General Information of Target

Target ID LDTP10715
Target Name BTB/POZ domain-containing protein 9 (BTBD9)
Gene Name BTBD9
Gene ID 114781
Synonyms
KIAA1880; BTB/POZ domain-containing protein 9
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MSAPDEGRRDPPKPKGKTLGSFFGSLPGFSSARNLVANAHSSARARPAADPTGAPAAEAA
QPQAQVAAHPEQTAPWTEKELQPSEKMVSGAKDLVCSKMSRAKDAVSSGVASVVDVAKGV
VQGGLDTTRSALTGTKEVVSSGVTGAMDMAKGAVQGGLDTSKAVLTGTKDTVSTGLTGAV
NVAKGTVQAGVDTTKTVLTGTKDTVTTGVMGAVNLAKGTVQTGVETSKAVLTGTKDAVST
GLTGAVNVARGSIQTGVDTSKTVLTGTKDTVCSGVTGAMNVAKGTIQTGVDTSKTVLTGT
KDTVCSGVTGAMNVAKGTIQTGVDTSKTVLTGTKDTVCSGVTGAMNVAKGTIQTGVDTTK
TVLTGTKNTVCSGVTGAVNLAKEAIQGGLDTTKSMVMGTKDTMSTGLTGAANVAKGAMQT
GLNTTQNIATGTKDTVCSGVTGAMNLARGTIQTGVDTTKIVLTGTKDTVCSGVTGAANVA
KGAVQGGLDTTKSVLTGTKDAVSTGLTGAVNVAKGTVQTGVDTTKTVLTGTKDTVCSGVT
SAVNVAKGAVQGGLDTTKSVVIGTKDTMSTGLTGAANVAKGAVQTGVDTAKTVLTGTKDT
VTTGLVGAVNVAKGTVQTGMDTTKTVLTGTKDTIYSGVTSAVNVAKGAVQTGLKTTQNIA
TGTKNTFGSGVTSAVNVAKGAAQTGVDTAKTVLTGTKDTVTTGLMGAVNVAKGTVQTSVD
TTKTVLTGTKDTVCSGVTGAANVAKGAIQGGLDTTKSVLTGTKDAVSTGLTGAVKLAKGT
VQTGMDTTKTVLTGTKDAVCSGVTGAANVAKGAVQMGVDTAKTVLTGTKDTVCSGVTGAA
NVAKGAVQTGLKTTQNIATGTKNTLGSGVTGAAKVAKGAVQGGLDTTKSVLTGTKDAVST
GLTGAVNLAKGTVQTGVDTSKTVLTGTKDTVCSGVTGAVNVAKGTVQTGVDTAKTVLSGA
KDAVTTGVTGAVNVAKGTVQTGVDASKAVLMGTKDTVFSGVTGAMSMAKGAVQGGLDTTK
TVLTGTKDAVSAGLMGSGNVATGATHTGLSTFQNWLPSTPATSWGGLTSSRTTDNGGEQT
ALSPQEAPFSGISTPPDVLSVGPEPAWEAAATTKGLATDVATFTQGAAPGREDTGLLATT
HGPEEAPRLAMLQNELEGLGDIFHPMNAEEQAQLAASQPGPKVLSAEQGSYFVRLGDLGP
SFRQRAFEHAVSHLQHGQFQARDTLAQLQDCFRLIEKAQQAPEGQPRLDQGSGASAEDAA
VQEERDAGVLSRVCGLLRQLHTAYSGLVSSLQGLPAELQQPVGRARHSLCELYGIVASAG
SVEELPAERLVQSREGVHQAWQGLEQLLEGLQHNPPLSWLVGPFALPAGGQ
Target Bioclass
Other
Uniprot ID
Q96Q07
Ensemble ID
ENST00000314100.10
HGNC ID
HGNC:21228

Target Site Mutations in Different Cell Lines

Cell line Mutation details Probe for labeling this protein in this cell
CAL62 SNV: p.A28T .
CCK81 SNV: p.D341G .
HCT15 SNV: p.T145N .
IGROV1 SNV: p.G601C .
LNCaP clone FGC SNV: p.N411S .
MFE319 SNV: p.H5R .
RL952 SNV: p.R442Q .
SUPT1 SNV: p.E323K .
SW1271 SNV: p.P600Q .

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 2 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
DBIA
 Probe Info 
C318(1.00)  LDD0531  [1]
IA-alkyne
 Probe Info 
N.A.  LDD0165  [2]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0214  AC1 HCT 116 C318(1.00)  LDD0531  [1]
 LDCM0215  AC10 PaTu 8988t C210(0.87)  LDD1094  [1]
 LDCM0226  AC11 PaTu 8988t C210(0.81)  LDD1105  [1]
 LDCM0230  AC113 PaTu 8988t C210(1.06)  LDD1109  [1]
 LDCM0231  AC114 PaTu 8988t C210(1.13)  LDD1110  [1]
 LDCM0232  AC115 PaTu 8988t C210(1.07)  LDD1111  [1]
 LDCM0233  AC116 PaTu 8988t C210(0.96)  LDD1112  [1]
 LDCM0234  AC117 PaTu 8988t C210(1.14)  LDD1113  [1]
 LDCM0235  AC118 PaTu 8988t C210(1.08)  LDD1114  [1]
 LDCM0236  AC119 PaTu 8988t C210(1.08)  LDD1115  [1]
 LDCM0237  AC12 PaTu 8988t C210(0.81)  LDD1116  [1]
 LDCM0238  AC120 PaTu 8988t C210(1.13)  LDD1117  [1]
 LDCM0239  AC121 PaTu 8988t C210(0.92)  LDD1118  [1]
 LDCM0240  AC122 PaTu 8988t C210(1.09)  LDD1119  [1]
 LDCM0241  AC123 PaTu 8988t C210(1.04)  LDD1120  [1]
 LDCM0242  AC124 PaTu 8988t C210(1.13)  LDD1121  [1]
 LDCM0243  AC125 PaTu 8988t C210(0.96)  LDD1122  [1]
 LDCM0244  AC126 PaTu 8988t C210(1.36)  LDD1123  [1]
 LDCM0245  AC127 PaTu 8988t C210(1.08)  LDD1124  [1]
 LDCM0246  AC128 PaTu 8988t C210(0.87)  LDD1125  [1]
 LDCM0247  AC129 PaTu 8988t C210(0.83)  LDD1126  [1]
 LDCM0249  AC130 PaTu 8988t C210(1.04)  LDD1128  [1]
 LDCM0250  AC131 PaTu 8988t C210(1.07)  LDD1129  [1]
 LDCM0251  AC132 PaTu 8988t C210(0.96)  LDD1130  [1]
 LDCM0252  AC133 PaTu 8988t C210(0.92)  LDD1131  [1]
 LDCM0253  AC134 PaTu 8988t C210(0.98)  LDD1132  [1]
 LDCM0254  AC135 PaTu 8988t C210(0.92)  LDD1133  [1]
 LDCM0255  AC136 PaTu 8988t C210(0.91)  LDD1134  [1]
 LDCM0256  AC137 PaTu 8988t C210(0.94)  LDD1135  [1]
 LDCM0257  AC138 PaTu 8988t C210(0.79)  LDD1136  [1]
 LDCM0258  AC139 PaTu 8988t C210(1.09)  LDD1137  [1]
 LDCM0259  AC14 PaTu 8988t C210(0.93)  LDD1138  [1]
 LDCM0260  AC140 PaTu 8988t C210(0.78)  LDD1139  [1]
 LDCM0261  AC141 PaTu 8988t C210(0.84)  LDD1140  [1]
 LDCM0262  AC142 PaTu 8988t C210(0.86)  LDD1141  [1]
 LDCM0270  AC15 PaTu 8988t C210(0.84)  LDD1149  [1]
 LDCM0276  AC17 PaTu 8988t C210(0.78); C318(1.01)  LDD1155  [1]
 LDCM0277  AC18 PaTu 8988t C210(0.69); C318(1.18)  LDD1156  [1]
 LDCM0278  AC19 PaTu 8988t C210(0.76); C318(1.13)  LDD1157  [1]
 LDCM0279  AC2 HCT 116 C318(1.14)  LDD0596  [1]
 LDCM0280  AC20 PaTu 8988t C210(0.71); C318(1.16)  LDD1159  [1]
 LDCM0281  AC21 PaTu 8988t C210(0.69); C318(1.21)  LDD1160  [1]
 LDCM0282  AC22 PaTu 8988t C210(0.77); C318(1.36)  LDD1161  [1]
 LDCM0283  AC23 PaTu 8988t C210(0.67); C318(1.32)  LDD1162  [1]
 LDCM0284  AC24 PaTu 8988t C210(0.76); C318(1.19)  LDD1163  [1]
 LDCM0285  AC25 PaTu 8988t C210(0.84); C318(0.91)  LDD1164  [1]
 LDCM0286  AC26 PaTu 8988t C210(0.82); C318(1.05)  LDD1165  [1]
 LDCM0287  AC27 PaTu 8988t C210(0.85); C318(1.00)  LDD1166  [1]
 LDCM0288  AC28 PaTu 8988t C210(0.72); C318(1.11)  LDD1167  [1]
 LDCM0289  AC29 PaTu 8988t C210(0.79); C318(1.12)  LDD1168  [1]
 LDCM0290  AC3 HCT 116 C318(1.06)  LDD0607  [1]
 LDCM0291  AC30 PaTu 8988t C210(0.83); C318(1.05)  LDD1170  [1]
 LDCM0292  AC31 PaTu 8988t C210(0.92); C318(0.92)  LDD1171  [1]
 LDCM0293  AC32 PaTu 8988t C210(0.93); C318(1.01)  LDD1172  [1]
 LDCM0294  AC33 PaTu 8988t C210(0.68); C318(1.04)  LDD1173  [1]
 LDCM0295  AC34 PaTu 8988t C210(0.79); C318(1.14)  LDD1174  [1]
 LDCM0296  AC35 PaTu 8988t C210(0.75); C318(0.79)  LDD1175  [1]
 LDCM0297  AC36 PaTu 8988t C210(0.64); C318(1.14)  LDD1176  [1]
 LDCM0298  AC37 PaTu 8988t C210(0.67); C318(1.17)  LDD1177  [1]
 LDCM0299  AC38 PaTu 8988t C210(0.83); C318(1.06)  LDD1178  [1]
 LDCM0300  AC39 PaTu 8988t C210(0.71); C318(1.08)  LDD1179  [1]
 LDCM0301  AC4 HCT 116 C318(1.08)  LDD0618  [1]
 LDCM0302  AC40 PaTu 8988t C210(0.73); C318(1.19)  LDD1181  [1]
 LDCM0303  AC41 PaTu 8988t C210(0.76); C318(1.13)  LDD1182  [1]
 LDCM0304  AC42 PaTu 8988t C210(0.79); C318(1.29)  LDD1183  [1]
 LDCM0305  AC43 PaTu 8988t C210(0.73); C318(1.06)  LDD1184  [1]
 LDCM0306  AC44 PaTu 8988t C210(0.61); C318(1.42)  LDD1185  [1]
 LDCM0307  AC45 PaTu 8988t C210(0.74); C318(1.42)  LDD1186  [1]
 LDCM0308  AC46 PaTu 8988t C210(0.82); C318(1.02)  LDD1187  [1]
 LDCM0309  AC47 PaTu 8988t C210(0.82); C318(1.14)  LDD1188  [1]
 LDCM0310  AC48 PaTu 8988t C210(0.76); C318(1.31)  LDD1189  [1]
 LDCM0311  AC49 PaTu 8988t C210(0.79); C318(1.42)  LDD1190  [1]
 LDCM0312  AC5 HCT 116 C318(1.16)  LDD0629  [1]
 LDCM0313  AC50 PaTu 8988t C210(0.72); C318(1.35)  LDD1192  [1]
 LDCM0314  AC51 PaTu 8988t C210(0.76); C318(0.32)  LDD1193  [1]
 LDCM0315  AC52 PaTu 8988t C210(0.82); C318(1.28)  LDD1194  [1]
 LDCM0316  AC53 PaTu 8988t C210(0.72); C318(1.36)  LDD1195  [1]
 LDCM0317  AC54 PaTu 8988t C210(0.83); C318(1.46)  LDD1196  [1]
 LDCM0318  AC55 PaTu 8988t C210(0.72); C318(1.25)  LDD1197  [1]
 LDCM0319  AC56 PaTu 8988t C210(0.90); C318(1.57)  LDD1198  [1]
 LDCM0320  AC57 PaTu 8988t C210(1.04)  LDD1199  [1]
 LDCM0321  AC58 PaTu 8988t C210(0.97)  LDD1200  [1]
 LDCM0322  AC59 PaTu 8988t C210(1.01)  LDD1201  [1]
 LDCM0323  AC6 PaTu 8988t C210(0.89)  LDD1202  [1]
 LDCM0324  AC60 PaTu 8988t C210(0.98)  LDD1203  [1]
 LDCM0325  AC61 PaTu 8988t C210(1.03)  LDD1204  [1]
 LDCM0326  AC62 PaTu 8988t C210(1.05)  LDD1205  [1]
 LDCM0327  AC63 PaTu 8988t C210(1.01)  LDD1206  [1]
 LDCM0328  AC64 PaTu 8988t C210(1.03)  LDD1207  [1]
 LDCM0329  AC65 PaTu 8988t C210(1.02)  LDD1208  [1]
 LDCM0330  AC66 PaTu 8988t C210(0.95)  LDD1209  [1]
 LDCM0331  AC67 PaTu 8988t C210(1.11)  LDD1210  [1]
 LDCM0332  AC68 PaTu 8988t C318(1.07)  LDD1211  [1]
 LDCM0333  AC69 PaTu 8988t C318(0.98)  LDD1212  [1]
 LDCM0334  AC7 PaTu 8988t C210(1.03)  LDD1213  [1]
 LDCM0335  AC70 PaTu 8988t C318(0.91)  LDD1214  [1]
 LDCM0336  AC71 PaTu 8988t C318(0.92)  LDD1215  [1]
 LDCM0337  AC72 PaTu 8988t C318(1.12)  LDD1216  [1]
 LDCM0338  AC73 PaTu 8988t C318(0.93)  LDD1217  [1]
 LDCM0339  AC74 PaTu 8988t C318(1.08)  LDD1218  [1]
 LDCM0340  AC75 PaTu 8988t C318(1.16)  LDD1219  [1]
 LDCM0341  AC76 PaTu 8988t C318(1.20)  LDD1220  [1]
 LDCM0342  AC77 PaTu 8988t C318(1.21)  LDD1221  [1]
 LDCM0343  AC78 PaTu 8988t C318(1.26)  LDD1222  [1]
 LDCM0344  AC79 PaTu 8988t C318(1.20)  LDD1223  [1]
 LDCM0345  AC8 PaTu 8988t C210(1.09)  LDD1224  [1]
 LDCM0346  AC80 PaTu 8988t C318(1.14)  LDD1225  [1]
 LDCM0347  AC81 PaTu 8988t C318(2.95)  LDD1226  [1]
 LDCM0348  AC82 PaTu 8988t C318(1.21)  LDD1227  [1]
 LDCM0248  AKOS034007472 PaTu 8988t C210(0.89)  LDD1127  [1]
 LDCM0356  AKOS034007680 PaTu 8988t C210(0.91)  LDD1235  [1]
 LDCM0275  AKOS034007705 PaTu 8988t C210(0.83)  LDD1154  [1]
 LDCM0367  CL1 PaTu 8988t C318(1.11)  LDD1246  [1]
 LDCM0368  CL10 PaTu 8988t C318(1.16)  LDD1247  [1]
 LDCM0369  CL100 HCT 116 C318(1.00)  LDD0686  [1]
 LDCM0370  CL101 PaTu 8988t C210(0.91)  LDD1249  [1]
 LDCM0371  CL102 PaTu 8988t C210(0.93)  LDD1250  [1]
 LDCM0372  CL103 PaTu 8988t C210(0.95)  LDD1251  [1]
 LDCM0373  CL104 PaTu 8988t C210(1.00)  LDD1252  [1]
 LDCM0374  CL105 PaTu 8988t C210(0.76); C318(0.92)  LDD1253  [1]
 LDCM0375  CL106 PaTu 8988t C210(0.81); C318(0.97)  LDD1254  [1]
 LDCM0376  CL107 PaTu 8988t C210(0.74); C318(0.92)  LDD1255  [1]
 LDCM0377  CL108 PaTu 8988t C210(0.77); C318(0.94)  LDD1256  [1]
 LDCM0378  CL109 PaTu 8988t C210(0.74); C318(0.94)  LDD1257  [1]
 LDCM0379  CL11 PaTu 8988t C318(1.33)  LDD1258  [1]
 LDCM0380  CL110 PaTu 8988t C210(0.65); C318(0.94)  LDD1259  [1]
 LDCM0381  CL111 PaTu 8988t C210(0.69); C318(1.20)  LDD1260  [1]
 LDCM0382  CL112 PaTu 8988t C210(0.82); C318(0.92)  LDD1261  [1]
 LDCM0383  CL113 PaTu 8988t C210(0.76); C318(1.01)  LDD1262  [1]
 LDCM0384  CL114 PaTu 8988t C210(0.75); C318(1.00)  LDD1263  [1]
 LDCM0385  CL115 PaTu 8988t C210(0.74); C318(0.96)  LDD1264  [1]
 LDCM0386  CL116 PaTu 8988t C210(0.84); C318(1.00)  LDD1265  [1]
 LDCM0387  CL117 PaTu 8988t C210(0.78); C318(1.19)  LDD1266  [1]
 LDCM0388  CL118 PaTu 8988t C210(0.91); C318(1.12)  LDD1267  [1]
 LDCM0389  CL119 PaTu 8988t C210(0.64); C318(1.08)  LDD1268  [1]
 LDCM0390  CL12 PaTu 8988t C318(1.43)  LDD1269  [1]
 LDCM0391  CL120 PaTu 8988t C210(0.64); C318(0.89)  LDD1270  [1]
 LDCM0392  CL121 PaTu 8988t C210(0.85); C318(0.99)  LDD1271  [1]
 LDCM0393  CL122 PaTu 8988t C210(0.91); C318(1.22)  LDD1272  [1]
 LDCM0394  CL123 PaTu 8988t C210(0.87); C318(1.33)  LDD1273  [1]
 LDCM0395  CL124 PaTu 8988t C210(0.77); C318(1.64)  LDD1274  [1]
 LDCM0396  CL125 PaTu 8988t C210(1.00)  LDD1275  [1]
 LDCM0397  CL126 PaTu 8988t C210(1.00)  LDD1276  [1]
 LDCM0398  CL127 PaTu 8988t C210(1.01)  LDD1277  [1]
 LDCM0399  CL128 PaTu 8988t C210(1.04)  LDD1278  [1]
 LDCM0400  CL13 PaTu 8988t C318(1.54)  LDD1279  [1]
 LDCM0401  CL14 PaTu 8988t C318(1.97)  LDD1280  [1]
 LDCM0402  CL15 PaTu 8988t C318(1.91)  LDD1281  [1]
 LDCM0403  CL16 PaTu 8988t C318(1.12)  LDD1282  [1]
 LDCM0404  CL17 PaTu 8988t C318(1.12)  LDD1283  [1]
 LDCM0405  CL18 PaTu 8988t C318(1.23)  LDD1284  [1]
 LDCM0406  CL19 PaTu 8988t C318(1.11)  LDD1285  [1]
 LDCM0407  CL2 PaTu 8988t C318(2.38)  LDD1286  [1]
 LDCM0408  CL20 PaTu 8988t C318(1.05)  LDD1287  [1]
 LDCM0409  CL21 PaTu 8988t C318(1.20)  LDD1288  [1]
 LDCM0410  CL22 PaTu 8988t C318(1.15)  LDD1289  [1]
 LDCM0411  CL23 PaTu 8988t C318(1.37)  LDD1290  [1]
 LDCM0412  CL24 PaTu 8988t C318(1.10)  LDD1291  [1]
 LDCM0413  CL25 PaTu 8988t C318(1.07)  LDD1292  [1]
 LDCM0414  CL26 PaTu 8988t C318(1.23)  LDD1293  [1]
 LDCM0415  CL27 PaTu 8988t C318(1.28)  LDD1294  [1]
 LDCM0416  CL28 PaTu 8988t C318(1.38)  LDD1295  [1]
 LDCM0417  CL29 PaTu 8988t C318(1.01)  LDD1296  [1]
 LDCM0418  CL3 PaTu 8988t C318(1.29)  LDD1297  [1]
 LDCM0419  CL30 PaTu 8988t C318(1.06)  LDD1298  [1]
 LDCM0420  CL31 HCT 116 C318(0.93)  LDD0737  [1]
 LDCM0421  CL32 HCT 116 C318(0.99)  LDD0738  [1]
 LDCM0422  CL33 HCT 116 C318(1.05)  LDD0739  [1]
 LDCM0423  CL34 HCT 116 C318(1.10)  LDD0740  [1]
 LDCM0424  CL35 HCT 116 C318(1.05)  LDD0741  [1]
 LDCM0425  CL36 HCT 116 C318(0.98)  LDD0742  [1]
 LDCM0426  CL37 HCT 116 C318(0.93)  LDD0743  [1]
 LDCM0428  CL39 HCT 116 C318(0.97)  LDD0745  [1]
 LDCM0429  CL4 PaTu 8988t C318(1.64)  LDD1308  [1]
 LDCM0430  CL40 HCT 116 C318(0.88)  LDD0747  [1]
 LDCM0431  CL41 HCT 116 C318(0.93)  LDD0748  [1]
 LDCM0432  CL42 HCT 116 C318(0.95)  LDD0749  [1]
 LDCM0433  CL43 HCT 116 C318(0.91)  LDD0750  [1]
 LDCM0434  CL44 HCT 116 C318(0.94)  LDD0751  [1]
 LDCM0435  CL45 HCT 116 C318(0.92)  LDD0752  [1]
 LDCM0436  CL46 HCT 116 C318(1.00)  LDD0753  [1]
 LDCM0437  CL47 HCT 116 C318(1.19)  LDD0754  [1]
 LDCM0438  CL48 HCT 116 C318(1.04)  LDD0755  [1]
 LDCM0439  CL49 HCT 116 C318(1.03)  LDD0756  [1]
 LDCM0440  CL5 PaTu 8988t C318(1.32)  LDD1319  [1]
 LDCM0441  CL50 HCT 116 C318(0.93)  LDD0758  [1]
 LDCM0442  CL51 HCT 116 C318(0.90)  LDD0759  [1]
 LDCM0443  CL52 HCT 116 C318(1.03)  LDD0760  [1]
 LDCM0444  CL53 HCT 116 C318(0.91)  LDD0761  [1]
 LDCM0445  CL54 HCT 116 C318(0.94)  LDD0762  [1]
 LDCM0446  CL55 HCT 116 C318(0.89)  LDD0763  [1]
 LDCM0447  CL56 HCT 116 C318(1.01)  LDD0764  [1]
 LDCM0448  CL57 HCT 116 C318(0.91)  LDD0765  [1]
 LDCM0449  CL58 HCT 116 C318(1.03)  LDD0766  [1]
 LDCM0450  CL59 HCT 116 C318(0.97)  LDD0767  [1]
 LDCM0451  CL6 PaTu 8988t C318(1.29)  LDD1330  [1]
 LDCM0452  CL60 HCT 116 C318(0.99)  LDD0769  [1]
 LDCM0453  CL61 PaTu 8988t C210(0.90)  LDD1332  [1]
 LDCM0454  CL62 PaTu 8988t C210(1.04)  LDD1333  [1]
 LDCM0455  CL63 PaTu 8988t C210(1.04)  LDD1334  [1]
 LDCM0456  CL64 PaTu 8988t C210(0.86)  LDD1335  [1]
 LDCM0457  CL65 PaTu 8988t C210(0.94)  LDD1336  [1]
 LDCM0458  CL66 PaTu 8988t C210(0.84)  LDD1337  [1]
 LDCM0459  CL67 PaTu 8988t C210(1.04)  LDD1338  [1]
 LDCM0460  CL68 PaTu 8988t C210(0.80)  LDD1339  [1]
 LDCM0461  CL69 PaTu 8988t C210(0.86)  LDD1340  [1]
 LDCM0462  CL7 PaTu 8988t C318(1.49)  LDD1341  [1]
 LDCM0463  CL70 PaTu 8988t C210(1.01)  LDD1342  [1]
 LDCM0464  CL71 PaTu 8988t C210(0.87)  LDD1343  [1]
 LDCM0465  CL72 PaTu 8988t C210(1.00)  LDD1344  [1]
 LDCM0466  CL73 PaTu 8988t C210(0.92)  LDD1345  [1]
 LDCM0467  CL74 PaTu 8988t C210(1.24)  LDD1346  [1]
 LDCM0469  CL76 HCT 116 C318(1.11)  LDD0786  [1]
 LDCM0470  CL77 HCT 116 C318(0.90)  LDD0787  [1]
 LDCM0471  CL78 HCT 116 C318(1.01)  LDD0788  [1]
 LDCM0472  CL79 HCT 116 C318(0.98)  LDD0789  [1]
 LDCM0473  CL8 PaTu 8988t C318(1.97)  LDD1352  [1]
 LDCM0474  CL80 HCT 116 C318(0.94)  LDD0791  [1]
 LDCM0475  CL81 HCT 116 C318(0.98)  LDD0792  [1]
 LDCM0476  CL82 HCT 116 C318(0.95)  LDD0793  [1]
 LDCM0477  CL83 HCT 116 C318(0.90)  LDD0794  [1]
 LDCM0478  CL84 HCT 116 C318(0.90)  LDD0795  [1]
 LDCM0479  CL85 HCT 116 C318(0.83)  LDD0796  [1]
 LDCM0480  CL86 HCT 116 C318(0.83)  LDD0797  [1]
 LDCM0481  CL87 HCT 116 C318(0.86)  LDD0798  [1]
 LDCM0482  CL88 HCT 116 C318(0.77)  LDD0799  [1]
 LDCM0483  CL89 HCT 116 C318(0.58)  LDD0800  [1]
 LDCM0484  CL9 PaTu 8988t C318(1.62)  LDD1363  [1]
 LDCM0485  CL90 HCT 116 C318(0.74)  LDD0802  [1]
 LDCM0486  CL91 HCT 116 C318(0.82)  LDD0803  [1]
 LDCM0487  CL92 HCT 116 C318(1.26)  LDD0804  [1]
 LDCM0488  CL93 HCT 116 C318(1.09)  LDD0805  [1]
 LDCM0489  CL94 HCT 116 C318(1.00)  LDD0806  [1]
 LDCM0490  CL95 HCT 116 C318(1.08)  LDD0807  [1]
 LDCM0491  CL96 HCT 116 C318(1.24)  LDD0808  [1]
 LDCM0492  CL97 HCT 116 C318(1.27)  LDD0809  [1]
 LDCM0493  CL98 HCT 116 C318(1.18)  LDD0810  [1]
 LDCM0494  CL99 HCT 116 C318(1.15)  LDD0811  [1]
 LDCM0495  E2913 HEK-293T C210(1.10)  LDD1698  [3]
 LDCM0468  Fragment33 PaTu 8988t C210(1.13)  LDD1347  [1]
 LDCM0427  Fragment51 HCT 116 C318(0.76)  LDD0744  [1]
 LDCM0022  KB02 HEK-293T C318(0.90); C210(0.96)  LDD1492  [3]
 LDCM0023  KB03 HEK-293T C318(1.01); C210(1.03)  LDD1497  [3]
 LDCM0024  KB05 IGR37 C371(3.12)  LDD3314  [4]

The Interaction Atlas With This Target

The Protein(s) Related To This Target

Enzyme
Click To Hide/Show 2 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Caspase-6 (CASP6) Peptidase C14A family P55212
GTP-binding nuclear protein Ran (RAN) Ran family P62826

References

1 Reimagining high-throughput profiling of reactive cysteines for cell-based screening of large electrophile libraries. Nat Biotechnol. 2021 May;39(5):630-641. doi: 10.1038/s41587-020-00778-3. Epub 2021 Jan 4.
2 SP3-FAIMS Chemoproteomics for High-Coverage Profiling of the Human Cysteinome*. Chembiochem. 2021 May 14;22(10):1841-1851. doi: 10.1002/cbic.202000870. Epub 2021 Feb 18.
Mass spectrometry data entry: PXD023056 , PXD023059 , PXD023058 , PXD023057 , PXD023060
3 Accelerating multiplexed profiling of protein-ligand interactions: High-throughput plate-based reactive cysteine profiling with minimal input. Cell Chem Biol. 2024 Mar 21;31(3):565-576.e4. doi: 10.1016/j.chembiol.2023.11.015. Epub 2023 Dec 19.
Mass spectrometry data entry: PXD044402
4 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840