General Information of Target

Target ID LDTP05175
Target Name Small ribosomal subunit protein mS22 (MRPS22)
Gene Name MRPS22
Gene ID 56945
Synonyms
C3orf5; RPMS22; Small ribosomal subunit protein mS22; 28S ribosomal protein S22, mitochondrial; MRP-S22; S22mt
3D Structure
Download
2D Sequence (FASTA)
Download
3D Structure (PDB)
Download
Sequence
MAPLGTTVLLWSLLRSSPGVERVCFRARIQPWHGGLLQPLPCSFEMGLPRRRFSSEAAES
GSPETKKPTFMDEEVQSILTKMTGLNLQKTFKPAIQELKPPTYKLMTQAQLEEATRQAVE
AAKVRLKMPPVLEERVPINDVLAEDKILEGTETTKYVFTDISYSIPHRERFIVVREPSGT
LRKASWEERDRMIQVYFPKEGRKILTPIIFKEENLRTMYSQDRHVDVLNLCFAQFEPDST
EYIKVHHKTYEDIDKRGKYDLLRSTRYFGGMVWYFVNNKKIDGLLIDQIQRDLIDDATNL
VQLYHVLHPDGQSAQGAKDQAAEGINLIKVFAKTEAQKGAYIELTLQTYQEALSRHSAAS
Target Bioclass
Other
Family
Mitochondrion-specific ribosomal protein mS22 family
Subcellular location
Mitochondrion
Uniprot ID
P82650
Ensemble ID
ENST00000495075.5
HGNC ID
HGNC:14508

Target Site Mutations in Different Cell Lines

Cell line Mutation details Probe for labeling this protein in this cell
AN3CA SNV: p.F158L .
CAL148 SNV: p.E134K .
HCC44 SNV: p.M106V .
KATOIII Insertion: p.A58_S60dup DBIA    Probe Info 

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 15 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
STPyne
 Probe Info 
K203(8.33); K329(10.00)  LDD0277  [1]
HHS-475
 Probe Info 
Y163(0.69)  LDD0264  [2]
DBIA
 Probe Info 
C231(0.54)  LDD0532  [3]
ATP probe
 Probe Info 
N.A.  LDD0199  [4]
4-Iodoacetamidophenylacetylene
 Probe Info 
N.A.  LDD0038  [5]
IA-alkyne
 Probe Info 
N.A.  LDD0032  [6]
IPIAA_H
 Probe Info 
N.A.  LDD0030  [7]
IPIAA_L
 Probe Info 
N.A.  LDD0031  [7]
Lodoacetamide azide
 Probe Info 
N.A.  LDD0037  [5]
NHS
 Probe Info 
N.A.  LDD0010  [8]
SF
 Probe Info 
Y163(0.00); Y103(0.00)  LDD0028  [9]
1c-yne
 Probe Info 
K338(0.00); K81(0.00)  LDD0228  [10]
1d-yne
 Probe Info 
N.A.  LDD0357  [10]
NAIA_5
 Probe Info 
N.A.  LDD2223  [11]
HHS-465
 Probe Info 
N.A.  LDD2240  [12]
PAL-AfBPP Probe
Click To Hide/Show 3 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
C280
 Probe Info 
14.22  LDD1950  [13]
FFF probe13
 Probe Info 
20.00  LDD0475  [14]
FFF probe3
 Probe Info 
13.74  LDD0464  [14]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0214  AC1 PaTu 8988t C231(0.24)  LDD1093  [3]
 LDCM0215  AC10 HCT 116 C231(0.54)  LDD0532  [3]
 LDCM0216  AC100 HEK-293T C231(1.14)  LDD0814  [3]
 LDCM0217  AC101 HEK-293T C231(1.00)  LDD0815  [3]
 LDCM0218  AC102 HEK-293T C231(1.31)  LDD0816  [3]
 LDCM0219  AC103 HEK-293T C231(1.00)  LDD0817  [3]
 LDCM0220  AC104 HEK-293T C231(0.85)  LDD0818  [3]
 LDCM0221  AC105 HEK-293T C231(1.20)  LDD0819  [3]
 LDCM0222  AC106 HEK-293T C231(1.71)  LDD0820  [3]
 LDCM0223  AC107 HEK-293T C231(1.03)  LDD0821  [3]
 LDCM0224  AC108 HEK-293T C231(1.13)  LDD0822  [3]
 LDCM0225  AC109 HEK-293T C231(1.38)  LDD0823  [3]
 LDCM0226  AC11 HCT 116 C231(0.65)  LDD0543  [3]
 LDCM0227  AC110 HEK-293T C231(0.40)  LDD0825  [3]
 LDCM0228  AC111 HEK-293T C231(0.24)  LDD0826  [3]
 LDCM0229  AC112 HEK-293T C231(0.33)  LDD0827  [3]
 LDCM0230  AC113 PaTu 8988t C231(1.23)  LDD1109  [3]
 LDCM0231  AC114 PaTu 8988t C231(1.11)  LDD1110  [3]
 LDCM0232  AC115 PaTu 8988t C231(1.33)  LDD1111  [3]
 LDCM0233  AC116 PaTu 8988t C231(1.07)  LDD1112  [3]
 LDCM0234  AC117 PaTu 8988t C231(1.11)  LDD1113  [3]
 LDCM0235  AC118 PaTu 8988t C231(0.97)  LDD1114  [3]
 LDCM0236  AC119 PaTu 8988t C231(0.47)  LDD1115  [3]
 LDCM0237  AC12 HCT 116 C231(0.92)  LDD0554  [3]
 LDCM0238  AC120 PaTu 8988t C231(0.72)  LDD1117  [3]
 LDCM0239  AC121 PaTu 8988t C231(0.34)  LDD1118  [3]
 LDCM0240  AC122 PaTu 8988t C231(1.05)  LDD1119  [3]
 LDCM0241  AC123 PaTu 8988t C231(0.77)  LDD1120  [3]
 LDCM0242  AC124 PaTu 8988t C231(0.32)  LDD1121  [3]
 LDCM0243  AC125 PaTu 8988t C231(0.77)  LDD1122  [3]
 LDCM0244  AC126 PaTu 8988t C231(1.11)  LDD1123  [3]
 LDCM0245  AC127 PaTu 8988t C231(0.46)  LDD1124  [3]
 LDCM0246  AC128 PaTu 8988t C231(0.52)  LDD1125  [3]
 LDCM0247  AC129 PaTu 8988t C231(0.30)  LDD1126  [3]
 LDCM0249  AC130 PaTu 8988t C231(0.51)  LDD1128  [3]
 LDCM0250  AC131 PaTu 8988t C231(0.40)  LDD1129  [3]
 LDCM0251  AC132 PaTu 8988t C231(0.48)  LDD1130  [3]
 LDCM0252  AC133 PaTu 8988t C231(0.22)  LDD1131  [3]
 LDCM0253  AC134 PaTu 8988t C231(0.21)  LDD1132  [3]
 LDCM0254  AC135 PaTu 8988t C231(0.27)  LDD1133  [3]
 LDCM0255  AC136 PaTu 8988t C231(0.22)  LDD1134  [3]
 LDCM0256  AC137 PaTu 8988t C231(0.24)  LDD1135  [3]
 LDCM0257  AC138 PaTu 8988t C231(0.39)  LDD1136  [3]
 LDCM0258  AC139 PaTu 8988t C231(0.30)  LDD1137  [3]
 LDCM0259  AC14 HCT 116 C231(0.68)  LDD0576  [3]
 LDCM0260  AC140 PaTu 8988t C231(0.50)  LDD1139  [3]
 LDCM0261  AC141 PaTu 8988t C231(0.60)  LDD1140  [3]
 LDCM0262  AC142 PaTu 8988t C231(0.32)  LDD1141  [3]
 LDCM0263  AC143 HCT 116 C231(0.73)  LDD0580  [3]
 LDCM0264  AC144 HCT 116 C231(0.27)  LDD0581  [3]
 LDCM0265  AC145 HCT 116 C231(0.49)  LDD0582  [3]
 LDCM0266  AC146 HCT 116 C231(0.35)  LDD0583  [3]
 LDCM0267  AC147 HCT 116 C231(0.23)  LDD0584  [3]
 LDCM0268  AC148 HCT 116 C231(0.16)  LDD0585  [3]
 LDCM0269  AC149 HCT 116 C231(0.20)  LDD0586  [3]
 LDCM0270  AC15 HCT 116 C231(0.54)  LDD0587  [3]
 LDCM0271  AC150 HCT 116 C231(0.61)  LDD0588  [3]
 LDCM0272  AC151 HCT 116 C231(0.59)  LDD0589  [3]
 LDCM0273  AC152 HCT 116 C231(0.19)  LDD0590  [3]
 LDCM0274  AC153 HCT 116 C231(0.16)  LDD0591  [3]
 LDCM0621  AC154 HCT 116 C231(0.32)  LDD2158  [3]
 LDCM0622  AC155 HCT 116 C231(0.34)  LDD2159  [3]
 LDCM0623  AC156 HCT 116 C231(0.76)  LDD2160  [3]
 LDCM0624  AC157 HCT 116 C231(0.84)  LDD2161  [3]
 LDCM0276  AC17 PaTu 8988t C231(0.77)  LDD1155  [3]
 LDCM0277  AC18 PaTu 8988t C231(0.38)  LDD1156  [3]
 LDCM0278  AC19 PaTu 8988t C231(0.63)  LDD1157  [3]
 LDCM0279  AC2 PaTu 8988t C231(0.46)  LDD1158  [3]
 LDCM0280  AC20 PaTu 8988t C231(0.46)  LDD1159  [3]
 LDCM0281  AC21 PaTu 8988t C231(0.27)  LDD1160  [3]
 LDCM0282  AC22 PaTu 8988t C231(0.27)  LDD1161  [3]
 LDCM0283  AC23 PaTu 8988t C231(0.30)  LDD1162  [3]
 LDCM0284  AC24 PaTu 8988t C231(0.75)  LDD1163  [3]
 LDCM0285  AC25 PaTu 8988t C231(1.70)  LDD1164  [3]
 LDCM0286  AC26 PaTu 8988t C231(1.14)  LDD1165  [3]
 LDCM0287  AC27 PaTu 8988t C231(0.88)  LDD1166  [3]
 LDCM0288  AC28 PaTu 8988t C231(0.77)  LDD1167  [3]
 LDCM0289  AC29 PaTu 8988t C231(0.87)  LDD1168  [3]
 LDCM0290  AC3 PaTu 8988t C231(0.55)  LDD1169  [3]
 LDCM0291  AC30 PaTu 8988t C231(0.96)  LDD1170  [3]
 LDCM0292  AC31 PaTu 8988t C231(1.56)  LDD1171  [3]
 LDCM0293  AC32 PaTu 8988t C231(0.97)  LDD1172  [3]
 LDCM0294  AC33 PaTu 8988t C231(0.85)  LDD1173  [3]
 LDCM0295  AC34 PaTu 8988t C231(0.37)  LDD1174  [3]
 LDCM0296  AC35 PaTu 8988t C231(0.65)  LDD1175  [3]
 LDCM0297  AC36 PaTu 8988t C231(0.46)  LDD1176  [3]
 LDCM0298  AC37 PaTu 8988t C231(0.53)  LDD1177  [3]
 LDCM0299  AC38 PaTu 8988t C231(0.67)  LDD1178  [3]
 LDCM0300  AC39 PaTu 8988t C231(0.47)  LDD1179  [3]
 LDCM0301  AC4 PaTu 8988t C231(0.78)  LDD1180  [3]
 LDCM0302  AC40 PaTu 8988t C231(0.45)  LDD1181  [3]
 LDCM0303  AC41 PaTu 8988t C231(0.75)  LDD1182  [3]
 LDCM0304  AC42 PaTu 8988t C231(0.78)  LDD1183  [3]
 LDCM0305  AC43 PaTu 8988t C231(0.73)  LDD1184  [3]
 LDCM0306  AC44 PaTu 8988t C231(0.52)  LDD1185  [3]
 LDCM0307  AC45 PaTu 8988t C231(0.78)  LDD1186  [3]
 LDCM0308  AC46 HEK-293T C231(0.89)  LDD0906  [3]
 LDCM0309  AC47 HEK-293T C231(1.03)  LDD0907  [3]
 LDCM0310  AC48 HEK-293T C231(0.89)  LDD0908  [3]
 LDCM0311  AC49 HEK-293T C231(0.97)  LDD0909  [3]
 LDCM0312  AC5 PaTu 8988t C231(0.25)  LDD1191  [3]
 LDCM0313  AC50 HEK-293T C231(0.77)  LDD0911  [3]
 LDCM0314  AC51 HEK-293T C231(0.85)  LDD0912  [3]
 LDCM0315  AC52 HEK-293T C231(1.01)  LDD0913  [3]
 LDCM0316  AC53 HEK-293T C231(0.96)  LDD0914  [3]
 LDCM0317  AC54 HEK-293T C231(0.83)  LDD0915  [3]
 LDCM0318  AC55 HEK-293T C231(0.93)  LDD0916  [3]
 LDCM0319  AC56 HEK-293T C231(0.72)  LDD0917  [3]
 LDCM0320  AC57 HEK-293T C231(0.93)  LDD0918  [3]
 LDCM0321  AC58 HEK-293T C231(0.90)  LDD0919  [3]
 LDCM0322  AC59 HEK-293T C231(0.80)  LDD0920  [3]
 LDCM0323  AC6 HCT 116 C231(0.63)  LDD0640  [3]
 LDCM0324  AC60 HEK-293T C231(0.92)  LDD0922  [3]
 LDCM0325  AC61 HEK-293T C231(1.06)  LDD0923  [3]
 LDCM0326  AC62 HEK-293T C231(0.76)  LDD0924  [3]
 LDCM0327  AC63 HEK-293T C231(0.73)  LDD0925  [3]
 LDCM0328  AC64 HEK-293T C231(0.87)  LDD0926  [3]
 LDCM0329  AC65 HEK-293T C231(1.12)  LDD0927  [3]
 LDCM0330  AC66 HEK-293T C231(0.79)  LDD0928  [3]
 LDCM0331  AC67 HEK-293T C231(0.97)  LDD0929  [3]
 LDCM0332  AC68 HEK-293T C231(1.12)  LDD0930  [3]
 LDCM0333  AC69 HEK-293T C231(1.02)  LDD0931  [3]
 LDCM0334  AC7 HCT 116 C231(0.85)  LDD0651  [3]
 LDCM0335  AC70 HEK-293T C231(1.04)  LDD0933  [3]
 LDCM0336  AC71 HEK-293T C231(1.15)  LDD0934  [3]
 LDCM0337  AC72 HEK-293T C231(1.39)  LDD0935  [3]
 LDCM0338  AC73 HEK-293T C231(1.30)  LDD0936  [3]
 LDCM0339  AC74 HEK-293T C231(1.54)  LDD0937  [3]
 LDCM0340  AC75 HEK-293T C231(1.43)  LDD0938  [3]
 LDCM0341  AC76 HEK-293T C231(1.12)  LDD0939  [3]
 LDCM0342  AC77 HEK-293T C231(1.47)  LDD0940  [3]
 LDCM0343  AC78 HEK-293T C231(1.23)  LDD0941  [3]
 LDCM0344  AC79 HEK-293T C231(0.96)  LDD0942  [3]
 LDCM0345  AC8 HCT 116 C231(0.75)  LDD0662  [3]
 LDCM0346  AC80 HEK-293T C231(1.36)  LDD0944  [3]
 LDCM0347  AC81 HEK-293T C231(1.31)  LDD0945  [3]
 LDCM0348  AC82 HEK-293T C231(1.20)  LDD0946  [3]
 LDCM0349  AC83 HEK-293T C231(1.18)  LDD0947  [3]
 LDCM0350  AC84 HEK-293T C231(1.43)  LDD0948  [3]
 LDCM0351  AC85 HEK-293T C231(1.20)  LDD0949  [3]
 LDCM0352  AC86 HEK-293T C231(1.32)  LDD0950  [3]
 LDCM0353  AC87 HEK-293T C231(1.41)  LDD0951  [3]
 LDCM0354  AC88 HEK-293T C231(1.45)  LDD0952  [3]
 LDCM0355  AC89 HEK-293T C231(1.43)  LDD0953  [3]
 LDCM0357  AC90 HEK-293T C231(1.16)  LDD0955  [3]
 LDCM0358  AC91 HEK-293T C231(1.13)  LDD0956  [3]
 LDCM0359  AC92 HEK-293T C231(1.30)  LDD0957  [3]
 LDCM0360  AC93 HEK-293T C231(1.83)  LDD0958  [3]
 LDCM0361  AC94 HEK-293T C231(1.16)  LDD0959  [3]
 LDCM0362  AC95 HEK-293T C231(1.19)  LDD0960  [3]
 LDCM0363  AC96 HEK-293T C231(1.49)  LDD0961  [3]
 LDCM0364  AC97 HEK-293T C231(0.41)  LDD0962  [3]
 LDCM0365  AC98 HEK-293T C231(1.28)  LDD0963  [3]
 LDCM0366  AC99 HEK-293T C231(1.17)  LDD0964  [3]
 LDCM0248  AKOS034007472 HCT 116 C231(0.76)  LDD0565  [3]
 LDCM0356  AKOS034007680 HCT 116 C231(0.65)  LDD0673  [3]
 LDCM0275  AKOS034007705 HCT 116 C231(0.25)  LDD0592  [3]
 LDCM0367  CL1 HCT 116 C231(1.22)  LDD0684  [3]
 LDCM0368  CL10 HCT 116 C231(0.43)  LDD0685  [3]
 LDCM0369  CL100 PaTu 8988t C231(0.74)  LDD1248  [3]
 LDCM0370  CL101 HCT 116 C231(0.58)  LDD0687  [3]
 LDCM0371  CL102 HCT 116 C231(1.16)  LDD0688  [3]
 LDCM0372  CL103 HCT 116 C231(1.04)  LDD0689  [3]
 LDCM0373  CL104 HCT 116 C231(0.72)  LDD0690  [3]
 LDCM0374  CL105 PaTu 8988t C231(0.87)  LDD1253  [3]
 LDCM0375  CL106 PaTu 8988t C231(0.74)  LDD1254  [3]
 LDCM0376  CL107 PaTu 8988t C231(0.86)  LDD1255  [3]
 LDCM0377  CL108 PaTu 8988t C231(0.74)  LDD1256  [3]
 LDCM0378  CL109 PaTu 8988t C231(0.60)  LDD1257  [3]
 LDCM0379  CL11 HCT 116 C231(0.31)  LDD0696  [3]
 LDCM0380  CL110 PaTu 8988t C231(0.53)  LDD1259  [3]
 LDCM0381  CL111 PaTu 8988t C231(0.27)  LDD1260  [3]
 LDCM0382  CL112 PaTu 8988t C231(1.36)  LDD1261  [3]
 LDCM0383  CL113 PaTu 8988t C231(1.40)  LDD1262  [3]
 LDCM0384  CL114 PaTu 8988t C231(1.23)  LDD1263  [3]
 LDCM0385  CL115 PaTu 8988t C231(1.49)  LDD1264  [3]
 LDCM0386  CL116 PaTu 8988t C231(1.49)  LDD1265  [3]
 LDCM0387  CL117 PaTu 8988t C231(0.97)  LDD1266  [3]
 LDCM0388  CL118 PaTu 8988t C231(1.27)  LDD1267  [3]
 LDCM0389  CL119 PaTu 8988t C231(0.64)  LDD1268  [3]
 LDCM0390  CL12 HCT 116 C231(0.28)  LDD0707  [3]
 LDCM0391  CL120 PaTu 8988t C231(0.43)  LDD1270  [3]
 LDCM0392  CL121 HEK-293T C231(1.00)  LDD0990  [3]
 LDCM0393  CL122 HEK-293T C231(1.03)  LDD0991  [3]
 LDCM0394  CL123 HEK-293T C231(0.83)  LDD0992  [3]
 LDCM0395  CL124 HEK-293T C231(0.87)  LDD0993  [3]
 LDCM0396  CL125 HEK-293T C231(0.82)  LDD0994  [3]
 LDCM0397  CL126 HEK-293T C231(0.89)  LDD0995  [3]
 LDCM0398  CL127 HEK-293T C231(0.83)  LDD0996  [3]
 LDCM0399  CL128 HEK-293T C231(1.19)  LDD0997  [3]
 LDCM0400  CL13 HCT 116 C231(0.50)  LDD0717  [3]
 LDCM0401  CL14 HCT 116 C231(0.83)  LDD0718  [3]
 LDCM0402  CL15 HCT 116 C231(0.58)  LDD0719  [3]
 LDCM0403  CL16 HEK-293T C231(0.91)  LDD1001  [3]
 LDCM0404  CL17 HEK-293T C231(0.70)  LDD1002  [3]
 LDCM0405  CL18 HEK-293T C231(0.85)  LDD1003  [3]
 LDCM0406  CL19 HEK-293T C231(0.86)  LDD1004  [3]
 LDCM0407  CL2 HCT 116 C231(1.22)  LDD0724  [3]
 LDCM0408  CL20 HEK-293T C231(0.99)  LDD1006  [3]
 LDCM0409  CL21 HEK-293T C231(1.07)  LDD1007  [3]
 LDCM0410  CL22 HEK-293T C231(0.87)  LDD1008  [3]
 LDCM0411  CL23 HEK-293T C231(0.66)  LDD1009  [3]
 LDCM0412  CL24 HEK-293T C231(0.94)  LDD1010  [3]
 LDCM0413  CL25 HEK-293T C231(0.83)  LDD1011  [3]
 LDCM0414  CL26 HEK-293T C231(0.87)  LDD1012  [3]
 LDCM0415  CL27 HEK-293T C231(0.87)  LDD1013  [3]
 LDCM0416  CL28 HEK-293T C231(0.79)  LDD1014  [3]
 LDCM0417  CL29 HEK-293T C231(0.94)  LDD1015  [3]
 LDCM0418  CL3 HCT 116 C231(0.86)  LDD0735  [3]
 LDCM0419  CL30 HEK-293T C231(0.69)  LDD1017  [3]
 LDCM0420  CL31 HCT 116 C231(0.68)  LDD0737  [3]
 LDCM0421  CL32 HCT 116 C231(0.72)  LDD0738  [3]
 LDCM0422  CL33 HCT 116 C231(0.90)  LDD0739  [3]
 LDCM0423  CL34 HCT 116 C231(0.31)  LDD0740  [3]
 LDCM0424  CL35 HCT 116 C231(0.31)  LDD0741  [3]
 LDCM0425  CL36 HCT 116 C231(0.35)  LDD0742  [3]
 LDCM0426  CL37 HCT 116 C231(0.28)  LDD0743  [3]
 LDCM0428  CL39 HCT 116 C231(0.28)  LDD0745  [3]
 LDCM0429  CL4 HCT 116 C231(0.85)  LDD0746  [3]
 LDCM0430  CL40 HCT 116 C231(0.36)  LDD0747  [3]
 LDCM0431  CL41 HCT 116 C231(0.40)  LDD0748  [3]
 LDCM0432  CL42 HCT 116 C231(0.30)  LDD0749  [3]
 LDCM0433  CL43 HCT 116 C231(0.29)  LDD0750  [3]
 LDCM0434  CL44 HCT 116 C231(0.53)  LDD0751  [3]
 LDCM0435  CL45 HCT 116 C231(0.34)  LDD0752  [3]
 LDCM0436  CL46 HEK-293T C231(1.00)  LDD1640  [15]
 LDCM0438  CL48 HEK-293T C231(1.06)  LDD1642  [15]
 LDCM0439  CL49 HEK-293T C231(1.28)  LDD1643  [15]
 LDCM0440  CL5 HCT 116 C231(0.72)  LDD0757  [3]
 LDCM0441  CL50 HEK-293T C231(1.01)  LDD1645  [15]
 LDCM0444  CL53 HEK-293T C231(0.87)  LDD1647  [15]
 LDCM0445  CL54 HEK-293T C231(1.00)  LDD1648  [15]
 LDCM0448  CL57 HEK-293T C231(0.95)  LDD1651  [15]
 LDCM0449  CL58 HEK-293T C231(1.02)  LDD1652  [15]
 LDCM0451  CL6 HCT 116 C231(0.70)  LDD0768  [3]
 LDCM0452  CL60 HEK-293T C231(1.11)  LDD1655  [15]
 LDCM0453  CL61 HEK-293T C231(1.42)  LDD1051  [3]
 LDCM0454  CL62 HEK-293T C231(1.46)  LDD1052  [3]
 LDCM0455  CL63 HEK-293T C231(1.60)  LDD1053  [3]
 LDCM0456  CL64 HEK-293T C231(1.26)  LDD1054  [3]
 LDCM0457  CL65 HEK-293T C231(1.43)  LDD1055  [3]
 LDCM0458  CL66 HEK-293T C231(1.37)  LDD1056  [3]
 LDCM0459  CL67 HEK-293T C231(1.01)  LDD1057  [3]
 LDCM0460  CL68 HEK-293T C231(1.17)  LDD1058  [3]
 LDCM0461  CL69 HEK-293T C231(1.23)  LDD1059  [3]
 LDCM0462  CL7 HCT 116 C231(0.37)  LDD0779  [3]
 LDCM0463  CL70 HEK-293T C231(1.22)  LDD1061  [3]
 LDCM0464  CL71 HEK-293T C231(1.54)  LDD1062  [3]
 LDCM0465  CL72 HEK-293T C231(1.37)  LDD1063  [3]
 LDCM0466  CL73 HEK-293T C231(1.35)  LDD1064  [3]
 LDCM0467  CL74 HEK-293T C231(1.14)  LDD1065  [3]
 LDCM0469  CL76 HCT 116 C231(0.92)  LDD0786  [3]
 LDCM0470  CL77 HCT 116 C231(0.81)  LDD0787  [3]
 LDCM0471  CL78 HCT 116 C231(0.70)  LDD0788  [3]
 LDCM0472  CL79 HCT 116 C231(0.44)  LDD0789  [3]
 LDCM0473  CL8 HCT 116 C231(0.29)  LDD0790  [3]
 LDCM0474  CL80 HCT 116 C231(0.95)  LDD0791  [3]
 LDCM0475  CL81 HCT 116 C231(0.64)  LDD0792  [3]
 LDCM0476  CL82 HCT 116 C231(0.33)  LDD0793  [3]
 LDCM0477  CL83 HCT 116 C231(0.35)  LDD0794  [3]
 LDCM0478  CL84 HCT 116 C231(0.37)  LDD0795  [3]
 LDCM0479  CL85 HCT 116 C231(0.67)  LDD0796  [3]
 LDCM0480  CL86 HCT 116 C231(0.84)  LDD0797  [3]
 LDCM0481  CL87 HCT 116 C231(0.67)  LDD0798  [3]
 LDCM0482  CL88 HCT 116 C231(0.38)  LDD0799  [3]
 LDCM0483  CL89 HCT 116 C231(0.41)  LDD0800  [3]
 LDCM0484  CL9 HCT 116 C231(0.53)  LDD0801  [3]
 LDCM0485  CL90 HCT 116 C231(0.85)  LDD0802  [3]
 LDCM0486  CL91 PaTu 8988t C231(0.87)  LDD1365  [3]
 LDCM0487  CL92 PaTu 8988t C231(0.47)  LDD1366  [3]
 LDCM0488  CL93 PaTu 8988t C231(0.46)  LDD1367  [3]
 LDCM0489  CL94 PaTu 8988t C231(0.43)  LDD1368  [3]
 LDCM0490  CL95 PaTu 8988t C231(0.29)  LDD1369  [3]
 LDCM0491  CL96 PaTu 8988t C231(0.54)  LDD1370  [3]
 LDCM0492  CL97 PaTu 8988t C231(0.55)  LDD1371  [3]
 LDCM0493  CL98 PaTu 8988t C231(0.32)  LDD1372  [3]
 LDCM0494  CL99 PaTu 8988t C231(0.48)  LDD1373  [3]
 LDCM0495  E2913 HEK-293T C231(0.94)  LDD1698  [15]
 LDCM0468  Fragment33 HEK-293T C231(1.58)  LDD1066  [3]
 LDCM0427  Fragment51 HCT 116 C231(0.28)  LDD0744  [3]
 LDCM0116  HHS-0101 DM93 Y163(0.69)  LDD0264  [2]
 LDCM0117  HHS-0201 DM93 Y163(2.41)  LDD0265  [2]
 LDCM0118  HHS-0301 DM93 Y163(1.45)  LDD0266  [2]
 LDCM0119  HHS-0401 DM93 Y163(2.65)  LDD0267  [2]
 LDCM0120  HHS-0701 DM93 Y163(10.78)  LDD0268  [2]
 LDCM0022  KB02 HEK-293T C231(0.95)  LDD1492  [15]
 LDCM0023  KB03 HEK-293T C231(1.04)  LDD1497  [15]
 LDCM0024  KB05 IGR37 C231(3.55)  LDD3314  [16]

References

1 A Paal-Knorr agent for chemoproteomic profiling of targets of isoketals in cells. Chem Sci. 2021 Oct 15;12(43):14557-14563. doi: 10.1039/d1sc02230j. eCollection 2021 Nov 10.
Mass spectrometry data entry: PXD028270
2 Discovery of a Cell-Active SuTEx Ligand of Prostaglandin Reductase 2. Chembiochem. 2021 Jun 15;22(12):2134-2139. doi: 10.1002/cbic.202000879. Epub 2021 Apr 29.
3 Reimagining high-throughput profiling of reactive cysteines for cell-based screening of large electrophile libraries. Nat Biotechnol. 2021 May;39(5):630-641. doi: 10.1038/s41587-020-00778-3. Epub 2021 Jan 4.
4 Targeted Proteomic Approaches for Proteome-Wide Characterizations of the AMP-Binding Capacities of Kinases. J Proteome Res. 2022 Aug 5;21(8):2063-2070. doi: 10.1021/acs.jproteome.2c00225. Epub 2022 Jul 12.
5 Enhancing Cysteine Chemoproteomic Coverage through Systematic Assessment of Click Chemistry Product Fragmentation. Anal Chem. 2022 Mar 8;94(9):3800-3810. doi: 10.1021/acs.analchem.1c04402. Epub 2022 Feb 23.
Mass spectrometry data entry: PXD028853
6 SP3-FAIMS Chemoproteomics for High-Coverage Profiling of the Human Cysteinome*. Chembiochem. 2021 May 14;22(10):1841-1851. doi: 10.1002/cbic.202000870. Epub 2021 Feb 18.
Mass spectrometry data entry: PXD023056 , PXD023059 , PXD023058 , PXD023057 , PXD023060
7 SP3-Enabled Rapid and High Coverage Chemoproteomic Identification of Cell-State-Dependent Redox-Sensitive Cysteines. Mol Cell Proteomics. 2022 Apr;21(4):100218. doi: 10.1016/j.mcpro.2022.100218. Epub 2022 Feb 25.
Mass spectrometry data entry: PXD029500 , PXD031647
8 A modification-centric assessment tool for the performance of chemoproteomic probes. Nat Chem Biol. 2022 Aug;18(8):904-912. doi: 10.1038/s41589-022-01074-8. Epub 2022 Jul 21.
Mass spectrometry data entry: PXD027758 , PXD027755 , PXD027760 , PXD027762 , PXD027756 , PXD027591 , PXD007149 , PXD030064 , PXD032392 , PXD027789 , PXD027767 , PXD027764
9 Solid Phase Synthesis of Fluorosulfate Containing Macrocycles for Chemoproteomic Workflows. bioRxiv [Preprint]. 2023 Feb 18:2023.02.17.529022. doi: 10.1101/2023.02.17.529022.
Mass spectrometry data entry: PXD039931
10 Tunable Amine-Reactive Electrophiles for Selective Profiling of Lysine. Angew Chem Int Ed Engl. 2022 Jan 26;61(5):e202112107. doi: 10.1002/anie.202112107. Epub 2021 Dec 16.
11 N-Acryloylindole-alkyne (NAIA) enables imaging and profiling new ligandable cysteines and oxidized thiols by chemoproteomics. Nat Commun. 2023 Jun 15;14(1):3564. doi: 10.1038/s41467-023-39268-w.
Mass spectrometry data entry: PXD041264
12 Global profiling identifies a stress-responsive tyrosine site on EDC3 regulating biomolecular condensate formation. Cell Chem Biol. 2022 Dec 15;29(12):1709-1720.e7. doi: 10.1016/j.chembiol.2022.11.008. Epub 2022 Dec 6.
Mass spectrometry data entry: PXD038010
13 Large-scale chemoproteomics expedites ligand discovery and predicts ligand behavior in cells. Science. 2024 Apr 26;384(6694):eadk5864. doi: 10.1126/science.adk5864. Epub 2024 Apr 26.
Mass spectrometry data entry: PXD041587
14 Ligand and Target Discovery by Fragment-Based Screening in Human Cells. Cell. 2017 Jan 26;168(3):527-541.e29. doi: 10.1016/j.cell.2016.12.029. Epub 2017 Jan 19.
15 Accelerating multiplexed profiling of protein-ligand interactions: High-throughput plate-based reactive cysteine profiling with minimal input. Cell Chem Biol. 2024 Mar 21;31(3):565-576.e4. doi: 10.1016/j.chembiol.2023.11.015. Epub 2023 Dec 19.
Mass spectrometry data entry: PXD044402
16 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840