Details of the Target
General Information of Target
Target ID | LDTP04223 | |||||
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Target Name | DNA polymerase delta subunit 2 (POLD2) | |||||
Gene Name | POLD2 | |||||
Gene ID | 5425 | |||||
Synonyms |
DNA polymerase delta subunit 2; DNA polymerase delta subunit p50 |
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3D Structure | ||||||
Sequence |
MFSEQAAQRAHTLLSPPSANNATFARVPVATYTNSSQPFRLGERSFSRQYAHIYATRLIQ
MRPFLENRAQQHWGSGVGVKKLCELQPEEKCCVVGTLFKAMPLQPSILREVSEEHNLLPQ PPRSKYIHPDDELVLEDELQRIKLKGTIDVSKLVTGTVLAVFGSVRDDGKFLVEDYCFAD LAPQKPAPPLDTDRFVLLVSGLGLGGGGGESLLGTQLLVDVVTGQLGDEGEQCSAAHVSR VILAGNLLSHSTQSRDSINKAKYLTKKTQAASVEAVKMLDEILLQLSASVPVDVMPGEFD PTNYTLPQQPLHPCMFPLATAYSTLQLVTNPYQATIDGVRFLGTSGQNVSDIFRYSSMED HLEILEWTLRVRHISPTAPDTLGCYPFYKTDPFIFPECPHVYFCGNTPSFGSKIIRGPED QTVLLVTVPDFSATQTACLVNLRSLACQPISFSGFGAEDDDLGGLGLGP |
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Target Bioclass |
Enzyme
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Family |
DNA polymerase delta/II small subunit family
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Subcellular location |
Nucleus
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Function |
Accessory component of both the DNA polymerase delta complex and the DNA polymerase zeta complex. As a component of the trimeric and tetrameric DNA polymerase delta complexes (Pol-delta3 and Pol-delta4, respectively), plays a role in high fidelity genome replication, including in lagging strand synthesis, and repair. Pol-delta3 and Pol-delta4 are characterized by the absence or the presence of POLD4. They exhibit differences in catalytic activity. Most notably, Pol-delta3 shows higher proofreading activity than Pol-delta4. Although both Pol-delta3 and Pol-delta4 process Okazaki fragments in vitro, Pol-delta3 may also be better suited to fulfill this task, exhibiting near-absence of strand displacement activity compared to Pol-delta4 and stalling on encounter with the 5'-blocking oligonucleotides. Pol-delta3 idling process may avoid the formation of a gap, while maintaining a nick that can be readily ligated. Along with DNA polymerase kappa, DNA polymerase delta carries out approximately half of nucleotide excision repair (NER) synthesis following UV irradiation. Under conditions of DNA replication stress, required for the repair of broken replication forks through break-induced replication (BIR). Involved in the translesion synthesis (TLS) of templates carrying O6-methylguanine or abasic sites performed by Pol-delta4, independently of DNA polymerase zeta (REV3L) or eta (POLH). Facilitates abasic site bypass by DNA polymerase delta by promoting extension from the nucleotide inserted opposite the lesion. Also involved in TLS as a component of the DNA polymerase zeta complex. Along with POLD3, dramatically increases the efficiency and processivity of DNA synthesis of the DNA polymerase zeta complex compared to the minimal zeta complex, consisting of only REV3L and REV7.
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Uniprot ID | ||||||
Ensemble ID | ||||||
HGNC ID | ||||||
ChEMBL ID |
Probe(s) Labeling This Target
ABPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
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m-APA Probe Info |
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14.67 | LDD0402 | [1] | |
TH211 Probe Info |
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Y32(8.78) | LDD0257 | [2] | |
Probe 1 Probe Info |
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Y32(5.49) | LDD3495 | [3] | |
DBIA Probe Info |
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C91(9.03); C92(9.03); C83(1.24) | LDD0080 | [4] | |
5E-2FA Probe Info |
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H72(0.00); H400(0.00); H250(0.00) | LDD2235 | [5] | |
4-Iodoacetamidophenylacetylene Probe Info |
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C384(0.00); C83(0.00); C447(0.00); C438(0.00) | LDD0038 | [6] | |
IA-alkyne Probe Info |
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C91(0.00); C92(0.00); C438(0.00); C384(0.00) | LDD0036 | [6] | |
Lodoacetamide azide Probe Info |
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C177(0.00); C384(0.00); C83(0.00); C447(0.00) | LDD0037 | [6] | |
BTD Probe Info |
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N.A. | LDD0004 | [7] | |
NAIA_4 Probe Info |
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N.A. | LDD2226 | [8] | |
TFBX Probe Info |
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N.A. | LDD0027 | [9] | |
Compound 10 Probe Info |
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N.A. | LDD2216 | [10] | |
ENE Probe Info |
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N.A. | LDD0006 | [7] | |
IPM Probe Info |
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N.A. | LDD0005 | [7] | |
VSF Probe Info |
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N.A. | LDD0007 | [7] | |
Phosphinate-6 Probe Info |
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N.A. | LDD0018 | [11] | |
Acrolein Probe Info |
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N.A. | LDD0217 | [12] | |
AOyne Probe Info |
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6.20 | LDD0443 | [13] | |
NAIA_5 Probe Info |
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N.A. | LDD2223 | [8] |
Competitor(s) Related to This Target
Competitor ID | Name | Cell line | Binding Site(Ratio) | Interaction ID | Ref |
---|---|---|---|---|---|
LDCM0510 | 3-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-3-oxopropanenitrile | MDA-MB-231 | C83(0.97) | LDD2103 | [14] |
LDCM0539 | 3-(4-Isopropylpiperazin-1-yl)-3-oxopropanenitrile | MDA-MB-231 | C83(0.73) | LDD2132 | [14] |
LDCM0214 | AC1 | HCT 116 | C91(1.12); C92(1.12) | LDD0531 | [4] |
LDCM0215 | AC10 | HCT 116 | C91(1.26); C92(1.26) | LDD0532 | [4] |
LDCM0216 | AC100 | HCT 116 | C91(0.99); C92(0.99) | LDD0533 | [4] |
LDCM0217 | AC101 | HCT 116 | C91(0.81); C92(0.81) | LDD0534 | [4] |
LDCM0218 | AC102 | HCT 116 | C91(0.95); C92(0.95) | LDD0535 | [4] |
LDCM0219 | AC103 | HCT 116 | C91(0.78); C92(0.78) | LDD0536 | [4] |
LDCM0220 | AC104 | HCT 116 | C91(0.97); C92(0.97) | LDD0537 | [4] |
LDCM0221 | AC105 | HCT 116 | C91(0.83); C92(0.83) | LDD0538 | [4] |
LDCM0222 | AC106 | HCT 116 | C91(0.87); C92(0.87) | LDD0539 | [4] |
LDCM0223 | AC107 | HCT 116 | C91(0.84); C92(0.84) | LDD0540 | [4] |
LDCM0224 | AC108 | HCT 116 | C91(0.81); C92(0.81) | LDD0541 | [4] |
LDCM0225 | AC109 | HCT 116 | C91(1.06); C92(1.06) | LDD0542 | [4] |
LDCM0226 | AC11 | HCT 116 | C91(1.41); C92(1.41) | LDD0543 | [4] |
LDCM0227 | AC110 | HCT 116 | C91(0.78); C92(0.78) | LDD0544 | [4] |
LDCM0228 | AC111 | HCT 116 | C91(0.77); C92(0.77) | LDD0545 | [4] |
LDCM0229 | AC112 | HCT 116 | C91(0.79); C92(0.79) | LDD0546 | [4] |
LDCM0230 | AC113 | HCT 116 | C91(0.89); C92(0.89) | LDD0547 | [4] |
LDCM0231 | AC114 | HCT 116 | C91(0.88); C92(0.75) | LDD0548 | [4] |
LDCM0232 | AC115 | HCT 116 | C91(1.19); C92(0.76) | LDD0549 | [4] |
LDCM0233 | AC116 | HCT 116 | C91(0.77); C92(0.89) | LDD0550 | [4] |
LDCM0234 | AC117 | HCT 116 | C91(0.90); C92(0.84) | LDD0551 | [4] |
LDCM0235 | AC118 | HCT 116 | C91(0.97); C92(0.93) | LDD0552 | [4] |
LDCM0236 | AC119 | HCT 116 | C91(1.08); C92(0.87) | LDD0553 | [4] |
LDCM0237 | AC12 | HCT 116 | C91(1.46); C92(1.46) | LDD0554 | [4] |
LDCM0238 | AC120 | HCT 116 | C91(1.29); C92(0.91) | LDD0555 | [4] |
LDCM0239 | AC121 | HCT 116 | C91(0.82); C92(0.99) | LDD0556 | [4] |
LDCM0240 | AC122 | HCT 116 | C91(0.74); C92(0.91) | LDD0557 | [4] |
LDCM0241 | AC123 | HCT 116 | C91(0.77); C92(0.86) | LDD0558 | [4] |
LDCM0242 | AC124 | HCT 116 | C91(0.90); C92(0.99) | LDD0559 | [4] |
LDCM0243 | AC125 | HCT 116 | C91(0.93); C92(0.81) | LDD0560 | [4] |
LDCM0244 | AC126 | HCT 116 | C91(0.96); C92(0.84) | LDD0561 | [4] |
LDCM0245 | AC127 | HCT 116 | C91(0.89); C92(0.89) | LDD0562 | [4] |
LDCM0246 | AC128 | HCT 116 | C91(0.89); C92(0.89) | LDD0563 | [4] |
LDCM0247 | AC129 | HCT 116 | C91(1.06); C92(1.06) | LDD0564 | [4] |
LDCM0249 | AC130 | HCT 116 | C91(0.76); C92(0.76) | LDD0566 | [4] |
LDCM0250 | AC131 | HCT 116 | C91(1.06); C92(1.06) | LDD0567 | [4] |
LDCM0251 | AC132 | HCT 116 | C91(0.90); C92(0.90) | LDD0568 | [4] |
LDCM0252 | AC133 | HCT 116 | C91(0.80); C92(0.80) | LDD0569 | [4] |
LDCM0253 | AC134 | HCT 116 | C91(0.74); C92(0.74) | LDD0570 | [4] |
LDCM0254 | AC135 | HCT 116 | C91(0.77); C92(0.77) | LDD0571 | [4] |
LDCM0255 | AC136 | HCT 116 | C91(0.78); C92(0.78) | LDD0572 | [4] |
LDCM0256 | AC137 | HCT 116 | C91(0.85); C92(0.85) | LDD0573 | [4] |
LDCM0257 | AC138 | HCT 116 | C91(0.74); C92(0.74) | LDD0574 | [4] |
LDCM0258 | AC139 | HCT 116 | C91(0.77); C92(0.77) | LDD0575 | [4] |
LDCM0259 | AC14 | HCT 116 | C91(1.48); C92(1.48) | LDD0576 | [4] |
LDCM0260 | AC140 | HCT 116 | C91(0.74); C92(0.74) | LDD0577 | [4] |
LDCM0261 | AC141 | HCT 116 | C91(0.78); C92(0.78) | LDD0578 | [4] |
LDCM0262 | AC142 | HCT 116 | C91(0.72); C92(0.72) | LDD0579 | [4] |
LDCM0263 | AC143 | HCT 116 | C83(1.03) | LDD0580 | [4] |
LDCM0264 | AC144 | HCT 116 | C83(1.12) | LDD0581 | [4] |
LDCM0265 | AC145 | HCT 116 | C83(1.02) | LDD0582 | [4] |
LDCM0266 | AC146 | HCT 116 | C83(0.94) | LDD0583 | [4] |
LDCM0267 | AC147 | HCT 116 | C83(1.05) | LDD0584 | [4] |
LDCM0268 | AC148 | HCT 116 | C83(1.08) | LDD0585 | [4] |
LDCM0269 | AC149 | HCT 116 | C83(0.98) | LDD0586 | [4] |
LDCM0270 | AC15 | HCT 116 | C91(1.25); C92(1.25) | LDD0587 | [4] |
LDCM0271 | AC150 | HCT 116 | C83(0.89) | LDD0588 | [4] |
LDCM0272 | AC151 | HCT 116 | C83(1.03) | LDD0589 | [4] |
LDCM0273 | AC152 | HCT 116 | C83(0.85) | LDD0590 | [4] |
LDCM0274 | AC153 | HCT 116 | C83(0.98) | LDD0591 | [4] |
LDCM0621 | AC154 | HCT 116 | C83(1.09) | LDD2158 | [4] |
LDCM0622 | AC155 | HCT 116 | C83(1.08) | LDD2159 | [4] |
LDCM0623 | AC156 | HCT 116 | C83(1.03) | LDD2160 | [4] |
LDCM0624 | AC157 | HCT 116 | C83(0.96) | LDD2161 | [4] |
LDCM0276 | AC17 | HCT 116 | C91(0.89); C92(0.89) | LDD0593 | [4] |
LDCM0277 | AC18 | HCT 116 | C91(0.55); C92(0.55) | LDD0594 | [4] |
LDCM0278 | AC19 | HCT 116 | C91(0.75); C92(0.75) | LDD0595 | [4] |
LDCM0279 | AC2 | HCT 116 | C91(0.99); C92(0.99) | LDD0596 | [4] |
LDCM0280 | AC20 | HCT 116 | C91(0.55); C92(0.55) | LDD0597 | [4] |
LDCM0281 | AC21 | HCT 116 | C91(0.72); C92(0.72) | LDD0598 | [4] |
LDCM0282 | AC22 | HCT 116 | C91(0.69); C92(0.69) | LDD0599 | [4] |
LDCM0283 | AC23 | HCT 116 | C91(0.81); C92(0.81) | LDD0600 | [4] |
LDCM0284 | AC24 | HCT 116 | C91(1.14); C92(1.14) | LDD0601 | [4] |
LDCM0285 | AC25 | HCT 116 | C91(1.00); C92(1.00) | LDD0602 | [4] |
LDCM0286 | AC26 | HCT 116 | C91(0.79); C92(0.79) | LDD0603 | [4] |
LDCM0287 | AC27 | HCT 116 | C91(0.76); C92(0.76) | LDD0604 | [4] |
LDCM0288 | AC28 | HCT 116 | C91(0.76); C92(0.76) | LDD0605 | [4] |
LDCM0289 | AC29 | HCT 116 | C91(0.66); C92(0.66) | LDD0606 | [4] |
LDCM0290 | AC3 | HCT 116 | C91(1.18); C92(1.18) | LDD0607 | [4] |
LDCM0291 | AC30 | HCT 116 | C91(0.64); C92(0.64) | LDD0608 | [4] |
LDCM0292 | AC31 | HCT 116 | C91(0.60); C92(0.60) | LDD0609 | [4] |
LDCM0293 | AC32 | HCT 116 | C91(0.62); C92(0.62) | LDD0610 | [4] |
LDCM0294 | AC33 | HCT 116 | C91(0.68); C92(0.68) | LDD0611 | [4] |
LDCM0295 | AC34 | HCT 116 | C91(0.63); C92(0.63) | LDD0612 | [4] |
LDCM0296 | AC35 | HCT 116 | C83(0.89) | LDD0613 | [4] |
LDCM0297 | AC36 | HCT 116 | C83(0.89) | LDD0614 | [4] |
LDCM0298 | AC37 | HCT 116 | C83(1.02) | LDD0615 | [4] |
LDCM0299 | AC38 | HCT 116 | C83(1.02) | LDD0616 | [4] |
LDCM0300 | AC39 | HCT 116 | C83(1.20) | LDD0617 | [4] |
LDCM0301 | AC4 | HCT 116 | C91(1.13); C92(1.13) | LDD0618 | [4] |
LDCM0302 | AC40 | HCT 116 | C83(1.09) | LDD0619 | [4] |
LDCM0303 | AC41 | HCT 116 | C83(1.03) | LDD0620 | [4] |
LDCM0304 | AC42 | HCT 116 | C83(1.08) | LDD0621 | [4] |
LDCM0305 | AC43 | HCT 116 | C83(1.09) | LDD0622 | [4] |
LDCM0306 | AC44 | HCT 116 | C83(1.13) | LDD0623 | [4] |
LDCM0307 | AC45 | HCT 116 | C83(1.16) | LDD0624 | [4] |
LDCM0308 | AC46 | HCT 116 | C91(0.72); C92(0.72) | LDD0625 | [4] |
LDCM0309 | AC47 | HCT 116 | C91(0.82); C92(0.82) | LDD0626 | [4] |
LDCM0310 | AC48 | HCT 116 | C91(0.52); C92(0.52) | LDD0627 | [4] |
LDCM0311 | AC49 | HCT 116 | C91(0.57); C92(0.57) | LDD0628 | [4] |
LDCM0312 | AC5 | HCT 116 | C91(1.22); C92(1.22) | LDD0629 | [4] |
LDCM0313 | AC50 | HCT 116 | C91(0.61); C92(0.61) | LDD0630 | [4] |
LDCM0314 | AC51 | HCT 116 | C91(0.82); C92(0.82) | LDD0631 | [4] |
LDCM0315 | AC52 | HCT 116 | C91(0.79); C92(0.79) | LDD0632 | [4] |
LDCM0316 | AC53 | HCT 116 | C91(0.87); C92(0.87) | LDD0633 | [4] |
LDCM0317 | AC54 | HCT 116 | C91(0.77); C92(0.77) | LDD0634 | [4] |
LDCM0318 | AC55 | HCT 116 | C91(0.88); C92(0.88) | LDD0635 | [4] |
LDCM0319 | AC56 | HCT 116 | C91(0.59); C92(0.59) | LDD0636 | [4] |
LDCM0320 | AC57 | HCT 116 | C91(0.66); C92(0.66); C83(1.17) | LDD0637 | [4] |
LDCM0321 | AC58 | HCT 116 | C91(0.61); C92(0.61); C83(1.37) | LDD0638 | [4] |
LDCM0322 | AC59 | HCT 116 | C91(0.65); C92(0.65); C83(1.32) | LDD0639 | [4] |
LDCM0323 | AC6 | HCT 116 | C91(0.93); C92(0.93) | LDD0640 | [4] |
LDCM0324 | AC60 | HCT 116 | C91(0.51); C92(0.51); C83(1.23) | LDD0641 | [4] |
LDCM0325 | AC61 | HCT 116 | C91(0.52); C92(0.52); C83(1.00) | LDD0642 | [4] |
LDCM0326 | AC62 | HCT 116 | C91(0.62); C92(0.62); C83(1.33) | LDD0643 | [4] |
LDCM0327 | AC63 | HCT 116 | C91(0.64); C92(0.64); C83(1.07) | LDD0644 | [4] |
LDCM0328 | AC64 | HCT 116 | C91(0.59); C92(0.59); C83(1.44) | LDD0645 | [4] |
LDCM0329 | AC65 | HCT 116 | C91(0.52); C92(0.52); C83(1.47) | LDD0646 | [4] |
LDCM0330 | AC66 | HCT 116 | C91(0.56); C92(0.56); C83(1.11) | LDD0647 | [4] |
LDCM0331 | AC67 | HCT 116 | C91(0.39); C92(0.39); C83(0.94) | LDD0648 | [4] |
LDCM0332 | AC68 | HCT 116 | C91(0.70); C92(0.70); C83(1.03) | LDD0649 | [4] |
LDCM0333 | AC69 | HCT 116 | C91(0.77); C92(0.77); C83(1.06) | LDD0650 | [4] |
LDCM0334 | AC7 | HCT 116 | C91(1.06); C92(1.06) | LDD0651 | [4] |
LDCM0335 | AC70 | HCT 116 | C91(0.81); C92(0.81); C83(0.95) | LDD0652 | [4] |
LDCM0336 | AC71 | HCT 116 | C91(0.84); C92(0.84); C83(0.99) | LDD0653 | [4] |
LDCM0337 | AC72 | HCT 116 | C91(0.81); C92(0.81); C83(0.91) | LDD0654 | [4] |
LDCM0338 | AC73 | HCT 116 | C91(0.66); C92(0.66); C83(1.02) | LDD0655 | [4] |
LDCM0339 | AC74 | HCT 116 | C91(0.65); C92(0.65); C83(1.02) | LDD0656 | [4] |
LDCM0340 | AC75 | HCT 116 | C91(0.69); C92(0.69); C83(0.97) | LDD0657 | [4] |
LDCM0341 | AC76 | HCT 116 | C91(0.76); C92(0.76); C83(0.96) | LDD0658 | [4] |
LDCM0342 | AC77 | HCT 116 | C91(0.75); C92(0.75); C83(1.01) | LDD0659 | [4] |
LDCM0343 | AC78 | HCT 116 | C91(0.69); C92(0.69); C83(0.96) | LDD0660 | [4] |
LDCM0344 | AC79 | HCT 116 | C91(0.81); C92(0.81); C83(1.03) | LDD0661 | [4] |
LDCM0345 | AC8 | HCT 116 | C91(1.01); C92(1.01) | LDD0662 | [4] |
LDCM0346 | AC80 | HCT 116 | C91(0.75); C92(0.75); C83(0.99) | LDD0663 | [4] |
LDCM0347 | AC81 | HCT 116 | C91(1.02); C92(1.02); C83(1.04) | LDD0664 | [4] |
LDCM0348 | AC82 | HCT 116 | C91(0.63); C92(0.63); C83(0.94) | LDD0665 | [4] |
LDCM0349 | AC83 | HCT 116 | C91(0.74); C92(0.74) | LDD0666 | [4] |
LDCM0350 | AC84 | HCT 116 | C91(0.76); C92(0.76) | LDD0667 | [4] |
LDCM0351 | AC85 | HCT 116 | C91(0.84); C92(0.84) | LDD0668 | [4] |
LDCM0352 | AC86 | HCT 116 | C91(0.92); C92(0.92) | LDD0669 | [4] |
LDCM0353 | AC87 | HCT 116 | C91(0.92); C92(0.92) | LDD0670 | [4] |
LDCM0354 | AC88 | HCT 116 | C91(0.94); C92(0.94) | LDD0671 | [4] |
LDCM0355 | AC89 | HCT 116 | C91(0.86); C92(0.86) | LDD0672 | [4] |
LDCM0357 | AC90 | HCT 116 | C91(1.16); C92(1.16) | LDD0674 | [4] |
LDCM0358 | AC91 | HCT 116 | C91(0.99); C92(0.99) | LDD0675 | [4] |
LDCM0359 | AC92 | HCT 116 | C91(1.02); C92(1.02) | LDD0676 | [4] |
LDCM0360 | AC93 | HCT 116 | C91(1.01); C92(1.01) | LDD0677 | [4] |
LDCM0361 | AC94 | HCT 116 | C91(1.16); C92(1.16) | LDD0678 | [4] |
LDCM0362 | AC95 | HCT 116 | C91(0.72); C92(0.72) | LDD0679 | [4] |
LDCM0363 | AC96 | HCT 116 | C91(1.17); C92(1.17) | LDD0680 | [4] |
LDCM0364 | AC97 | HCT 116 | C91(0.84); C92(0.84) | LDD0681 | [4] |
LDCM0365 | AC98 | HCT 116 | C91(0.69); C92(0.69) | LDD0682 | [4] |
LDCM0366 | AC99 | HCT 116 | C91(0.76); C92(0.76) | LDD0683 | [4] |
LDCM0545 | Acetamide | MDA-MB-231 | C83(0.44) | LDD2138 | [14] |
LDCM0520 | AKOS000195272 | MDA-MB-231 | C83(0.71) | LDD2113 | [14] |
LDCM0248 | AKOS034007472 | HCT 116 | C91(1.33); C92(1.33) | LDD0565 | [4] |
LDCM0356 | AKOS034007680 | HCT 116 | C91(1.52); C92(1.52) | LDD0673 | [4] |
LDCM0275 | AKOS034007705 | HCT 116 | C91(1.05); C92(1.05) | LDD0592 | [4] |
LDCM0156 | Aniline | NCI-H1299 | 10.20 | LDD0403 | [1] |
LDCM0498 | BS-3668 | MDA-MB-231 | C83(0.51) | LDD2091 | [14] |
LDCM0108 | Chloroacetamide | HeLa | C384(0.00); C83(0.00) | LDD0222 | [12] |
LDCM0367 | CL1 | HCT 116 | C91(1.08); C92(1.08) | LDD0684 | [4] |
LDCM0368 | CL10 | HCT 116 | C91(0.63); C92(0.63) | LDD0685 | [4] |
LDCM0369 | CL100 | HCT 116 | C91(1.06); C92(1.06) | LDD0686 | [4] |
LDCM0370 | CL101 | HCT 116 | C91(1.04); C92(1.04) | LDD0687 | [4] |
LDCM0371 | CL102 | HCT 116 | C91(1.19); C92(1.19) | LDD0688 | [4] |
LDCM0372 | CL103 | HCT 116 | C91(1.66); C92(1.66) | LDD0689 | [4] |
LDCM0373 | CL104 | HCT 116 | C91(1.16); C92(1.16) | LDD0690 | [4] |
LDCM0374 | CL105 | HCT 116 | C91(0.68); C92(0.68) | LDD0691 | [4] |
LDCM0375 | CL106 | HCT 116 | C91(0.63); C92(0.63) | LDD0692 | [4] |
LDCM0376 | CL107 | HCT 116 | C91(0.50); C92(0.50) | LDD0693 | [4] |
LDCM0377 | CL108 | HCT 116 | C91(1.07); C92(1.07) | LDD0694 | [4] |
LDCM0378 | CL109 | HCT 116 | C91(0.48); C92(0.48) | LDD0695 | [4] |
LDCM0379 | CL11 | HCT 116 | C91(0.76); C92(0.76) | LDD0696 | [4] |
LDCM0380 | CL110 | HCT 116 | C91(1.03); C92(1.03) | LDD0697 | [4] |
LDCM0381 | CL111 | HCT 116 | C91(0.48); C92(0.48) | LDD0698 | [4] |
LDCM0382 | CL112 | HCT 116 | C91(0.85); C92(0.85) | LDD0699 | [4] |
LDCM0383 | CL113 | HCT 116 | C91(0.68); C92(0.68) | LDD0700 | [4] |
LDCM0384 | CL114 | HCT 116 | C91(0.66); C92(0.66) | LDD0701 | [4] |
LDCM0385 | CL115 | HCT 116 | C91(0.68); C92(0.68) | LDD0702 | [4] |
LDCM0386 | CL116 | HCT 116 | C91(0.75); C92(0.75) | LDD0703 | [4] |
LDCM0387 | CL117 | HCT 116 | C83(1.00) | LDD0704 | [4] |
LDCM0388 | CL118 | HCT 116 | C83(1.08) | LDD0705 | [4] |
LDCM0389 | CL119 | HCT 116 | C83(1.08) | LDD0706 | [4] |
LDCM0390 | CL12 | HCT 116 | C91(0.75); C92(0.75) | LDD0707 | [4] |
LDCM0391 | CL120 | HCT 116 | C83(1.07) | LDD0708 | [4] |
LDCM0392 | CL121 | HCT 116 | C91(0.90); C92(0.90) | LDD0709 | [4] |
LDCM0393 | CL122 | HCT 116 | C91(0.58); C92(0.58) | LDD0710 | [4] |
LDCM0394 | CL123 | HCT 116 | C91(0.78); C92(0.78) | LDD0711 | [4] |
LDCM0395 | CL124 | HCT 116 | C91(0.63); C92(0.63) | LDD0712 | [4] |
LDCM0396 | CL125 | HCT 116 | C91(0.85); C92(0.85); C83(1.10) | LDD0713 | [4] |
LDCM0397 | CL126 | HCT 116 | C91(0.71); C92(0.71); C83(1.31) | LDD0714 | [4] |
LDCM0398 | CL127 | HCT 116 | C91(0.69); C92(0.69); C83(0.93) | LDD0715 | [4] |
LDCM0399 | CL128 | HCT 116 | C91(0.69); C92(0.69); C83(1.55) | LDD0716 | [4] |
LDCM0400 | CL13 | HCT 116 | C91(0.66); C92(0.66) | LDD0717 | [4] |
LDCM0401 | CL14 | HCT 116 | C91(0.86); C92(0.86) | LDD0718 | [4] |
LDCM0402 | CL15 | HCT 116 | C91(0.66); C92(0.66) | LDD0719 | [4] |
LDCM0403 | CL16 | HCT 116 | C91(0.78); C92(0.78) | LDD0720 | [4] |
LDCM0404 | CL17 | HCT 116 | C91(0.51); C92(0.51) | LDD0721 | [4] |
LDCM0405 | CL18 | HCT 116 | C91(0.35); C92(0.35) | LDD0722 | [4] |
LDCM0406 | CL19 | HCT 116 | C91(0.43); C92(0.43) | LDD0723 | [4] |
LDCM0407 | CL2 | HCT 116 | C91(0.95); C92(0.95) | LDD0724 | [4] |
LDCM0408 | CL20 | HCT 116 | C91(0.61); C92(0.61) | LDD0725 | [4] |
LDCM0409 | CL21 | HCT 116 | C91(0.46); C92(0.46) | LDD0726 | [4] |
LDCM0410 | CL22 | HCT 116 | C91(0.35); C92(0.35) | LDD0727 | [4] |
LDCM0411 | CL23 | HCT 116 | C91(0.69); C92(0.69) | LDD0728 | [4] |
LDCM0412 | CL24 | HCT 116 | C91(0.56); C92(0.56) | LDD0729 | [4] |
LDCM0413 | CL25 | HCT 116 | C91(0.60); C92(0.60) | LDD0730 | [4] |
LDCM0414 | CL26 | HCT 116 | C91(0.57); C92(0.57) | LDD0731 | [4] |
LDCM0415 | CL27 | HCT 116 | C91(0.79); C92(0.79) | LDD0732 | [4] |
LDCM0416 | CL28 | HCT 116 | C91(0.55); C92(0.55) | LDD0733 | [4] |
LDCM0417 | CL29 | HCT 116 | C91(0.54); C92(0.54) | LDD0734 | [4] |
LDCM0418 | CL3 | HCT 116 | C91(0.94); C92(0.94) | LDD0735 | [4] |
LDCM0419 | CL30 | HCT 116 | C91(0.75); C92(0.75) | LDD0736 | [4] |
LDCM0420 | CL31 | HCT 116 | C91(1.01); C92(1.01) | LDD0737 | [4] |
LDCM0421 | CL32 | HCT 116 | C91(0.53); C92(0.53) | LDD0738 | [4] |
LDCM0422 | CL33 | HCT 116 | C91(0.75); C92(0.75) | LDD0739 | [4] |
LDCM0423 | CL34 | HCT 116 | C91(0.58); C92(0.58) | LDD0740 | [4] |
LDCM0424 | CL35 | HCT 116 | C91(0.69); C92(0.69) | LDD0741 | [4] |
LDCM0425 | CL36 | HCT 116 | C91(0.84); C92(0.84) | LDD0742 | [4] |
LDCM0426 | CL37 | HCT 116 | C91(0.86); C92(0.86) | LDD0743 | [4] |
LDCM0428 | CL39 | HCT 116 | C91(0.68); C92(0.68) | LDD0745 | [4] |
LDCM0429 | CL4 | HCT 116 | C91(0.94); C92(0.94) | LDD0746 | [4] |
LDCM0430 | CL40 | HCT 116 | C91(0.86); C92(0.86) | LDD0747 | [4] |
LDCM0431 | CL41 | HCT 116 | C91(0.98); C92(0.98) | LDD0748 | [4] |
LDCM0432 | CL42 | HCT 116 | C91(0.72); C92(0.72) | LDD0749 | [4] |
LDCM0433 | CL43 | HCT 116 | C91(0.79); C92(0.79) | LDD0750 | [4] |
LDCM0434 | CL44 | HCT 116 | C91(0.86); C92(0.86) | LDD0751 | [4] |
LDCM0435 | CL45 | HCT 116 | C91(0.63); C92(0.63) | LDD0752 | [4] |
LDCM0436 | CL46 | HCT 116 | C91(1.00); C92(1.00) | LDD0753 | [4] |
LDCM0437 | CL47 | HCT 116 | C91(0.87); C92(0.87) | LDD0754 | [4] |
LDCM0438 | CL48 | HCT 116 | C91(0.96); C92(0.96) | LDD0755 | [4] |
LDCM0439 | CL49 | HCT 116 | C91(1.14); C92(1.14) | LDD0756 | [4] |
LDCM0440 | CL5 | HCT 116 | C91(0.84); C92(0.84) | LDD0757 | [4] |
LDCM0441 | CL50 | HCT 116 | C91(1.14); C92(1.14) | LDD0758 | [4] |
LDCM0442 | CL51 | HCT 116 | C91(1.02); C92(1.02) | LDD0759 | [4] |
LDCM0443 | CL52 | HCT 116 | C91(0.84); C92(0.84) | LDD0760 | [4] |
LDCM0444 | CL53 | HCT 116 | C91(1.02); C92(1.02) | LDD0761 | [4] |
LDCM0445 | CL54 | HCT 116 | C91(1.32); C92(1.32) | LDD0762 | [4] |
LDCM0446 | CL55 | HCT 116 | C91(1.20); C92(1.20) | LDD0763 | [4] |
LDCM0447 | CL56 | HCT 116 | C91(1.16); C92(1.16) | LDD0764 | [4] |
LDCM0448 | CL57 | HCT 116 | C91(1.21); C92(1.21) | LDD0765 | [4] |
LDCM0449 | CL58 | HCT 116 | C91(1.02); C92(1.02) | LDD0766 | [4] |
LDCM0450 | CL59 | HCT 116 | C91(1.19); C92(1.19) | LDD0767 | [4] |
LDCM0451 | CL6 | HCT 116 | C91(0.55); C92(0.55) | LDD0768 | [4] |
LDCM0452 | CL60 | HCT 116 | C91(0.97); C92(0.97) | LDD0769 | [4] |
LDCM0453 | CL61 | HCT 116 | C83(1.23); C91(1.05); C92(1.05) | LDD0770 | [4] |
LDCM0454 | CL62 | HCT 116 | C83(1.02); C91(0.95); C92(0.95) | LDD0771 | [4] |
LDCM0455 | CL63 | HCT 116 | C83(1.06); C91(0.90); C92(0.90) | LDD0772 | [4] |
LDCM0456 | CL64 | HCT 116 | C83(1.14); C91(0.90); C92(0.90) | LDD0773 | [4] |
LDCM0457 | CL65 | HCT 116 | C83(1.04); C91(0.84); C92(0.84) | LDD0774 | [4] |
LDCM0458 | CL66 | HCT 116 | C83(1.05); C91(0.63); C92(0.63) | LDD0775 | [4] |
LDCM0459 | CL67 | HCT 116 | C83(1.01); C91(0.72); C92(0.72) | LDD0776 | [4] |
LDCM0460 | CL68 | HCT 116 | C83(0.98); C91(0.57); C92(0.57) | LDD0777 | [4] |
LDCM0461 | CL69 | HCT 116 | C83(1.00); C91(0.59); C92(0.59) | LDD0778 | [4] |
LDCM0462 | CL7 | HCT 116 | C91(0.72); C92(0.72) | LDD0779 | [4] |
LDCM0463 | CL70 | HCT 116 | C83(1.06); C91(0.59); C92(0.59) | LDD0780 | [4] |
LDCM0464 | CL71 | HCT 116 | C83(1.03); C91(0.93); C92(0.93) | LDD0781 | [4] |
LDCM0465 | CL72 | HCT 116 | C83(0.90); C91(0.97); C92(0.97) | LDD0782 | [4] |
LDCM0466 | CL73 | HCT 116 | C83(1.04); C91(0.81); C92(0.81) | LDD0783 | [4] |
LDCM0467 | CL74 | HCT 116 | C83(1.02); C91(0.85); C92(0.85) | LDD0784 | [4] |
LDCM0469 | CL76 | HCT 116 | C91(1.02); C92(1.02) | LDD0786 | [4] |
LDCM0470 | CL77 | HCT 116 | C91(1.23); C92(1.23) | LDD0787 | [4] |
LDCM0471 | CL78 | HCT 116 | C91(0.85); C92(0.85) | LDD0788 | [4] |
LDCM0472 | CL79 | HCT 116 | C91(1.24); C92(1.24) | LDD0789 | [4] |
LDCM0473 | CL8 | HCT 116 | C91(0.76); C92(0.76) | LDD0790 | [4] |
LDCM0474 | CL80 | HCT 116 | C91(0.99); C92(0.99) | LDD0791 | [4] |
LDCM0475 | CL81 | HCT 116 | C91(1.48); C92(1.48) | LDD0792 | [4] |
LDCM0476 | CL82 | HCT 116 | C91(1.54); C92(1.54) | LDD0793 | [4] |
LDCM0477 | CL83 | HCT 116 | C91(1.42); C92(1.42) | LDD0794 | [4] |
LDCM0478 | CL84 | HCT 116 | C91(1.13); C92(1.13) | LDD0795 | [4] |
LDCM0479 | CL85 | HCT 116 | C91(1.01); C92(1.01) | LDD0796 | [4] |
LDCM0480 | CL86 | HCT 116 | C91(1.14); C92(1.14) | LDD0797 | [4] |
LDCM0481 | CL87 | HCT 116 | C91(1.48); C92(1.48) | LDD0798 | [4] |
LDCM0482 | CL88 | HCT 116 | C91(1.88); C92(1.88) | LDD0799 | [4] |
LDCM0483 | CL89 | HCT 116 | C91(1.11); C92(1.11) | LDD0800 | [4] |
LDCM0484 | CL9 | HCT 116 | C91(0.85); C92(0.85) | LDD0801 | [4] |
LDCM0485 | CL90 | HCT 116 | C91(1.39); C92(1.39) | LDD0802 | [4] |
LDCM0486 | CL91 | HCT 116 | C91(0.83); C92(0.83) | LDD0803 | [4] |
LDCM0487 | CL92 | HCT 116 | C91(0.71); C92(0.71) | LDD0804 | [4] |
LDCM0488 | CL93 | HCT 116 | C91(0.93); C92(0.93) | LDD0805 | [4] |
LDCM0489 | CL94 | HCT 116 | C91(0.87); C92(0.87) | LDD0806 | [4] |
LDCM0490 | CL95 | HCT 116 | C91(0.98); C92(0.98) | LDD0807 | [4] |
LDCM0491 | CL96 | HCT 116 | C91(1.01); C92(1.01) | LDD0808 | [4] |
LDCM0492 | CL97 | HCT 116 | C91(1.11); C92(1.11) | LDD0809 | [4] |
LDCM0493 | CL98 | HCT 116 | C91(0.75); C92(0.75) | LDD0810 | [4] |
LDCM0494 | CL99 | HCT 116 | C91(0.76); C92(0.76) | LDD0811 | [4] |
LDCM0495 | E2913 | HEK-293T | C83(1.13); C384(0.98); C438(0.91); C447(1.29) | LDD1698 | [15] |
LDCM0625 | F8 | Ramos | C384(1.30); C83(1.13) | LDD2187 | [16] |
LDCM0572 | Fragment10 | Ramos | C384(1.30); C83(1.06) | LDD2189 | [16] |
LDCM0573 | Fragment11 | Ramos | C384(0.71); C83(0.12); 5.89 | LDD2190 | [16] |
LDCM0574 | Fragment12 | Ramos | C384(0.93); C83(0.55) | LDD2191 | [16] |
LDCM0575 | Fragment13 | Ramos | C384(0.92); C83(0.70) | LDD2192 | [16] |
LDCM0576 | Fragment14 | Ramos | C384(1.09); C83(0.60); 1.18 | LDD2193 | [16] |
LDCM0579 | Fragment20 | Ramos | C384(1.27); C83(0.71) | LDD2194 | [16] |
LDCM0580 | Fragment21 | Ramos | C384(0.86); C83(0.83) | LDD2195 | [16] |
LDCM0582 | Fragment23 | Ramos | C384(1.16); C83(0.60) | LDD2196 | [16] |
LDCM0578 | Fragment27 | Ramos | C384(1.03); C83(0.47) | LDD2197 | [16] |
LDCM0586 | Fragment28 | Ramos | C384(0.65); C83(0.75); 0.85 | LDD2198 | [16] |
LDCM0588 | Fragment30 | Ramos | C384(1.13); C83(0.87) | LDD2199 | [16] |
LDCM0589 | Fragment31 | Ramos | C384(1.01); C83(0.84) | LDD2200 | [16] |
LDCM0590 | Fragment32 | Ramos | C384(0.99); C83(0.96) | LDD2201 | [16] |
LDCM0468 | Fragment33 | HCT 116 | C83(1.16); C91(0.82); C92(0.82) | LDD0785 | [4] |
LDCM0596 | Fragment38 | Ramos | C384(0.90); C83(0.20) | LDD2203 | [16] |
LDCM0566 | Fragment4 | Ramos | C384(0.94); C83(0.95) | LDD2184 | [16] |
LDCM0427 | Fragment51 | HCT 116 | C91(0.65); C92(0.65) | LDD0744 | [4] |
LDCM0610 | Fragment52 | Ramos | C384(1.09); C83(0.73) | LDD2204 | [16] |
LDCM0614 | Fragment56 | Ramos | C384(1.10); C83(0.97) | LDD2205 | [16] |
LDCM0569 | Fragment7 | Ramos | C384(0.97); C83(2.07) | LDD2186 | [16] |
LDCM0571 | Fragment9 | Ramos | C384(1.15); C83(1.09) | LDD2188 | [16] |
LDCM0107 | IAA | HeLa | H250(0.00); H128(0.00) | LDD0221 | [12] |
LDCM0022 | KB02 | HCT 116 | C91(9.03); C92(9.03); C83(1.24) | LDD0080 | [4] |
LDCM0023 | KB03 | HCT 116 | C91(10.36); C92(10.36); C83(1.20) | LDD0081 | [4] |
LDCM0024 | KB05 | HCT 116 | C91(4.14); C92(4.14); C83(1.14) | LDD0082 | [4] |
LDCM0109 | NEM | HeLa | H250(0.00); H128(0.00); H373(0.00) | LDD0223 | [12] |
LDCM0496 | Nucleophilic fragment 11a | MDA-MB-231 | C83(0.68) | LDD2089 | [14] |
LDCM0497 | Nucleophilic fragment 11b | MDA-MB-231 | C83(1.11) | LDD2090 | [14] |
LDCM0499 | Nucleophilic fragment 12b | MDA-MB-231 | C83(0.87) | LDD2092 | [14] |
LDCM0501 | Nucleophilic fragment 13b | MDA-MB-231 | C83(1.13) | LDD2094 | [14] |
LDCM0505 | Nucleophilic fragment 15b | MDA-MB-231 | C83(0.99) | LDD2098 | [14] |
LDCM0512 | Nucleophilic fragment 19a | MDA-MB-231 | C83(1.28) | LDD2105 | [14] |
LDCM0544 | Nucleophilic fragment 39 | MDA-MB-231 | C83(0.94) | LDD2137 | [14] |
LDCM0556 | Nucleophilic fragment 8a | MDA-MB-231 | C83(0.43) | LDD2150 | [14] |
LDCM0628 | OTUB2-COV-1 | HEK-293T | C384(1.02) | LDD2207 | [17] |
LDCM0131 | RA190 | MM1.R | C384(1.33) | LDD0304 | [18] |
The Interaction Atlas With This Target
The Protein(s) Related To This Target
Enzyme
Other
Protein name | Family | Uniprot ID | |||
---|---|---|---|---|---|
Proliferating cell nuclear antigen (PCNA) | PCNA family | P12004 | |||
DNA polymerase delta subunit 3 (POLD3) | . | Q15054 |
References