Details of the Target

General Information of Target

Target ID LDTP04734
Target Name Myc-associated zinc finger protein (MAZ)
Gene Name MAZ
Gene ID 4150
Synonyms
ZNF801; Myc-associated zinc finger protein; MAZI; Pur-1; Purine-binding transcription factor; Serum amyloid A-activating factor-1; SAF-1; Transcription factor Zif87; ZF87; Zinc finger protein 801
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MFPVFPCTLLAPPFPVLGLDSRGVGGLMNSFPPPQGHAQNPLQVGAELQSRFFASQGCAQ
SPFQAAPAPPPTPQAPAAEPLQVDLLPVLAAAQESAAAAAAAAAAAAAVAAAPPAPAAAS
TVDTAALKQPPAPPPPPPPVSAPAAEAAPPASAATIAAAAATAVVAPTSTVAVAPVASAL
EKKTKSKGPYICALCAKEFKNGYNLRRHEAIHTGAKAGRVPSGAMKMPTMVPLSLLSVPQ
LSGAGGGGGEAGAGGGAAAVAAGGVVTTTASGKRIRKNHACEMCGKAFRDVYHLNRHKLS
HSDEKPYQCPVCQQRFKRKDRMSYHVRSHDGAVHKPYNCSHCGKSFSRPDHLNSHVRQVH
STERPFKCEKCEAAFATKDRLRAHTVRHEEKVPCHVCGKMLSSAYISDHMKVHSQGPHHV
CELCNKGTGEVCPMAAAAAAAAAAAAAAVAAPPTAVGSLSGAEGVPVSSQPLPSQPW
Target Type
Literature-reported
Target Bioclass
Transcription factor
Subcellular location
Nucleus
Function
Transcriptional regulator, potentially with dual roles in transcription initiation and termination.; [Isoform 1]: Binds DNA and functions as a transcriptional activator. Binds to two G/A-rich sites, ME1a1 and ME1a2, within the MYC promoter having greater affinity for the former. Also binds to multiple G/C-rich sites within the promoter of the Sp1 family of transcription factors.; [Isoform 2]: Binds DNA and functions as a transcriptional activator. Inhibits MAZ isoform 1-mediated transcription.; [Isoform 3]: Binds DNA and functions as a transcriptional activator.
TTD ID
T60042
Uniprot ID
P56270
DrugMap ID
TT059DA
Ensemble ID
ENST00000219782.11
HGNC ID
HGNC:6914

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 11 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
TH211
 Probe Info  		Y307(20.00); Y337(20.00); Y405(7.01)  LDD0257  [1]
DBIA
 Probe Info  		C66(1.01)  LDD3315  [2]
m-APA
 Probe Info  		N.A.  LDD2231  [3]
IA-alkyne
 Probe Info  		C371(0.00); C309(0.00); C421(0.00)  LDD0165  [4]
TFBX
 Probe Info  		N.A.  LDD0027  [5]
IPM
 Probe Info  		C424(0.00); C421(0.00)  LDD0005  [6]
OSF
 Probe Info  		N.A.  LDD0029  [7]
SF
 Probe Info  		N.A.  LDD0028  [7]
Phosphinate-6
 Probe Info  		C397(0.00); C394(0.00); C368(0.00); C342(0.00)  LDD0018  [8]
Acrolein
 Probe Info  		C421(0.00); C424(0.00)  LDD0217  [9]
W1
 Probe Info  		C281(0.00); C284(0.00)  LDD0236  [10]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0025  4SU-RNA HEK-293T C421(2.15)  LDD0371  [11]
 LDCM0214  AC1 HEK-293T C424(1.02)  LDD1507  [12]
 LDCM0215  AC10 HEK-293T C421(1.21)  LDD1508  [12]
 LDCM0226  AC11 HEK-293T C421(0.98)  LDD1509  [12]
 LDCM0237  AC12 HEK-293T C394(1.03)  LDD1510  [12]
 LDCM0259  AC14 HEK-293T C394(1.09)  LDD1512  [12]
 LDCM0270  AC15 HEK-293T C421(1.07); C397(0.91)  LDD1513  [12]
 LDCM0276  AC17 HEK-293T C424(1.03)  LDD1515  [12]
 LDCM0277  AC18 HEK-293T C421(1.10)  LDD1516  [12]
 LDCM0278  AC19 HEK-293T C421(0.56)  LDD1517  [12]
 LDCM0279  AC2 HEK-293T C421(1.09)  LDD1518  [12]
 LDCM0280  AC20 HEK-293T C394(0.99)  LDD1519  [12]
 LDCM0281  AC21 HEK-293T C432(0.75); C424(0.92)  LDD1520  [12]
 LDCM0282  AC22 HEK-293T C394(0.99)  LDD1521  [12]
 LDCM0283  AC23 HEK-293T C421(1.04); C397(1.00)  LDD1522  [12]
 LDCM0284  AC24 HEK-293T C424(1.18)  LDD1523  [12]
 LDCM0285  AC25 HEK-293T C424(1.10)  LDD1524  [12]
 LDCM0286  AC26 HEK-293T C421(1.15)  LDD1525  [12]
 LDCM0287  AC27 HEK-293T C421(1.05)  LDD1526  [12]
 LDCM0288  AC28 HEK-293T C394(0.98)  LDD1527  [12]
 LDCM0289  AC29 HEK-293T C432(0.80); C424(0.92)  LDD1528  [12]
 LDCM0290  AC3 HEK-293T C421(1.03)  LDD1529  [12]
 LDCM0291  AC30 HEK-293T C394(0.98)  LDD1530  [12]
 LDCM0292  AC31 HEK-293T C421(1.12); C397(0.86)  LDD1531  [12]
 LDCM0293  AC32 HEK-293T C424(1.05)  LDD1532  [12]
 LDCM0294  AC33 HEK-293T C424(1.11)  LDD1533  [12]
 LDCM0295  AC34 HEK-293T C421(1.14)  LDD1534  [12]
 LDCM0296  AC35 HEK-293T C421(1.10)  LDD1535  [12]
 LDCM0297  AC36 HEK-293T C394(1.02)  LDD1536  [12]
 LDCM0298  AC37 HEK-293T C432(0.82); C424(0.90)  LDD1537  [12]
 LDCM0299  AC38 HEK-293T C394(1.12)  LDD1538  [12]
 LDCM0300  AC39 HEK-293T C421(1.13); C397(0.96)  LDD1539  [12]
 LDCM0301  AC4 HEK-293T C394(0.94)  LDD1540  [12]
 LDCM0302  AC40 HEK-293T C424(1.13)  LDD1541  [12]
 LDCM0303  AC41 HEK-293T C424(1.06)  LDD1542  [12]
 LDCM0304  AC42 HEK-293T C421(1.19)  LDD1543  [12]
 LDCM0305  AC43 HEK-293T C421(1.02)  LDD1544  [12]
 LDCM0306  AC44 HEK-293T C394(1.01)  LDD1545  [12]
 LDCM0307  AC45 HEK-293T C432(0.87); C424(0.92)  LDD1546  [12]
 LDCM0308  AC46 HEK-293T C394(1.04)  LDD1547  [12]
 LDCM0309  AC47 HEK-293T C421(1.07); C397(0.96)  LDD1548  [12]
 LDCM0310  AC48 HEK-293T C424(1.16)  LDD1549  [12]
 LDCM0311  AC49 HEK-293T C424(1.06)  LDD1550  [12]
 LDCM0312  AC5 HEK-293T C432(0.74); C424(0.88)  LDD1551  [12]
 LDCM0313  AC50 HEK-293T C421(1.10)  LDD1552  [12]
 LDCM0314  AC51 HEK-293T C421(1.00)  LDD1553  [12]
 LDCM0315  AC52 HEK-293T C394(0.92)  LDD1554  [12]
 LDCM0316  AC53 HEK-293T C432(0.81); C424(0.89)  LDD1555  [12]
 LDCM0317  AC54 HEK-293T C394(0.96)  LDD1556  [12]
 LDCM0318  AC55 HEK-293T C421(1.04); C397(0.97)  LDD1557  [12]
 LDCM0319  AC56 HEK-293T C424(1.13)  LDD1558  [12]
 LDCM0320  AC57 HEK-293T C424(1.07)  LDD1559  [12]
 LDCM0321  AC58 HEK-293T C421(0.98)  LDD1560  [12]
 LDCM0322  AC59 HEK-293T C421(0.97)  LDD1561  [12]
 LDCM0323  AC6 HEK-293T C394(0.97)  LDD1562  [12]
 LDCM0324  AC60 HEK-293T C394(0.98)  LDD1563  [12]
 LDCM0325  AC61 HEK-293T C432(0.79); C424(0.87)  LDD1564  [12]
 LDCM0326  AC62 HEK-293T C394(1.06)  LDD1565  [12]
 LDCM0327  AC63 HEK-293T C421(0.99); C397(1.00)  LDD1566  [12]
 LDCM0328  AC64 HEK-293T C424(1.01)  LDD1567  [12]
 LDCM0334  AC7 HEK-293T C421(1.04); C397(0.81)  LDD1568  [12]
 LDCM0345  AC8 HEK-293T C424(1.11)  LDD1569  [12]
 LDCM0248  AKOS034007472 HEK-293T C432(0.78); C424(0.95)  LDD1511  [12]
 LDCM0356  AKOS034007680 HEK-293T C424(1.12)  LDD1570  [12]
 LDCM0275  AKOS034007705 HEK-293T C424(1.23)  LDD1514  [12]
 LDCM0108  Chloroacetamide HeLa N.A.  LDD0222  [9]
 LDCM0367  CL1 HEK-293T C424(0.93); C421(0.95)  LDD1571  [12]
 LDCM0368  CL10 HEK-293T C394(0.84)  LDD1572  [12]
 LDCM0370  CL101 HEK-293T C424(1.07); C421(1.07)  LDD1574  [12]
 LDCM0371  CL102 HEK-293T C421(0.91)  LDD1575  [12]
 LDCM0372  CL103 HEK-293T C432(1.22)  LDD1576  [12]
 LDCM0374  CL105 HEK-293T C424(0.95); C421(1.08)  LDD1578  [12]
 LDCM0375  CL106 HEK-293T C421(0.93)  LDD1579  [12]
 LDCM0376  CL107 HEK-293T C432(1.64)  LDD1580  [12]
 LDCM0378  CL109 HEK-293T C424(0.99); C421(0.99)  LDD1582  [12]
 LDCM0379  CL11 HEK-293T C421(1.13); C397(1.05)  LDD1583  [12]
 LDCM0380  CL110 HEK-293T C421(0.97)  LDD1584  [12]
 LDCM0381  CL111 HEK-293T C432(1.16)  LDD1585  [12]
 LDCM0383  CL113 HEK-293T C424(1.07); C421(1.02)  LDD1587  [12]
 LDCM0384  CL114 HEK-293T C421(0.84)  LDD1588  [12]
 LDCM0385  CL115 HEK-293T C432(0.90)  LDD1589  [12]
 LDCM0387  CL117 HEK-293T C424(1.01); C421(0.95)  LDD1591  [12]
 LDCM0388  CL118 HEK-293T C421(0.87)  LDD1592  [12]
 LDCM0389  CL119 HEK-293T C432(1.66)  LDD1593  [12]
 LDCM0390  CL12 HEK-293T C424(1.00)  LDD1594  [12]
 LDCM0392  CL121 HEK-293T C424(1.00); C421(0.90)  LDD1596  [12]
 LDCM0393  CL122 HEK-293T C421(0.93)  LDD1597  [12]
 LDCM0394  CL123 HEK-293T C432(1.33)  LDD1598  [12]
 LDCM0396  CL125 HEK-293T C424(0.84); C421(0.78)  LDD1600  [12]
 LDCM0397  CL126 HEK-293T C421(0.90)  LDD1601  [12]
 LDCM0398  CL127 HEK-293T C432(1.08)  LDD1602  [12]
 LDCM0400  CL13 HEK-293T C424(0.81); C421(0.92)  LDD1604  [12]
 LDCM0401  CL14 HEK-293T C421(1.00)  LDD1605  [12]
 LDCM0402  CL15 HEK-293T C432(0.84)  LDD1606  [12]
 LDCM0404  CL17 HEK-293T C424(0.95)  LDD1608  [12]
 LDCM0405  CL18 HEK-293T C421(1.04)  LDD1609  [12]
 LDCM0406  CL19 HEK-293T C421(0.93)  LDD1610  [12]
 LDCM0407  CL2 HEK-293T C421(0.91)  LDD1611  [12]
 LDCM0408  CL20 HEK-293T C394(1.06)  LDD1612  [12]
 LDCM0409  CL21 HEK-293T C432(0.73); C424(0.85)  LDD1613  [12]
 LDCM0410  CL22 HEK-293T C394(1.24)  LDD1614  [12]
 LDCM0411  CL23 HEK-293T C421(1.15); C397(1.13)  LDD1615  [12]
 LDCM0412  CL24 HEK-293T C424(1.21)  LDD1616  [12]
 LDCM0413  CL25 HEK-293T C424(0.83); C421(0.88)  LDD1617  [12]
 LDCM0414  CL26 HEK-293T C421(1.00)  LDD1618  [12]
 LDCM0415  CL27 HEK-293T C432(1.06)  LDD1619  [12]
 LDCM0417  CL29 HEK-293T C424(1.00)  LDD1621  [12]
 LDCM0418  CL3 HEK-293T C432(0.95)  LDD1622  [12]
 LDCM0419  CL30 HEK-293T C421(1.02)  LDD1623  [12]
 LDCM0420  CL31 HEK-293T C421(0.98)  LDD1624  [12]
 LDCM0421  CL32 HEK-293T C394(1.01)  LDD1625  [12]
 LDCM0422  CL33 HEK-293T C432(0.65); C424(0.82)  LDD1626  [12]
 LDCM0423  CL34 HEK-293T C394(1.08)  LDD1627  [12]
 LDCM0424  CL35 HEK-293T C421(1.15); C397(1.11)  LDD1628  [12]
 LDCM0425  CL36 HEK-293T C424(1.23)  LDD1629  [12]
 LDCM0426  CL37 HEK-293T C424(0.99); C421(0.79)  LDD1630  [12]
 LDCM0428  CL39 HEK-293T C432(1.36)  LDD1632  [12]
 LDCM0431  CL41 HEK-293T C424(1.06)  LDD1635  [12]
 LDCM0432  CL42 HEK-293T C421(0.95)  LDD1636  [12]
 LDCM0433  CL43 HEK-293T C421(1.04)  LDD1637  [12]
 LDCM0434  CL44 HEK-293T C394(1.05)  LDD1638  [12]
 LDCM0435  CL45 HEK-293T C432(0.81); C424(0.87)  LDD1639  [12]
 LDCM0436  CL46 HEK-293T C394(1.08)  LDD1640  [12]
 LDCM0437  CL47 HEK-293T C421(1.12); C397(0.99)  LDD1641  [12]
 LDCM0438  CL48 HEK-293T C424(1.11)  LDD1642  [12]
 LDCM0439  CL49 HEK-293T C424(1.01); C421(0.79)  LDD1643  [12]
 LDCM0440  CL5 HEK-293T C424(1.04)  LDD1644  [12]
 LDCM0441  CL50 HEK-293T C421(1.00)  LDD1645  [12]
 LDCM0444  CL53 HEK-293T C424(1.08)  LDD1647  [12]
 LDCM0445  CL54 HEK-293T C421(0.93)  LDD1648  [12]
 LDCM0446  CL55 HEK-293T C421(1.04)  LDD1649  [12]
 LDCM0447  CL56 HEK-293T C394(1.02)  LDD1650  [12]
 LDCM0448  CL57 HEK-293T C432(0.79); C424(0.84)  LDD1651  [12]
 LDCM0449  CL58 HEK-293T C394(1.13)  LDD1652  [12]
 LDCM0450  CL59 HEK-293T C421(1.05); C397(0.96)  LDD1653  [12]
 LDCM0451  CL6 HEK-293T C421(0.89)  LDD1654  [12]
 LDCM0452  CL60 HEK-293T C424(1.07)  LDD1655  [12]
 LDCM0453  CL61 HEK-293T C424(0.88); C421(0.86)  LDD1656  [12]
 LDCM0454  CL62 HEK-293T C421(0.96)  LDD1657  [12]
 LDCM0455  CL63 HEK-293T C432(1.30)  LDD1658  [12]
 LDCM0457  CL65 HEK-293T C424(1.08)  LDD1660  [12]
 LDCM0458  CL66 HEK-293T C421(1.09)  LDD1661  [12]
 LDCM0459  CL67 HEK-293T C421(1.10)  LDD1662  [12]
 LDCM0460  CL68 HEK-293T C394(1.01)  LDD1663  [12]
 LDCM0461  CL69 HEK-293T C432(0.56); C424(0.95)  LDD1664  [12]
 LDCM0462  CL7 HEK-293T C421(0.96)  LDD1665  [12]
 LDCM0463  CL70 HEK-293T C394(1.15)  LDD1666  [12]
 LDCM0464  CL71 HEK-293T C421(1.08); C397(1.05)  LDD1667  [12]
 LDCM0465  CL72 HEK-293T C424(1.21)  LDD1668  [12]
 LDCM0466  CL73 HEK-293T C424(0.94); C421(0.95)  LDD1669  [12]
 LDCM0467  CL74 HEK-293T C421(0.88)  LDD1670  [12]
 LDCM0470  CL77 HEK-293T C424(0.95)  LDD1673  [12]
 LDCM0471  CL78 HEK-293T C421(1.10)  LDD1674  [12]
 LDCM0472  CL79 HEK-293T C421(1.01)  LDD1675  [12]
 LDCM0473  CL8 HEK-293T C394(0.79)  LDD1676  [12]
 LDCM0474  CL80 HEK-293T C394(1.12)  LDD1677  [12]
 LDCM0475  CL81 HEK-293T C432(0.77); C424(0.86)  LDD1678  [12]
 LDCM0476  CL82 HEK-293T C394(1.10)  LDD1679  [12]
 LDCM0477  CL83 HEK-293T C421(1.06); C397(1.04)  LDD1680  [12]
 LDCM0478  CL84 HEK-293T C424(1.04)  LDD1681  [12]
 LDCM0479  CL85 HEK-293T C424(0.84); C421(0.90)  LDD1682  [12]
 LDCM0480  CL86 HEK-293T C421(0.69)  LDD1683  [12]
 LDCM0481  CL87 HEK-293T C432(1.14)  LDD1684  [12]
 LDCM0483  CL89 HEK-293T C424(0.86)  LDD1686  [12]
 LDCM0484  CL9 HEK-293T C432(0.71); C424(0.86)  LDD1687  [12]
 LDCM0485  CL90 HEK-293T C421(0.78)  LDD1688  [12]
 LDCM0486  CL91 HEK-293T C421(0.85)  LDD1689  [12]
 LDCM0487  CL92 HEK-293T C394(0.99)  LDD1690  [12]
 LDCM0488  CL93 HEK-293T C432(0.66); C424(0.83)  LDD1691  [12]
 LDCM0489  CL94 HEK-293T C394(1.08)  LDD1692  [12]
 LDCM0490  CL95 HEK-293T C421(0.85); C397(0.84)  LDD1693  [12]
 LDCM0491  CL96 HEK-293T C424(0.82)  LDD1694  [12]
 LDCM0492  CL97 HEK-293T C424(1.03); C421(0.97)  LDD1695  [12]
 LDCM0493  CL98 HEK-293T C421(1.06)  LDD1696  [12]
 LDCM0494  CL99 HEK-293T C432(0.93)  LDD1697  [12]
 LDCM0495  E2913 HEK-293T C432(1.72)  LDD1698  [12]
 LDCM0625  F8 Ramos C432(0.53)  LDD2187  [13]
 LDCM0572  Fragment10 Ramos C432(0.52)  LDD2189  [13]
 LDCM0573  Fragment11 Ramos C432(0.43)  LDD2190  [13]
 LDCM0574  Fragment12 Ramos C432(0.81)  LDD2191  [13]
 LDCM0575  Fragment13 Ramos C432(0.63)  LDD2192  [13]
 LDCM0576  Fragment14 Ramos C432(0.53)  LDD2193  [13]
 LDCM0579  Fragment20 Ramos C432(0.54)  LDD2194  [13]
 LDCM0580  Fragment21 Ramos C432(0.64)  LDD2195  [13]
 LDCM0582  Fragment23 Ramos C432(0.34)  LDD2196  [13]
 LDCM0578  Fragment27 Ramos C432(0.15)  LDD2197  [13]
 LDCM0586  Fragment28 Ramos C432(0.34)  LDD2198  [13]
 LDCM0588  Fragment30 Ramos C432(0.59)  LDD2199  [13]
 LDCM0589  Fragment31 Ramos C432(1.26)  LDD2200  [13]
 LDCM0590  Fragment32 Ramos C432(0.43)  LDD2201  [13]
 LDCM0468  Fragment33 HEK-293T C432(1.14)  LDD1671  [12]
 LDCM0596  Fragment38 Ramos C432(0.49)  LDD2203  [13]
 LDCM0566  Fragment4 Ramos C432(1.33)  LDD2184  [13]
 LDCM0427  Fragment51 HEK-293T C421(0.98)  LDD1631  [12]
 LDCM0610  Fragment52 Ramos C432(0.44)  LDD2204  [13]
 LDCM0614  Fragment56 Ramos C432(0.41)  LDD2205  [13]
 LDCM0569  Fragment7 Ramos C432(0.41)  LDD2186  [13]
 LDCM0571  Fragment9 Ramos C432(0.82)  LDD2188  [13]
 LDCM0022  KB02 Ramos C432(0.78)  LDD2182  [13]
 LDCM0023  KB03 Ramos C432(1.22)  LDD2183  [13]
 LDCM0024  KB05 IGR39 C66(1.01)  LDD3315  [2]

The Interaction Atlas With This Target

The Protein(s) Related To This Target

Transporter and channel
Click To Hide/Show 1 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Huntingtin (HTT) Huntingtin family P42858
Immunoglobulin
Click To Hide/Show 1 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Netrin receptor DCC (DCC) DCC family P43146
Other
Click To Hide/Show 2 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Keratin-associated protein 10-9 (KRTAP10-9) KRTAP type 10 family P60411
PRKCA-binding protein (PICK1) . Q9NRD5

References

1 Chemoproteomic profiling of kinases in live cells using electrophilic sulfonyl triazole probes. Chem Sci. 2021 Jan 21;12(9):3295-3307. doi: 10.1039/d0sc06623k.
2 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840
3 Global profiling of functional histidines in live cells using small-molecule photosensitizer and chemical probe relay labelling. Nat Chem. 2024 Jun 4. doi: 10.1038/s41557-024-01545-6. Online ahead of print.
Mass spectrometry data entry: PXD042377
4 SP3-FAIMS Chemoproteomics for High-Coverage Profiling of the Human Cysteinome*. Chembiochem. 2021 May 14;22(10):1841-1851. doi: 10.1002/cbic.202000870. Epub 2021 Feb 18.
Mass spectrometry data entry: PXD023056 , PXD023059 , PXD023058 , PXD023057 , PXD023060
5 Chemoproteomic Profiling by Cysteine Fluoroalkylation Reveals Myrocin G as an Inhibitor of the Nonhomologous End Joining DNA Repair Pathway. J Am Chem Soc. 2021 Dec 8;143(48):20332-20342. doi: 10.1021/jacs.1c09724. Epub 2021 Nov 24.
Mass spectrometry data entry: PXD029255
6 A modification-centric assessment tool for the performance of chemoproteomic probes. Nat Chem Biol. 2022 Aug;18(8):904-912. doi: 10.1038/s41589-022-01074-8. Epub 2022 Jul 21.
Mass spectrometry data entry: PXD027758 , PXD027755 , PXD027760 , PXD027762 , PXD027756 , PXD027591 , PXD007149 , PXD030064 , PXD032392 , PXD027789 , PXD027767 , PXD027764
7 Solid Phase Synthesis of Fluorosulfate Containing Macrocycles for Chemoproteomic Workflows. bioRxiv [Preprint]. 2023 Feb 18:2023.02.17.529022. doi: 10.1101/2023.02.17.529022.
Mass spectrometry data entry: PXD039931
8 DFT-Guided Discovery of Ethynyl-Triazolyl-Phosphinates as Modular Electrophiles for Chemoselective Cysteine Bioconjugation and Profiling. Angew Chem Int Ed Engl. 2022 Oct 10;61(41):e202205348. doi: 10.1002/anie.202205348. Epub 2022 Aug 22.
Mass spectrometry data entry: PXD033004
9 ACR-Based Probe for the Quantitative Profiling of Histidine Reactivity in the Human Proteome. J Am Chem Soc. 2023 Mar 8;145(9):5252-5260. doi: 10.1021/jacs.2c12653. Epub 2023 Feb 27.
10 Oxidant-Induced Bioconjugation for Protein Labeling in Live Cells. ACS Chem Biol. 2023 Jan 20;18(1):112-122. doi: 10.1021/acschembio.2c00740. Epub 2022 Dec 21.
11 Chemoproteomic capture of RNA binding activity in living cells. Nat Commun. 2023 Oct 7;14(1):6282. doi: 10.1038/s41467-023-41844-z.
Mass spectrometry data entry: PXD044625
12 Accelerating multiplexed profiling of protein-ligand interactions: High-throughput plate-based reactive cysteine profiling with minimal input. Cell Chem Biol. 2024 Mar 21;31(3):565-576.e4. doi: 10.1016/j.chembiol.2023.11.015. Epub 2023 Dec 19.
Mass spectrometry data entry: PXD044402
13 Site-specific quantitative cysteine profiling with data-independent acquisition-based mass spectrometry. Methods Enzymol. 2023;679:295-322. doi: 10.1016/bs.mie.2022.07.037. Epub 2022 Sep 7.
Mass spectrometry data entry: PXD027578