General Information of Target

Target ID LDTP11588
Target Name GREB1-like protein (GREB1L)
Gene Name GREB1L
Gene ID 80000
Synonyms
C18orf6; KIAA1772; GREB1-like protein; Growth regulation by estrogen in breast cancer 1-like protein
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MSKLWRRGSTSGAMEAPEPGEALELSLAGAHGHGVHKKKHKKHKKKHKKKHHQEEDAGPT
QPSPAKPQLKLKIKLGGQVLGTKSVPTFTVIPEGPRSPSPLMVVDNEEEPMEGVPLEQYR
AWLDEDSNLSPSPLRDLSGGLGGQEEEEEQRWLDALEKGELDDNGDLKKEINERLLTARQ
RALLQKARSQPSPMLPLPVAEGCPPPALTEEMLLKREERARKRRLQAARRAEEHKNQTIE
RLTKTAATSGRGGRGGARGERRGGRAAAPAPMVRYCSGAQGSTLSFPPGVPAPTAVSQRP
SPSGPPPRCSVPGCPHPRRYACSRTGQALCSLQCYRINLQMRLGGPEGPGSPLLAT
Target Bioclass
Other
Family
GREB1 family
Subcellular location
Membrane
Function Plays a major role in early metanephros and genital development.
Uniprot ID
Q9C091
Ensemble ID
ENST00000269218.10
HGNC ID
HGNC:31042

Target Site Mutations in Different Cell Lines

Cell line Mutation details Probe for labeling this protein in this cell
A431 SNV: p.L1883S .
AN3CA SNV: p.R1607C .
COLO679 Substitution: p.P1258L .
HCT15 SNV: p.S788R; p.K1274N .
IPC298 SNV: p.P1042L .
J82 SNV: p.P1229L .
KYSE410 SNV: p.R1503Q .
MCC13 SNV: p.S530F .
MEWO SNV: p.K327I; p.D1450N .
NCIH716 SNV: p.E93Q .
NUGC3 Insertion: p.M627NfsTer18 .
ONS76 SNV: p.L1623V
Substitution: p.L982P
.
SG231 SNV: p.K1097E .
SHSY5Y SNV: p.N1563S .
SISO SNV: p.M1449I .
SKNSH SNV: p.N1563S .
TE10 SNV: p.M627L .
TE4 Deletion: p.A17LfsTer6
SNV: p.A17P
.
YSCCC SNV: p.E843Q .

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 2 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
DBIA
 Probe Info 
C234(1.90)  LDD3395  [1]
AOyne
 Probe Info 
13.80  LDD0443  [2]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0214  AC1 HEK-293T C121(0.84)  LDD0812  [3]
 LDCM0215  AC10 HEK-293T C121(0.85)  LDD0813  [3]
 LDCM0216  AC100 HEK-293T C121(1.10)  LDD0814  [3]
 LDCM0217  AC101 HEK-293T C121(1.00)  LDD0815  [3]
 LDCM0218  AC102 HEK-293T C121(1.12)  LDD0816  [3]
 LDCM0219  AC103 HEK-293T C121(1.26)  LDD0817  [3]
 LDCM0220  AC104 HEK-293T C121(1.21)  LDD0818  [3]
 LDCM0221  AC105 HEK-293T C121(0.86)  LDD0819  [3]
 LDCM0222  AC106 HEK-293T C121(0.81)  LDD0820  [3]
 LDCM0223  AC107 HEK-293T C121(1.05)  LDD0821  [3]
 LDCM0224  AC108 HEK-293T C121(0.88)  LDD0822  [3]
 LDCM0225  AC109 HEK-293T C121(1.04)  LDD0823  [3]
 LDCM0226  AC11 HEK-293T C121(0.90)  LDD0824  [3]
 LDCM0227  AC110 HEK-293T C121(1.46)  LDD0825  [3]
 LDCM0228  AC111 HEK-293T C121(1.93)  LDD0826  [3]
 LDCM0229  AC112 HEK-293T C121(1.48)  LDD0827  [3]
 LDCM0237  AC12 HEK-293T C121(0.88)  LDD0835  [3]
 LDCM0246  AC128 HEK-293T C121(0.74)  LDD0844  [3]
 LDCM0247  AC129 HEK-293T C121(0.82)  LDD0845  [3]
 LDCM0249  AC130 HEK-293T C121(1.06)  LDD0847  [3]
 LDCM0250  AC131 HEK-293T C121(0.83)  LDD0848  [3]
 LDCM0251  AC132 HEK-293T C121(0.99)  LDD0849  [3]
 LDCM0252  AC133 HEK-293T C121(1.10)  LDD0850  [3]
 LDCM0253  AC134 HEK-293T C121(1.07)  LDD0851  [3]
 LDCM0254  AC135 HEK-293T C121(1.42)  LDD0852  [3]
 LDCM0255  AC136 HEK-293T C121(1.39)  LDD0853  [3]
 LDCM0256  AC137 HEK-293T C121(1.44)  LDD0854  [3]
 LDCM0257  AC138 HEK-293T C121(1.78)  LDD0855  [3]
 LDCM0258  AC139 HEK-293T C121(1.31)  LDD0856  [3]
 LDCM0259  AC14 HEK-293T C121(1.00)  LDD0857  [3]
 LDCM0260  AC140 HEK-293T C121(1.36)  LDD0858  [3]
 LDCM0261  AC141 HEK-293T C121(1.50)  LDD0859  [3]
 LDCM0262  AC142 HEK-293T C121(1.15)  LDD0860  [3]
 LDCM0270  AC15 HEK-293T C121(1.45)  LDD0868  [3]
 LDCM0276  AC17 HEK-293T C499(0.93); C1033(1.14)  LDD1515  [4]
 LDCM0277  AC18 HEK-293T C499(0.99); C1033(0.77)  LDD1516  [4]
 LDCM0278  AC19 HEK-293T C499(1.07)  LDD1517  [4]
 LDCM0279  AC2 HEK-293T C121(1.12)  LDD0877  [3]
 LDCM0280  AC20 HEK-293T C499(0.85)  LDD1519  [4]
 LDCM0281  AC21 HEK-293T C499(1.01)  LDD1520  [4]
 LDCM0282  AC22 HEK-293T C499(0.95)  LDD1521  [4]
 LDCM0283  AC23 HEK-293T C499(1.08)  LDD1522  [4]
 LDCM0284  AC24 HEK-293T C247(1.09); C499(1.15); C1033(1.01); C28(0.86)  LDD1523  [4]
 LDCM0285  AC25 HEK-293T C499(0.85); C1033(1.17)  LDD1524  [4]
 LDCM0286  AC26 HEK-293T C499(0.94); C1033(1.02)  LDD1525  [4]
 LDCM0287  AC27 HEK-293T C499(1.01)  LDD1526  [4]
 LDCM0288  AC28 HEK-293T C499(1.09)  LDD1527  [4]
 LDCM0289  AC29 HEK-293T C499(1.03)  LDD1528  [4]
 LDCM0290  AC3 HEK-293T C121(0.65)  LDD0888  [3]
 LDCM0291  AC30 HEK-293T C499(0.84)  LDD1530  [4]
 LDCM0292  AC31 HEK-293T C499(0.79)  LDD1531  [4]
 LDCM0293  AC32 HEK-293T C247(1.07); C499(1.07); C1033(0.96); C28(0.93)  LDD1532  [4]
 LDCM0294  AC33 HEK-293T C499(0.95); C1033(1.21)  LDD1533  [4]
 LDCM0295  AC34 HEK-293T C499(1.08); C1033(0.94)  LDD1534  [4]
 LDCM0296  AC35 HEK-293T C499(1.24)  LDD1535  [4]
 LDCM0297  AC36 HEK-293T C499(0.91)  LDD1536  [4]
 LDCM0298  AC37 HEK-293T C499(0.86)  LDD1537  [4]
 LDCM0299  AC38 HEK-293T C499(0.68)  LDD1538  [4]
 LDCM0300  AC39 HEK-293T C499(1.01)  LDD1539  [4]
 LDCM0301  AC4 HEK-293T C121(1.05)  LDD0899  [3]
 LDCM0302  AC40 HEK-293T C247(1.07); C499(0.90); C1033(0.91); C28(1.04)  LDD1541  [4]
 LDCM0303  AC41 HEK-293T C499(0.98); C1033(1.24)  LDD1542  [4]
 LDCM0304  AC42 HEK-293T C499(1.14); C1033(0.83)  LDD1543  [4]
 LDCM0305  AC43 HEK-293T C499(1.14)  LDD1544  [4]
 LDCM0306  AC44 HEK-293T C499(1.07)  LDD1545  [4]
 LDCM0307  AC45 HEK-293T C499(0.82)  LDD1546  [4]
 LDCM0308  AC46 HEK-293T C499(0.85)  LDD1547  [4]
 LDCM0309  AC47 HEK-293T C499(0.84)  LDD1548  [4]
 LDCM0310  AC48 HEK-293T C247(1.29); C499(0.91); C1033(1.06); C28(1.04)  LDD1549  [4]
 LDCM0311  AC49 HEK-293T C499(1.24); C1033(1.14)  LDD1550  [4]
 LDCM0312  AC5 HEK-293T C121(0.57)  LDD0910  [3]
 LDCM0313  AC50 HEK-293T C499(1.14); C1033(1.00)  LDD1552  [4]
 LDCM0314  AC51 HEK-293T C499(0.99)  LDD1553  [4]
 LDCM0315  AC52 HEK-293T C499(0.86)  LDD1554  [4]
 LDCM0316  AC53 HEK-293T C499(0.98)  LDD1555  [4]
 LDCM0317  AC54 HEK-293T C499(0.87)  LDD1556  [4]
 LDCM0318  AC55 HEK-293T C499(0.92)  LDD1557  [4]
 LDCM0319  AC56 HEK-293T C247(1.01); C499(1.04); C1033(1.29); C28(1.22)  LDD1558  [4]
 LDCM0320  AC57 HEK-293T C499(1.03); C1033(1.33)  LDD1559  [4]
 LDCM0321  AC58 HEK-293T C499(1.01); C1033(0.96)  LDD1560  [4]
 LDCM0322  AC59 HEK-293T C499(1.22)  LDD1561  [4]
 LDCM0323  AC6 HEK-293T C121(0.84)  LDD0921  [3]
 LDCM0324  AC60 HEK-293T C499(1.04)  LDD1563  [4]
 LDCM0325  AC61 HEK-293T C499(1.17)  LDD1564  [4]
 LDCM0326  AC62 HEK-293T C499(1.13)  LDD1565  [4]
 LDCM0327  AC63 HEK-293T C499(0.94)  LDD1566  [4]
 LDCM0328  AC64 HEK-293T C247(1.01); C499(1.01); C1033(0.95); C28(0.98)  LDD1567  [4]
 LDCM0334  AC7 HEK-293T C121(1.07)  LDD0932  [3]
 LDCM0345  AC8 HEK-293T C121(1.44)  LDD0943  [3]
 LDCM0349  AC83 HEK-293T C121(0.65)  LDD0947  [3]
 LDCM0350  AC84 HEK-293T C121(0.88)  LDD0948  [3]
 LDCM0351  AC85 HEK-293T C121(0.72)  LDD0949  [3]
 LDCM0352  AC86 HEK-293T C121(0.79)  LDD0950  [3]
 LDCM0353  AC87 HEK-293T C121(0.67)  LDD0951  [3]
 LDCM0354  AC88 HEK-293T C121(1.10)  LDD0952  [3]
 LDCM0355  AC89 HEK-293T C121(0.93)  LDD0953  [3]
 LDCM0357  AC90 HEK-293T C121(1.28)  LDD0955  [3]
 LDCM0358  AC91 HEK-293T C121(0.79)  LDD0956  [3]
 LDCM0359  AC92 HEK-293T C121(0.79)  LDD0957  [3]
 LDCM0360  AC93 HEK-293T C121(0.81)  LDD0958  [3]
 LDCM0361  AC94 HEK-293T C121(1.17)  LDD0959  [3]
 LDCM0362  AC95 HEK-293T C121(0.98)  LDD0960  [3]
 LDCM0363  AC96 HEK-293T C121(1.26)  LDD0961  [3]
 LDCM0364  AC97 HEK-293T C121(1.62)  LDD0962  [3]
 LDCM0365  AC98 HEK-293T C121(0.94)  LDD0963  [3]
 LDCM0366  AC99 HEK-293T C121(0.97)  LDD0964  [3]
 LDCM0248  AKOS034007472 HEK-293T C121(1.09)  LDD0846  [3]
 LDCM0356  AKOS034007680 HEK-293T C121(1.47)  LDD0954  [3]
 LDCM0275  AKOS034007705 HEK-293T C121(1.17)  LDD0873  [3]
 LDCM0367  CL1 HEK-293T C247(1.07); C499(0.84)  LDD1571  [4]
 LDCM0368  CL10 HEK-293T C499(0.81)  LDD1572  [4]
 LDCM0369  CL100 HEK-293T C121(0.64)  LDD0967  [3]
 LDCM0370  CL101 HEK-293T C121(1.28)  LDD0968  [3]
 LDCM0371  CL102 HEK-293T C121(1.33)  LDD0969  [3]
 LDCM0372  CL103 HEK-293T C121(0.94)  LDD0970  [3]
 LDCM0373  CL104 HEK-293T C121(1.13)  LDD0971  [3]
 LDCM0374  CL105 HEK-293T C247(1.15); C499(0.91)  LDD1578  [4]
 LDCM0375  CL106 HEK-293T C247(1.14); C499(0.78)  LDD1579  [4]
 LDCM0376  CL107 HEK-293T C499(0.98)  LDD1580  [4]
 LDCM0377  CL108 HEK-293T C499(1.20)  LDD1581  [4]
 LDCM0378  CL109 HEK-293T C247(0.91); C499(0.96)  LDD1582  [4]
 LDCM0379  CL11 HEK-293T C499(0.79)  LDD1583  [4]
 LDCM0380  CL110 HEK-293T C247(1.22); C499(0.99)  LDD1584  [4]
 LDCM0381  CL111 HEK-293T C499(0.93)  LDD1585  [4]
 LDCM0382  CL112 HEK-293T C499(0.91)  LDD1586  [4]
 LDCM0383  CL113 HEK-293T C247(1.28); C499(1.03)  LDD1587  [4]
 LDCM0384  CL114 HEK-293T C247(0.91); C499(0.85)  LDD1588  [4]
 LDCM0385  CL115 HEK-293T C499(0.96)  LDD1589  [4]
 LDCM0386  CL116 HEK-293T C499(1.05)  LDD1590  [4]
 LDCM0387  CL117 HEK-293T C247(1.16); C499(1.07)  LDD1591  [4]
 LDCM0388  CL118 HEK-293T C247(0.67); C499(0.90)  LDD1592  [4]
 LDCM0389  CL119 HEK-293T C499(0.84)  LDD1593  [4]
 LDCM0390  CL12 HEK-293T C247(0.92); C499(1.11); C1033(1.17); C28(1.56)  LDD1594  [4]
 LDCM0391  CL120 HEK-293T C499(1.22)  LDD1595  [4]
 LDCM0392  CL121 HEK-293T C247(0.99); C499(1.04)  LDD1596  [4]
 LDCM0393  CL122 HEK-293T C247(0.83); C499(1.09)  LDD1597  [4]
 LDCM0394  CL123 HEK-293T C499(1.11)  LDD1598  [4]
 LDCM0395  CL124 HEK-293T C499(1.01)  LDD1599  [4]
 LDCM0396  CL125 HEK-293T C247(0.89); C499(0.92)  LDD1600  [4]
 LDCM0397  CL126 HEK-293T C247(0.80); C499(0.96)  LDD1601  [4]
 LDCM0398  CL127 HEK-293T C499(0.96)  LDD1602  [4]
 LDCM0399  CL128 HEK-293T C499(1.00)  LDD1603  [4]
 LDCM0400  CL13 HEK-293T C247(0.88); C499(1.09)  LDD1604  [4]
 LDCM0401  CL14 HEK-293T C247(0.88); C499(1.12)  LDD1605  [4]
 LDCM0402  CL15 HEK-293T C499(0.94)  LDD1606  [4]
 LDCM0403  CL16 HEK-293T C121(0.96)  LDD1001  [3]
 LDCM0404  CL17 HEK-293T C121(0.87)  LDD1002  [3]
 LDCM0405  CL18 HEK-293T C121(0.91)  LDD1003  [3]
 LDCM0406  CL19 HEK-293T C121(1.06)  LDD1004  [3]
 LDCM0407  CL2 HEK-293T C247(1.03); C499(1.10)  LDD1611  [4]
 LDCM0408  CL20 HEK-293T C121(1.04)  LDD1006  [3]
 LDCM0409  CL21 HEK-293T C121(1.23)  LDD1007  [3]
 LDCM0410  CL22 HEK-293T C121(1.08)  LDD1008  [3]
 LDCM0411  CL23 HEK-293T C121(0.98)  LDD1009  [3]
 LDCM0412  CL24 HEK-293T C121(0.90)  LDD1010  [3]
 LDCM0413  CL25 HEK-293T C121(1.02)  LDD1011  [3]
 LDCM0414  CL26 HEK-293T C121(0.96)  LDD1012  [3]
 LDCM0415  CL27 HEK-293T C121(1.11)  LDD1013  [3]
 LDCM0416  CL28 HEK-293T C121(1.02)  LDD1014  [3]
 LDCM0417  CL29 HEK-293T C121(0.99)  LDD1015  [3]
 LDCM0418  CL3 HEK-293T C499(0.78)  LDD1622  [4]
 LDCM0419  CL30 HEK-293T C121(1.32)  LDD1017  [3]
 LDCM0420  CL31 HEK-293T C121(0.95)  LDD1018  [3]
 LDCM0421  CL32 HEK-293T C121(1.07)  LDD1019  [3]
 LDCM0422  CL33 HEK-293T C121(1.19)  LDD1020  [3]
 LDCM0423  CL34 HEK-293T C121(1.10)  LDD1021  [3]
 LDCM0424  CL35 HEK-293T C121(1.20)  LDD1022  [3]
 LDCM0425  CL36 HEK-293T C121(1.19)  LDD1023  [3]
 LDCM0426  CL37 HEK-293T C121(1.22)  LDD1024  [3]
 LDCM0428  CL39 HEK-293T C121(1.73)  LDD1026  [3]
 LDCM0429  CL4 HEK-293T C499(0.40)  LDD1633  [4]
 LDCM0430  CL40 HEK-293T C121(1.26)  LDD1028  [3]
 LDCM0431  CL41 HEK-293T C121(1.48)  LDD1029  [3]
 LDCM0432  CL42 HEK-293T C121(1.58)  LDD1030  [3]
 LDCM0433  CL43 HEK-293T C121(1.90)  LDD1031  [3]
 LDCM0434  CL44 HEK-293T C121(1.15)  LDD1032  [3]
 LDCM0435  CL45 HEK-293T C121(1.66)  LDD1033  [3]
 LDCM0436  CL46 HEK-293T C121(1.17)  LDD1034  [3]
 LDCM0437  CL47 HEK-293T C121(1.12)  LDD1035  [3]
 LDCM0438  CL48 HEK-293T C121(1.05)  LDD1036  [3]
 LDCM0439  CL49 HEK-293T C121(1.10)  LDD1037  [3]
 LDCM0440  CL5 HEK-293T C499(0.96); C1033(1.07)  LDD1644  [4]
 LDCM0441  CL50 HEK-293T C121(1.52)  LDD1039  [3]
 LDCM0442  CL51 HEK-293T C121(1.15)  LDD1040  [3]
 LDCM0443  CL52 HEK-293T C121(0.94)  LDD1041  [3]
 LDCM0444  CL53 HEK-293T C121(1.03)  LDD1042  [3]
 LDCM0445  CL54 HEK-293T C121(1.05)  LDD1043  [3]
 LDCM0446  CL55 HEK-293T C121(1.21)  LDD1044  [3]
 LDCM0447  CL56 HEK-293T C121(0.97)  LDD1045  [3]
 LDCM0448  CL57 HEK-293T C121(1.14)  LDD1046  [3]
 LDCM0449  CL58 HEK-293T C121(1.22)  LDD1047  [3]
 LDCM0450  CL59 HEK-293T C121(1.43)  LDD1048  [3]
 LDCM0451  CL6 HEK-293T C499(1.16); C1033(0.87)  LDD1654  [4]
 LDCM0452  CL60 HEK-293T C121(1.49)  LDD1050  [3]
 LDCM0453  CL61 HEK-293T C121(1.23)  LDD1051  [3]
 LDCM0454  CL62 HEK-293T C121(1.04)  LDD1052  [3]
 LDCM0455  CL63 HEK-293T C121(1.22)  LDD1053  [3]
 LDCM0456  CL64 HEK-293T C121(1.05)  LDD1054  [3]
 LDCM0457  CL65 HEK-293T C121(1.26)  LDD1055  [3]
 LDCM0458  CL66 HEK-293T C121(1.16)  LDD1056  [3]
 LDCM0459  CL67 HEK-293T C121(1.11)  LDD1057  [3]
 LDCM0460  CL68 HEK-293T C121(1.14)  LDD1058  [3]
 LDCM0461  CL69 HEK-293T C121(1.07)  LDD1059  [3]
 LDCM0462  CL7 HEK-293T C499(1.21)  LDD1665  [4]
 LDCM0463  CL70 HEK-293T C121(1.07)  LDD1061  [3]
 LDCM0464  CL71 HEK-293T C121(1.12)  LDD1062  [3]
 LDCM0465  CL72 HEK-293T C121(1.05)  LDD1063  [3]
 LDCM0466  CL73 HEK-293T C121(1.14)  LDD1064  [3]
 LDCM0467  CL74 HEK-293T C121(1.69)  LDD1065  [3]
 LDCM0469  CL76 HEK-293T C121(1.18)  LDD1067  [3]
 LDCM0470  CL77 HEK-293T C121(1.03)  LDD1068  [3]
 LDCM0471  CL78 HEK-293T C121(1.64)  LDD1069  [3]
 LDCM0472  CL79 HEK-293T C121(1.43)  LDD1070  [3]
 LDCM0473  CL8 HEK-293T C499(0.67)  LDD1676  [4]
 LDCM0474  CL80 HEK-293T C121(1.39)  LDD1072  [3]
 LDCM0475  CL81 HEK-293T C121(1.28)  LDD1073  [3]
 LDCM0476  CL82 HEK-293T C121(1.07)  LDD1074  [3]
 LDCM0477  CL83 HEK-293T C121(1.12)  LDD1075  [3]
 LDCM0478  CL84 HEK-293T C121(1.60)  LDD1076  [3]
 LDCM0479  CL85 HEK-293T C121(1.45)  LDD1077  [3]
 LDCM0480  CL86 HEK-293T C121(1.85)  LDD1078  [3]
 LDCM0481  CL87 HEK-293T C121(1.50)  LDD1079  [3]
 LDCM0482  CL88 HEK-293T C121(1.26)  LDD1080  [3]
 LDCM0483  CL89 HEK-293T C121(1.51)  LDD1081  [3]
 LDCM0484  CL9 HEK-293T C499(1.05)  LDD1687  [4]
 LDCM0485  CL90 HEK-293T C121(1.28)  LDD1083  [3]
 LDCM0486  CL91 HEK-293T C121(0.60)  LDD1084  [3]
 LDCM0487  CL92 HEK-293T C121(0.54)  LDD1085  [3]
 LDCM0488  CL93 HEK-293T C121(0.48)  LDD1086  [3]
 LDCM0489  CL94 HEK-293T C121(0.53)  LDD1087  [3]
 LDCM0490  CL95 HEK-293T C121(0.69)  LDD1088  [3]
 LDCM0491  CL96 HEK-293T C121(0.55)  LDD1089  [3]
 LDCM0492  CL97 HEK-293T C121(0.54)  LDD1090  [3]
 LDCM0493  CL98 HEK-293T C121(0.51)  LDD1091  [3]
 LDCM0494  CL99 HEK-293T C121(0.89)  LDD1092  [3]
 LDCM0495  E2913 HEK-293T C499(0.93)  LDD1698  [4]
 LDCM0468  Fragment33 HEK-293T C121(1.58)  LDD1066  [3]
 LDCM0427  Fragment51 HEK-293T C121(1.16)  LDD1025  [3]
 LDCM0022  KB02 HEK-293T C499(1.04)  LDD1492  [4]
 LDCM0023  KB03 HEK-293T C499(0.91)  LDD1497  [4]
 LDCM0024  KB05 PC-3 C234(1.90)  LDD3395  [1]

References

1 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840
2 Chemoproteomic profiling of targets of lipid-derived electrophiles by bioorthogonal aminooxy probe. Redox Biol. 2017 Aug;12:712-718. doi: 10.1016/j.redox.2017.04.001. Epub 2017 Apr 5.
3 Reimagining high-throughput profiling of reactive cysteines for cell-based screening of large electrophile libraries. Nat Biotechnol. 2021 May;39(5):630-641. doi: 10.1038/s41587-020-00778-3. Epub 2021 Jan 4.
4 Accelerating multiplexed profiling of protein-ligand interactions: High-throughput plate-based reactive cysteine profiling with minimal input. Cell Chem Biol. 2024 Mar 21;31(3):565-576.e4. doi: 10.1016/j.chembiol.2023.11.015. Epub 2023 Dec 19.
Mass spectrometry data entry: PXD044402