General Information of Target

Target ID LDTP09753
Target Name Cortactin-binding protein 2 (CTTNBP2)
Gene Name CTTNBP2
Gene ID 83992
Synonyms
C7orf8; CORTBP2; KIAA1758; Cortactin-binding protein 2; CortBP2
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MWATCCNWFCLDGQPEEVPPPQGARMQAYSNPGYSSFPSPTGLEPSCKSCGAHFANTARK
QTCLDCKKNFCMTCSSQVGNGPRLCLLCQRFRATAFQREELMKMKVKDLRDYLSLHDIST
EMCREKEELVLLVLGQQPVISQEDRTRASTLSPDFPEQQAFLTQPHSSMVPPTSPNLPSS
SAQATSVPPAQVQENQQANGHVSQDQEEPVYLESVARVPAEDETQSIDSEDSFVPGRRAS
LSDLTDLEDIEGLTVRQLKEILARNFVNYKGCCEKWELMERVTRLYKDQKGLQHLVSGAE
DQNGGAVPSGLEENLCKICMDSPIDCVLLECGHMVTCTKCGKRMNECPICRQYVIRAVHV
FRS
Target Bioclass
Other
Subcellular location
Cytoplasm, cell cortex
Function Regulates the dendritic spine distribution of CTTN/cortactin in hippocampal neurons, thus controls dendritic spinogenesis and dendritic spine maintenance.
Uniprot ID
Q8WZ74
Ensemble ID
ENST00000160373.8
HGNC ID
HGNC:15679

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 4 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
DBIA
 Probe Info 
C1225(0.97)  LDD0547  [1]
IPM
 Probe Info 
N.A.  LDD0005  [2]
YN-1
 Probe Info 
N.A.  LDD0447  [3]
AOyne
 Probe Info 
15.00  LDD0443  [4]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0214  AC1 HEK-293T C1623(1.17); C346(1.04); C104(1.15)  LDD1507  [5]
 LDCM0215  AC10 HEK-293T C346(0.80); C104(0.98); C104(1.06); C118(1.06)  LDD1508  [5]
 LDCM0226  AC11 HEK-293T C1623(1.13); C346(0.96); C1415(0.99); C1538(0.89)  LDD1509  [5]
 LDCM0230  AC113 HCT 116 C1225(0.97)  LDD0547  [1]
 LDCM0231  AC114 HCT 116 C1225(0.95)  LDD0548  [1]
 LDCM0232  AC115 HCT 116 C1225(0.88)  LDD0549  [1]
 LDCM0233  AC116 HCT 116 C1225(0.88)  LDD0550  [1]
 LDCM0234  AC117 HCT 116 C1225(1.00)  LDD0551  [1]
 LDCM0235  AC118 HCT 116 C1225(0.92)  LDD0552  [1]
 LDCM0236  AC119 HCT 116 C1225(0.99)  LDD0553  [1]
 LDCM0237  AC12 HEK-293T C346(1.08); C307(1.07)  LDD1510  [5]
 LDCM0238  AC120 HCT 116 C1225(0.93)  LDD0555  [1]
 LDCM0239  AC121 HCT 116 C1225(0.84)  LDD0556  [1]
 LDCM0240  AC122 HCT 116 C1225(0.91)  LDD0557  [1]
 LDCM0241  AC123 HCT 116 C1225(0.85)  LDD0558  [1]
 LDCM0242  AC124 HCT 116 C1225(0.88)  LDD0559  [1]
 LDCM0243  AC125 HCT 116 C1225(0.90)  LDD0560  [1]
 LDCM0244  AC126 HCT 116 C1225(0.88)  LDD0561  [1]
 LDCM0245  AC127 HCT 116 C1225(0.86)  LDD0562  [1]
 LDCM0259  AC14 HEK-293T C1623(0.85); C346(0.99)  LDD1512  [5]
 LDCM0270  AC15 HEK-293T C346(1.03); C104(1.11); C104(0.76); C118(0.76)  LDD1513  [5]
 LDCM0276  AC17 HEK-293T C1623(1.39); C346(1.00); C104(0.91)  LDD1515  [5]
 LDCM0277  AC18 HEK-293T C346(1.00); C104(1.18); C104(1.08); C118(1.08)  LDD1516  [5]
 LDCM0278  AC19 HEK-293T C1623(1.48); C346(1.13); C1415(1.05); C1538(0.94)  LDD1517  [5]
 LDCM0279  AC2 HEK-293T C346(0.88); C104(0.93); C104(1.15); C118(1.15)  LDD1518  [5]
 LDCM0280  AC20 HEK-293T C346(0.94); C307(1.20)  LDD1519  [5]
 LDCM0281  AC21 HEK-293T C1623(0.99); C346(1.00); C104(1.13); C104(0.81)  LDD1520  [5]
 LDCM0282  AC22 HEK-293T C1623(0.95); C346(1.00)  LDD1521  [5]
 LDCM0283  AC23 HEK-293T C346(1.09); C104(0.85); C104(0.85); C118(0.85)  LDD1522  [5]
 LDCM0284  AC24 HEK-293T C346(1.08); C104(1.24)  LDD1523  [5]
 LDCM0285  AC25 HEK-293T C1623(1.23); C346(0.92); C104(0.87)  LDD1524  [5]
 LDCM0286  AC26 HEK-293T C346(0.96); C104(0.90); C104(1.09); C118(1.09)  LDD1525  [5]
 LDCM0287  AC27 HEK-293T C1623(0.96); C346(0.95); C1415(0.98); C1538(0.92)  LDD1526  [5]
 LDCM0288  AC28 HEK-293T C346(1.00); C307(1.07)  LDD1527  [5]
 LDCM0289  AC29 HEK-293T C1623(0.87); C346(1.03); C104(1.00); C104(0.87)  LDD1528  [5]
 LDCM0290  AC3 HEK-293T C1623(1.04); C346(0.99); C1415(1.00); C1538(0.98)  LDD1529  [5]
 LDCM0291  AC30 HEK-293T C1623(1.18); C346(1.06)  LDD1530  [5]
 LDCM0292  AC31 HEK-293T C346(1.06); C104(0.92); C104(0.97); C118(0.97)  LDD1531  [5]
 LDCM0293  AC32 HEK-293T C346(1.11); C104(1.25)  LDD1532  [5]
 LDCM0294  AC33 HEK-293T C1623(1.21); C346(0.99); C104(0.97)  LDD1533  [5]
 LDCM0295  AC34 HEK-293T C346(0.88); C104(0.99); C104(1.12); C118(1.12)  LDD1534  [5]
 LDCM0296  AC35 HEK-293T C1623(0.96); C346(0.93); C1415(0.93); C1538(0.94)  LDD1535  [5]
 LDCM0297  AC36 HEK-293T C346(0.96); C307(1.24)  LDD1536  [5]
 LDCM0298  AC37 HEK-293T C1623(0.99); C346(1.00); C104(0.95); C104(0.83)  LDD1537  [5]
 LDCM0299  AC38 HEK-293T C1623(0.99); C346(0.98)  LDD1538  [5]
 LDCM0300  AC39 HEK-293T C346(1.11); C104(0.96); C104(0.95); C118(0.95)  LDD1539  [5]
 LDCM0301  AC4 HEK-293T C346(0.92); C307(1.14)  LDD1540  [5]
 LDCM0302  AC40 HEK-293T C346(1.03); C104(2.24)  LDD1541  [5]
 LDCM0303  AC41 HEK-293T C1623(1.22); C346(1.00); C104(1.02)  LDD1542  [5]
 LDCM0304  AC42 HEK-293T C346(1.12); C104(0.81); C104(1.05); C118(1.05)  LDD1543  [5]
 LDCM0305  AC43 HEK-293T C1623(1.28); C346(0.98); C1415(0.99); C1538(0.92)  LDD1544  [5]
 LDCM0306  AC44 HEK-293T C346(0.98); C307(1.21)  LDD1545  [5]
 LDCM0307  AC45 HEK-293T C1623(0.78); C346(1.11); C104(0.96); C104(1.00)  LDD1546  [5]
 LDCM0308  AC46 HEK-293T C1623(0.98); C346(0.94)  LDD1547  [5]
 LDCM0309  AC47 HEK-293T C346(1.05); C104(1.08); C104(0.97); C118(0.97)  LDD1548  [5]
 LDCM0310  AC48 HEK-293T C346(1.05); C104(2.54)  LDD1549  [5]
 LDCM0311  AC49 HEK-293T C1623(1.00); C346(1.09); C104(0.93)  LDD1550  [5]
 LDCM0312  AC5 HEK-293T C1623(0.77); C346(1.02); C104(1.02); C104(0.98)  LDD1551  [5]
 LDCM0313  AC50 HEK-293T C346(0.81); C104(0.80); C104(1.07); C118(1.07)  LDD1552  [5]
 LDCM0314  AC51 HEK-293T C1623(0.94); C346(0.98); C1415(0.93); C1538(0.93)  LDD1553  [5]
 LDCM0315  AC52 HEK-293T C346(1.00); C307(1.10)  LDD1554  [5]
 LDCM0316  AC53 HEK-293T C1623(0.94); C346(1.06); C104(1.01); C104(1.01)  LDD1555  [5]
 LDCM0317  AC54 HEK-293T C1623(1.13); C346(1.09)  LDD1556  [5]
 LDCM0318  AC55 HEK-293T C346(1.06); C104(0.89); C104(0.93); C118(0.93)  LDD1557  [5]
 LDCM0319  AC56 HEK-293T C346(1.11); C104(1.27)  LDD1558  [5]
 LDCM0320  AC57 HEK-293T C1623(1.11); C346(1.09); C104(1.08)  LDD1559  [5]
 LDCM0321  AC58 HEK-293T C346(0.81); C104(0.93); C104(1.09); C118(1.09)  LDD1560  [5]
 LDCM0322  AC59 HEK-293T C1623(1.11); C346(1.03); C1415(1.00); C1538(0.98)  LDD1561  [5]
 LDCM0323  AC6 HEK-293T C1623(0.86); C346(1.04)  LDD1562  [5]
 LDCM0324  AC60 HEK-293T C346(0.98); C307(1.14)  LDD1563  [5]
 LDCM0325  AC61 HEK-293T C1623(1.07); C346(1.04); C104(1.01); C104(1.01)  LDD1564  [5]
 LDCM0326  AC62 HEK-293T C1623(1.18); C346(1.14)  LDD1565  [5]
 LDCM0327  AC63 HEK-293T C346(1.07); C104(1.06); C104(1.00); C118(1.00)  LDD1566  [5]
 LDCM0328  AC64 HEK-293T C346(1.06); C104(1.22)  LDD1567  [5]
 LDCM0334  AC7 HEK-293T C346(1.08); C104(1.01); C104(1.06); C118(1.06)  LDD1568  [5]
 LDCM0345  AC8 HEK-293T C346(1.13); C104(1.62)  LDD1569  [5]
 LDCM0248  AKOS034007472 HEK-293T C1623(0.95); C346(1.09); C104(0.91); C104(0.91)  LDD1511  [5]
 LDCM0356  AKOS034007680 HEK-293T C1623(1.07); C346(1.03); C104(0.87)  LDD1570  [5]
 LDCM0275  AKOS034007705 HEK-293T C346(0.99); C104(1.64)  LDD1514  [5]
 LDCM0367  CL1 HEK-293T C1623(0.93); C104(1.19)  LDD1571  [5]
 LDCM0368  CL10 HEK-293T C1623(1.12); C346(0.90)  LDD1572  [5]
 LDCM0369  CL100 HEK-293T C346(1.13); C104(1.26)  LDD1573  [5]
 LDCM0370  CL101 HEK-293T C1623(1.01); C104(1.04)  LDD1574  [5]
 LDCM0371  CL102 HEK-293T C346(1.04)  LDD1575  [5]
 LDCM0372  CL103 HEK-293T C1623(0.89); C346(1.09); C104(1.04)  LDD1576  [5]
 LDCM0373  CL104 HEK-293T C346(0.96); C104(1.01)  LDD1577  [5]
 LDCM0374  CL105 HEK-293T C1623(1.01); C104(1.11)  LDD1578  [5]
 LDCM0375  CL106 HEK-293T C346(0.99)  LDD1579  [5]
 LDCM0376  CL107 HEK-293T C1623(0.94); C346(0.98); C104(0.99)  LDD1580  [5]
 LDCM0377  CL108 HEK-293T C346(1.17); C104(1.08)  LDD1581  [5]
 LDCM0378  CL109 HEK-293T C1623(0.91); C104(1.09)  LDD1582  [5]
 LDCM0379  CL11 HEK-293T C346(0.97); C104(0.89); C104(0.83); C118(0.83)  LDD1583  [5]
 LDCM0380  CL110 HEK-293T C346(1.00)  LDD1584  [5]
 LDCM0381  CL111 HEK-293T C1623(1.00); C346(1.09); C104(0.83)  LDD1585  [5]
 LDCM0382  CL112 HEK-293T C346(1.19); C104(1.29)  LDD1586  [5]
 LDCM0383  CL113 HEK-293T C1623(0.97); C104(1.09)  LDD1587  [5]
 LDCM0384  CL114 HEK-293T C346(1.14)  LDD1588  [5]
 LDCM0385  CL115 HEK-293T C1623(1.12); C346(1.19); C104(1.01)  LDD1589  [5]
 LDCM0386  CL116 HEK-293T C346(0.96); C104(1.10)  LDD1590  [5]
 LDCM0387  CL117 HEK-293T C1623(0.99); C104(1.10)  LDD1591  [5]
 LDCM0388  CL118 HEK-293T C346(1.22)  LDD1592  [5]
 LDCM0389  CL119 HEK-293T C1623(1.00); C346(1.02); C104(1.15)  LDD1593  [5]
 LDCM0390  CL12 HEK-293T C346(0.93); C104(0.91)  LDD1594  [5]
 LDCM0391  CL120 HEK-293T C346(1.00); C104(1.13)  LDD1595  [5]
 LDCM0392  CL121 HEK-293T C1623(0.99); C104(1.33)  LDD1596  [5]
 LDCM0393  CL122 HEK-293T C346(0.93)  LDD1597  [5]
 LDCM0394  CL123 HEK-293T C1623(1.17); C346(1.02); C104(0.89)  LDD1598  [5]
 LDCM0395  CL124 HEK-293T C346(1.07); C104(0.97)  LDD1599  [5]
 LDCM0396  CL125 HEK-293T C1623(1.01); C104(1.19)  LDD1600  [5]
 LDCM0397  CL126 HEK-293T C346(0.98)  LDD1601  [5]
 LDCM0398  CL127 HEK-293T C1623(1.04); C346(1.26); C104(1.30)  LDD1602  [5]
 LDCM0399  CL128 HEK-293T C346(1.04); C104(1.33)  LDD1603  [5]
 LDCM0400  CL13 HEK-293T C1623(0.96); C104(1.23)  LDD1604  [5]
 LDCM0401  CL14 HEK-293T C346(1.04)  LDD1605  [5]
 LDCM0402  CL15 HEK-293T C1623(1.02); C346(1.00); C104(1.00)  LDD1606  [5]
 LDCM0403  CL16 HEK-293T C346(0.95); C104(0.96)  LDD1607  [5]
 LDCM0404  CL17 HEK-293T C1623(1.14); C346(0.85); C104(0.98)  LDD1608  [5]
 LDCM0405  CL18 HEK-293T C346(0.94); C104(0.99); C104(1.00); C118(1.00)  LDD1609  [5]
 LDCM0406  CL19 HEK-293T C1623(1.03); C346(1.15); C1415(1.02); C1538(0.89)  LDD1610  [5]
 LDCM0407  CL2 HEK-293T C346(0.98)  LDD1611  [5]
 LDCM0408  CL20 HEK-293T C346(0.94); C307(1.10)  LDD1612  [5]
 LDCM0409  CL21 HEK-293T C1623(1.05); C346(1.00); C104(0.89); C104(0.68)  LDD1613  [5]
 LDCM0410  CL22 HEK-293T C1623(0.87); C346(0.83)  LDD1614  [5]
 LDCM0411  CL23 HEK-293T C346(1.00); C104(0.71); C104(0.70); C118(0.70)  LDD1615  [5]
 LDCM0412  CL24 HEK-293T C346(1.14); C104(1.09)  LDD1616  [5]
 LDCM0413  CL25 HEK-293T C1623(0.94); C104(1.10)  LDD1617  [5]
 LDCM0414  CL26 HEK-293T C346(0.95)  LDD1618  [5]
 LDCM0415  CL27 HEK-293T C1623(0.84); C346(1.18); C104(0.93)  LDD1619  [5]
 LDCM0416  CL28 HEK-293T C346(0.95); C104(1.00)  LDD1620  [5]
 LDCM0417  CL29 HEK-293T C1623(1.17); C346(1.15); C104(0.87)  LDD1621  [5]
 LDCM0418  CL3 HEK-293T C1623(1.04); C346(0.92); C104(1.09)  LDD1622  [5]
 LDCM0419  CL30 HEK-293T C346(0.95); C104(0.85); C104(0.76); C118(0.76)  LDD1623  [5]
 LDCM0420  CL31 HCT 116 C1225(1.13)  LDD0737  [1]
 LDCM0421  CL32 HCT 116 C1225(0.96)  LDD0738  [1]
 LDCM0422  CL33 HCT 116 C1225(1.04)  LDD0739  [1]
 LDCM0423  CL34 HCT 116 C1225(1.15)  LDD0740  [1]
 LDCM0424  CL35 HCT 116 C1225(1.06)  LDD0741  [1]
 LDCM0425  CL36 HCT 116 C1225(1.08)  LDD0742  [1]
 LDCM0426  CL37 HCT 116 C1225(1.12)  LDD0743  [1]
 LDCM0428  CL39 HCT 116 C1225(1.14)  LDD0745  [1]
 LDCM0429  CL4 HEK-293T C346(1.00); C104(1.08)  LDD1633  [5]
 LDCM0430  CL40 HCT 116 C1225(1.20)  LDD0747  [1]
 LDCM0431  CL41 HCT 116 C1225(1.13)  LDD0748  [1]
 LDCM0432  CL42 HCT 116 C1225(1.05)  LDD0749  [1]
 LDCM0433  CL43 HCT 116 C1225(0.99)  LDD0750  [1]
 LDCM0434  CL44 HCT 116 C1225(1.11)  LDD0751  [1]
 LDCM0435  CL45 HCT 116 C1225(1.27)  LDD0752  [1]
 LDCM0436  CL46 HCT 116 C1225(1.09)  LDD0753  [1]
 LDCM0437  CL47 HCT 116 C1225(1.05)  LDD0754  [1]
 LDCM0438  CL48 HCT 116 C1225(0.93)  LDD0755  [1]
 LDCM0439  CL49 HCT 116 C1225(1.02)  LDD0756  [1]
 LDCM0440  CL5 HEK-293T C1623(1.56); C346(1.11); C104(0.85)  LDD1644  [5]
 LDCM0441  CL50 HCT 116 C1225(1.08)  LDD0758  [1]
 LDCM0442  CL51 HCT 116 C1225(1.07)  LDD0759  [1]
 LDCM0443  CL52 HCT 116 C1225(1.25)  LDD0760  [1]
 LDCM0444  CL53 HCT 116 C1225(0.94)  LDD0761  [1]
 LDCM0445  CL54 HCT 116 C1225(1.08)  LDD0762  [1]
 LDCM0446  CL55 HCT 116 C1225(1.02)  LDD0763  [1]
 LDCM0447  CL56 HCT 116 C1225(1.02)  LDD0764  [1]
 LDCM0448  CL57 HCT 116 C1225(1.05)  LDD0765  [1]
 LDCM0449  CL58 HCT 116 C1225(1.18)  LDD0766  [1]
 LDCM0450  CL59 HCT 116 C1225(1.05)  LDD0767  [1]
 LDCM0451  CL6 HEK-293T C346(0.84); C104(0.72); C104(0.86); C118(0.86)  LDD1654  [5]
 LDCM0452  CL60 HCT 116 C1225(1.07)  LDD0769  [1]
 LDCM0453  CL61 HCT 116 C1225(1.14)  LDD0770  [1]
 LDCM0454  CL62 HCT 116 C1225(1.14)  LDD0771  [1]
 LDCM0455  CL63 HCT 116 C1225(1.00)  LDD0772  [1]
 LDCM0456  CL64 HCT 116 C1225(1.12)  LDD0773  [1]
 LDCM0457  CL65 HCT 116 C1225(1.20)  LDD0774  [1]
 LDCM0458  CL66 HCT 116 C1225(1.06)  LDD0775  [1]
 LDCM0459  CL67 HCT 116 C1225(0.99)  LDD0776  [1]
 LDCM0460  CL68 HCT 116 C1225(1.09)  LDD0777  [1]
 LDCM0461  CL69 HCT 116 C1225(1.12)  LDD0778  [1]
 LDCM0462  CL7 HEK-293T C1623(1.09); C346(0.95); C1415(0.96); C1538(0.85)  LDD1665  [5]
 LDCM0463  CL70 HCT 116 C1225(0.98)  LDD0780  [1]
 LDCM0464  CL71 HCT 116 C1225(0.94)  LDD0781  [1]
 LDCM0465  CL72 HCT 116 C1225(1.07)  LDD0782  [1]
 LDCM0466  CL73 HCT 116 C1225(1.15)  LDD0783  [1]
 LDCM0467  CL74 HCT 116 C1225(1.09)  LDD0784  [1]
 LDCM0469  CL76 HCT 116 C1225(0.93)  LDD0786  [1]
 LDCM0470  CL77 HCT 116 C1225(1.04)  LDD0787  [1]
 LDCM0471  CL78 HCT 116 C1225(0.92)  LDD0788  [1]
 LDCM0472  CL79 HCT 116 C1225(1.04)  LDD0789  [1]
 LDCM0473  CL8 HEK-293T C346(0.84); C307(1.00)  LDD1676  [5]
 LDCM0474  CL80 HCT 116 C1225(1.09)  LDD0791  [1]
 LDCM0475  CL81 HCT 116 C1225(0.96)  LDD0792  [1]
 LDCM0476  CL82 HCT 116 C1225(0.88)  LDD0793  [1]
 LDCM0477  CL83 HCT 116 C1225(0.94)  LDD0794  [1]
 LDCM0478  CL84 HCT 116 C1225(0.96)  LDD0795  [1]
 LDCM0479  CL85 HCT 116 C1225(0.95)  LDD0796  [1]
 LDCM0480  CL86 HCT 116 C1225(0.87)  LDD0797  [1]
 LDCM0481  CL87 HCT 116 C1225(0.90)  LDD0798  [1]
 LDCM0482  CL88 HCT 116 C1225(0.88)  LDD0799  [1]
 LDCM0483  CL89 HCT 116 C1225(0.91)  LDD0800  [1]
 LDCM0484  CL9 HEK-293T C1623(0.83); C346(0.97); C104(1.02); C104(0.69)  LDD1687  [5]
 LDCM0485  CL90 HCT 116 C1225(1.03)  LDD0802  [1]
 LDCM0486  CL91 HEK-293T C1623(0.98); C346(1.08); C1415(1.17); C1538(0.89)  LDD1689  [5]
 LDCM0487  CL92 HEK-293T C346(0.99); C307(1.17)  LDD1690  [5]
 LDCM0488  CL93 HEK-293T C1623(0.98); C346(1.13); C104(0.98); C104(0.79)  LDD1691  [5]
 LDCM0489  CL94 HEK-293T C1623(1.02); C346(1.05)  LDD1692  [5]
 LDCM0490  CL95 HEK-293T C346(1.05); C104(1.33); C104(0.51); C118(0.51)  LDD1693  [5]
 LDCM0491  CL96 HEK-293T C346(1.10); C104(1.06)  LDD1694  [5]
 LDCM0492  CL97 HEK-293T C1623(1.02); C104(1.17)  LDD1695  [5]
 LDCM0493  CL98 HEK-293T C346(0.86)  LDD1696  [5]
 LDCM0494  CL99 HEK-293T C1623(1.10); C346(1.22); C104(1.24)  LDD1697  [5]
 LDCM0495  E2913 HEK-293T C1623(1.40); C346(1.19); C104(1.02)  LDD1698  [5]
 LDCM0468  Fragment33 HCT 116 C1225(1.15)  LDD0785  [1]
 LDCM0427  Fragment51 HCT 116 C1225(1.44)  LDD0744  [1]
 LDCM0022  KB02 HEK-293T C346(0.90); C1623(1.01)  LDD1492  [5]
 LDCM0023  KB03 HEK-293T C346(1.04); C1623(1.04)  LDD1497  [5]
 LDCM0024  KB05 RVH-421 C1623(1.60)  LDD3413  [6]

The Interaction Atlas With This Target

The Protein(s) Related To This Target

Transcription factor
Click To Hide/Show 1 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Homeobox protein PKNOX2 (PKNOX2) TALE/MEIS homeobox family Q96KN3
Other
Click To Hide/Show 5 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Protein INCA1 (INCA1) INCA family Q0VD86
Keratin, type I cytoskeletal 14 (KRT14) Intermediate filament family P02533
Meiosis-specific protein MEI4 (MEI4) MEI4L family A8MW99
Heat shock factor 2-binding protein (HSF2BP) . O75031
Melanoma-associated antigen 11 (MAGEA11) . P43364

References

1 Reimagining high-throughput profiling of reactive cysteines for cell-based screening of large electrophile libraries. Nat Biotechnol. 2021 May;39(5):630-641. doi: 10.1038/s41587-020-00778-3. Epub 2021 Jan 4.
2 A modification-centric assessment tool for the performance of chemoproteomic probes. Nat Chem Biol. 2022 Aug;18(8):904-912. doi: 10.1038/s41589-022-01074-8. Epub 2022 Jul 21.
Mass spectrometry data entry: PXD027758 , PXD027755 , PXD027760 , PXD027762 , PXD027756 , PXD027591 , PXD007149 , PXD030064 , PXD032392 , PXD027789 , PXD027767 , PXD027764
3 Ynamide Electrophile for the Profiling of Ligandable Carboxyl Residues in Live Cells and the Development of New Covalent Inhibitors. J Med Chem. 2022 Aug 11;65(15):10408-10418. doi: 10.1021/acs.jmedchem.2c00272. Epub 2022 Jul 26.
4 Chemoproteomic profiling of targets of lipid-derived electrophiles by bioorthogonal aminooxy probe. Redox Biol. 2017 Aug;12:712-718. doi: 10.1016/j.redox.2017.04.001. Epub 2017 Apr 5.
5 Accelerating multiplexed profiling of protein-ligand interactions: High-throughput plate-based reactive cysteine profiling with minimal input. Cell Chem Biol. 2024 Mar 21;31(3):565-576.e4. doi: 10.1016/j.chembiol.2023.11.015. Epub 2023 Dec 19.
Mass spectrometry data entry: PXD044402
6 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840