 Jan 19.
11 Design and synthesis of minimalist terminal alkyne-containing diazirine photo-crosslinkers and their incorporation into kinase inhibitors for cell- and tissue-based proteome profiling. Angew Chem Int Ed Engl. 2013 Aug 12;52(33):8551-6. doi: 10.1002/anie.201300683. Epub 2013 Jun 10.
12 Covalent Ligand Screening Uncovers a RNF4 E3 Ligase Recruiter for Targeted Protein Degradation Applications. ACS Chem Biol. 2019 Nov 15;14(11):2430-2440. doi: 10.1021/acschembio.8b01083. Epub 2019 May 13.
13 Accelerating multiplexed profiling of protein-ligand interactions: High-throughput plate-based reactive cysteine profiling with minimal input. Cell Chem Biol. 2024 Mar 21;31(3):565-576.e4. doi: 10.1016/j.chembiol.2023.11.015. Epub 2023 Dec 19.
Mass spectrometry data entry: PXD044402
14 Site-specific quantitative cysteine profiling with data-independent acquisition-based mass spectrometry. Methods Enzymol. 2023;679:295-322. doi: 10.1016/bs.mie.2022.07.037. Epub 2022 Sep 7.
Mass spectrometry data entry: PXD027578
15 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840