Details of the Target
General Information of Target
Probe(s) Labeling This Target
ABPP Probe
Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
---|---|---|---|---|---|
STPyne Probe Info |
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K141(8.80) | LDD0277 | [1] | |
m-APA Probe Info |
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12.30 | LDD0403 | [2] | |
DBIA Probe Info |
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C72(4.21) | LDD3332 | [3] | |
BTD Probe Info |
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C72(1.67) | LDD2090 | [4] | |
HHS-482 Probe Info |
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Y172(0.89) | LDD0285 | [5] | |
HHS-475 Probe Info |
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Y127(0.21); Y172(1.50) | LDD0264 | [6] | |
W1 Probe Info |
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C72(0.99) | LDD0239 | [7] | |
NAIA_4 Probe Info |
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N.A. | LDD2226 | [8] | |
ENE Probe Info |
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N.A. | LDD0006 | [9] | |
IPM Probe Info |
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N.A. | LDD0005 | [9] |
Competitor(s) Related to This Target
Competitor ID | Name | Cell line | Binding Site(Ratio) | Interaction ID | Ref |
---|---|---|---|---|---|
LDCM0548 | 1-(4-(Benzo[d][1,3]dioxol-5-ylmethyl)piperazin-1-yl)-2-nitroethan-1-one | MDA-MB-231 | C72(1.24) | LDD2142 | [4] |
LDCM0519 | 1-(6-methoxy-3,4-dihydroquinolin-1(2H)-yl)-2-nitroethan-1-one | MDA-MB-231 | C72(1.17) | LDD2112 | [4] |
LDCM0510 | 3-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-3-oxopropanenitrile | MDA-MB-231 | C72(1.01) | LDD2103 | [4] |
LDCM0156 | Aniline | NCI-H1299 | 12.30 | LDD0403 | [2] |
LDCM0116 | HHS-0101 | DM93 | Y127(0.21); Y172(1.50) | LDD0264 | [6] |
LDCM0117 | HHS-0201 | DM93 | Y127(0.29); Y172(1.46) | LDD0265 | [6] |
LDCM0118 | HHS-0301 | DM93 | Y127(0.18); Y172(1.47) | LDD0266 | [6] |
LDCM0119 | HHS-0401 | DM93 | Y127(0.27); Y172(1.58) | LDD0267 | [6] |
LDCM0120 | HHS-0701 | DM93 | Y127(0.42); Y172(1.51) | LDD0268 | [6] |
LDCM0123 | JWB131 | DM93 | Y172(0.89) | LDD0285 | [5] |
LDCM0124 | JWB142 | DM93 | Y172(1.33) | LDD0286 | [5] |
LDCM0125 | JWB146 | DM93 | Y172(1.00) | LDD0287 | [5] |
LDCM0126 | JWB150 | DM93 | Y172(4.22) | LDD0288 | [5] |
LDCM0127 | JWB152 | DM93 | Y172(1.97) | LDD0289 | [5] |
LDCM0128 | JWB198 | DM93 | Y172(1.27) | LDD0290 | [5] |
LDCM0129 | JWB202 | DM93 | Y172(0.97) | LDD0291 | [5] |
LDCM0130 | JWB211 | DM93 | Y172(0.96) | LDD0292 | [5] |
LDCM0022 | KB02 | 22RV1 | C72(2.53) | LDD2243 | [3] |
LDCM0023 | KB03 | 22RV1 | C72(3.01) | LDD2660 | [3] |
LDCM0024 | KB05 | MKN45 | C72(4.21) | LDD3332 | [3] |
LDCM0497 | Nucleophilic fragment 11b | MDA-MB-231 | C72(1.67) | LDD2090 | [4] |
LDCM0507 | Nucleophilic fragment 16b | MDA-MB-231 | C72(3.03) | LDD2100 | [4] |
LDCM0511 | Nucleophilic fragment 18b | MDA-MB-231 | C72(1.61) | LDD2104 | [4] |
LDCM0513 | Nucleophilic fragment 19b | MDA-MB-231 | C72(1.68) | LDD2106 | [4] |
LDCM0544 | Nucleophilic fragment 39 | MDA-MB-231 | C72(1.14) | LDD2137 | [4] |
LDCM0547 | Nucleophilic fragment 41 | MDA-MB-231 | C72(1.36) | LDD2141 | [4] |
LDCM0112 | W16 | Hep-G2 | C72(0.99) | LDD0239 | [7] |
References