General Information of Target

Target ID LDTP04669
Target Name Microfibril-associated glycoprotein 3 (MFAP3)
Gene Name MFAP3
Gene ID 4238
Synonyms
Microfibril-associated glycoprotein 3
3D Structure
Download
2D Sequence (FASTA)
Download
3D Structure (PDB)
Download
Sequence
MKLHCCLFTLVASIIVPAAFVLEDVDFDQMVSLEANRSSYNASFPSSFELSASSHSDDDV
IIAKEGTSVSIECLLTASHYEDVHWHNSKGQQLDGRSRGGKWLVSDNFLNITNVAFDDRG
LYTCFVTSPIRASYSVTLRVIFTSGDMSVYYMIVCLIAFTITLILNVTRLCMMSSHLRKT
EKAINEFFRTEGAEKLQKAFEIAKRIPIITSAKTLELAKVTQFKTMEFARYIEELARSVP
LPPLILNCRAFVEEMFEAVRVDDPDDLGERIKERPALNAQGGIYVINPEMGRSNSPGGDS
DDGSLNEQGQEIAVQVSVHLQSETKSIDTESQGSSHFSPPDDIGSAESNCNYKDGAYENC
QL
Target Bioclass
Immunoglobulin
Subcellular location
Cell membrane
Function Component of the elastin-associated microfibrils.
Uniprot ID
P55082
Ensemble ID
ENST00000322602.9
HGNC ID
HGNC:7034

Target Site Mutations in Different Cell Lines

Cell line Mutation details Probe for labeling this protein in this cell
COLO792 SNV: p.L177F .
HCT15 SNV: p.W85L .
YSCCC SNV: p.E358K .

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 6 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
STPyne
 Probe Info 
K204(0.86)  LDD0277  [1]
Acrolein
 Probe Info 
C171(0.00); H176(0.00)  LDD0227  [2]
DBIA
 Probe Info 
C248(2.26); C360(1.57)  LDD0080  [3]
IA-alkyne
 Probe Info 
N.A.  LDD0165  [4]
JW-RF-010
 Probe Info 
N.A.  LDD0026  [5]
TFBX
 Probe Info 
N.A.  LDD0027  [5]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0214  AC1 HCT 116 C248(1.10)  LDD0531  [3]
 LDCM0215  AC10 HCT 116 C248(0.82)  LDD0532  [3]
 LDCM0216  AC100 HEK-293T C360(0.94)  LDD0814  [3]
 LDCM0217  AC101 HEK-293T C360(1.02)  LDD0815  [3]
 LDCM0218  AC102 HEK-293T C360(1.08)  LDD0816  [3]
 LDCM0219  AC103 HEK-293T C360(0.90)  LDD0817  [3]
 LDCM0220  AC104 HEK-293T C360(1.07)  LDD0818  [3]
 LDCM0221  AC105 HEK-293T C360(1.12)  LDD0819  [3]
 LDCM0222  AC106 HEK-293T C360(1.01)  LDD0820  [3]
 LDCM0223  AC107 HEK-293T C360(1.07)  LDD0821  [3]
 LDCM0224  AC108 HEK-293T C360(0.90)  LDD0822  [3]
 LDCM0225  AC109 HEK-293T C360(0.99)  LDD0823  [3]
 LDCM0226  AC11 HCT 116 C248(1.22)  LDD0543  [3]
 LDCM0227  AC110 HEK-293T C360(1.05)  LDD0825  [3]
 LDCM0228  AC111 HEK-293T C360(1.28)  LDD0826  [3]
 LDCM0229  AC112 HEK-293T C360(1.21)  LDD0827  [3]
 LDCM0230  AC113 HCT 116 C248(1.13)  LDD0547  [3]
 LDCM0231  AC114 HCT 116 C248(1.11)  LDD0548  [3]
 LDCM0232  AC115 HCT 116 C248(1.41)  LDD0549  [3]
 LDCM0233  AC116 HCT 116 C248(1.22)  LDD0550  [3]
 LDCM0234  AC117 HCT 116 C248(1.08)  LDD0551  [3]
 LDCM0235  AC118 HCT 116 C248(1.14)  LDD0552  [3]
 LDCM0236  AC119 HCT 116 C248(1.10)  LDD0553  [3]
 LDCM0237  AC12 HCT 116 C248(0.99)  LDD0554  [3]
 LDCM0238  AC120 HCT 116 C248(1.04)  LDD0555  [3]
 LDCM0239  AC121 HCT 116 C248(1.03)  LDD0556  [3]
 LDCM0240  AC122 HCT 116 C248(1.19)  LDD0557  [3]
 LDCM0241  AC123 HCT 116 C248(1.01)  LDD0558  [3]
 LDCM0242  AC124 HCT 116 C248(1.24)  LDD0559  [3]
 LDCM0243  AC125 HCT 116 C248(1.00)  LDD0560  [3]
 LDCM0244  AC126 HCT 116 C248(1.20)  LDD0561  [3]
 LDCM0245  AC127 HCT 116 C248(1.22)  LDD0562  [3]
 LDCM0259  AC14 HCT 116 C248(0.97)  LDD0576  [3]
 LDCM0270  AC15 HCT 116 C248(0.99)  LDD0587  [3]
 LDCM0276  AC17 HEK-293T C248(1.00)  LDD1515  [6]
 LDCM0277  AC18 HEK-293T C248(1.12)  LDD1516  [6]
 LDCM0278  AC19 HEK-293T C248(0.82)  LDD1517  [6]
 LDCM0279  AC2 HCT 116 C248(1.16)  LDD0596  [3]
 LDCM0280  AC20 HEK-293T C248(0.98)  LDD1519  [6]
 LDCM0281  AC21 HEK-293T C248(0.99)  LDD1520  [6]
 LDCM0282  AC22 HEK-293T C248(0.88)  LDD1521  [6]
 LDCM0283  AC23 HEK-293T C248(0.99)  LDD1522  [6]
 LDCM0284  AC24 HEK-293T C248(1.04)  LDD1523  [6]
 LDCM0285  AC25 HEK-293T C360(1.29)  LDD0883  [3]
 LDCM0286  AC26 HEK-293T C360(1.12)  LDD0884  [3]
 LDCM0287  AC27 HEK-293T C360(1.07)  LDD0885  [3]
 LDCM0288  AC28 HEK-293T C360(1.34)  LDD0886  [3]
 LDCM0289  AC29 HEK-293T C360(1.24)  LDD0887  [3]
 LDCM0290  AC3 HCT 116 C248(1.42)  LDD0607  [3]
 LDCM0291  AC30 HEK-293T C360(1.19)  LDD0889  [3]
 LDCM0292  AC31 HEK-293T C360(1.10)  LDD0890  [3]
 LDCM0293  AC32 HEK-293T C360(1.10)  LDD0891  [3]
 LDCM0294  AC33 HEK-293T C360(1.22)  LDD0892  [3]
 LDCM0295  AC34 HEK-293T C360(1.43)  LDD0893  [3]
 LDCM0296  AC35 HEK-293T C248(0.90)  LDD1535  [6]
 LDCM0297  AC36 HEK-293T C248(0.94)  LDD1536  [6]
 LDCM0298  AC37 HEK-293T C248(0.93)  LDD1537  [6]
 LDCM0299  AC38 HEK-293T C248(0.88)  LDD1538  [6]
 LDCM0300  AC39 HEK-293T C248(0.98)  LDD1539  [6]
 LDCM0301  AC4 HCT 116 C248(1.18)  LDD0618  [3]
 LDCM0302  AC40 HEK-293T C248(0.93)  LDD1541  [6]
 LDCM0303  AC41 HEK-293T C248(0.92)  LDD1542  [6]
 LDCM0304  AC42 HEK-293T C248(1.04)  LDD1543  [6]
 LDCM0305  AC43 HEK-293T C248(0.93)  LDD1544  [6]
 LDCM0306  AC44 HEK-293T C248(1.20)  LDD1545  [6]
 LDCM0307  AC45 HEK-293T C248(0.93)  LDD1546  [6]
 LDCM0308  AC46 HEK-293T C248(0.97)  LDD1547  [6]
 LDCM0309  AC47 HEK-293T C248(0.89)  LDD1548  [6]
 LDCM0310  AC48 HEK-293T C248(1.02)  LDD1549  [6]
 LDCM0311  AC49 HEK-293T C248(0.98)  LDD1550  [6]
 LDCM0312  AC5 HCT 116 C248(1.17)  LDD0629  [3]
 LDCM0313  AC50 HEK-293T C248(0.93)  LDD1552  [6]
 LDCM0314  AC51 HEK-293T C248(0.85)  LDD1553  [6]
 LDCM0315  AC52 HEK-293T C248(0.92)  LDD1554  [6]
 LDCM0316  AC53 HEK-293T C248(0.96)  LDD1555  [6]
 LDCM0317  AC54 HEK-293T C248(1.04)  LDD1556  [6]
 LDCM0318  AC55 HEK-293T C248(0.91)  LDD1557  [6]
 LDCM0319  AC56 HEK-293T C248(1.12)  LDD1558  [6]
 LDCM0320  AC57 HEK-293T C248(1.00); C360(0.95)  LDD0918  [3]
 LDCM0321  AC58 HEK-293T C248(0.83); C360(0.87)  LDD0919  [3]
 LDCM0322  AC59 HEK-293T C248(1.15); C360(0.85)  LDD0920  [3]
 LDCM0323  AC6 HCT 116 C248(0.98)  LDD0640  [3]
 LDCM0324  AC60 HEK-293T C248(0.63); C360(0.94)  LDD0922  [3]
 LDCM0325  AC61 HEK-293T C248(0.86); C360(0.99)  LDD0923  [3]
 LDCM0326  AC62 HEK-293T C248(0.80); C360(0.99)  LDD0924  [3]
 LDCM0327  AC63 HEK-293T C248(0.95); C360(0.91)  LDD0925  [3]
 LDCM0328  AC64 HEK-293T C248(0.69); C360(1.29)  LDD0926  [3]
 LDCM0329  AC65 HEK-293T C248(0.97); C360(1.10)  LDD0927  [3]
 LDCM0330  AC66 HEK-293T C248(0.94); C360(1.10)  LDD0928  [3]
 LDCM0331  AC67 HEK-293T C248(1.21); C360(1.01)  LDD0929  [3]
 LDCM0334  AC7 HCT 116 C248(1.05)  LDD0651  [3]
 LDCM0345  AC8 HCT 116 C248(1.12)  LDD0662  [3]
 LDCM0349  AC83 HEK-293T C360(1.25)  LDD0947  [3]
 LDCM0350  AC84 HEK-293T C360(1.01)  LDD0948  [3]
 LDCM0351  AC85 HEK-293T C360(1.08)  LDD0949  [3]
 LDCM0352  AC86 HEK-293T C360(1.03)  LDD0950  [3]
 LDCM0353  AC87 HEK-293T C360(1.14)  LDD0951  [3]
 LDCM0354  AC88 HEK-293T C360(0.91)  LDD0952  [3]
 LDCM0355  AC89 HEK-293T C360(1.07)  LDD0953  [3]
 LDCM0357  AC90 HEK-293T C360(0.94)  LDD0955  [3]
 LDCM0358  AC91 HEK-293T C360(1.02)  LDD0956  [3]
 LDCM0359  AC92 HEK-293T C360(1.12)  LDD0957  [3]
 LDCM0360  AC93 HEK-293T C360(1.20)  LDD0958  [3]
 LDCM0361  AC94 HEK-293T C360(1.23)  LDD0959  [3]
 LDCM0362  AC95 HEK-293T C360(0.94)  LDD0960  [3]
 LDCM0363  AC96 HEK-293T C360(1.00)  LDD0961  [3]
 LDCM0364  AC97 HEK-293T C360(1.09)  LDD0962  [3]
 LDCM0365  AC98 HEK-293T C360(0.84)  LDD0963  [3]
 LDCM0366  AC99 HEK-293T C360(0.87)  LDD0964  [3]
 LDCM0248  AKOS034007472 HCT 116 C248(1.14)  LDD0565  [3]
 LDCM0356  AKOS034007680 HCT 116 C248(1.04)  LDD0673  [3]
 LDCM0275  AKOS034007705 HCT 116 C248(1.10)  LDD0592  [3]
 LDCM0367  CL1 HEK-293T C248(1.47)  LDD0965  [3]
 LDCM0368  CL10 HEK-293T C248(1.59)  LDD0966  [3]
 LDCM0369  CL100 HCT 116 C248(1.05)  LDD0686  [3]
 LDCM0370  CL101 HCT 116 C248(0.79)  LDD0687  [3]
 LDCM0371  CL102 HCT 116 C248(0.99)  LDD0688  [3]
 LDCM0372  CL103 HCT 116 C248(1.12)  LDD0689  [3]
 LDCM0373  CL104 HCT 116 C248(1.13)  LDD0690  [3]
 LDCM0374  CL105 HEK-293T C248(1.01)  LDD1578  [6]
 LDCM0375  CL106 HEK-293T C248(1.05)  LDD1579  [6]
 LDCM0376  CL107 HEK-293T C248(0.98)  LDD1580  [6]
 LDCM0377  CL108 HEK-293T C248(1.04)  LDD1581  [6]
 LDCM0378  CL109 HEK-293T C248(1.18)  LDD1582  [6]
 LDCM0379  CL11 HEK-293T C248(1.12)  LDD0977  [3]
 LDCM0380  CL110 HEK-293T C248(1.30)  LDD1584  [6]
 LDCM0381  CL111 HEK-293T C248(0.88)  LDD1585  [6]
 LDCM0382  CL112 HEK-293T C360(1.30)  LDD0980  [3]
 LDCM0383  CL113 HEK-293T C360(1.25)  LDD0981  [3]
 LDCM0384  CL114 HEK-293T C360(1.03)  LDD0982  [3]
 LDCM0385  CL115 HEK-293T C360(1.39)  LDD0983  [3]
 LDCM0386  CL116 HEK-293T C360(1.42)  LDD0984  [3]
 LDCM0387  CL117 HEK-293T C248(0.97)  LDD1591  [6]
 LDCM0388  CL118 HEK-293T C248(0.97)  LDD1592  [6]
 LDCM0389  CL119 HEK-293T C248(0.99)  LDD1593  [6]
 LDCM0390  CL12 HEK-293T C248(0.99)  LDD0988  [3]
 LDCM0391  CL120 HEK-293T C248(0.93)  LDD1595  [6]
 LDCM0392  CL121 HEK-293T C248(0.98)  LDD1596  [6]
 LDCM0393  CL122 HEK-293T C248(1.07)  LDD1597  [6]
 LDCM0394  CL123 HEK-293T C248(0.89)  LDD1598  [6]
 LDCM0395  CL124 HEK-293T C248(1.19)  LDD1599  [6]
 LDCM0396  CL125 HEK-293T C248(0.97); C360(0.87)  LDD0994  [3]
 LDCM0397  CL126 HEK-293T C248(0.76); C360(1.03)  LDD0995  [3]
 LDCM0398  CL127 HEK-293T C248(0.59); C360(1.22)  LDD0996  [3]
 LDCM0399  CL128 HEK-293T C248(0.94); C360(0.89)  LDD0997  [3]
 LDCM0400  CL13 HEK-293T C248(0.91)  LDD0998  [3]
 LDCM0401  CL14 HEK-293T C248(0.96)  LDD0999  [3]
 LDCM0402  CL15 HEK-293T C248(1.14)  LDD1000  [3]
 LDCM0403  CL16 HEK-293T C248(0.94)  LDD1001  [3]
 LDCM0404  CL17 HEK-293T C248(0.77)  LDD1002  [3]
 LDCM0405  CL18 HEK-293T C248(1.16)  LDD1003  [3]
 LDCM0406  CL19 HEK-293T C248(0.95)  LDD1004  [3]
 LDCM0407  CL2 HEK-293T C248(0.81)  LDD1005  [3]
 LDCM0408  CL20 HEK-293T C248(0.92)  LDD1006  [3]
 LDCM0409  CL21 HEK-293T C248(0.82)  LDD1007  [3]
 LDCM0410  CL22 HEK-293T C248(0.79)  LDD1008  [3]
 LDCM0411  CL23 HEK-293T C248(0.45)  LDD1009  [3]
 LDCM0412  CL24 HEK-293T C248(0.79)  LDD1010  [3]
 LDCM0413  CL25 HEK-293T C248(0.73)  LDD1011  [3]
 LDCM0414  CL26 HEK-293T C248(0.85)  LDD1012  [3]
 LDCM0415  CL27 HEK-293T C248(0.83)  LDD1013  [3]
 LDCM0416  CL28 HEK-293T C248(0.71)  LDD1014  [3]
 LDCM0417  CL29 HEK-293T C248(0.75)  LDD1015  [3]
 LDCM0418  CL3 HEK-293T C248(1.65)  LDD1016  [3]
 LDCM0419  CL30 HEK-293T C248(0.84)  LDD1017  [3]
 LDCM0420  CL31 HEK-293T C248(1.44)  LDD1018  [3]
 LDCM0421  CL32 HEK-293T C248(1.49)  LDD1019  [3]
 LDCM0422  CL33 HEK-293T C248(1.41)  LDD1020  [3]
 LDCM0423  CL34 HEK-293T C248(1.00)  LDD1021  [3]
 LDCM0424  CL35 HEK-293T C248(1.35)  LDD1022  [3]
 LDCM0425  CL36 HEK-293T C248(1.14)  LDD1023  [3]
 LDCM0426  CL37 HEK-293T C248(1.14)  LDD1024  [3]
 LDCM0428  CL39 HEK-293T C248(1.45)  LDD1026  [3]
 LDCM0429  CL4 HEK-293T C248(1.03)  LDD1027  [3]
 LDCM0430  CL40 HEK-293T C248(1.04)  LDD1028  [3]
 LDCM0431  CL41 HEK-293T C248(1.19)  LDD1029  [3]
 LDCM0432  CL42 HEK-293T C248(1.36)  LDD1030  [3]
 LDCM0433  CL43 HEK-293T C248(1.25)  LDD1031  [3]
 LDCM0434  CL44 HEK-293T C248(1.31)  LDD1032  [3]
 LDCM0435  CL45 HEK-293T C248(1.23)  LDD1033  [3]
 LDCM0436  CL46 HCT 116 C248(0.59)  LDD0753  [3]
 LDCM0437  CL47 HCT 116 C248(0.54)  LDD0754  [3]
 LDCM0438  CL48 HCT 116 C248(0.54)  LDD0755  [3]
 LDCM0439  CL49 HCT 116 C248(0.65)  LDD0756  [3]
 LDCM0440  CL5 HEK-293T C248(1.19)  LDD1038  [3]
 LDCM0441  CL50 HCT 116 C248(0.70)  LDD0758  [3]
 LDCM0442  CL51 HCT 116 C248(0.71)  LDD0759  [3]
 LDCM0443  CL52 HCT 116 C248(0.69)  LDD0760  [3]
 LDCM0444  CL53 HCT 116 C248(0.62)  LDD0761  [3]
 LDCM0445  CL54 HCT 116 C248(0.53)  LDD0762  [3]
 LDCM0446  CL55 HCT 116 C248(0.61)  LDD0763  [3]
 LDCM0447  CL56 HCT 116 C248(0.72)  LDD0764  [3]
 LDCM0448  CL57 HCT 116 C248(0.64)  LDD0765  [3]
 LDCM0449  CL58 HCT 116 C248(0.60)  LDD0766  [3]
 LDCM0450  CL59 HCT 116 C248(0.72)  LDD0767  [3]
 LDCM0451  CL6 HEK-293T C248(0.72)  LDD1049  [3]
 LDCM0452  CL60 HCT 116 C248(0.79)  LDD0769  [3]
 LDCM0453  CL61 HCT 116 C248(1.04)  LDD0770  [3]
 LDCM0454  CL62 HCT 116 C248(1.04)  LDD0771  [3]
 LDCM0455  CL63 HCT 116 C248(1.24)  LDD0772  [3]
 LDCM0456  CL64 HCT 116 C248(1.27)  LDD0773  [3]
 LDCM0457  CL65 HCT 116 C248(1.09)  LDD0774  [3]
 LDCM0458  CL66 HCT 116 C248(1.75)  LDD0775  [3]
 LDCM0459  CL67 HCT 116 C248(1.40)  LDD0776  [3]
 LDCM0460  CL68 HCT 116 C248(1.27)  LDD0777  [3]
 LDCM0461  CL69 HCT 116 C248(0.92)  LDD0778  [3]
 LDCM0462  CL7 HEK-293T C248(1.58)  LDD1060  [3]
 LDCM0463  CL70 HCT 116 C248(1.09)  LDD0780  [3]
 LDCM0464  CL71 HCT 116 C248(1.22)  LDD0781  [3]
 LDCM0465  CL72 HCT 116 C248(1.07)  LDD0782  [3]
 LDCM0466  CL73 HCT 116 C248(1.22)  LDD0783  [3]
 LDCM0467  CL74 HCT 116 C248(1.23)  LDD0784  [3]
 LDCM0469  CL76 HEK-293T C248(1.32)  LDD1067  [3]
 LDCM0470  CL77 HEK-293T C248(1.31)  LDD1068  [3]
 LDCM0471  CL78 HEK-293T C248(1.94)  LDD1069  [3]
 LDCM0472  CL79 HEK-293T C248(1.67)  LDD1070  [3]
 LDCM0473  CL8 HEK-293T C248(0.67)  LDD1071  [3]
 LDCM0474  CL80 HEK-293T C248(1.34)  LDD1072  [3]
 LDCM0475  CL81 HEK-293T C248(0.98)  LDD1073  [3]
 LDCM0476  CL82 HEK-293T C248(0.83)  LDD1074  [3]
 LDCM0477  CL83 HEK-293T C248(1.06)  LDD1075  [3]
 LDCM0478  CL84 HEK-293T C248(2.18)  LDD1076  [3]
 LDCM0479  CL85 HEK-293T C248(1.43)  LDD1077  [3]
 LDCM0480  CL86 HEK-293T C248(1.45)  LDD1078  [3]
 LDCM0481  CL87 HEK-293T C248(1.37)  LDD1079  [3]
 LDCM0482  CL88 HEK-293T C248(1.16)  LDD1080  [3]
 LDCM0483  CL89 HEK-293T C248(1.32)  LDD1081  [3]
 LDCM0484  CL9 HEK-293T C248(1.51)  LDD1082  [3]
 LDCM0485  CL90 HEK-293T C248(1.45)  LDD1083  [3]
 LDCM0486  CL91 HCT 116 C248(1.20)  LDD0803  [3]
 LDCM0487  CL92 HCT 116 C248(0.88)  LDD0804  [3]
 LDCM0488  CL93 HCT 116 C248(0.78)  LDD0805  [3]
 LDCM0489  CL94 HCT 116 C248(0.71)  LDD0806  [3]
 LDCM0490  CL95 HCT 116 C248(0.99)  LDD0807  [3]
 LDCM0491  CL96 HCT 116 C248(1.23)  LDD0808  [3]
 LDCM0492  CL97 HCT 116 C248(1.16)  LDD0809  [3]
 LDCM0493  CL98 HCT 116 C248(1.34)  LDD0810  [3]
 LDCM0494  CL99 HCT 116 C248(1.23)  LDD0811  [3]
 LDCM0495  E2913 HEK-293T C248(1.00)  LDD1698  [6]
 LDCM0468  Fragment33 HCT 116 C248(1.16)  LDD0785  [3]
 LDCM0427  Fragment51 HEK-293T C248(1.27)  LDD1025  [3]
 LDCM0022  KB02 HCT 116 C248(2.26); C360(1.57)  LDD0080  [3]
 LDCM0023  KB03 HCT 116 C248(20.00); C360(1.18)  LDD0081  [3]
 LDCM0024  KB05 HCT 116 C248(7.90); C360(1.67)  LDD0082  [3]
 LDCM0109  NEM HeLa C171(0.00); H176(0.00)  LDD0227  [2]

References

1 A Paal-Knorr agent for chemoproteomic profiling of targets of isoketals in cells. Chem Sci. 2021 Oct 15;12(43):14557-14563. doi: 10.1039/d1sc02230j. eCollection 2021 Nov 10.
Mass spectrometry data entry: PXD028270
2 ACR-Based Probe for the Quantitative Profiling of Histidine Reactivity in the Human Proteome. J Am Chem Soc. 2023 Mar 8;145(9):5252-5260. doi: 10.1021/jacs.2c12653. Epub 2023 Feb 27.
3 Reimagining high-throughput profiling of reactive cysteines for cell-based screening of large electrophile libraries. Nat Biotechnol. 2021 May;39(5):630-641. doi: 10.1038/s41587-020-00778-3. Epub 2021 Jan 4.
4 SP3-FAIMS Chemoproteomics for High-Coverage Profiling of the Human Cysteinome*. Chembiochem. 2021 May 14;22(10):1841-1851. doi: 10.1002/cbic.202000870. Epub 2021 Feb 18.
Mass spectrometry data entry: PXD023056 , PXD023059 , PXD023058 , PXD023057 , PXD023060
5 Chemoproteomic Profiling by Cysteine Fluoroalkylation Reveals Myrocin G as an Inhibitor of the Nonhomologous End Joining DNA Repair Pathway. J Am Chem Soc. 2021 Dec 8;143(48):20332-20342. doi: 10.1021/jacs.1c09724. Epub 2021 Nov 24.
Mass spectrometry data entry: PXD029255
6 Accelerating multiplexed profiling of protein-ligand interactions: High-throughput plate-based reactive cysteine profiling with minimal input. Cell Chem Biol. 2024 Mar 21;31(3):565-576.e4. doi: 10.1016/j.chembiol.2023.11.015. Epub 2023 Dec 19.
Mass spectrometry data entry: PXD044402