General Information of Target

Target ID LDTP10195
Target Name G-protein coupled receptor-associated sorting protein 2 (GPRASP2)
Gene Name GPRASP2
Gene ID 100528062
Synonyms
G-protein coupled receptor-associated sorting protein 2; GASP-2
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
Download
Sequence
MVRILANGEIVQDDDPRVRTTTQPPRGSIPRQSFFNRGHGAPPGGPGPRQQQAGARLGAA
QSPFNDLNRQLVNMGFPQWHLGNHAVEPVTSILLLFLLMMLGVRGLLLVGLVYLVSHLSQ
R
Target Bioclass
Transcription factor
Family
GPRASP family
Function May play a role in regulation of a variety of G-protein coupled receptors.
Uniprot ID
Q96D09
Ensemble ID
ENST00000332262.10
HGNC ID
HGNC:25169

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 3 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
DBIA
 Probe Info 
C460(0.92); C466(0.92)  LDD0078  [1]
IPM
 Probe Info 
C325(0.00); C586(0.00)  LDD2156  [2]
AOyne
 Probe Info 
13.00  LDD0443  [3]
PAL-AfBPP Probe
Click To Hide/Show 2 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
C313
 Probe Info 
12.30  LDD1980  [4]
C314
 Probe Info 
12.21  LDD1981  [4]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0214  AC1 HEK-293T C460(1.06); C466(1.06); C584(0.90); C586(1.03)  LDD0812  [1]
 LDCM0215  AC10 HEK-293T C208(1.26); C460(1.34); C466(1.34); C584(1.08)  LDD0813  [1]
 LDCM0216  AC100 HEK-293T C208(0.62); C460(1.21); C466(1.12); C584(1.50)  LDD0814  [1]
 LDCM0217  AC101 HEK-293T C208(0.69); C460(2.23); C466(1.66); C584(1.44)  LDD0815  [1]
 LDCM0218  AC102 HEK-293T C208(0.61); C460(1.45); C466(1.32); C584(1.62)  LDD0816  [1]
 LDCM0219  AC103 HEK-293T C208(0.63); C460(1.37); C466(1.37); C584(1.69)  LDD0817  [1]
 LDCM0220  AC104 HEK-293T C208(0.81); C460(1.26); C466(1.39); C584(1.19)  LDD0818  [1]
 LDCM0221  AC105 HEK-293T C208(0.78); C460(1.92); C466(1.40); C584(1.24)  LDD0819  [1]
 LDCM0222  AC106 HEK-293T C208(0.48); C460(1.59); C466(1.32); C584(0.92)  LDD0820  [1]
 LDCM0223  AC107 HEK-293T C208(0.54); C460(1.55); C466(1.33); C584(1.09)  LDD0821  [1]
 LDCM0224  AC108 HEK-293T C208(0.61); C460(1.02); C466(1.01); C584(1.08)  LDD0822  [1]
 LDCM0225  AC109 HEK-293T C208(0.63); C460(1.19); C466(1.22); C584(1.36)  LDD0823  [1]
 LDCM0226  AC11 HEK-293T C208(1.30); C460(1.23); C466(1.23); C584(1.17)  LDD0824  [1]
 LDCM0227  AC110 HEK-293T C208(0.58); C460(2.51); C466(2.02); C584(1.71)  LDD0825  [1]
 LDCM0228  AC111 HEK-293T C208(0.67); C460(0.97); C466(1.05); C584(2.24)  LDD0826  [1]
 LDCM0229  AC112 HEK-293T C208(0.55); C460(1.05); C466(1.16); C584(2.43)  LDD0827  [1]
 LDCM0230  AC113 HEK-293T C208(1.12); C460(1.03); C466(1.03); C584(0.98)  LDD0828  [1]
 LDCM0231  AC114 HEK-293T C208(1.46); C460(1.01); C466(1.06); C584(0.79)  LDD0829  [1]
 LDCM0232  AC115 HEK-293T C208(0.72); C460(1.51); C466(1.32); C584(1.01)  LDD0830  [1]
 LDCM0233  AC116 HEK-293T C208(0.74); C460(0.64); C466(0.84); C584(0.98)  LDD0831  [1]
 LDCM0234  AC117 HEK-293T C208(0.82); C460(0.98); C466(1.10); C584(1.01)  LDD0832  [1]
 LDCM0235  AC118 HEK-293T C208(1.02); C460(0.93); C466(1.07); C584(1.11)  LDD0833  [1]
 LDCM0236  AC119 HEK-293T C208(0.68); C460(0.99); C466(1.12); C584(1.18)  LDD0834  [1]
 LDCM0237  AC12 HEK-293T C208(1.02); C460(1.46); C466(1.46); C584(1.19)  LDD0835  [1]
 LDCM0238  AC120 HEK-293T C208(0.96); C460(0.84); C466(1.04); C584(0.85)  LDD0836  [1]
 LDCM0239  AC121 HEK-293T C208(1.17); C460(0.69); C466(0.99); C584(1.12)  LDD0837  [1]
 LDCM0240  AC122 HEK-293T C208(1.04); C460(0.75); C466(1.08); C584(0.97)  LDD0838  [1]
 LDCM0241  AC123 HEK-293T C208(0.93); C460(0.68); C466(1.03); C584(0.89)  LDD0839  [1]
 LDCM0242  AC124 HEK-293T C208(0.96); C460(0.86); C466(1.09); C584(1.28)  LDD0840  [1]
 LDCM0243  AC125 HEK-293T C208(0.76); C460(1.17); C466(1.33); C584(1.43)  LDD0841  [1]
 LDCM0244  AC126 HEK-293T C208(0.87); C460(1.18); C466(1.31); C584(1.07)  LDD0842  [1]
 LDCM0245  AC127 HEK-293T C208(0.82); C460(0.92); C466(1.15); C584(1.34)  LDD0843  [1]
 LDCM0246  AC128 HEK-293T C460(0.89); C466(0.89); C584(1.19); C586(1.20)  LDD0844  [1]
 LDCM0247  AC129 HEK-293T C460(0.92); C466(0.92); C584(1.36); C586(1.31)  LDD0845  [1]
 LDCM0249  AC130 HEK-293T C460(0.78); C466(0.78); C584(1.09); C586(1.12)  LDD0847  [1]
 LDCM0250  AC131 HEK-293T C460(0.78); C466(0.78); C584(1.27); C586(1.39)  LDD0848  [1]
 LDCM0251  AC132 HEK-293T C460(0.88); C466(0.88); C584(1.47); C586(1.90)  LDD0849  [1]
 LDCM0252  AC133 HEK-293T C460(0.94); C466(0.94); C584(1.17); C586(1.20)  LDD0850  [1]
 LDCM0253  AC134 HEK-293T C460(0.77); C466(0.77); C584(1.12); C586(1.15)  LDD0851  [1]
 LDCM0254  AC135 HEK-293T C460(0.83); C466(0.83); C584(1.04); C586(1.06)  LDD0852  [1]
 LDCM0255  AC136 HEK-293T C460(1.38); C466(1.38); C584(1.16); C586(1.14)  LDD0853  [1]
 LDCM0256  AC137 HEK-293T C460(0.85); C466(0.85); C584(1.25); C586(1.39)  LDD0854  [1]
 LDCM0257  AC138 HEK-293T C460(0.73); C466(0.73); C584(1.24); C586(1.41)  LDD0855  [1]
 LDCM0258  AC139 HEK-293T C460(0.68); C466(0.68); C584(1.29); C586(1.36)  LDD0856  [1]
 LDCM0259  AC14 HEK-293T C208(1.46); C460(1.87); C466(1.87); C584(1.11)  LDD0857  [1]
 LDCM0260  AC140 HEK-293T C460(0.79); C466(0.79); C584(1.29); C586(1.36)  LDD0858  [1]
 LDCM0261  AC141 HEK-293T C460(0.81); C466(0.81); C584(1.25); C586(1.32)  LDD0859  [1]
 LDCM0262  AC142 HEK-293T C460(0.62); C466(0.62); C584(1.24); C586(1.70)  LDD0860  [1]
 LDCM0263  AC143 HEK-293T C208(1.16); C460(0.90); C466(0.90); C584(0.85)  LDD0861  [1]
 LDCM0264  AC144 HEK-293T C208(1.21); C460(0.89); C466(0.89); C584(0.92)  LDD0862  [1]
 LDCM0265  AC145 HEK-293T C208(1.44); C460(0.58); C466(0.58); C584(1.09)  LDD0863  [1]
 LDCM0266  AC146 HEK-293T C208(1.28); C460(0.55); C466(0.55); C584(1.02)  LDD0864  [1]
 LDCM0267  AC147 HEK-293T C208(1.30); C460(0.46); C466(0.46); C584(1.13)  LDD0865  [1]
 LDCM0268  AC148 HEK-293T C208(1.11); C460(0.61); C466(0.61); C584(0.97)  LDD0866  [1]
 LDCM0269  AC149 HEK-293T C208(0.98); C460(0.72); C466(0.72); C584(0.82)  LDD0867  [1]
 LDCM0270  AC15 HEK-293T C208(1.06); C460(1.11); C466(1.11); C584(0.94)  LDD0868  [1]
 LDCM0271  AC150 HEK-293T C208(0.86); C460(0.72); C466(0.72); C584(0.96)  LDD0869  [1]
 LDCM0272  AC151 HEK-293T C208(1.11); C460(0.85); C466(0.85); C584(1.35)  LDD0870  [1]
 LDCM0273  AC152 HEK-293T C208(0.87); C460(0.79); C466(0.79); C584(1.26)  LDD0871  [1]
 LDCM0274  AC153 HEK-293T C208(0.99); C460(0.79); C466(0.79); C584(1.19)  LDD0872  [1]
 LDCM0621  AC154 HEK-293T C208(0.95); C460(0.69); C466(0.69); C584(0.91)  LDD2162  [1]
 LDCM0622  AC155 HEK-293T C208(1.12); C460(1.22); C466(1.22); C584(1.10)  LDD2163  [1]
 LDCM0623  AC156 HEK-293T C208(1.23); C460(0.92); C466(0.92); C584(1.50)  LDD2164  [1]
 LDCM0624  AC157 HEK-293T C208(1.77); C460(0.62); C466(0.62); C584(1.23)  LDD2165  [1]
 LDCM0276  AC17 HEK-293T C208(1.57); C460(1.05); C466(1.05); C584(1.08)  LDD0874  [1]
 LDCM0277  AC18 HEK-293T C208(1.38); C460(1.18); C466(1.18); C584(1.04)  LDD0875  [1]
 LDCM0278  AC19 HEK-293T C208(1.20); C460(1.13); C466(1.13); C584(1.11)  LDD0876  [1]
 LDCM0279  AC2 HEK-293T C460(1.27); C466(1.27); C584(1.24); C586(1.41)  LDD0877  [1]
 LDCM0280  AC20 HEK-293T C208(1.44); C460(1.19); C466(1.19); C584(1.00)  LDD0878  [1]
 LDCM0281  AC21 HEK-293T C208(0.93); C460(1.43); C466(1.43); C584(1.63)  LDD0879  [1]
 LDCM0282  AC22 HEK-293T C208(1.16); C460(1.20); C466(1.20); C584(1.15)  LDD0880  [1]
 LDCM0283  AC23 HEK-293T C208(1.15); C460(1.82); C466(1.82); C584(1.13)  LDD0881  [1]
 LDCM0284  AC24 HEK-293T C208(1.43); C460(1.27); C466(1.27); C584(0.97)  LDD0882  [1]
 LDCM0285  AC25 HEK-293T C460(0.37); C466(0.62); C584(0.73); C586(0.86)  LDD0883  [1]
 LDCM0286  AC26 HEK-293T C460(0.35); C466(0.68); C584(0.77); C586(0.98)  LDD0884  [1]
 LDCM0287  AC27 HEK-293T C460(0.45); C466(0.77); C584(0.66); C586(0.87)  LDD0885  [1]
 LDCM0288  AC28 HEK-293T C460(0.38); C466(0.94); C584(0.69); C586(1.42)  LDD0886  [1]
 LDCM0289  AC29 HEK-293T C460(0.64); C466(0.87); C584(0.68); C586(0.96)  LDD0887  [1]
 LDCM0290  AC3 HEK-293T C460(0.93); C466(0.93); C584(0.88); C586(0.93)  LDD0888  [1]
 LDCM0291  AC30 HEK-293T C460(0.44); C466(0.74); C584(0.89); C586(1.06)  LDD0889  [1]
 LDCM0292  AC31 HEK-293T C460(0.51); C466(0.70); C584(0.69); C586(0.84)  LDD0890  [1]
 LDCM0293  AC32 HEK-293T C460(0.62); C466(0.78); C584(0.72); C586(0.83)  LDD0891  [1]
 LDCM0294  AC33 HEK-293T C460(0.42); C466(0.81); C584(0.76); C586(0.89)  LDD0892  [1]
 LDCM0295  AC34 HEK-293T C460(0.55); C466(0.85); C584(0.78); C586(0.89)  LDD0893  [1]
 LDCM0296  AC35 HEK-293T C208(1.29); C584(1.12); C586(0.99); C589(0.99)  LDD0894  [1]
 LDCM0297  AC36 HEK-293T C208(1.31); C584(1.07); C586(0.88); C589(0.88)  LDD0895  [1]
 LDCM0298  AC37 HEK-293T C208(2.16); C584(0.89); C586(0.82); C589(0.82)  LDD0896  [1]
 LDCM0299  AC38 HEK-293T C208(2.21); C584(1.15); C586(1.15); C589(1.15)  LDD0897  [1]
 LDCM0300  AC39 HEK-293T C208(1.72); C584(1.49); C586(1.28); C589(1.28)  LDD0898  [1]
 LDCM0301  AC4 HEK-293T C460(1.28); C466(1.28); C584(1.02); C586(1.03)  LDD0899  [1]
 LDCM0302  AC40 HEK-293T C208(1.61); C584(0.99); C586(0.85); C589(0.85)  LDD0900  [1]
 LDCM0303  AC41 HEK-293T C208(1.38); C584(1.15); C586(1.17); C589(1.17)  LDD0901  [1]
 LDCM0304  AC42 HEK-293T C208(1.57); C584(1.15); C586(1.30); C589(1.30)  LDD0902  [1]
 LDCM0305  AC43 HEK-293T C208(1.82); C584(1.30); C586(1.16); C589(1.16)  LDD0903  [1]
 LDCM0306  AC44 HEK-293T C208(1.18); C584(1.12); C586(1.11); C589(1.11)  LDD0904  [1]
 LDCM0307  AC45 HEK-293T C208(1.42); C584(1.26); C586(1.05); C589(1.05)  LDD0905  [1]
 LDCM0308  AC46 HEK-293T C208(0.83); C460(0.59); C466(0.76); C584(1.69)  LDD0906  [1]
 LDCM0309  AC47 HEK-293T C208(0.98); C460(0.68); C466(0.87); C584(1.58)  LDD0907  [1]
 LDCM0310  AC48 HEK-293T C208(1.01); C460(0.66); C466(0.80); C584(1.34)  LDD0908  [1]
 LDCM0311  AC49 HEK-293T C208(1.36); C460(0.97); C466(1.03); C584(1.44)  LDD0909  [1]
 LDCM0312  AC5 HEK-293T C460(1.00); C466(1.00); C584(1.03); C586(1.12)  LDD0910  [1]
 LDCM0313  AC50 HEK-293T C208(0.97); C460(0.70); C466(0.81); C584(0.91)  LDD0911  [1]
 LDCM0314  AC51 HEK-293T C208(1.06); C460(0.85); C466(0.92); C584(1.07)  LDD0912  [1]
 LDCM0315  AC52 HEK-293T C208(1.05); C460(0.70); C466(0.89); C584(1.33)  LDD0913  [1]
 LDCM0316  AC53 HEK-293T C208(0.95); C460(0.63); C466(0.77); C584(1.46)  LDD0914  [1]
 LDCM0317  AC54 HEK-293T C208(1.13); C460(0.64); C466(0.84); C584(1.12)  LDD0915  [1]
 LDCM0318  AC55 HEK-293T C208(1.15); C460(0.90); C466(0.97); C584(1.99)  LDD0916  [1]
 LDCM0319  AC56 HEK-293T C208(1.08); C460(0.82); C466(0.80); C584(1.38)  LDD0917  [1]
 LDCM0320  AC57 HEK-293T C208(0.81); C584(0.81); C586(0.91); C589(0.96)  LDD0918  [1]
 LDCM0321  AC58 HEK-293T C208(0.57); C584(1.18); C586(1.07); C589(1.08)  LDD0919  [1]
 LDCM0322  AC59 HEK-293T C208(0.59); C584(0.64); C586(0.96); C589(0.96)  LDD0920  [1]
 LDCM0323  AC6 HEK-293T C208(1.14); C460(1.03); C466(1.03); C584(1.03)  LDD0921  [1]
 LDCM0324  AC60 HEK-293T C208(0.40); C584(0.93); C586(1.04); C589(1.08)  LDD0922  [1]
 LDCM0325  AC61 HEK-293T C208(0.30); C584(0.93); C586(0.93); C589(1.02)  LDD0923  [1]
 LDCM0326  AC62 HEK-293T C208(0.27); C584(1.13); C586(1.06); C589(1.20)  LDD0924  [1]
 LDCM0327  AC63 HEK-293T C208(0.30); C584(0.81); C586(0.94); C589(1.05)  LDD0925  [1]
 LDCM0328  AC64 HEK-293T C208(0.38); C584(0.88); C586(1.14); C589(1.29)  LDD0926  [1]
 LDCM0329  AC65 HEK-293T C208(0.32); C584(0.99); C586(1.13); C589(1.14)  LDD0927  [1]
 LDCM0330  AC66 HEK-293T C208(0.33); C584(0.96); C586(1.00); C589(1.07)  LDD0928  [1]
 LDCM0331  AC67 HEK-293T C208(0.38); C584(0.93); C586(0.96); C589(1.03)  LDD0929  [1]
 LDCM0332  AC68 HEK-293T C208(1.09); C460(1.00); C466(1.04); C584(0.80)  LDD0930  [1]
 LDCM0333  AC69 HEK-293T C208(1.13); C460(1.89); C466(1.47); C584(0.79)  LDD0931  [1]
 LDCM0334  AC7 HEK-293T C208(0.90); C460(1.03); C466(1.03); C584(0.82)  LDD0932  [1]
 LDCM0335  AC70 HEK-293T C208(0.90); C460(1.40); C466(1.31); C584(0.74)  LDD0933  [1]
 LDCM0336  AC71 HEK-293T C208(1.27); C460(1.13); C466(1.09); C584(0.70)  LDD0934  [1]
 LDCM0337  AC72 HEK-293T C208(1.19); C460(1.39); C466(1.26); C584(0.81)  LDD0935  [1]
 LDCM0338  AC73 HEK-293T C208(1.27); C460(1.41); C466(1.33); C584(0.73)  LDD0936  [1]
 LDCM0339  AC74 HEK-293T C208(1.10); C460(1.24); C466(1.21); C584(1.00)  LDD0937  [1]
 LDCM0340  AC75 HEK-293T C208(1.23); C460(0.87); C466(0.92); C584(1.12)  LDD0938  [1]
 LDCM0341  AC76 HEK-293T C208(1.31); C460(0.93); C466(0.96); C584(0.81)  LDD0939  [1]
 LDCM0342  AC77 HEK-293T C208(1.41); C460(1.55); C466(1.33); C584(0.95)  LDD0940  [1]
 LDCM0343  AC78 HEK-293T C208(1.20); C460(0.98); C466(1.05); C584(0.84)  LDD0941  [1]
 LDCM0344  AC79 HEK-293T C208(1.20); C460(0.87); C466(0.98); C584(0.95)  LDD0942  [1]
 LDCM0345  AC8 HEK-293T C208(0.70); C460(1.03); C466(1.03); C584(1.19)  LDD0943  [1]
 LDCM0346  AC80 HEK-293T C208(1.81); C460(0.79); C466(1.01); C584(1.08)  LDD0944  [1]
 LDCM0347  AC81 HEK-293T C208(1.82); C460(1.10); C466(1.16); C584(0.93)  LDD0945  [1]
 LDCM0348  AC82 HEK-293T C208(1.67); C460(1.88); C466(1.70); C584(1.48)  LDD0946  [1]
 LDCM0349  AC83 HEK-293T C466(1.06); C584(0.87); C586(0.87); C589(0.94)  LDD0947  [1]
 LDCM0350  AC84 HEK-293T C466(1.21); C584(0.91); C586(0.91); C589(1.09)  LDD0948  [1]
 LDCM0351  AC85 HEK-293T C466(1.14); C584(0.86); C586(0.86); C589(0.93)  LDD0949  [1]
 LDCM0352  AC86 HEK-293T C466(1.07); C584(1.15); C586(1.15); C589(1.01)  LDD0950  [1]
 LDCM0353  AC87 HEK-293T C466(1.09); C584(1.10); C586(1.10); C589(1.13)  LDD0951  [1]
 LDCM0354  AC88 HEK-293T C466(1.44); C584(0.84); C586(0.84); C589(1.08)  LDD0952  [1]
 LDCM0355  AC89 HEK-293T C466(1.51); C584(0.99); C586(0.99); C589(1.13)  LDD0953  [1]
 LDCM0357  AC90 HEK-293T C466(1.44); C584(0.97); C586(0.97); C589(1.04)  LDD0955  [1]
 LDCM0358  AC91 HEK-293T C466(1.17); C584(0.92); C586(0.92); C589(1.16)  LDD0956  [1]
 LDCM0359  AC92 HEK-293T C466(1.29); C584(0.85); C586(0.85); C589(0.94)  LDD0957  [1]
 LDCM0360  AC93 HEK-293T C466(1.53); C584(0.89); C586(0.89); C589(0.92)  LDD0958  [1]
 LDCM0361  AC94 HEK-293T C466(1.39); C584(1.01); C586(1.01); C589(1.14)  LDD0959  [1]
 LDCM0362  AC95 HEK-293T C466(1.23); C584(0.74); C586(0.74); C589(0.91)  LDD0960  [1]
 LDCM0363  AC96 HEK-293T C466(1.40); C584(0.92); C586(0.92); C589(1.09)  LDD0961  [1]
 LDCM0364  AC97 HEK-293T C466(2.04); C584(0.80); C586(0.80); C589(1.15)  LDD0962  [1]
 LDCM0365  AC98 HEK-293T C208(0.46); C460(1.15); C466(1.16); C584(1.35)  LDD0963  [1]
 LDCM0366  AC99 HEK-293T C208(0.59); C460(1.01); C466(0.99); C584(1.19)  LDD0964  [1]
 LDCM0248  AKOS034007472 HEK-293T C208(1.31); C460(1.22); C466(1.22); C584(1.00)  LDD0846  [1]
 LDCM0356  AKOS034007680 HEK-293T C208(1.15); C460(1.39); C466(1.39); C584(1.07)  LDD0954  [1]
 LDCM0275  AKOS034007705 HEK-293T C208(2.23); C460(1.62); C466(1.62); C584(1.26)  LDD0873  [1]
 LDCM0020  ARS-1620 HCC44 C460(0.92); C466(0.92)  LDD0078  [1]
 LDCM0367  CL1 HEK-293T C208(1.04); C584(0.75); C586(0.97); C589(0.84)  LDD0965  [1]
 LDCM0368  CL10 HEK-293T C208(1.30); C584(1.07); C586(1.29); C589(1.02)  LDD0966  [1]
 LDCM0369  CL100 HEK-293T C460(1.10); C466(1.10); C584(0.80); C586(0.82)  LDD0967  [1]
 LDCM0370  CL101 HEK-293T C208(0.92); C460(0.96); C466(0.96); C584(0.85)  LDD0968  [1]
 LDCM0371  CL102 HEK-293T C208(1.18); C460(1.10); C466(1.10); C584(1.02)  LDD0969  [1]
 LDCM0372  CL103 HEK-293T C208(0.90); C460(1.05); C466(1.05); C584(0.87)  LDD0970  [1]
 LDCM0373  CL104 HEK-293T C208(0.85); C460(0.99); C466(0.99); C584(0.77)  LDD0971  [1]
 LDCM0374  CL105 HEK-293T C208(1.41); C460(1.86); C466(1.86); C584(0.77)  LDD0972  [1]
 LDCM0375  CL106 HEK-293T C208(1.29); C460(1.64); C466(1.64); C584(0.77)  LDD0973  [1]
 LDCM0376  CL107 HEK-293T C208(1.26); C460(1.56); C466(1.56); C584(0.91)  LDD0974  [1]
 LDCM0377  CL108 HEK-293T C208(0.99); C460(0.66); C466(0.66); C584(0.91)  LDD0975  [1]
 LDCM0378  CL109 HEK-293T C208(1.41); C460(1.94); C466(1.94); C584(1.01)  LDD0976  [1]
 LDCM0379  CL11 HEK-293T C208(1.15); C584(0.44); C586(1.04); C589(0.63)  LDD0977  [1]
 LDCM0380  CL110 HEK-293T C208(1.53); C460(1.33); C466(1.33); C584(1.07)  LDD0978  [1]
 LDCM0381  CL111 HEK-293T C208(1.14); C460(2.45); C466(2.45); C584(1.45)  LDD0979  [1]
 LDCM0382  CL112 HEK-293T C460(0.60); C466(0.74); C584(0.76); C586(0.92)  LDD0980  [1]
 LDCM0383  CL113 HEK-293T C460(0.37); C466(0.75); C584(0.76); C586(0.96)  LDD0981  [1]
 LDCM0384  CL114 HEK-293T C460(0.55); C466(0.83); C584(0.87); C586(1.09)  LDD0982  [1]
 LDCM0385  CL115 HEK-293T C460(0.60); C466(0.84); C584(0.92); C586(0.94)  LDD0983  [1]
 LDCM0386  CL116 HEK-293T C460(0.44); C466(0.75); C584(0.73); C586(0.97)  LDD0984  [1]
 LDCM0387  CL117 HEK-293T C208(2.00); C584(2.13); C586(1.78); C589(1.78)  LDD0985  [1]
 LDCM0388  CL118 HEK-293T C208(1.00); C584(0.97); C586(0.89); C589(0.89)  LDD0986  [1]
 LDCM0389  CL119 HEK-293T C208(1.23); C584(1.05); C586(0.86); C589(0.86)  LDD0987  [1]
 LDCM0390  CL12 HEK-293T C208(1.31); C584(0.52); C586(0.81); C589(0.70)  LDD0988  [1]
 LDCM0391  CL120 HEK-293T C208(1.27); C584(1.33); C586(1.12); C589(1.12)  LDD0989  [1]
 LDCM0392  CL121 HEK-293T C208(1.30); C460(0.54); C466(0.80); C584(1.22)  LDD0990  [1]
 LDCM0393  CL122 HEK-293T C208(1.11); C460(0.72); C466(0.83); C584(1.87)  LDD0991  [1]
 LDCM0394  CL123 HEK-293T C208(1.48); C460(1.36); C466(1.13); C584(1.37)  LDD0992  [1]
 LDCM0395  CL124 HEK-293T C208(1.15); C460(0.80); C466(0.93); C584(2.90)  LDD0993  [1]
 LDCM0396  CL125 HEK-293T C208(0.85); C584(0.99); C586(1.11); C589(1.12)  LDD0994  [1]
 LDCM0397  CL126 HEK-293T C208(1.19); C584(0.75); C586(1.09); C589(1.11)  LDD0995  [1]
 LDCM0398  CL127 HEK-293T C208(0.71); C584(0.87); C586(0.99); C589(1.04)  LDD0996  [1]
 LDCM0399  CL128 HEK-293T C208(0.80); C584(1.03); C586(1.17); C589(1.27)  LDD0997  [1]
 LDCM0400  CL13 HEK-293T C208(0.88); C584(0.49); C586(0.72); C589(0.60)  LDD0998  [1]
 LDCM0401  CL14 HEK-293T C208(0.96); C584(0.70); C586(0.91); C589(0.73)  LDD0999  [1]
 LDCM0402  CL15 HEK-293T C208(1.27); C584(0.57); C586(0.94); C589(0.70)  LDD1000  [1]
 LDCM0403  CL16 HEK-293T C460(0.94); C466(0.94); C584(1.06); C586(1.01)  LDD1001  [1]
 LDCM0404  CL17 HEK-293T C460(1.02); C466(1.02); C584(1.17); C586(1.02)  LDD1002  [1]
 LDCM0405  CL18 HEK-293T C460(1.10); C466(1.10); C584(1.24); C586(1.22)  LDD1003  [1]
 LDCM0406  CL19 HEK-293T C460(1.06); C466(1.06); C584(1.40); C586(1.27)  LDD1004  [1]
 LDCM0407  CL2 HEK-293T C208(0.93); C584(0.51); C586(0.70); C589(0.72)  LDD1005  [1]
 LDCM0408  CL20 HEK-293T C460(0.93); C466(0.93); C584(1.24); C586(1.17)  LDD1006  [1]
 LDCM0409  CL21 HEK-293T C460(1.29); C466(1.29); C584(1.32); C586(1.25)  LDD1007  [1]
 LDCM0410  CL22 HEK-293T C460(0.95); C466(0.95); C584(1.21); C586(1.14)  LDD1008  [1]
 LDCM0411  CL23 HEK-293T C460(0.60); C466(0.60); C584(1.11); C586(1.06)  LDD1009  [1]
 LDCM0412  CL24 HEK-293T C460(0.99); C466(0.99); C584(1.49); C586(1.29)  LDD1010  [1]
 LDCM0413  CL25 HEK-293T C460(0.97); C466(0.97); C584(1.49); C586(1.30)  LDD1011  [1]
 LDCM0414  CL26 HEK-293T C460(0.94); C466(0.94); C584(1.27); C586(1.23)  LDD1012  [1]
 LDCM0415  CL27 HEK-293T C460(0.91); C466(0.91); C584(1.12); C586(1.11)  LDD1013  [1]
 LDCM0416  CL28 HEK-293T C460(1.08); C466(1.08); C584(1.66); C586(1.31)  LDD1014  [1]
 LDCM0417  CL29 HEK-293T C460(0.84); C466(0.84); C584(1.47); C586(1.21)  LDD1015  [1]
 LDCM0418  CL3 HEK-293T C208(0.83); C584(0.64); C586(0.78); C589(0.74)  LDD1016  [1]
 LDCM0419  CL30 HEK-293T C460(1.01); C466(1.01); C584(1.45); C586(1.30)  LDD1017  [1]
 LDCM0420  CL31 HEK-293T C208(1.00); C460(0.96); C466(0.96); C584(0.98)  LDD1018  [1]
 LDCM0421  CL32 HEK-293T C208(0.99); C460(0.78); C466(0.78); C584(0.88)  LDD1019  [1]
 LDCM0422  CL33 HEK-293T C208(1.06); C460(1.20); C466(1.20); C584(0.89)  LDD1020  [1]
 LDCM0423  CL34 HEK-293T C208(1.06); C460(0.84); C466(0.84); C584(0.95)  LDD1021  [1]
 LDCM0424  CL35 HEK-293T C208(1.04); C460(1.09); C466(1.09); C584(1.37)  LDD1022  [1]
 LDCM0425  CL36 HEK-293T C208(1.15); C460(1.03); C466(1.03); C584(1.25)  LDD1023  [1]
 LDCM0426  CL37 HEK-293T C208(1.08); C460(1.21); C466(1.21); C584(1.36)  LDD1024  [1]
 LDCM0428  CL39 HEK-293T C208(1.29); C460(1.18); C466(1.18); C584(0.87)  LDD1026  [1]
 LDCM0429  CL4 HEK-293T C208(1.29); C584(0.67); C586(0.97); C589(0.89)  LDD1027  [1]
 LDCM0430  CL40 HEK-293T C208(0.96); C460(0.91); C466(0.91); C584(0.80)  LDD1028  [1]
 LDCM0431  CL41 HEK-293T C208(1.12); C460(1.08); C466(1.08); C584(1.05)  LDD1029  [1]
 LDCM0432  CL42 HEK-293T C208(1.26); C460(0.84); C466(0.84); C584(1.03)  LDD1030  [1]
 LDCM0433  CL43 HEK-293T C208(1.02); C460(0.87); C466(0.87); C584(0.99)  LDD1031  [1]
 LDCM0434  CL44 HEK-293T C208(1.30); C460(1.34); C466(1.34); C584(1.03)  LDD1032  [1]
 LDCM0435  CL45 HEK-293T C208(1.13); C460(1.18); C466(1.18); C584(1.20)  LDD1033  [1]
 LDCM0436  CL46 HEK-293T C208(1.49); C460(0.94); C466(0.96); C584(1.05)  LDD1034  [1]
 LDCM0437  CL47 HEK-293T C208(0.92); C460(0.82); C466(0.97); C584(1.23)  LDD1035  [1]
 LDCM0438  CL48 HEK-293T C208(0.83); C460(0.84); C466(0.89); C584(1.18)  LDD1036  [1]
 LDCM0439  CL49 HEK-293T C208(0.89); C460(0.76); C466(1.03); C584(1.08)  LDD1037  [1]
 LDCM0440  CL5 HEK-293T C208(1.04); C584(0.59); C586(0.95); C589(0.85)  LDD1038  [1]
 LDCM0441  CL50 HEK-293T C208(1.19); C460(0.90); C466(1.39); C584(1.14)  LDD1039  [1]
 LDCM0442  CL51 HEK-293T C208(1.22); C460(0.99); C466(1.11); C584(0.93)  LDD1040  [1]
 LDCM0443  CL52 HEK-293T C208(1.20); C460(0.73); C466(0.68); C584(1.22)  LDD1041  [1]
 LDCM0444  CL53 HEK-293T C208(1.00); C460(0.84); C466(0.90); C584(1.10)  LDD1042  [1]
 LDCM0445  CL54 HEK-293T C208(1.33); C460(1.14); C466(0.96); C584(0.98)  LDD1043  [1]
 LDCM0446  CL55 HEK-293T C208(0.89); C460(0.94); C466(1.13); C584(0.96)  LDD1044  [1]
 LDCM0447  CL56 HEK-293T C208(0.83); C460(0.72); C466(0.79); C584(1.09)  LDD1045  [1]
 LDCM0448  CL57 HEK-293T C208(1.74); C460(0.90); C466(1.26); C584(1.45)  LDD1046  [1]
 LDCM0449  CL58 HEK-293T C208(0.95); C460(1.26); C466(1.29); C584(1.30)  LDD1047  [1]
 LDCM0450  CL59 HEK-293T C208(1.14); C460(1.19); C466(1.12); C584(1.35)  LDD1048  [1]
 LDCM0451  CL6 HEK-293T C208(0.99); C584(0.52); C586(1.06); C589(0.83)  LDD1049  [1]
 LDCM0452  CL60 HEK-293T C208(1.30); C460(1.15); C466(1.44); C584(1.10)  LDD1050  [1]
 LDCM0453  CL61 HEK-293T C208(0.84); C460(1.44); C466(1.44); C584(0.97)  LDD1051  [1]
 LDCM0454  CL62 HEK-293T C208(0.98); C460(1.15); C466(1.15); C584(0.96)  LDD1052  [1]
 LDCM0455  CL63 HEK-293T C208(0.88); C460(1.23); C466(1.23); C584(0.88)  LDD1053  [1]
 LDCM0456  CL64 HEK-293T C208(1.31); C460(2.33); C466(2.33); C584(0.91)  LDD1054  [1]
 LDCM0457  CL65 HEK-293T C208(1.07); C460(1.45); C466(1.45); C584(1.08)  LDD1055  [1]
 LDCM0458  CL66 HEK-293T C208(0.91); C460(1.23); C466(1.23); C584(0.91)  LDD1056  [1]
 LDCM0459  CL67 HEK-293T C208(1.09); C460(1.68); C466(1.68); C584(1.02)  LDD1057  [1]
 LDCM0460  CL68 HEK-293T C208(1.19); C460(2.70); C466(2.70); C584(1.24)  LDD1058  [1]
 LDCM0461  CL69 HEK-293T C208(1.08); C460(1.72); C466(1.72); C584(0.95)  LDD1059  [1]
 LDCM0462  CL7 HEK-293T C208(0.86); C584(0.51); C586(1.11); C589(0.65)  LDD1060  [1]
 LDCM0463  CL70 HEK-293T C208(1.05); C460(2.04); C466(2.04); C584(1.03)  LDD1061  [1]
 LDCM0464  CL71 HEK-293T C208(1.08); C460(2.81); C466(2.81); C584(0.97)  LDD1062  [1]
 LDCM0465  CL72 HEK-293T C208(1.19); C460(1.40); C466(1.40); C584(1.11)  LDD1063  [1]
 LDCM0466  CL73 HEK-293T C208(1.23); C460(1.53); C466(1.53); C584(0.85)  LDD1064  [1]
 LDCM0467  CL74 HEK-293T C208(1.00); C460(1.73); C466(1.73); C584(0.94)  LDD1065  [1]
 LDCM0469  CL76 HEK-293T C208(0.92); C460(1.15); C466(1.15); C584(1.16)  LDD1067  [1]
 LDCM0470  CL77 HEK-293T C208(1.18); C460(1.15); C466(1.15); C584(0.98)  LDD1068  [1]
 LDCM0471  CL78 HEK-293T C208(1.12); C460(1.07); C466(1.07); C584(0.99)  LDD1069  [1]
 LDCM0472  CL79 HEK-293T C208(0.94); C460(1.12); C466(1.12); C584(0.99)  LDD1070  [1]
 LDCM0473  CL8 HEK-293T C208(1.10); C584(1.16); C586(1.00); C589(0.84)  LDD1071  [1]
 LDCM0474  CL80 HEK-293T C208(1.08); C460(0.82); C466(0.82); C584(1.09)  LDD1072  [1]
 LDCM0475  CL81 HEK-293T C208(1.12); C460(1.27); C466(1.27); C584(0.97)  LDD1073  [1]
 LDCM0476  CL82 HEK-293T C208(1.09); C460(1.28); C466(1.28); C584(0.93)  LDD1074  [1]
 LDCM0477  CL83 HEK-293T C208(1.26); C460(1.14); C466(1.14); C584(0.90)  LDD1075  [1]
 LDCM0478  CL84 HEK-293T C208(0.84); C460(0.81); C466(0.81); C584(1.10)  LDD1076  [1]
 LDCM0479  CL85 HEK-293T C208(1.04); C460(0.88); C466(0.88); C584(1.08)  LDD1077  [1]
 LDCM0480  CL86 HEK-293T C208(0.66); C460(0.82); C466(0.82); C584(1.10)  LDD1078  [1]
 LDCM0481  CL87 HEK-293T C208(1.07); C460(0.99); C466(0.99); C584(1.20)  LDD1079  [1]
 LDCM0482  CL88 HEK-293T C208(0.67); C460(0.84); C466(0.84); C584(1.35)  LDD1080  [1]
 LDCM0483  CL89 HEK-293T C208(1.30); C460(1.06); C466(1.06); C584(0.96)  LDD1081  [1]
 LDCM0484  CL9 HEK-293T C208(1.33); C584(0.63); C586(1.16); C589(0.88)  LDD1082  [1]
 LDCM0485  CL90 HEK-293T C208(1.27); C460(1.12); C466(1.12); C584(1.05)  LDD1083  [1]
 LDCM0486  CL91 HEK-293T C460(0.94); C466(0.94); C584(0.94); C586(1.12)  LDD1084  [1]
 LDCM0487  CL92 HEK-293T C460(1.33); C466(1.33); C584(0.93); C586(1.01)  LDD1085  [1]
 LDCM0488  CL93 HEK-293T C460(1.08); C466(1.08); C584(1.09); C586(0.96)  LDD1086  [1]
 LDCM0489  CL94 HEK-293T C460(1.27); C466(1.27); C584(1.45); C586(1.38)  LDD1087  [1]
 LDCM0490  CL95 HEK-293T C460(1.47); C466(1.47); C584(1.02); C586(1.26)  LDD1088  [1]
 LDCM0491  CL96 HEK-293T C460(0.86); C466(0.86); C584(0.93); C586(0.95)  LDD1089  [1]
 LDCM0492  CL97 HEK-293T C460(0.93); C466(0.93); C584(1.11); C586(1.17)  LDD1090  [1]
 LDCM0493  CL98 HEK-293T C460(1.29); C466(1.29); C584(0.95); C586(1.10)  LDD1091  [1]
 LDCM0494  CL99 HEK-293T C460(1.44); C466(1.44); C584(1.17); C586(1.03)  LDD1092  [1]
 LDCM0495  E2913 HEK-293T C325(1.05); C407(1.27); C208(0.94)  LDD1698  [5]
 LDCM0468  Fragment33 HEK-293T C208(1.06); C460(1.81); C466(1.81); C584(1.12)  LDD1066  [1]
 LDCM0427  Fragment51 HEK-293T C208(1.22); C460(1.36); C466(1.36); C584(0.92)  LDD1025  [1]
 LDCM0022  KB02 HCT 116 C586(2.45); C584(1.96); C589(1.96)  LDD0080  [1]
 LDCM0023  KB03 HCT 116 C586(8.30); C584(4.21); C589(4.21)  LDD0081  [1]
 LDCM0024  KB05 HCT 116 C586(3.49); C584(2.53); C589(2.53)  LDD0082  [1]

The Interaction Atlas With This Target

The Protein(s) Related To This Target

Enzyme
Click To Hide/Show 3 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
FAST kinase domain-containing protein 4 (TBRG4) FAST kinase family Q969Z0
E3 ubiquitin-protein ligase RNF8 (RNF8) RNF8 family O76064
Thioredoxin, mitochondrial (TXN2) Thioredoxin family Q99757
Transporter and channel
Click To Hide/Show 2 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
14-3-3 protein gamma (YWHAG) 14-3-3 family P61981
Huntingtin (HTT) Huntingtin family P42858
Transcription factor
Click To Hide/Show 2 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Ribosome quality control complex subunit TCF25 (TCF25) TCF25 family Q9BQ70
Forkhead box protein D4-like 1 (FOXD4L1) . Q9NU39
Other
Click To Hide/Show 15 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Caveolae-associated protein 3 (CAVIN3) CAVIN family Q969G5
Cilia- and flagella-associated protein 206 (CFAP206) CFAP206 family Q8IYR0
Methyl-CpG-binding domain protein 3-like 2 (MBD3L2) MBD3L family Q8NHZ7
Large ribosomal subunit protein mL64 (GADD45GIP1) Mitochondrion-specific ribosomal protein mL64 family Q8TAE8
PIH1 domain-containing protein 2 (PIH1D2) PIH1 family Q8WWB5
Placenta-specific protein 9 (PLAC9) PLAC9 family Q5JTB6
Rhophilin-1 (RHPN1) RHPN family Q8TCX5
Splicing regulatory glutamine/lysine-rich protein 1 (SREK1) Splicing factor SR family Q8WXA9
Chromobox protein homolog 8 (CBX8) . Q9HC52
Coiled-coil domain-containing protein 146 (CCDC146) . Q8IYE0
Putative uncharacterized protein MGC163334 . Q5W150
Required for excision 1-B domain-containing protein (REX1BD) . Q96EN9
SH2 domain-containing protein 4A (SH2D4A) . Q9H788
Suppressor APC domain-containing protein 2 (SAPCD2) . Q86UD0
U4/U6 small nuclear ribonucleoprotein Prp3 (PRPF3) . O43395

References

1 Reimagining high-throughput profiling of reactive cysteines for cell-based screening of large electrophile libraries. Nat Biotechnol. 2021 May;39(5):630-641. doi: 10.1038/s41587-020-00778-3. Epub 2021 Jan 4.
2 Benchmarking Cleavable Biotin Tags for Peptide-Centric Chemoproteomics. J Proteome Res. 2022 May 6;21(5):1349-1358. doi: 10.1021/acs.jproteome.2c00174. Epub 2022 Apr 25.
Mass spectrometry data entry: PXD031019
3 Chemoproteomic profiling of targets of lipid-derived electrophiles by bioorthogonal aminooxy probe. Redox Biol. 2017 Aug;12:712-718. doi: 10.1016/j.redox.2017.04.001. Epub 2017 Apr 5.
4 Large-scale chemoproteomics expedites ligand discovery and predicts ligand behavior in cells. Science. 2024 Apr 26;384(6694):eadk5864. doi: 10.1126/science.adk5864. Epub 2024 Apr 26.
Mass spectrometry data entry: PXD041587
5 Accelerating multiplexed profiling of protein-ligand interactions: High-throughput plate-based reactive cysteine profiling with minimal input. Cell Chem Biol. 2024 Mar 21;31(3):565-576.e4. doi: 10.1016/j.chembiol.2023.11.015. Epub 2023 Dec 19.
Mass spectrometry data entry: PXD044402