General Information of Target

Target ID LDTP14589
Target Name Large ribosomal subunit protein uL3m (MRPL3)
Gene Name MRPL3
Gene ID 11222
Synonyms
MRL3; RPML3; Large ribosomal subunit protein uL3m; 39S ribosomal protein L3, mitochondrial; L3mt; MRP-L3
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MDPNCSCTTGGSCACAGSCKCKECKCTSCKKCCCSCCPVGCAKCAQGCVCKGSSEKCRCC
A
Target Bioclass
Other
Family
Universal ribosomal protein uL3 family
Subcellular location
Mitochondrion
Uniprot ID
P09001
Ensemble ID
ENST00000264995.8
HGNC ID
HGNC:10379

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 13 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
m-APA
 Probe Info 
14.40  LDD0402  [1]
N1
 Probe Info 
100.00  LDD0242  [2]
STPyne
 Probe Info 
K235(10.00)  LDD0277  [3]
Acrolein
 Probe Info 
N.A.  LDD0222  [4]
DBIA
 Probe Info 
C127(1.24)  LDD0580  [5]
ATP probe
 Probe Info 
K209(0.00); K157(0.00); K235(0.00)  LDD0199  [6]
4-Iodoacetamidophenylacetylene
 Probe Info 
N.A.  LDD0038  [7]
IA-alkyne
 Probe Info 
N.A.  LDD0032  [8]
Lodoacetamide azide
 Probe Info 
C127(0.00); C78(0.00)  LDD0037  [7]
IPM
 Probe Info 
N.A.  LDD0147  [9]
1c-yne
 Probe Info 
K188(0.00); K81(0.00)  LDD0228  [10]
NAIA_5
 Probe Info 
C127(0.00); C295(0.00); C78(0.00); C138(0.00)  LDD2223  [11]
TPP-AC
 Probe Info 
N.A.  LDD0427  [12]
PAL-AfBPP Probe
Click To Hide/Show 1 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
VE-P
 Probe Info 
N.A.  LDD0396  [13]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0214  AC1 HEK-293T C127(1.03); C78(1.32)  LDD1507  [14]
 LDCM0215  AC10 HEK-293T C127(1.19); C78(1.58)  LDD1508  [14]
 LDCM0226  AC11 HEK-293T C127(0.92); C78(1.32)  LDD1509  [14]
 LDCM0237  AC12 HEK-293T C127(1.10); C78(1.22)  LDD1510  [14]
 LDCM0246  AC128 PaTu 8988t C127(0.89)  LDD1125  [5]
 LDCM0247  AC129 PaTu 8988t C127(0.54)  LDD1126  [5]
 LDCM0249  AC130 PaTu 8988t C127(0.64)  LDD1128  [5]
 LDCM0250  AC131 PaTu 8988t C127(0.66)  LDD1129  [5]
 LDCM0251  AC132 PaTu 8988t C127(0.78)  LDD1130  [5]
 LDCM0252  AC133 PaTu 8988t C127(0.41)  LDD1131  [5]
 LDCM0253  AC134 PaTu 8988t C127(0.49)  LDD1132  [5]
 LDCM0254  AC135 PaTu 8988t C127(0.45)  LDD1133  [5]
 LDCM0255  AC136 PaTu 8988t C127(0.46)  LDD1134  [5]
 LDCM0256  AC137 PaTu 8988t C127(0.40)  LDD1135  [5]
 LDCM0257  AC138 PaTu 8988t C127(0.58)  LDD1136  [5]
 LDCM0258  AC139 PaTu 8988t C127(0.59)  LDD1137  [5]
 LDCM0259  AC14 HEK-293T C127(0.96); C78(1.63)  LDD1512  [14]
 LDCM0260  AC140 PaTu 8988t C127(0.63)  LDD1139  [5]
 LDCM0261  AC141 PaTu 8988t C127(0.74)  LDD1140  [5]
 LDCM0262  AC142 PaTu 8988t C127(0.55)  LDD1141  [5]
 LDCM0263  AC143 HCT 116 C127(1.24)  LDD0580  [5]
 LDCM0264  AC144 HCT 116 C127(0.79)  LDD0581  [5]
 LDCM0265  AC145 HCT 116 C127(0.98)  LDD0582  [5]
 LDCM0266  AC146 HCT 116 C127(1.15)  LDD0583  [5]
 LDCM0267  AC147 HCT 116 C127(0.81)  LDD0584  [5]
 LDCM0268  AC148 HCT 116 C127(0.56)  LDD0585  [5]
 LDCM0269  AC149 HCT 116 C127(0.72)  LDD0586  [5]
 LDCM0270  AC15 HEK-293T C127(0.98); C78(1.27)  LDD1513  [14]
 LDCM0271  AC150 HCT 116 C127(0.86)  LDD0588  [5]
 LDCM0272  AC151 HCT 116 C127(1.12)  LDD0589  [5]
 LDCM0273  AC152 HCT 116 C127(0.72)  LDD0590  [5]
 LDCM0274  AC153 HCT 116 C127(0.52)  LDD0591  [5]
 LDCM0621  AC154 HCT 116 C127(0.79)  LDD2158  [5]
 LDCM0622  AC155 HCT 116 C127(0.82)  LDD2159  [5]
 LDCM0623  AC156 HCT 116 C127(1.11)  LDD2160  [5]
 LDCM0624  AC157 HCT 116 C127(0.88)  LDD2161  [5]
 LDCM0276  AC17 HEK-293T C127(1.09); C78(1.51)  LDD1515  [14]
 LDCM0277  AC18 HEK-293T C127(1.12); C78(1.16)  LDD1516  [14]
 LDCM0278  AC19 HEK-293T C127(0.88); C78(1.15)  LDD1517  [14]
 LDCM0279  AC2 HEK-293T C127(1.03); C78(1.49)  LDD1518  [14]
 LDCM0280  AC20 HEK-293T C127(0.99); C78(1.30)  LDD1519  [14]
 LDCM0281  AC21 HEK-293T C127(0.94); C78(1.21)  LDD1520  [14]
 LDCM0282  AC22 HEK-293T C127(1.02); C78(1.58)  LDD1521  [14]
 LDCM0283  AC23 HEK-293T C127(0.93); C78(1.79)  LDD1522  [14]
 LDCM0284  AC24 HEK-293T C127(1.03); C78(1.25)  LDD1523  [14]
 LDCM0285  AC25 HEK-293T C127(0.96); C78(1.91)  LDD1524  [14]
 LDCM0286  AC26 HEK-293T C127(1.24); C78(1.32)  LDD1525  [14]
 LDCM0287  AC27 HEK-293T C127(0.99); C78(1.35)  LDD1526  [14]
 LDCM0288  AC28 HEK-293T C127(1.00); C78(1.25)  LDD1527  [14]
 LDCM0289  AC29 HEK-293T C127(0.97); C78(1.31)  LDD1528  [14]
 LDCM0290  AC3 HEK-293T C127(0.99); C78(1.33)  LDD1529  [14]
 LDCM0291  AC30 HEK-293T C127(0.99); C78(1.34)  LDD1530  [14]
 LDCM0292  AC31 HEK-293T C127(0.95); C78(1.22)  LDD1531  [14]
 LDCM0293  AC32 HEK-293T C127(1.13); C78(1.26)  LDD1532  [14]
 LDCM0294  AC33 HEK-293T C127(1.04); C78(1.74)  LDD1533  [14]
 LDCM0295  AC34 HEK-293T C127(0.98); C78(1.46)  LDD1534  [14]
 LDCM0296  AC35 HEK-293T C127(1.02); C78(1.57)  LDD1535  [14]
 LDCM0297  AC36 HEK-293T C127(1.05); C78(1.36)  LDD1536  [14]
 LDCM0298  AC37 HEK-293T C127(1.02); C78(1.24)  LDD1537  [14]
 LDCM0299  AC38 HEK-293T C127(0.98); C78(1.43)  LDD1538  [14]
 LDCM0300  AC39 HEK-293T C127(1.06); C78(1.26)  LDD1539  [14]
 LDCM0301  AC4 HEK-293T C127(1.02); C78(1.19)  LDD1540  [14]
 LDCM0302  AC40 HEK-293T C127(1.01); C78(1.23)  LDD1541  [14]
 LDCM0303  AC41 HEK-293T C127(1.04); C78(1.40)  LDD1542  [14]
 LDCM0304  AC42 HEK-293T C127(0.86); C78(1.65)  LDD1543  [14]
 LDCM0305  AC43 HEK-293T C127(1.12); C78(1.34)  LDD1544  [14]
 LDCM0306  AC44 HEK-293T C127(1.05); C78(1.27)  LDD1545  [14]
 LDCM0307  AC45 HEK-293T C127(0.91); C78(1.26)  LDD1546  [14]
 LDCM0308  AC46 PaTu 8988t C127(0.93)  LDD1187  [5]
 LDCM0309  AC47 PaTu 8988t C127(0.80)  LDD1188  [5]
 LDCM0310  AC48 PaTu 8988t C127(0.59)  LDD1189  [5]
 LDCM0311  AC49 PaTu 8988t C127(0.61)  LDD1190  [5]
 LDCM0312  AC5 HEK-293T C127(1.01); C78(1.28)  LDD1551  [14]
 LDCM0313  AC50 PaTu 8988t C127(0.59)  LDD1192  [5]
 LDCM0314  AC51 PaTu 8988t C127(0.95)  LDD1193  [5]
 LDCM0315  AC52 PaTu 8988t C127(0.57)  LDD1194  [5]
 LDCM0316  AC53 PaTu 8988t C127(0.47)  LDD1195  [5]
 LDCM0317  AC54 PaTu 8988t C127(0.39)  LDD1196  [5]
 LDCM0318  AC55 PaTu 8988t C127(0.80)  LDD1197  [5]
 LDCM0319  AC56 PaTu 8988t C127(0.80)  LDD1198  [5]
 LDCM0320  AC57 HCT 116 C127(0.79)  LDD0637  [5]
 LDCM0321  AC58 HCT 116 C127(0.85)  LDD0638  [5]
 LDCM0322  AC59 HCT 116 C127(0.62)  LDD0639  [5]
 LDCM0323  AC6 HEK-293T C127(0.99); C78(1.27)  LDD1562  [14]
 LDCM0324  AC60 HCT 116 C127(1.15)  LDD0641  [5]
 LDCM0325  AC61 HCT 116 C127(1.40)  LDD0642  [5]
 LDCM0326  AC62 HCT 116 C127(0.61)  LDD0643  [5]
 LDCM0327  AC63 HCT 116 C127(0.89)  LDD0644  [5]
 LDCM0328  AC64 HCT 116 C127(0.68)  LDD0645  [5]
 LDCM0329  AC65 HCT 116 C127(1.13)  LDD0646  [5]
 LDCM0330  AC66 HCT 116 C127(1.16)  LDD0647  [5]
 LDCM0331  AC67 HCT 116 C127(0.56)  LDD0648  [5]
 LDCM0334  AC7 HEK-293T C127(0.97); C78(1.33)  LDD1568  [14]
 LDCM0345  AC8 HEK-293T C127(1.11); C78(1.10)  LDD1569  [14]
 LDCM0248  AKOS034007472 HEK-293T C127(0.89); C78(1.17)  LDD1511  [14]
 LDCM0356  AKOS034007680 HEK-293T C127(1.14); C78(1.64)  LDD1570  [14]
 LDCM0275  AKOS034007705 HEK-293T C127(1.00); C78(1.20)  LDD1514  [14]
 LDCM0108  Chloroacetamide HeLa N.A.  LDD0222  [4]
 LDCM0632  CL-Sc Hep-G2 C78(1.52); C138(1.07)  LDD2227  [11]
 LDCM0367  CL1 HCT 116 C127(0.82)  LDD0684  [5]
 LDCM0368  CL10 HCT 116 C127(0.89)  LDD0685  [5]
 LDCM0369  CL100 HEK-293T C127(1.00); C78(1.67)  LDD1573  [14]
 LDCM0370  CL101 HEK-293T C127(1.01); C78(1.36)  LDD1574  [14]
 LDCM0371  CL102 HEK-293T C127(1.02); C78(1.22)  LDD1575  [14]
 LDCM0372  CL103 HEK-293T C127(1.06); C78(1.33)  LDD1576  [14]
 LDCM0373  CL104 HEK-293T C127(0.99); C78(1.48)  LDD1577  [14]
 LDCM0374  CL105 HEK-293T C127(1.02); C78(1.26)  LDD1578  [14]
 LDCM0375  CL106 HEK-293T C127(1.03); C78(1.15)  LDD1579  [14]
 LDCM0376  CL107 HEK-293T C127(0.99); C78(1.28)  LDD1580  [14]
 LDCM0377  CL108 HEK-293T C127(1.19); C78(1.45)  LDD1581  [14]
 LDCM0378  CL109 HEK-293T C127(1.04); C78(1.36)  LDD1582  [14]
 LDCM0379  CL11 HCT 116 C127(0.89)  LDD0696  [5]
 LDCM0380  CL110 HEK-293T C127(1.01); C78(1.21)  LDD1584  [14]
 LDCM0381  CL111 HEK-293T C127(1.02); C78(1.21)  LDD1585  [14]
 LDCM0382  CL112 HEK-293T C127(1.06); C78(1.66)  LDD1586  [14]
 LDCM0383  CL113 HEK-293T C127(1.07); C78(1.44)  LDD1587  [14]
 LDCM0384  CL114 HEK-293T C127(1.05); C78(1.32)  LDD1588  [14]
 LDCM0385  CL115 HEK-293T C127(1.13); C78(1.13)  LDD1589  [14]
 LDCM0386  CL116 HEK-293T C127(1.00); C78(1.71)  LDD1590  [14]
 LDCM0387  CL117 HEK-293T C127(1.03); C78(1.42)  LDD1591  [14]
 LDCM0388  CL118 HEK-293T C127(0.92); C78(1.11)  LDD1592  [14]
 LDCM0389  CL119 HEK-293T C127(1.09); C78(1.36)  LDD1593  [14]
 LDCM0390  CL12 HCT 116 C127(0.73)  LDD0707  [5]
 LDCM0391  CL120 HEK-293T C127(1.10); C78(1.53)  LDD1595  [14]
 LDCM0392  CL121 PaTu 8988t C127(0.86)  LDD1271  [5]
 LDCM0393  CL122 PaTu 8988t C127(0.79)  LDD1272  [5]
 LDCM0394  CL123 PaTu 8988t C127(0.57)  LDD1273  [5]
 LDCM0395  CL124 PaTu 8988t C127(0.64)  LDD1274  [5]
 LDCM0396  CL125 HCT 116 C127(1.42)  LDD0713  [5]
 LDCM0397  CL126 HCT 116 C127(1.11)  LDD0714  [5]
 LDCM0398  CL127 HCT 116 C127(1.16)  LDD0715  [5]
 LDCM0399  CL128 HCT 116 C127(0.65)  LDD0716  [5]
 LDCM0400  CL13 HCT 116 C127(0.95)  LDD0717  [5]
 LDCM0401  CL14 HCT 116 C127(1.01)  LDD0718  [5]
 LDCM0402  CL15 HCT 116 C127(1.14)  LDD0719  [5]
 LDCM0403  CL16 PaTu 8988t C127(0.80)  LDD1282  [5]
 LDCM0404  CL17 PaTu 8988t C127(0.69)  LDD1283  [5]
 LDCM0405  CL18 PaTu 8988t C127(0.58)  LDD1284  [5]
 LDCM0406  CL19 PaTu 8988t C127(0.72)  LDD1285  [5]
 LDCM0407  CL2 HCT 116 C127(0.98)  LDD0724  [5]
 LDCM0408  CL20 PaTu 8988t C127(0.74)  LDD1287  [5]
 LDCM0409  CL21 PaTu 8988t C127(0.68)  LDD1288  [5]
 LDCM0410  CL22 PaTu 8988t C127(0.73)  LDD1289  [5]
 LDCM0411  CL23 PaTu 8988t C127(0.78)  LDD1290  [5]
 LDCM0412  CL24 PaTu 8988t C127(1.11)  LDD1291  [5]
 LDCM0413  CL25 PaTu 8988t C127(0.96)  LDD1292  [5]
 LDCM0414  CL26 PaTu 8988t C127(0.60)  LDD1293  [5]
 LDCM0415  CL27 PaTu 8988t C127(0.87)  LDD1294  [5]
 LDCM0416  CL28 PaTu 8988t C127(0.78)  LDD1295  [5]
 LDCM0417  CL29 PaTu 8988t C127(0.87)  LDD1296  [5]
 LDCM0418  CL3 HCT 116 C127(0.97)  LDD0735  [5]
 LDCM0419  CL30 PaTu 8988t C127(1.15)  LDD1298  [5]
 LDCM0420  CL31 PaTu 8988t C127(1.08)  LDD1299  [5]
 LDCM0421  CL32 PaTu 8988t C127(0.92)  LDD1300  [5]
 LDCM0422  CL33 PaTu 8988t C127(0.82)  LDD1301  [5]
 LDCM0423  CL34 PaTu 8988t C127(1.06)  LDD1302  [5]
 LDCM0424  CL35 PaTu 8988t C127(0.67)  LDD1303  [5]
 LDCM0425  CL36 PaTu 8988t C127(1.17)  LDD1304  [5]
 LDCM0426  CL37 PaTu 8988t C127(0.71)  LDD1305  [5]
 LDCM0428  CL39 PaTu 8988t C127(1.04)  LDD1307  [5]
 LDCM0429  CL4 HCT 116 C127(1.05)  LDD0746  [5]
 LDCM0430  CL40 PaTu 8988t C127(0.95)  LDD1309  [5]
 LDCM0431  CL41 PaTu 8988t C127(0.60)  LDD1310  [5]
 LDCM0432  CL42 PaTu 8988t C127(0.51)  LDD1311  [5]
 LDCM0433  CL43 PaTu 8988t C127(0.72)  LDD1312  [5]
 LDCM0434  CL44 PaTu 8988t C127(0.81)  LDD1313  [5]
 LDCM0435  CL45 PaTu 8988t C127(0.99)  LDD1314  [5]
 LDCM0436  CL46 HEK-293T C127(1.07); C78(0.42)  LDD1640  [14]
 LDCM0437  CL47 HEK-293T C127(1.06); C78(0.30)  LDD1641  [14]
 LDCM0438  CL48 HEK-293T C127(1.16); C78(0.25)  LDD1642  [14]
 LDCM0439  CL49 HEK-293T C127(1.22); C78(1.27)  LDD1643  [14]
 LDCM0440  CL5 HCT 116 C127(0.92)  LDD0757  [5]
 LDCM0441  CL50 HEK-293T C127(0.88); C78(1.17)  LDD1645  [14]
 LDCM0443  CL52 HEK-293T C127(1.12); C78(1.29)  LDD1646  [14]
 LDCM0444  CL53 HEK-293T C127(1.06); C78(1.09)  LDD1647  [14]
 LDCM0445  CL54 HEK-293T C127(1.00); C78(0.76)  LDD1648  [14]
 LDCM0446  CL55 HEK-293T C127(1.13); C78(0.58)  LDD1649  [14]
 LDCM0447  CL56 HEK-293T C127(1.05); C78(0.59)  LDD1650  [14]
 LDCM0448  CL57 HEK-293T C127(0.91); C78(0.41)  LDD1651  [14]
 LDCM0449  CL58 HEK-293T C127(0.99); C78(0.36)  LDD1652  [14]
 LDCM0450  CL59 HEK-293T C127(1.12); C78(0.32)  LDD1653  [14]
 LDCM0451  CL6 HCT 116 C127(1.24)  LDD0768  [5]
 LDCM0452  CL60 HEK-293T C127(1.01); C78(0.32)  LDD1655  [14]
 LDCM0453  CL61 PaTu 8988t C127(1.16)  LDD1332  [5]
 LDCM0454  CL62 PaTu 8988t C127(1.08)  LDD1333  [5]
 LDCM0455  CL63 PaTu 8988t C127(1.17)  LDD1334  [5]
 LDCM0456  CL64 PaTu 8988t C127(0.86)  LDD1335  [5]
 LDCM0457  CL65 PaTu 8988t C127(0.72)  LDD1336  [5]
 LDCM0458  CL66 PaTu 8988t C127(0.76)  LDD1337  [5]
 LDCM0459  CL67 PaTu 8988t C127(0.41)  LDD1338  [5]
 LDCM0460  CL68 PaTu 8988t C127(0.38)  LDD1339  [5]
 LDCM0461  CL69 PaTu 8988t C127(0.40)  LDD1340  [5]
 LDCM0462  CL7 HCT 116 C127(0.94)  LDD0779  [5]
 LDCM0463  CL70 PaTu 8988t C127(0.40)  LDD1342  [5]
 LDCM0464  CL71 PaTu 8988t C127(1.23)  LDD1343  [5]
 LDCM0465  CL72 PaTu 8988t C127(1.39)  LDD1344  [5]
 LDCM0466  CL73 PaTu 8988t C127(0.43)  LDD1345  [5]
 LDCM0467  CL74 PaTu 8988t C127(1.52)  LDD1346  [5]
 LDCM0469  CL76 HCT 116 C127(1.08)  LDD0786  [5]
 LDCM0470  CL77 HCT 116 C127(0.92)  LDD0787  [5]
 LDCM0471  CL78 HCT 116 C127(0.96)  LDD0788  [5]
 LDCM0472  CL79 HCT 116 C127(0.61)  LDD0789  [5]
 LDCM0473  CL8 HCT 116 C127(0.77)  LDD0790  [5]
 LDCM0474  CL80 HCT 116 C127(0.86)  LDD0791  [5]
 LDCM0475  CL81 HCT 116 C127(0.86)  LDD0792  [5]
 LDCM0476  CL82 HCT 116 C127(0.51)  LDD0793  [5]
 LDCM0477  CL83 HCT 116 C127(0.58)  LDD0794  [5]
 LDCM0478  CL84 HCT 116 C127(0.52)  LDD0795  [5]
 LDCM0479  CL85 HCT 116 C127(0.94)  LDD0796  [5]
 LDCM0480  CL86 HCT 116 C127(1.03)  LDD0797  [5]
 LDCM0481  CL87 HCT 116 C127(0.83)  LDD0798  [5]
 LDCM0482  CL88 HCT 116 C127(0.62)  LDD0799  [5]
 LDCM0483  CL89 HCT 116 C127(0.61)  LDD0800  [5]
 LDCM0484  CL9 HCT 116 C127(0.92)  LDD0801  [5]
 LDCM0485  CL90 HCT 116 C127(0.99)  LDD0802  [5]
 LDCM0486  CL91 HEK-293T C127(1.10); C78(0.76)  LDD1689  [14]
 LDCM0487  CL92 HEK-293T C127(1.12); C78(0.75)  LDD1690  [14]
 LDCM0488  CL93 HEK-293T C127(1.03); C78(0.53)  LDD1691  [14]
 LDCM0489  CL94 HEK-293T C127(1.05); C78(0.64)  LDD1692  [14]
 LDCM0490  CL95 HEK-293T C127(0.95); C78(0.54)  LDD1693  [14]
 LDCM0491  CL96 HEK-293T C127(1.09); C78(0.57)  LDD1694  [14]
 LDCM0492  CL97 HEK-293T C127(1.08); C78(1.35)  LDD1695  [14]
 LDCM0493  CL98 HEK-293T C127(1.18); C78(1.21)  LDD1696  [14]
 LDCM0494  CL99 HEK-293T C127(1.11); C78(1.14)  LDD1697  [14]
 LDCM0495  E2913 HEK-293T C127(1.15); C78(1.13)  LDD1698  [14]
 LDCM0625  F8 Ramos C138(1.57); C78(1.49)  LDD2187  [15]
 LDCM0572  Fragment10 Ramos C138(0.49); C78(1.24)  LDD2189  [15]
 LDCM0573  Fragment11 Ramos C138(20.00); C78(1.02)  LDD2190  [15]
 LDCM0574  Fragment12 Ramos C138(0.40); C78(0.78)  LDD2191  [15]
 LDCM0575  Fragment13 Ramos C138(0.77); C78(0.85)  LDD2192  [15]
 LDCM0576  Fragment14 Ramos C138(0.59); C78(0.69)  LDD2193  [15]
 LDCM0579  Fragment20 Ramos C138(0.39); C78(0.50)  LDD2194  [15]
 LDCM0580  Fragment21 Ramos C138(0.95); C78(0.67)  LDD2195  [15]
 LDCM0582  Fragment23 Ramos C138(0.55); C78(1.24)  LDD2196  [15]
 LDCM0578  Fragment27 Ramos C138(0.79); C78(0.91)  LDD2197  [15]
 LDCM0586  Fragment28 Ramos C138(0.37); C78(1.02)  LDD2198  [15]
 LDCM0588  Fragment30 Ramos C138(0.87); C78(0.74)  LDD2199  [15]
 LDCM0589  Fragment31 Ramos C138(0.52); C78(0.49)  LDD2200  [15]
 LDCM0590  Fragment32 Ramos C138(0.52); C78(1.10)  LDD2201  [15]
 LDCM0468  Fragment33 PaTu 8988t C127(0.66)  LDD1347  [5]
 LDCM0596  Fragment38 Ramos C138(0.55); C78(1.50)  LDD2203  [15]
 LDCM0566  Fragment4 Ramos C138(0.59); C78(0.77)  LDD2184  [15]
 LDCM0427  Fragment51 PaTu 8988t C127(0.78)  LDD1306  [5]
 LDCM0610  Fragment52 Ramos C138(0.85); C78(0.80)  LDD2204  [15]
 LDCM0614  Fragment56 Ramos C138(1.07); C78(0.69)  LDD2205  [15]
 LDCM0569  Fragment7 Ramos C138(0.48); C78(0.85)  LDD2186  [15]
 LDCM0571  Fragment9 Ramos C138(0.46); C78(1.16)  LDD2188  [15]
 LDCM0022  KB02 HEK-293T C127(0.95); C78(1.01); C338(1.16)  LDD1492  [14]
 LDCM0023  KB03 HEK-293T C127(0.90); C78(0.91); C338(1.16)  LDD1497  [14]
 LDCM0024  KB05 COLO792 C127(1.28)  LDD3310  [16]
 LDCM0627  NUDT7-COV-1 HEK-293T C78(0.09)  LDD2206  [17]
 LDCM0628  OTUB2-COV-1 HEK-293T C78(0.15)  LDD2207  [17]

References

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2 Cyclopropenone, Cyclopropeniminium Ion, and Cyclopropenethione as Novel Electrophilic Warheads for Potential Target Discovery of Triple-Negative Breast Cancer. J Med Chem. 2023 Feb 23;66(4):2851-2864. doi: 10.1021/acs.jmedchem.2c01889. Epub 2023 Feb 10.
3 A Paal-Knorr agent for chemoproteomic profiling of targets of isoketals in cells. Chem Sci. 2021 Oct 15;12(43):14557-14563. doi: 10.1039/d1sc02230j. eCollection 2021 Nov 10.
Mass spectrometry data entry: PXD028270
4 ACR-Based Probe for the Quantitative Profiling of Histidine Reactivity in the Human Proteome. J Am Chem Soc. 2023 Mar 8;145(9):5252-5260. doi: 10.1021/jacs.2c12653. Epub 2023 Feb 27.
5 Reimagining high-throughput profiling of reactive cysteines for cell-based screening of large electrophile libraries. Nat Biotechnol. 2021 May;39(5):630-641. doi: 10.1038/s41587-020-00778-3. Epub 2021 Jan 4.
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Mass spectrometry data entry: PXD028853
8 SP3-FAIMS Chemoproteomics for High-Coverage Profiling of the Human Cysteinome*. Chembiochem. 2021 May 14;22(10):1841-1851. doi: 10.1002/cbic.202000870. Epub 2021 Feb 18.
Mass spectrometry data entry: PXD023056 , PXD023059 , PXD023058 , PXD023057 , PXD023060
9 Chemoproteomic Profiling by Cysteine Fluoroalkylation Reveals Myrocin G as an Inhibitor of the Nonhomologous End Joining DNA Repair Pathway. J Am Chem Soc. 2021 Dec 8;143(48):20332-20342. doi: 10.1021/jacs.1c09724. Epub 2021 Nov 24.
Mass spectrometry data entry: PXD029255
10 Tunable Amine-Reactive Electrophiles for Selective Profiling of Lysine. Angew Chem Int Ed Engl. 2022 Jan 26;61(5):e202112107. doi: 10.1002/anie.202112107. Epub 2021 Dec 16.
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Mass spectrometry data entry: PXD041264
12 Differently Tagged Probes for Protein Profiling of Mitochondria. Chembiochem. 2019 May 2;20(9):1155-1160. doi: 10.1002/cbic.201800735. Epub 2019 Mar 26.
13 Pharmacological Targeting of Vacuolar H(+)-ATPase via Subunit V1G Combats Multidrug-Resistant Cancer. Cell Chem Biol. 2020 Nov 19;27(11):1359-1370.e8. doi: 10.1016/j.chembiol.2020.06.011. Epub 2020 Jul 9.
14 Accelerating multiplexed profiling of protein-ligand interactions: High-throughput plate-based reactive cysteine profiling with minimal input. Cell Chem Biol. 2024 Mar 21;31(3):565-576.e4. doi: 10.1016/j.chembiol.2023.11.015. Epub 2023 Dec 19.
Mass spectrometry data entry: PXD044402
15 Site-specific quantitative cysteine profiling with data-independent acquisition-based mass spectrometry. Methods Enzymol. 2023;679:295-322. doi: 10.1016/bs.mie.2022.07.037. Epub 2022 Sep 7.
Mass spectrometry data entry: PXD027578
16 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840
17 Rapid Covalent-Probe Discovery by Electrophile-Fragment Screening. J Am Chem Soc. 2019 Jun 5;141(22):8951-8968. doi: 10.1021/jacs.9b02822. Epub 2019 May 22.