General Information of Target

Target ID LDTP12703
Target Name RNA-binding protein 28 (RBM28)
Gene Name RBM28
Gene ID 55131
Synonyms
RNA-binding protein 28; RNA-binding motif protein 28
3D Structure
Download
2D Sequence (FASTA)
Download
3D Structure (PDB)
Download
Sequence
MDVLAEEFGNLTPEQLAAPIPTVEEKWRLLPAFLKVKGLVKQHIDSFNYFINVEIKKIMK
ANEKVTSDADPMWYLKYLNIYVGLPDVEESFNVTRPVSPHECRLRDMTYSAPITVDIEYT
RGSQRIIRNALPIGRMPIMLRSSNCVLTGKTPAEFAKLNECPLDPGGYFIVKGVEKVILI
QEQLSKNRIIVEADRKGAVGASVTSSTHEKKSRTNMAVKQGRFYLRHNTLSEDIPIVIIF
KAMGVESDQEIVQMIGTEEHVMAAFGPSLEECQKAQIFTQMQALKYIGNKVRRQRMWGGG
PKKTKIEEARELLASTILTHVPVKEFNFRAKCIYTAVMVRRVILAQGDNKVDDRDYYGNK
RLELAGQLLSLLFEDLFKKFNSEMKKIADQVIPKQRAAQFDVVKHMRQDQITNGMVNAIS
TGNWSLKRFKMDRQGVTQVLSRLSYISALGMMTRISSQFEKTRKVSGPRSLQPSQWGMLC
PSDTPEGEACGLVKNLALMTHITTDMEDGPIVKLASNLGVEDVNLLCGEELSYPNVFLVF
LNGNILGVIRDHKKLVNTFRLMRRAGYINEFVSISTNLTDRCVYISSDGGRLCRPYIIVK
KQKPAVTNKHMEELAQGYRNFEDFLHESLVEYLDVNEENDCNIALYEHTINKDTTHLEIE
PFTLLGVCAGLIPYPHHNQSPRNTYQCAMGKQAMGTIGYNQRNRIDTLMYLLAYPQKPMV
KTKTIELIEFEKLPAGQNATVAVMSYSGYDIEDALVLNKASLDRGFGRCLVYKNAKCTLK
RYTNQTFDKVMGPMLDAATRKPIWRHEILDADGICSPGEKVENKQVLVNKSMPTVTQIPL
EGSNVPQQPQYKDVPITYKGATDSYIEKVMISSNAEDAFLIKMLLRQTRRPEIGDKFSSR
HGQKGVCGLIVPQEDMPFCDSGICPDIIMNPHGFPSRMTVGKLIELLAGKAGVLDGRFHY
GTAFGGSKVKDVCEDLVRHGYNYLGKDYVTSGITGEPLEAYIYFGPVYYQKLKHMVLDKM
HARARGPRAVLTRQPTEGRSRDGGLRLGEMERDCLIGYGASMLLLERLMISSDAFEVDVC
GQCGLLGYSGWCHYCKSSCHVSSLRIPYACKLLFQELQSMNIIPRLKLSKYNE
Target Bioclass
Other
Subcellular location
Nucleus, nucleolus
Function Nucleolar component of the spliceosomal ribonucleoprotein complexes.
Uniprot ID
Q9NW13
Ensemble ID
ENST00000223073.6
HGNC ID
HGNC:21863

Target Site Mutations in Different Cell Lines

Cell line Mutation details Probe for labeling this protein in this cell
AGS SNV: p.M174L; p.K177T DBIA    Probe Info 
G415 SNV: p.P603T DBIA    Probe Info 
HT115 SNV: p.D527Y DBIA    Probe Info 
IM95 Deletion: p.A721LfsTer69 DBIA    Probe Info 
LS180 Deletion: p.L554SfsTer12 DBIA    Probe Info 
MDAMB453 SNV: p.R640T DBIA    Probe Info 
SG231 SNV: p.D251E DBIA    Probe Info 

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 24 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
m-APA
 Probe Info 
9.94  LDD0402  [1]
BTD
 Probe Info 
C97(0.69)  LDD2092  [2]
DBIA
 Probe Info 
C97(1.28); C71(1.06)  LDD0078  [3]
ATP probe
 Probe Info 
K496(0.00); K501(0.00); K505(0.00); K478(0.00)  LDD0199  [4]
4-Iodoacetamidophenylacetylene
 Probe Info 
C392(0.00); C125(0.00); C71(0.00); C490(0.00)  LDD0038  [5]
IA-alkyne
 Probe Info 
C71(0.00); C33(0.00)  LDD0032  [6]
IPIAA_L
 Probe Info 
N.A.  LDD0031  [7]
Lodoacetamide azide
 Probe Info 
C392(0.00); C125(0.00); C71(0.00); C490(0.00)  LDD0037  [5]
WYneN
 Probe Info 
N.A.  LDD0021  [8]
Compound 10
 Probe Info 
C33(0.00); C71(0.00)  LDD2216  [9]
ENE
 Probe Info 
N.A.  LDD0006  [8]
IPM
 Probe Info 
N.A.  LDD0005  [8]
NHS
 Probe Info 
K505(0.00); K478(0.00)  LDD0010  [8]
SF
 Probe Info 
K196(0.00); Y737(0.00)  LDD0028  [10]
STPyne
 Probe Info 
N.A.  LDD0009  [8]
TFBX
 Probe Info 
C97(0.00); C490(0.00); C125(0.00); C71(0.00)  LDD0148  [11]
VSF
 Probe Info 
N.A.  LDD0007  [8]
Phosphinate-6
 Probe Info 
N.A.  LDD0018  [12]
1c-yne
 Probe Info 
N.A.  LDD0228  [13]
Acrolein
 Probe Info 
C71(0.00); C490(0.00); C97(0.00); H369(0.00)  LDD0217  [14]
Crotonaldehyde
 Probe Info 
N.A.  LDD0219  [14]
Methacrolein
 Probe Info 
C490(0.00); C97(0.00); C71(0.00)  LDD0218  [14]
W1
 Probe Info 
C71(0.00); C97(0.00)  LDD0236  [15]
NAIA_5
 Probe Info 
C71(0.00); C392(0.00); C490(0.00)  LDD2223  [16]
PAL-AfBPP Probe
Click To Hide/Show 2 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
FFF probe3
 Probe Info 
12.25  LDD0464  [17]
STS-1
 Probe Info 
N.A.  LDD0137  [18]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0548  1-(4-(Benzo[d][1,3]dioxol-5-ylmethyl)piperazin-1-yl)-2-nitroethan-1-one MDA-MB-231 C97(0.98)  LDD2142  [2]
 LDCM0524  2-Cyano-N-(2-morpholin-4-yl-ethyl)-acetamide MDA-MB-231 C97(1.16)  LDD2117  [2]
 LDCM0558  2-Cyano-N-phenylacetamide MDA-MB-231 C125(1.98)  LDD2152  [2]
 LDCM0214  AC1 HCT 116 C125(1.20); C33(1.30); C490(0.93); C71(1.22)  LDD0531  [3]
 LDCM0215  AC10 HCT 116 C125(0.98); C33(0.89); C490(1.32); C71(1.44)  LDD0532  [3]
 LDCM0216  AC100 HCT 116 C33(0.76); C490(1.64); C71(1.31); C97(1.33)  LDD0533  [3]
 LDCM0217  AC101 HCT 116 C33(0.81); C490(1.55); C71(1.47); C97(1.51)  LDD0534  [3]
 LDCM0218  AC102 HCT 116 C33(0.85); C490(1.50); C71(0.85); C97(1.24)  LDD0535  [3]
 LDCM0219  AC103 HCT 116 C33(0.69); C490(0.99); C71(1.24); C97(1.41)  LDD0536  [3]
 LDCM0220  AC104 HCT 116 C33(1.06); C490(1.17); C71(1.30); C97(1.30)  LDD0537  [3]
 LDCM0221  AC105 HCT 116 C33(0.85); C490(1.15); C71(1.10); C97(1.60)  LDD0538  [3]
 LDCM0222  AC106 HCT 116 C33(0.73); C490(1.14); C71(1.35); C97(1.78)  LDD0539  [3]
 LDCM0223  AC107 HCT 116 C33(0.76); C490(1.10); C71(1.22); C97(1.49)  LDD0540  [3]
 LDCM0224  AC108 HCT 116 C33(0.77); C490(0.83); C71(1.18); C97(1.36)  LDD0541  [3]
 LDCM0225  AC109 HCT 116 C33(1.11); C490(0.82); C71(0.99); C97(0.88)  LDD0542  [3]
 LDCM0226  AC11 HCT 116 C125(0.99); C33(0.91); C490(1.19); C71(1.41)  LDD0543  [3]
 LDCM0227  AC110 HCT 116 C33(0.70); C490(0.83); C71(1.21); C97(1.20)  LDD0544  [3]
 LDCM0228  AC111 HCT 116 C33(0.67); C490(0.89); C71(1.29); C97(1.54)  LDD0545  [3]
 LDCM0229  AC112 HCT 116 C33(0.72); C490(1.06); C71(1.05); C97(1.40)  LDD0546  [3]
 LDCM0230  AC113 HCT 116 C125(0.95); C33(1.22); C490(1.06); C71(1.17)  LDD0547  [3]
 LDCM0231  AC114 HCT 116 C125(1.06); C33(0.88); C490(1.41); C71(1.04)  LDD0548  [3]
 LDCM0232  AC115 HCT 116 C125(1.10); C33(0.88); C490(1.23); C71(1.09)  LDD0549  [3]
 LDCM0233  AC116 HCT 116 C125(1.09); C33(0.86); C490(1.11); C71(0.98)  LDD0550  [3]
 LDCM0234  AC117 HCT 116 C125(1.08); C33(1.35); C490(1.25); C71(1.14)  LDD0551  [3]
 LDCM0235  AC118 HCT 116 C125(1.02); C33(1.12); C490(1.29); C71(1.05)  LDD0552  [3]
 LDCM0236  AC119 HCT 116 C125(1.07); C33(0.98); C490(1.28); C71(1.24)  LDD0553  [3]
 LDCM0237  AC12 HCT 116 C125(0.71); C33(0.99); C490(1.12); C71(1.22)  LDD0554  [3]
 LDCM0238  AC120 HCT 116 C125(0.93); C33(0.82); C490(1.18); C71(1.00)  LDD0555  [3]
 LDCM0239  AC121 HCT 116 C125(0.99); C33(1.59); C490(1.12); C71(1.02)  LDD0556  [3]
 LDCM0240  AC122 HCT 116 C125(0.96); C33(0.82); C490(1.15); C71(1.03)  LDD0557  [3]
 LDCM0241  AC123 HCT 116 C125(0.75); C33(1.87); C490(0.94); C71(0.95)  LDD0558  [3]
 LDCM0242  AC124 HCT 116 C125(0.95); C33(1.27); C490(1.02); C71(0.98)  LDD0559  [3]
 LDCM0243  AC125 HCT 116 C125(1.00); C33(0.77); C490(1.21); C71(1.05)  LDD0560  [3]
 LDCM0244  AC126 HCT 116 C125(0.91); C33(0.84); C490(1.05); C71(1.00)  LDD0561  [3]
 LDCM0245  AC127 HCT 116 C125(0.86); C33(1.08); C490(1.06); C71(0.95)  LDD0562  [3]
 LDCM0246  AC128 HCT 116 C33(1.38); C71(0.93); C97(1.73)  LDD0563  [3]
 LDCM0247  AC129 HCT 116 C33(1.59); C71(0.96); C97(1.58)  LDD0564  [3]
 LDCM0249  AC130 HCT 116 C33(1.26); C71(1.15); C97(1.91)  LDD0566  [3]
 LDCM0250  AC131 HCT 116 C33(1.26); C71(0.96); C97(1.08)  LDD0567  [3]
 LDCM0251  AC132 HCT 116 C33(1.18); C71(0.97); C97(1.74)  LDD0568  [3]
 LDCM0252  AC133 HCT 116 C33(1.22); C71(1.12); C97(1.52)  LDD0569  [3]
 LDCM0253  AC134 HCT 116 C33(1.07); C71(1.33); C97(1.61)  LDD0570  [3]
 LDCM0254  AC135 HCT 116 C33(1.27); C71(1.16); C97(1.78)  LDD0571  [3]
 LDCM0255  AC136 HCT 116 C33(1.34); C71(1.15); C97(1.57)  LDD0572  [3]
 LDCM0256  AC137 HCT 116 C33(1.29); C71(0.96); C97(1.48)  LDD0573  [3]
 LDCM0257  AC138 HCT 116 C33(0.97); C71(1.17); C97(2.03)  LDD0574  [3]
 LDCM0258  AC139 HCT 116 C33(1.24); C71(1.14); C97(1.62)  LDD0575  [3]
 LDCM0259  AC14 HCT 116 C125(0.77); C33(1.08); C490(1.34); C71(1.28)  LDD0576  [3]
 LDCM0260  AC140 HCT 116 C33(1.17); C71(1.37); C97(1.90)  LDD0577  [3]
 LDCM0261  AC141 HCT 116 C33(1.06); C71(1.26); C97(1.65)  LDD0578  [3]
 LDCM0262  AC142 HCT 116 C33(1.27); C71(1.53); C97(1.46)  LDD0579  [3]
 LDCM0263  AC143 HCT 116 C378(0.90); C33(1.00); C97(1.08); C71(1.15)  LDD0580  [3]
 LDCM0264  AC144 HCT 116 C378(0.68); C97(0.97); C71(0.99); C33(1.15)  LDD0581  [3]
 LDCM0265  AC145 HCT 116 C33(0.82); C378(0.85); C97(0.95); C71(1.37)  LDD0582  [3]
 LDCM0266  AC146 HCT 116 C378(0.77); C33(0.81); C97(0.94); C71(1.16)  LDD0583  [3]
 LDCM0267  AC147 HCT 116 C378(0.60); C33(0.79); C97(0.94); C71(1.18)  LDD0584  [3]
 LDCM0268  AC148 HCT 116 C378(0.35); C33(0.83); C97(0.85); C490(1.09)  LDD0585  [3]
 LDCM0269  AC149 HCT 116 C378(0.59); C33(0.82); C97(1.06); C71(1.11)  LDD0586  [3]
 LDCM0270  AC15 HCT 116 C125(0.75); C33(0.89); C97(1.00); C71(1.16)  LDD0587  [3]
 LDCM0271  AC150 HCT 116 C378(0.88); C97(1.08); C71(1.15); C33(1.81)  LDD0588  [3]
 LDCM0272  AC151 HCT 116 C33(0.85); C378(0.89); C71(1.14); C97(1.25)  LDD0589  [3]
 LDCM0273  AC152 HCT 116 C378(0.54); C33(0.84); C97(0.92); C71(1.02)  LDD0590  [3]
 LDCM0274  AC153 HCT 116 C378(0.35); C97(0.94); C33(1.00); C490(1.20)  LDD0591  [3]
 LDCM0621  AC154 HCT 116 C33(1.06); C378(0.72); C490(1.50); C71(1.11)  LDD2158  [3]
 LDCM0622  AC155 HCT 116 C33(0.70); C378(0.77); C490(1.51); C71(1.02)  LDD2159  [3]
 LDCM0623  AC156 HCT 116 C33(1.61); C378(0.83); C490(1.24); C71(0.83)  LDD2160  [3]
 LDCM0624  AC157 HCT 116 C33(0.76); C378(0.87); C490(0.89); C71(1.01)  LDD2161  [3]
 LDCM0276  AC17 HCT 116 C71(1.02); C97(1.03); C125(1.05); C378(1.07)  LDD0593  [3]
 LDCM0277  AC18 HCT 116 C378(0.80); C125(0.86); C71(1.05); C97(1.24)  LDD0594  [3]
 LDCM0278  AC19 HCT 116 C378(0.80); C125(0.83); C490(0.91); C71(0.96)  LDD0595  [3]
 LDCM0279  AC2 HCT 116 C490(0.84); C33(1.07); C71(1.15); C97(1.25)  LDD0596  [3]
 LDCM0280  AC20 HCT 116 C125(0.90); C33(0.97); C97(1.00); C378(1.02)  LDD0597  [3]
 LDCM0281  AC21 HCT 116 C125(0.78); C71(0.99); C378(0.99); C97(1.03)  LDD0598  [3]
 LDCM0282  AC22 HCT 116 C125(0.81); C378(0.89); C33(0.92); C97(0.94)  LDD0599  [3]
 LDCM0283  AC23 HCT 116 C378(0.79); C125(0.79); C71(0.97); C33(1.04)  LDD0600  [3]
 LDCM0284  AC24 HCT 116 C97(0.86); C71(0.91); C33(0.93); C125(0.96)  LDD0601  [3]
 LDCM0285  AC25 HCT 116 C125(0.57); C33(0.94); C71(0.95); C97(1.14)  LDD0602  [3]
 LDCM0286  AC26 HCT 116 C125(0.50); C33(0.71); C71(1.05); C97(1.32)  LDD0603  [3]
 LDCM0287  AC27 HCT 116 C125(0.69); C33(0.71); C71(1.01); C490(1.25)  LDD0604  [3]
 LDCM0288  AC28 HCT 116 C125(0.62); C33(0.66); C71(1.00); C490(1.17)  LDD0605  [3]
 LDCM0289  AC29 HCT 116 C33(0.66); C125(0.77); C71(1.02); C490(1.20)  LDD0606  [3]
 LDCM0290  AC3 HCT 116 C490(0.94); C33(1.04); C71(1.18); C97(1.24)  LDD0607  [3]
 LDCM0291  AC30 HCT 116 C33(0.68); C125(0.74); C71(1.19); C97(1.26)  LDD0608  [3]
 LDCM0292  AC31 HCT 116 C33(0.71); C125(0.83); C71(1.08); C490(1.34)  LDD0609  [3]
 LDCM0293  AC32 HCT 116 C33(0.65); C125(0.80); C490(1.10); C71(1.15)  LDD0610  [3]
 LDCM0294  AC33 HCT 116 C33(0.66); C125(0.66); C490(1.01); C71(1.06)  LDD0611  [3]
 LDCM0295  AC34 HCT 116 C125(0.50); C33(0.56); C490(0.86); C71(1.10)  LDD0612  [3]
 LDCM0296  AC35 HCT 116 C97(0.71); C71(0.96); C125(1.10); C33(1.11)  LDD0613  [3]
 LDCM0297  AC36 HCT 116 C97(0.84); C125(1.03); C33(1.05); C71(1.11)  LDD0614  [3]
 LDCM0298  AC37 HCT 116 C71(1.04); C125(1.06); C97(1.14); C378(1.18)  LDD0615  [3]
 LDCM0299  AC38 HCT 116 C97(0.84); C71(0.92); C33(1.01); C125(1.10)  LDD0616  [3]
 LDCM0300  AC39 HCT 116 C378(0.85); C97(0.89); C33(0.98); C125(0.99)  LDD0617  [3]
 LDCM0301  AC4 HCT 116 C490(0.84); C33(0.97); C71(1.27); C97(1.50)  LDD0618  [3]
 LDCM0302  AC40 HCT 116 C378(0.58); C490(0.85); C71(0.90); C33(1.04)  LDD0619  [3]
 LDCM0303  AC41 HCT 116 C71(1.00); C33(1.09); C97(1.10); C378(1.18)  LDD0620  [3]
 LDCM0304  AC42 HCT 116 C378(0.92); C33(1.01); C97(1.03); C71(1.04)  LDD0621  [3]
 LDCM0305  AC43 HCT 116 C33(0.98); C71(1.04); C378(1.12); C97(1.30)  LDD0622  [3]
 LDCM0306  AC44 HCT 116 C378(0.85); C97(0.90); C71(0.97); C490(1.08)  LDD0623  [3]
 LDCM0307  AC45 HCT 116 C378(0.58); C490(0.91); C71(1.04); C97(1.06)  LDD0624  [3]
 LDCM0308  AC46 HCT 116 C33(0.98); C378(1.01); C71(1.09); C125(1.18)  LDD0625  [3]
 LDCM0309  AC47 HCT 116 C378(0.93); C33(0.99); C71(1.03); C490(1.06)  LDD0626  [3]
 LDCM0310  AC48 HCT 116 C33(1.08); C71(1.17); C125(1.21); C378(1.36)  LDD0627  [3]
 LDCM0311  AC49 HCT 116 C378(0.35); C33(0.81); C490(0.91); C125(1.00)  LDD0628  [3]
 LDCM0312  AC5 HCT 116 C490(0.86); C33(1.13); C71(1.35); C97(1.49)  LDD0629  [3]
 LDCM0313  AC50 HCT 116 C378(0.43); C33(0.78); C490(0.88); C125(1.04)  LDD0630  [3]
 LDCM0314  AC51 HCT 116 C125(0.93); C33(0.96); C71(1.00); C97(1.03)  LDD0631  [3]
 LDCM0315  AC52 HCT 116 C33(0.90); C378(0.99); C490(1.02); C71(1.06)  LDD0632  [3]
 LDCM0316  AC53 HCT 116 C378(0.59); C490(0.73); C33(0.87); C71(1.05)  LDD0633  [3]
 LDCM0317  AC54 HCT 116 C378(0.62); C33(0.88); C490(0.88); C71(0.99)  LDD0634  [3]
 LDCM0318  AC55 HCT 116 C378(0.38); C490(0.73); C33(0.90); C71(1.10)  LDD0635  [3]
 LDCM0319  AC56 HCT 116 C378(0.30); C490(0.80); C33(0.82); C125(1.06)  LDD0636  [3]
 LDCM0320  AC57 HCT 116 C71(1.05); C490(1.08); C33(1.20); C125(1.26)  LDD0637  [3]
 LDCM0321  AC58 HCT 116 C125(0.89); C71(0.97); C33(0.97); C490(1.00)  LDD0638  [3]
 LDCM0322  AC59 HCT 116 C490(1.15); C33(1.18); C71(1.21); C125(1.61)  LDD0639  [3]
 LDCM0323  AC6 HCT 116 C33(0.81); C125(0.99); C71(1.24); C490(1.36)  LDD0640  [3]
 LDCM0324  AC60 HCT 116 C33(1.04); C125(1.05); C490(1.06); C71(1.16)  LDD0641  [3]
 LDCM0325  AC61 HCT 116 C490(0.93); C33(1.12); C71(1.12); C125(1.48)  LDD0642  [3]
 LDCM0326  AC62 HCT 116 C490(0.99); C71(1.08); C125(1.08); C33(1.27)  LDD0643  [3]
 LDCM0327  AC63 HCT 116 C490(0.88); C71(0.99); C33(1.24); C125(1.43)  LDD0644  [3]
 LDCM0328  AC64 HCT 116 C490(0.88); C71(1.18); C125(1.26); C33(1.35)  LDD0645  [3]
 LDCM0329  AC65 HCT 116 C490(0.93); C71(0.95); C33(1.22); C125(1.39)  LDD0646  [3]
 LDCM0330  AC66 HCT 116 C71(0.87); C490(0.89); C33(1.19); C125(1.42)  LDD0647  [3]
 LDCM0331  AC67 HCT 116 C490(0.89); C33(1.02); C71(1.12); C125(1.39)  LDD0648  [3]
 LDCM0332  AC68 HCT 116 C378(0.67); C490(0.78); C125(0.85); C33(0.95)  LDD0649  [3]
 LDCM0333  AC69 HCT 116 C378(0.64); C490(0.79); C125(0.79); C71(0.91)  LDD0650  [3]
 LDCM0334  AC7 HCT 116 C33(1.00); C125(1.04); C71(1.15); C490(1.40)  LDD0651  [3]
 LDCM0335  AC70 HCT 116 C378(0.33); C125(0.66); C490(0.79); C33(0.82)  LDD0652  [3]
 LDCM0336  AC71 HCT 116 C71(0.93); C490(0.94); C378(1.05); C125(1.06)  LDD0653  [3]
 LDCM0337  AC72 HCT 116 C378(0.61); C125(0.82); C490(0.83); C33(0.87)  LDD0654  [3]
 LDCM0338  AC73 HCT 116 C378(0.29); C125(0.75); C490(0.79); C33(0.86)  LDD0655  [3]
 LDCM0339  AC74 HCT 116 C378(0.30); C125(0.79); C490(0.80); C33(0.96)  LDD0656  [3]
 LDCM0340  AC75 HCT 116 C378(0.26); C125(0.76); C490(0.81); C33(0.91)  LDD0657  [3]
 LDCM0341  AC76 HCT 116 C378(0.41); C490(0.68); C33(0.85); C125(0.85)  LDD0658  [3]
 LDCM0342  AC77 HCT 116 C378(0.39); C490(0.72); C125(0.80); C33(0.84)  LDD0659  [3]
 LDCM0343  AC78 HCT 116 C71(0.95); C97(0.96); C490(0.98); C125(1.02)  LDD0660  [3]
 LDCM0344  AC79 HCT 116 C378(0.73); C490(0.83); C71(0.88); C33(0.95)  LDD0661  [3]
 LDCM0345  AC8 HCT 116 C33(0.86); C125(1.02); C97(1.18); C71(1.21)  LDD0662  [3]
 LDCM0346  AC80 HCT 116 C378(0.59); C490(0.74); C125(0.77); C33(0.91)  LDD0663  [3]
 LDCM0347  AC81 HCT 116 C125(0.81); C490(0.99); C71(1.00); C378(1.05)  LDD0664  [3]
 LDCM0348  AC82 HCT 116 C378(0.26); C125(0.66); C490(0.81); C33(0.91)  LDD0665  [3]
 LDCM0349  AC83 HCT 116 C33(0.65); C125(0.74); C71(0.88); C490(1.06)  LDD0666  [3]
 LDCM0350  AC84 HCT 116 C33(0.73); C125(0.73); C71(0.85); C490(1.12)  LDD0667  [3]
 LDCM0351  AC85 HCT 116 C33(0.94); C71(1.01); C125(1.17); C97(1.42)  LDD0668  [3]
 LDCM0352  AC86 HCT 116 C33(0.79); C71(0.89); C125(0.98); C97(1.31)  LDD0669  [3]
 LDCM0353  AC87 HCT 116 C125(1.01); C71(1.01); C490(1.06); C97(1.15)  LDD0670  [3]
 LDCM0354  AC88 HCT 116 C33(0.76); C71(0.80); C125(0.87); C97(1.20)  LDD0671  [3]
 LDCM0355  AC89 HCT 116 C33(0.60); C125(0.95); C71(0.97); C490(1.10)  LDD0672  [3]
 LDCM0357  AC90 HCT 116 C125(1.11); C490(1.16); C71(1.23); C33(1.32)  LDD0674  [3]
 LDCM0358  AC91 HCT 116 C33(0.66); C125(0.76); C490(0.85); C71(0.95)  LDD0675  [3]
 LDCM0359  AC92 HCT 116 C33(0.64); C125(0.86); C71(0.93); C490(1.02)  LDD0676  [3]
 LDCM0360  AC93 HCT 116 C71(0.83); C125(0.84); C33(0.92); C97(1.09)  LDD0677  [3]
 LDCM0361  AC94 HCT 116 C71(0.81); C33(0.85); C125(0.87); C97(1.11)  LDD0678  [3]
 LDCM0362  AC95 HCT 116 C71(0.89); C490(0.94); C125(0.99); C33(1.12)  LDD0679  [3]
 LDCM0363  AC96 HCT 116 C33(0.70); C71(0.89); C125(0.97); C490(1.27)  LDD0680  [3]
 LDCM0364  AC97 HCT 116 C33(0.55); C71(0.83); C125(0.90); C490(0.99)  LDD0681  [3]
 LDCM0365  AC98 HCT 116 C33(0.69); C490(0.93); C71(1.62); C97(1.73)  LDD0682  [3]
 LDCM0366  AC99 HCT 116 C33(0.80); C71(1.24); C97(1.28); C490(1.39)  LDD0683  [3]
 LDCM0248  AKOS034007472 HCT 116 C125(0.85); C33(1.12); C490(1.22); C71(1.15)  LDD0565  [3]
 LDCM0356  AKOS034007680 HCT 116 C33(0.93); C125(1.04); C97(1.13); C71(1.25)  LDD0673  [3]
 LDCM0275  AKOS034007705 HCT 116 C33(0.67); C125(0.86); C490(1.02); C71(1.33)  LDD0592  [3]
 LDCM0020  ARS-1620 HCC44 C97(1.28); C71(1.06)  LDD0078  [3]
 LDCM0108  Chloroacetamide HeLa N.A.  LDD0222  [14]
 LDCM0632  CL-Sc Hep-G2 C97(0.74)  LDD2227  [16]
 LDCM0367  CL1 HCT 116 C490(0.95); C71(1.08); C97(1.11); C33(1.12)  LDD0684  [3]
 LDCM0368  CL10 HCT 116 C490(0.86); C33(0.93); C71(1.22); C97(1.53)  LDD0685  [3]
 LDCM0369  CL100 HCT 116 C33(1.04); C490(1.08); C125(1.19); C71(1.25)  LDD0686  [3]
 LDCM0370  CL101 HCT 116 C33(0.79); C125(0.87); C71(1.25); C97(1.25)  LDD0687  [3]
 LDCM0371  CL102 HCT 116 C33(1.00); C125(1.01); C97(1.06); C71(1.15)  LDD0688  [3]
 LDCM0372  CL103 HCT 116 C71(0.99); C33(1.00); C97(1.19); C490(1.21)  LDD0689  [3]
 LDCM0373  CL104 HCT 116 C33(0.91); C71(1.04); C125(1.10); C490(1.34)  LDD0690  [3]
 LDCM0374  CL105 HCT 116 C378(0.81); C71(0.94); C97(1.08); C125(1.12)  LDD0691  [3]
 LDCM0375  CL106 HCT 116 C378(0.70); C125(1.02); C71(1.11); C33(1.37)  LDD0692  [3]
 LDCM0376  CL107 HCT 116 C378(0.58); C125(0.99); C490(1.08); C71(1.11)  LDD0693  [3]
 LDCM0377  CL108 HCT 116 C378(0.48); C490(0.93); C125(1.09); C71(1.12)  LDD0694  [3]
 LDCM0378  CL109 HCT 116 C378(0.79); C125(0.83); C71(0.94); C33(1.00)  LDD0695  [3]
 LDCM0379  CL11 HCT 116 C490(0.71); C33(0.91); C71(1.06); C97(1.63)  LDD0696  [3]
 LDCM0380  CL110 HCT 116 C378(0.68); C125(0.84); C71(0.95); C33(1.05)  LDD0697  [3]
 LDCM0381  CL111 HCT 116 C378(0.75); C125(0.81); C33(0.96); C97(1.14)  LDD0698  [3]
 LDCM0382  CL112 HCT 116 C125(0.61); C33(0.79); C71(0.96); C490(1.15)  LDD0699  [3]
 LDCM0383  CL113 HCT 116 C125(0.60); C33(0.60); C490(1.09); C71(1.13)  LDD0700  [3]
 LDCM0384  CL114 HCT 116 C125(0.58); C33(0.63); C71(1.05); C490(1.44)  LDD0701  [3]
 LDCM0385  CL115 HCT 116 C125(0.61); C33(0.63); C71(1.07); C97(1.25)  LDD0702  [3]
 LDCM0386  CL116 HCT 116 C125(0.55); C33(0.72); C71(0.98); C490(1.47)  LDD0703  [3]
 LDCM0387  CL117 HCT 116 C378(0.39); C490(0.96); C71(1.03); C33(1.06)  LDD0704  [3]
 LDCM0388  CL118 HCT 116 C378(0.85); C97(0.92); C33(0.98); C71(1.00)  LDD0705  [3]
 LDCM0389  CL119 HCT 116 C378(0.78); C490(0.93); C33(0.98); C71(1.06)  LDD0706  [3]
 LDCM0390  CL12 HCT 116 C490(0.71); C33(0.88); C71(1.16); C97(1.65)  LDD0707  [3]
 LDCM0391  CL120 HCT 116 C33(0.96); C71(0.99); C97(1.10); C378(1.16)  LDD0708  [3]
 LDCM0392  CL121 HCT 116 C378(0.59); C33(0.73); C490(0.93); C125(1.19)  LDD0709  [3]
 LDCM0393  CL122 HCT 116 C33(0.90); C125(1.02); C378(1.09); C71(1.10)  LDD0710  [3]
 LDCM0394  CL123 HCT 116 C378(0.50); C33(0.79); C490(0.79); C71(1.07)  LDD0711  [3]
 LDCM0395  CL124 HCT 116 C378(0.44); C33(0.78); C490(0.84); C71(1.04)  LDD0712  [3]
 LDCM0396  CL125 HCT 116 C71(1.08); C490(1.12); C125(1.12); C33(1.18)  LDD0713  [3]
 LDCM0397  CL126 HCT 116 C33(1.05); C71(1.13); C490(1.14); C125(1.21)  LDD0714  [3]
 LDCM0398  CL127 HCT 116 C33(1.05); C71(1.13); C490(1.21); C125(1.24)  LDD0715  [3]
 LDCM0399  CL128 HCT 116 C125(1.00); C33(1.02); C490(1.14); C71(1.26)  LDD0716  [3]
 LDCM0400  CL13 HCT 116 C490(0.91); C71(1.02); C33(1.07); C97(1.27)  LDD0717  [3]
 LDCM0401  CL14 HCT 116 C490(0.88); C33(1.01); C71(1.09); C97(1.15)  LDD0718  [3]
 LDCM0402  CL15 HCT 116 C490(0.86); C71(0.87); C33(1.06); C97(1.35)  LDD0719  [3]
 LDCM0403  CL16 HCT 116 C33(0.89); C378(0.98); C490(1.03); C71(1.17)  LDD0720  [3]
 LDCM0404  CL17 HCT 116 C71(0.89); C378(0.91); C33(0.92); C490(1.19)  LDD0721  [3]
 LDCM0405  CL18 HCT 116 C71(0.98); C490(1.06); C33(1.06); C125(1.24)  LDD0722  [3]
 LDCM0406  CL19 HCT 116 C378(0.85); C71(0.95); C125(0.97); C33(1.00)  LDD0723  [3]
 LDCM0407  CL2 HCT 116 C490(1.00); C71(1.02); C97(1.14); C33(1.18)  LDD0724  [3]
 LDCM0408  CL20 HCT 116 C378(0.59); C490(0.84); C33(0.87); C71(1.04)  LDD0725  [3]
 LDCM0409  CL21 HCT 116 C378(0.39); C33(0.72); C490(0.81); C71(0.90)  LDD0726  [3]
 LDCM0410  CL22 HCT 116 C378(0.22); C490(0.85); C33(0.89); C125(0.95)  LDD0727  [3]
 LDCM0411  CL23 HCT 116 C378(0.65); C33(0.86); C490(0.91); C125(0.95)  LDD0728  [3]
 LDCM0412  CL24 HCT 116 C125(1.09); C33(0.78); C378(0.32); C490(0.83)  LDD0729  [3]
 LDCM0413  CL25 HCT 116 C125(1.18); C33(0.84); C378(0.39); C490(0.92)  LDD0730  [3]
 LDCM0414  CL26 HCT 116 C125(1.12); C33(0.96); C378(0.67); C490(0.95)  LDD0731  [3]
 LDCM0415  CL27 HCT 116 C125(1.07); C33(0.91); C378(0.64); C490(0.97)  LDD0732  [3]
 LDCM0416  CL28 HCT 116 C125(1.26); C33(0.85); C378(0.63); C490(0.94)  LDD0733  [3]
 LDCM0417  CL29 HCT 116 C125(1.04); C33(0.86); C378(0.57); C490(0.86)  LDD0734  [3]
 LDCM0418  CL3 HCT 116 C33(0.98); C490(0.88); C71(0.96); C97(1.03)  LDD0735  [3]
 LDCM0419  CL30 HCT 116 C125(1.09); C33(0.98); C378(0.84); C490(0.99)  LDD0736  [3]
 LDCM0420  CL31 HCT 116 C125(1.02); C33(0.78); C490(0.99); C71(0.93)  LDD0737  [3]
 LDCM0421  CL32 HCT 116 C125(0.91); C33(0.98); C490(0.90); C71(1.07)  LDD0738  [3]
 LDCM0422  CL33 HCT 116 C125(0.81); C33(0.74); C490(1.06); C71(1.04)  LDD0739  [3]
 LDCM0423  CL34 HCT 116 C125(0.89); C33(0.78); C490(0.90); C71(1.05)  LDD0740  [3]
 LDCM0424  CL35 HCT 116 C125(0.93); C33(0.66); C490(0.96); C71(1.05)  LDD0741  [3]
 LDCM0425  CL36 HCT 116 C125(0.92); C33(0.67); C490(0.98); C71(0.98)  LDD0742  [3]
 LDCM0426  CL37 HCT 116 C125(0.70); C33(0.63); C490(0.87); C71(1.05)  LDD0743  [3]
 LDCM0428  CL39 HCT 116 C125(0.72); C33(0.66); C490(0.74); C71(0.96)  LDD0745  [3]
 LDCM0429  CL4 HCT 116 C33(0.84); C490(0.82); C71(0.93); C97(1.11)  LDD0746  [3]
 LDCM0430  CL40 HCT 116 C125(0.72); C33(0.58); C490(0.66); C71(0.90)  LDD0747  [3]
 LDCM0431  CL41 HCT 116 C125(1.01); C33(0.71); C490(0.76); C71(0.93)  LDD0748  [3]
 LDCM0432  CL42 HCT 116 C125(0.78); C33(0.60); C490(0.76); C71(0.97)  LDD0749  [3]
 LDCM0433  CL43 HCT 116 C125(0.89); C33(0.64); C490(0.70); C71(0.94)  LDD0750  [3]
 LDCM0434  CL44 HCT 116 C125(0.85); C33(0.71); C490(0.84); C71(0.98)  LDD0751  [3]
 LDCM0435  CL45 HCT 116 C125(1.35); C33(0.67); C490(0.88); C71(0.96)  LDD0752  [3]
 LDCM0436  CL46 HCT 116 C125(1.03); C33(1.08); C71(1.06); C97(0.91)  LDD0753  [3]
 LDCM0437  CL47 HCT 116 C125(1.27); C33(0.93); C71(1.02); C97(0.90)  LDD0754  [3]
 LDCM0438  CL48 HCT 116 C125(1.05); C33(1.10); C71(1.04); C97(0.89)  LDD0755  [3]
 LDCM0439  CL49 HCT 116 C125(1.26); C33(1.32); C71(1.04); C97(0.89)  LDD0756  [3]
 LDCM0440  CL5 HCT 116 C33(1.08); C490(0.85); C71(1.03); C97(1.17)  LDD0757  [3]
 LDCM0441  CL50 HCT 116 C125(1.01); C33(1.09); C71(0.91); C97(0.85)  LDD0758  [3]
 LDCM0442  CL51 HCT 116 C125(1.09); C33(0.98); C71(0.97); C97(1.06)  LDD0759  [3]
 LDCM0443  CL52 HCT 116 C125(1.41); C33(1.02); C71(1.09); C97(1.11)  LDD0760  [3]
 LDCM0444  CL53 HCT 116 C125(0.85); C33(0.85); C71(0.95); C97(0.93)  LDD0761  [3]
 LDCM0445  CL54 HCT 116 C125(1.29); C33(1.07); C71(0.98); C97(0.93)  LDD0762  [3]
 LDCM0446  CL55 HCT 116 C125(1.16); C33(1.11); C71(0.91); C97(1.10)  LDD0763  [3]
 LDCM0447  CL56 HCT 116 C125(1.12); C33(0.98); C71(0.95); C97(1.07)  LDD0764  [3]
 LDCM0448  CL57 HCT 116 C125(1.21); C33(0.99); C71(0.97); C97(1.04)  LDD0765  [3]
 LDCM0449  CL58 HCT 116 C125(1.40); C33(1.12); C71(0.97); C97(1.12)  LDD0766  [3]
 LDCM0450  CL59 HCT 116 C125(1.43); C33(1.17); C71(0.95); C97(0.94)  LDD0767  [3]
 LDCM0451  CL6 HCT 116 C33(1.09); C490(1.01); C71(1.03); C97(1.14)  LDD0768  [3]
 LDCM0452  CL60 HCT 116 C125(1.36); C33(1.26); C71(0.96); C97(0.89)  LDD0769  [3]
 LDCM0453  CL61 HCT 116 C125(0.97); C33(0.92); C490(1.11); C71(0.97)  LDD0770  [3]
 LDCM0454  CL62 HCT 116 C125(0.94); C33(0.94); C490(1.19); C71(1.10)  LDD0771  [3]
 LDCM0455  CL63 HCT 116 C125(1.34); C33(0.92); C490(1.17); C71(1.17)  LDD0772  [3]
 LDCM0456  CL64 HCT 116 C125(0.92); C33(0.83); C490(0.99); C71(0.98)  LDD0773  [3]
 LDCM0457  CL65 HCT 116 C125(1.05); C33(0.99); C490(1.27); C71(1.24)  LDD0774  [3]
 LDCM0458  CL66 HCT 116 C125(0.93); C33(0.83); C490(0.98); C71(1.07)  LDD0775  [3]
 LDCM0459  CL67 HCT 116 C125(0.81); C33(0.81); C490(0.98); C71(1.07)  LDD0776  [3]
 LDCM0460  CL68 HCT 116 C125(1.06); C33(0.76); C490(1.20); C71(1.12)  LDD0777  [3]
 LDCM0461  CL69 HCT 116 C125(0.90); C33(0.91); C490(0.76); C71(0.98)  LDD0778  [3]
 LDCM0462  CL7 HCT 116 C33(0.92); C490(0.74); C71(1.18); C97(1.24)  LDD0779  [3]
 LDCM0463  CL70 HCT 116 C125(1.03); C33(0.95); C490(1.07); C71(0.99)  LDD0780  [3]
 LDCM0464  CL71 HCT 116 C125(0.97); C33(0.80); C490(0.93); C71(1.09)  LDD0781  [3]
 LDCM0465  CL72 HCT 116 C125(0.82); C33(0.86); C490(1.01); C71(1.00)  LDD0782  [3]
 LDCM0466  CL73 HCT 116 C125(0.90); C33(0.67); C490(0.92); C71(0.97)  LDD0783  [3]
 LDCM0467  CL74 HCT 116 C125(0.95); C33(0.78); C490(1.02); C71(1.12)  LDD0784  [3]
 LDCM0469  CL76 HCT 116 C125(1.00); C33(1.01); C490(1.26); C71(1.17)  LDD0786  [3]
 LDCM0470  CL77 HCT 116 C125(0.73); C33(0.81); C490(1.14); C71(1.12)  LDD0787  [3]
 LDCM0471  CL78 HCT 116 C125(1.05); C33(0.98); C490(1.14); C71(1.15)  LDD0788  [3]
 LDCM0472  CL79 HCT 116 C125(1.01); C33(0.90); C490(0.84); C71(1.22)  LDD0789  [3]
 LDCM0473  CL8 HCT 116 C33(0.93); C490(0.67); C71(1.12); C97(1.63)  LDD0790  [3]
 LDCM0474  CL80 HCT 116 C125(0.88); C33(1.04); C490(0.94); C71(1.20)  LDD0791  [3]
 LDCM0475  CL81 HCT 116 C125(1.06); C33(1.26); C490(0.99); C71(1.19)  LDD0792  [3]
 LDCM0476  CL82 HCT 116 C125(0.98); C33(1.07); C490(1.00); C71(1.43)  LDD0793  [3]
 LDCM0477  CL83 HCT 116 C125(0.84); C33(0.85); C490(1.05); C71(1.10)  LDD0794  [3]
 LDCM0478  CL84 HCT 116 C125(0.96); C33(1.08); C490(1.16); C71(1.40)  LDD0795  [3]
 LDCM0479  CL85 HCT 116 C125(1.03); C33(0.96); C490(1.08); C71(1.23)  LDD0796  [3]
 LDCM0480  CL86 HCT 116 C125(1.12); C33(1.23); C490(1.27); C71(1.17)  LDD0797  [3]
 LDCM0481  CL87 HCT 116 C125(0.89); C33(0.85); C490(1.08); C71(1.39)  LDD0798  [3]
 LDCM0482  CL88 HCT 116 C125(0.95); C33(0.88); C490(0.87); C71(1.38)  LDD0799  [3]
 LDCM0483  CL89 HCT 116 C125(0.86); C33(1.26); C490(1.34); C71(1.61)  LDD0800  [3]
 LDCM0484  CL9 HCT 116 C33(0.97); C490(0.80); C71(1.21); C97(1.35)  LDD0801  [3]
 LDCM0485  CL90 HCT 116 C125(0.71); C33(0.99); C490(0.73); C71(1.09)  LDD0802  [3]
 LDCM0486  CL91 HCT 116 C125(1.29); C33(1.00); C490(0.98); C71(1.33)  LDD0803  [3]
 LDCM0487  CL92 HCT 116 C125(0.98); C33(0.94); C490(0.81); C71(1.13)  LDD0804  [3]
 LDCM0488  CL93 HCT 116 C125(1.03); C33(0.95); C490(0.87); C71(1.19)  LDD0805  [3]
 LDCM0489  CL94 HCT 116 C125(1.06); C33(0.86); C490(0.85); C71(1.23)  LDD0806  [3]
 LDCM0490  CL95 HCT 116 C125(1.13); C33(0.90); C490(0.67); C71(1.37)  LDD0807  [3]
 LDCM0491  CL96 HCT 116 C125(1.22); C33(0.91); C490(0.85); C71(1.27)  LDD0808  [3]
 LDCM0492  CL97 HCT 116 C125(1.23); C33(1.06); C490(0.81); C71(1.15)  LDD0809  [3]
 LDCM0493  CL98 HCT 116 C125(1.39); C33(1.00); C490(0.90); C71(1.35)  LDD0810  [3]
 LDCM0494  CL99 HCT 116 C125(1.48); C33(1.08); C490(0.86); C71(1.42)  LDD0811  [3]
 LDCM0495  E2913 HEK-293T C97(1.17); C490(0.94); C33(1.09); C125(1.01)  LDD1698  [19]
 LDCM0213  Electrophilic fragment 2 MDA-MB-231 C33(1.04); C490(0.89)  LDD1702  [2]
 LDCM0468  Fragment33 HCT 116 C125(0.82); C33(0.90); C490(1.13); C71(1.14)  LDD0785  [3]
 LDCM0427  Fragment51 HCT 116 C125(0.56); C33(0.55); C490(0.74); C71(0.86)  LDD0744  [3]
 LDCM0107  IAA HeLa H374(0.00); H369(0.00)  LDD0221  [14]
 LDCM0022  KB02 HCT 116 C71(1.28); C97(1.88); C125(1.18); C490(1.11)  LDD0080  [3]
 LDCM0023  KB03 HCT 116 C71(1.38); C97(1.35); C125(1.49); C490(1.00)  LDD0081  [3]
 LDCM0024  KB05 HCT 116 C71(1.47); C97(1.46); C125(1.32); C490(1.03)  LDD0082  [3]
 LDCM0109  NEM HeLa H374(0.00); H369(0.00)  LDD0223  [14]
 LDCM0499  Nucleophilic fragment 12b MDA-MB-231 C97(0.69)  LDD2092  [2]
 LDCM0501  Nucleophilic fragment 13b MDA-MB-231 C97(1.50)  LDD2094  [2]
 LDCM0506  Nucleophilic fragment 16a MDA-MB-231 C490(1.54)  LDD2099  [2]
 LDCM0507  Nucleophilic fragment 16b MDA-MB-231 C490(0.50); C71(1.32)  LDD2100  [2]
 LDCM0511  Nucleophilic fragment 18b MDA-MB-231 C97(1.02)  LDD2104  [2]
 LDCM0514  Nucleophilic fragment 20a MDA-MB-231 C490(1.03)  LDD2107  [2]
 LDCM0516  Nucleophilic fragment 21a MDA-MB-231 C33(0.78)  LDD2109  [2]
 LDCM0521  Nucleophilic fragment 23b MDA-MB-231 C490(0.48)  LDD2114  [2]
 LDCM0526  Nucleophilic fragment 26a MDA-MB-231 C71(1.11)  LDD2119  [2]
 LDCM0529  Nucleophilic fragment 27b MDA-MB-231 C97(1.41)  LDD2122  [2]
 LDCM0532  Nucleophilic fragment 29a MDA-MB-231 C71(0.79); C33(0.94)  LDD2125  [2]
 LDCM0534  Nucleophilic fragment 30a MDA-MB-231 C490(1.03); C33(0.95)  LDD2127  [2]
 LDCM0541  Nucleophilic fragment 36 MDA-MB-231 C490(0.52)  LDD2134  [2]
 LDCM0543  Nucleophilic fragment 38 MDA-MB-231 C490(1.57); C33(1.19)  LDD2136  [2]
 LDCM0547  Nucleophilic fragment 41 MDA-MB-231 C97(1.00)  LDD2141  [2]
 LDCM0550  Nucleophilic fragment 5a MDA-MB-231 C490(1.73); C71(1.33)  LDD2144  [2]
 LDCM0552  Nucleophilic fragment 6a MDA-MB-231 C490(1.40)  LDD2146  [2]

References

1 Quantitative and Site-Specific Chemoproteomic Profiling of Targets of Acrolein. Chem Res Toxicol. 2019 Mar 18;32(3):467-473. doi: 10.1021/acs.chemrestox.8b00343. Epub 2019 Jan 15.
2 Nucleophilic covalent ligand discovery for the cysteine redoxome. Nat Chem Biol. 2023 Nov;19(11):1309-1319. doi: 10.1038/s41589-023-01330-5. Epub 2023 May 29.
Mass spectrometry data entry: PXD039908 , PXD029761
3 Reimagining high-throughput profiling of reactive cysteines for cell-based screening of large electrophile libraries. Nat Biotechnol. 2021 May;39(5):630-641. doi: 10.1038/s41587-020-00778-3. Epub 2021 Jan 4.
4 Targeted Proteomic Approaches for Proteome-Wide Characterizations of the AMP-Binding Capacities of Kinases. J Proteome Res. 2022 Aug 5;21(8):2063-2070. doi: 10.1021/acs.jproteome.2c00225. Epub 2022 Jul 12.
5 Enhancing Cysteine Chemoproteomic Coverage through Systematic Assessment of Click Chemistry Product Fragmentation. Anal Chem. 2022 Mar 8;94(9):3800-3810. doi: 10.1021/acs.analchem.1c04402. Epub 2022 Feb 23.
Mass spectrometry data entry: PXD028853
6 SP3-FAIMS Chemoproteomics for High-Coverage Profiling of the Human Cysteinome*. Chembiochem. 2021 May 14;22(10):1841-1851. doi: 10.1002/cbic.202000870. Epub 2021 Feb 18.
Mass spectrometry data entry: PXD023056 , PXD023059 , PXD023058 , PXD023057 , PXD023060
7 SP3-Enabled Rapid and High Coverage Chemoproteomic Identification of Cell-State-Dependent Redox-Sensitive Cysteines. Mol Cell Proteomics. 2022 Apr;21(4):100218. doi: 10.1016/j.mcpro.2022.100218. Epub 2022 Feb 25.
Mass spectrometry data entry: PXD029500 , PXD031647
8 A modification-centric assessment tool for the performance of chemoproteomic probes. Nat Chem Biol. 2022 Aug;18(8):904-912. doi: 10.1038/s41589-022-01074-8. Epub 2022 Jul 21.
Mass spectrometry data entry: PXD027758 , PXD027755 , PXD027760 , PXD027762 , PXD027756 , PXD027591 , PXD007149 , PXD030064 , PXD032392 , PXD027789 , PXD027767 , PXD027764
9 Multiplexed CuAAC Suzuki-Miyaura Labeling for Tandem Activity-Based Chemoproteomic Profiling. Anal Chem. 2021 Feb 2;93(4):2610-2618. doi: 10.1021/acs.analchem.0c04726. Epub 2021 Jan 20.
Mass spectrometry data entry: PXD022279
10 Solid Phase Synthesis of Fluorosulfate Containing Macrocycles for Chemoproteomic Workflows. bioRxiv [Preprint]. 2023 Feb 18:2023.02.17.529022. doi: 10.1101/2023.02.17.529022.
Mass spectrometry data entry: PXD039931
11 Chemoproteomic Profiling by Cysteine Fluoroalkylation Reveals Myrocin G as an Inhibitor of the Nonhomologous End Joining DNA Repair Pathway. J Am Chem Soc. 2021 Dec 8;143(48):20332-20342. doi: 10.1021/jacs.1c09724. Epub 2021 Nov 24.
Mass spectrometry data entry: PXD029255
12 DFT-Guided Discovery of Ethynyl-Triazolyl-Phosphinates as Modular Electrophiles for Chemoselective Cysteine Bioconjugation and Profiling. Angew Chem Int Ed Engl. 2022 Oct 10;61(41):e202205348. doi: 10.1002/anie.202205348. Epub 2022 Aug 22.
Mass spectrometry data entry: PXD033004
13 Tunable Amine-Reactive Electrophiles for Selective Profiling of Lysine. Angew Chem Int Ed Engl. 2022 Jan 26;61(5):e202112107. doi: 10.1002/anie.202112107. Epub 2021 Dec 16.
14 ACR-Based Probe for the Quantitative Profiling of Histidine Reactivity in the Human Proteome. J Am Chem Soc. 2023 Mar 8;145(9):5252-5260. doi: 10.1021/jacs.2c12653. Epub 2023 Feb 27.
15 Oxidant-Induced Bioconjugation for Protein Labeling in Live Cells. ACS Chem Biol. 2023 Jan 20;18(1):112-122. doi: 10.1021/acschembio.2c00740. Epub 2022 Dec 21.
16 N-Acryloylindole-alkyne (NAIA) enables imaging and profiling new ligandable cysteines and oxidized thiols by chemoproteomics. Nat Commun. 2023 Jun 15;14(1):3564. doi: 10.1038/s41467-023-39268-w.
Mass spectrometry data entry: PXD041264
17 Ligand and Target Discovery by Fragment-Based Screening in Human Cells. Cell. 2017 Jan 26;168(3):527-541.e29. doi: 10.1016/j.cell.2016.12.029. Epub 2017 Jan 19.
18 Design and synthesis of minimalist terminal alkyne-containing diazirine photo-crosslinkers and their incorporation into kinase inhibitors for cell- and tissue-based proteome profiling. Angew Chem Int Ed Engl. 2013 Aug 12;52(33):8551-6. doi: 10.1002/anie.201300683. Epub 2013 Jun 10.
19 Accelerating multiplexed profiling of protein-ligand interactions: High-throughput plate-based reactive cysteine profiling with minimal input. Cell Chem Biol. 2024 Mar 21;31(3):565-576.e4. doi: 10.1016/j.chembiol.2023.11.015. Epub 2023 Dec 19.
Mass spectrometry data entry: PXD044402