General Information of Target

Target ID LDTP07390
Target Name OTU domain-containing protein 7B (OTUD7B)
Gene Name OTUD7B
Gene ID 56957
Synonyms
ZA20D1; OTU domain-containing protein 7B; EC 3.4.19.12; Cellular zinc finger anti-NF-kappa-B protein; Cezanne; Zinc finger A20 domain-containing protein 1; Zinc finger protein Cezanne
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MTLDMDAVLSDFVRSTGAEPGLARDLLEGKNWDVNAALSDFEQLRQVHAGNLPPSFSEGS
GGSRTPEKGFSDREPTRPPRPILQRQDDIVQEKRLSRGISHASSSIVSLARSHVSSNGGG
GGSNEHPLEMPICAFQLPDLTVYNEDFRSFIERDLIEQSMLVALEQAGRLNWWVSVDPTS
QRLLPLATTGDGNCLLHAASLGMWGFHDRDLMLRKALYALMEKGVEKEALKRRWRWQQTQ
QNKESGLVYTEDEWQKEWNELIKLASSEPRMHLGTNGANCGGVESSEEPVYESLEEFHVF
VLAHVLRRPIVVVADTMLRDSGGEAFAPIPFGGIYLPLEVPASQCHRSPLVLAYDQAHFS
ALVSMEQKENTKEQAVIPLTDSEYKLLPLHFAVDPGKGWEWGKDDSDNVRLASVILSLEV
KLHLLHSYMNVKWIPLSSDAQAPLAQPESPTASAGDEPRSTPESGDSDKESVGSSSTSNE
GGRRKEKSKRDREKDKKRADSVANKLGSFGKTLGSKLKKNMGGLMHSKGSKPGGVGTGLG
GSSGTETLEKKKKNSLKSWKGGKEEAAGDGPVSEKPPAESVGNGGSKYSQEVMQSLSILR
TAMQGEGKFIFVGTLKMGHRHQYQEEMIQRYLSDAEERFLAEQKQKEAERKIMNGGIGGG
PPPAKKPEPDAREEQPTGPPAESRAMAFSTGYPGDFTIPRPSGGGVHCQEPRRQLAGGPC
VGGLPPYATFPRQCPPGRPYPHQDSIPSLEPGSHSKDGLHRGALLPPPYRVADSYSNGYR
EPPEPDGWAGGLRGLPPTQTKCKQPNCSFYGHPETNNFCSCCYREELRRREREPDGELLV
HRF
Target Bioclass
Enzyme
Family
Peptidase C64 family
Subcellular location
Cytoplasm
Function
Negative regulator of the non-canonical NF-kappa-B pathway that acts by mediating deubiquitination of TRAF3, an inhibitor of the NF-kappa-B pathway, thereby acting as a negative regulator of B-cell responses. In response to non-canonical NF-kappa-B stimuli, deubiquitinates 'Lys-48'-linked polyubiquitin chains of TRAF3, preventing TRAF3 proteolysis and over-activation of non-canonical NF-kappa-B. Negatively regulates mucosal immunity against infections. Deubiquitinates ZAP70, and thereby regulates T cell receptor (TCR) signaling that leads to the activation of NF-kappa-B. Plays a role in T cell homeostasis and is required for normal T cell responses, including production of IFNG and IL2. Mediates deubiquitination of EGFR. Has deubiquitinating activity toward 'Lys-11', 'Lys-48' and 'Lys-63'-linked polyubiquitin chains. Has a much higher catalytic rate with 'Lys-11'-linked polyubiquitin chains (in vitro); however the physiological significance of these data are unsure. Hydrolyzes both linear and branched forms of polyubiquitin.
Uniprot ID
Q6GQQ9
Ensemble ID
ENST00000581312.6
HGNC ID
HGNC:16683
ChEMBL ID
CHEMBL4630838

Target Site Mutations in Different Cell Lines

Cell line Mutation details Probe for labeling this protein in this cell
22RV1 Deletion: p.T451PfsTer74 .
G361 SNV: p.S774F .
KYSE410 SNV: p.S476F .
LNCaP clone FGC SNV: p.S437F .
NCIH1155 SNV: p.G190R .
NCIH1793 SNV: p.M617I; p.T729S .
P31FUJ SNV: p.N430I .
RL952 Deletion: p.Y769TfsTer59
SNV: p.A7V
.
SKMEL5 SNV: p.R45C .
WM2664 Insertion: p.R347PfsTer9 .

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 9 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
m-APA
 Probe Info 
15.00  LDD0402  [1]
Probe 1
 Probe Info 
Y384(9.22)  LDD3495  [2]
NAIA_5
 Probe Info 
C194(0.72)  LDD2227  [3]
DBIA
 Probe Info 
C708(1.02)  LDD1492  [4]
IA-alkyne
 Probe Info 
C345(0.00); C280(0.00)  LDD0162  [5]
Lodoacetamide azide
 Probe Info 
N.A.  LDD0037  [6]
IPM
 Probe Info 
N.A.  LDD0147  [7]
TFBX
 Probe Info 
N.A.  LDD0148  [7]
Phosphinate-6
 Probe Info 
N.A.  LDD0018  [8]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0214  AC1 HEK-293T C708(1.02)  LDD1507  [4]
 LDCM0215  AC10 HEK-293T C708(1.06)  LDD1508  [4]
 LDCM0226  AC11 HEK-293T C708(0.99); C720(1.15)  LDD1509  [4]
 LDCM0237  AC12 HEK-293T C708(1.10); C720(1.03)  LDD1510  [4]
 LDCM0259  AC14 HEK-293T C708(1.28); C720(0.98)  LDD1512  [4]
 LDCM0270  AC15 HEK-293T C708(1.07); C345(1.28); C720(1.01)  LDD1513  [4]
 LDCM0276  AC17 HEK-293T C708(1.03)  LDD1515  [4]
 LDCM0277  AC18 HEK-293T C708(0.90)  LDD1516  [4]
 LDCM0278  AC19 HEK-293T C708(1.68); C720(1.10)  LDD1517  [4]
 LDCM0279  AC2 HEK-293T C708(1.00)  LDD1518  [4]
 LDCM0280  AC20 HEK-293T C708(1.00); C720(0.98)  LDD1519  [4]
 LDCM0281  AC21 HEK-293T C708(0.91)  LDD1520  [4]
 LDCM0282  AC22 HEK-293T C708(1.08); C720(1.05)  LDD1521  [4]
 LDCM0283  AC23 HEK-293T C708(1.00); C345(0.93); C720(0.86)  LDD1522  [4]
 LDCM0284  AC24 HEK-293T C708(1.08); C720(0.92)  LDD1523  [4]
 LDCM0285  AC25 HEK-293T C708(1.14)  LDD1524  [4]
 LDCM0286  AC26 HEK-293T C708(0.93)  LDD1525  [4]
 LDCM0287  AC27 HEK-293T C708(1.10); C720(1.04)  LDD1526  [4]
 LDCM0288  AC28 HEK-293T C708(1.10); C720(1.05)  LDD1527  [4]
 LDCM0289  AC29 HEK-293T C708(0.93)  LDD1528  [4]
 LDCM0290  AC3 HEK-293T C708(1.06); C720(1.04)  LDD1529  [4]
 LDCM0291  AC30 HEK-293T C708(1.01); C720(0.99)  LDD1530  [4]
 LDCM0292  AC31 HEK-293T C708(1.00); C345(0.98); C720(1.03)  LDD1531  [4]
 LDCM0293  AC32 HEK-293T C708(1.00); C720(1.04)  LDD1532  [4]
 LDCM0294  AC33 HEK-293T C708(1.12)  LDD1533  [4]
 LDCM0295  AC34 HEK-293T C708(1.02)  LDD1534  [4]
 LDCM0296  AC35 HEK-293T C708(1.07); C720(0.94)  LDD1535  [4]
 LDCM0297  AC36 HEK-293T C708(1.04); C720(0.91)  LDD1536  [4]
 LDCM0298  AC37 HEK-293T C708(1.08)  LDD1537  [4]
 LDCM0299  AC38 HEK-293T C708(1.04); C720(1.10)  LDD1538  [4]
 LDCM0300  AC39 HEK-293T C708(1.11); C345(1.03); C720(1.05)  LDD1539  [4]
 LDCM0301  AC4 HEK-293T C708(1.04); C720(1.11)  LDD1540  [4]
 LDCM0302  AC40 HEK-293T C708(1.15); C720(1.21)  LDD1541  [4]
 LDCM0303  AC41 HEK-293T C708(1.11)  LDD1542  [4]
 LDCM0304  AC42 HEK-293T C708(1.31)  LDD1543  [4]
 LDCM0305  AC43 HEK-293T C708(1.08); C720(1.14)  LDD1544  [4]
 LDCM0306  AC44 HEK-293T C708(0.92); C720(1.04)  LDD1545  [4]
 LDCM0307  AC45 HEK-293T C708(1.02)  LDD1546  [4]
 LDCM0308  AC46 HEK-293T C708(1.05); C720(0.93)  LDD1547  [4]
 LDCM0309  AC47 HEK-293T C708(0.93); C345(1.05); C720(0.99)  LDD1548  [4]
 LDCM0310  AC48 HEK-293T C708(1.11); C720(1.10)  LDD1549  [4]
 LDCM0311  AC49 HEK-293T C708(1.07)  LDD1550  [4]
 LDCM0312  AC5 HEK-293T C708(0.92)  LDD1551  [4]
 LDCM0313  AC50 HEK-293T C708(0.93)  LDD1552  [4]
 LDCM0314  AC51 HEK-293T C708(1.08); C720(1.00)  LDD1553  [4]
 LDCM0315  AC52 HEK-293T C708(1.04); C720(0.99)  LDD1554  [4]
 LDCM0316  AC53 HEK-293T C708(0.90)  LDD1555  [4]
 LDCM0317  AC54 HEK-293T C708(1.06); C720(0.95)  LDD1556  [4]
 LDCM0318  AC55 HEK-293T C708(1.03); C345(1.01); C720(1.00)  LDD1557  [4]
 LDCM0319  AC56 HEK-293T C708(1.04); C720(0.90)  LDD1558  [4]
 LDCM0320  AC57 HEK-293T C708(0.98)  LDD1559  [4]
 LDCM0321  AC58 HEK-293T C708(0.99)  LDD1560  [4]
 LDCM0322  AC59 HEK-293T C708(0.97); C720(1.06)  LDD1561  [4]
 LDCM0323  AC6 HEK-293T C708(0.98); C720(0.95)  LDD1562  [4]
 LDCM0324  AC60 HEK-293T C708(1.03); C720(1.01)  LDD1563  [4]
 LDCM0325  AC61 HEK-293T C708(0.98)  LDD1564  [4]
 LDCM0326  AC62 HEK-293T C708(0.96); C720(1.20)  LDD1565  [4]
 LDCM0327  AC63 HEK-293T C708(0.96); C345(1.08); C720(1.01)  LDD1566  [4]
 LDCM0328  AC64 HEK-293T C708(1.08); C720(1.02)  LDD1567  [4]
 LDCM0334  AC7 HEK-293T C708(1.11); C345(1.25); C720(0.95)  LDD1568  [4]
 LDCM0345  AC8 HEK-293T C708(1.09); C720(1.18)  LDD1569  [4]
 LDCM0248  AKOS034007472 HEK-293T C708(1.08)  LDD1511  [4]
 LDCM0356  AKOS034007680 HEK-293T C708(1.10)  LDD1570  [4]
 LDCM0275  AKOS034007705 HEK-293T C708(1.16); C720(0.97)  LDD1514  [4]
 LDCM0632  CL-Sc Hep-G2 C194(0.72)  LDD2227  [3]
 LDCM0367  CL1 HEK-293T C708(1.03); C345(1.24)  LDD1571  [4]
 LDCM0368  CL10 HEK-293T C708(1.70); C720(1.21)  LDD1572  [4]
 LDCM0369  CL100 HEK-293T C708(1.08)  LDD1573  [4]
 LDCM0370  CL101 HEK-293T C708(0.99); C345(1.24)  LDD1574  [4]
 LDCM0371  CL102 HEK-293T C708(1.05)  LDD1575  [4]
 LDCM0372  CL103 HEK-293T C708(1.02)  LDD1576  [4]
 LDCM0373  CL104 HEK-293T C708(0.99)  LDD1577  [4]
 LDCM0374  CL105 HEK-293T C708(0.92); C345(1.14)  LDD1578  [4]
 LDCM0375  CL106 HEK-293T C708(1.06)  LDD1579  [4]
 LDCM0376  CL107 HEK-293T C708(1.04)  LDD1580  [4]
 LDCM0377  CL108 HEK-293T C708(1.01)  LDD1581  [4]
 LDCM0378  CL109 HEK-293T C708(1.04); C345(0.96)  LDD1582  [4]
 LDCM0379  CL11 HEK-293T C708(1.66); C345(0.84); C720(1.18)  LDD1583  [4]
 LDCM0380  CL110 HEK-293T C708(1.01)  LDD1584  [4]
 LDCM0381  CL111 HEK-293T C708(0.97)  LDD1585  [4]
 LDCM0382  CL112 HEK-293T C708(1.14)  LDD1586  [4]
 LDCM0383  CL113 HEK-293T C708(0.96); C345(1.01)  LDD1587  [4]
 LDCM0384  CL114 HEK-293T C708(1.10)  LDD1588  [4]
 LDCM0385  CL115 HEK-293T C708(1.06)  LDD1589  [4]
 LDCM0386  CL116 HEK-293T C708(1.23)  LDD1590  [4]
 LDCM0387  CL117 HEK-293T C708(0.96); C345(1.28)  LDD1591  [4]
 LDCM0388  CL118 HEK-293T C708(1.02)  LDD1592  [4]
 LDCM0389  CL119 HEK-293T C708(1.01)  LDD1593  [4]
 LDCM0390  CL12 HEK-293T C708(1.33); C720(1.16)  LDD1594  [4]
 LDCM0391  CL120 HEK-293T C708(1.01)  LDD1595  [4]
 LDCM0392  CL121 HEK-293T C708(0.94); C345(1.10)  LDD1596  [4]
 LDCM0393  CL122 HEK-293T C708(0.93)  LDD1597  [4]
 LDCM0394  CL123 HEK-293T C708(1.00)  LDD1598  [4]
 LDCM0395  CL124 HEK-293T C708(1.08)  LDD1599  [4]
 LDCM0396  CL125 HEK-293T C708(0.86); C345(1.33)  LDD1600  [4]
 LDCM0397  CL126 HEK-293T C708(0.97)  LDD1601  [4]
 LDCM0398  CL127 HEK-293T C708(0.84)  LDD1602  [4]
 LDCM0399  CL128 HEK-293T C708(0.91)  LDD1603  [4]
 LDCM0400  CL13 HEK-293T C708(1.26); C345(1.04)  LDD1604  [4]
 LDCM0401  CL14 HEK-293T C708(1.11)  LDD1605  [4]
 LDCM0402  CL15 HEK-293T C708(1.11)  LDD1606  [4]
 LDCM0403  CL16 HEK-293T C708(1.22)  LDD1607  [4]
 LDCM0404  CL17 HEK-293T C708(1.30)  LDD1608  [4]
 LDCM0405  CL18 HEK-293T C708(1.25)  LDD1609  [4]
 LDCM0406  CL19 HEK-293T C708(1.31); C720(0.89)  LDD1610  [4]
 LDCM0407  CL2 HEK-293T C708(0.99)  LDD1611  [4]
 LDCM0408  CL20 HEK-293T C708(1.40); C720(1.05)  LDD1612  [4]
 LDCM0409  CL21 HEK-293T C708(1.67)  LDD1613  [4]
 LDCM0410  CL22 HEK-293T C708(1.55); C720(1.01)  LDD1614  [4]
 LDCM0411  CL23 HEK-293T C708(1.97); C345(1.12); C720(1.00)  LDD1615  [4]
 LDCM0412  CL24 HEK-293T C708(1.57); C720(0.99)  LDD1616  [4]
 LDCM0413  CL25 HEK-293T C708(0.78); C345(0.81)  LDD1617  [4]
 LDCM0414  CL26 HEK-293T C708(0.95)  LDD1618  [4]
 LDCM0415  CL27 HEK-293T C708(0.97)  LDD1619  [4]
 LDCM0416  CL28 HEK-293T C708(1.03)  LDD1620  [4]
 LDCM0417  CL29 HEK-293T C708(1.17)  LDD1621  [4]
 LDCM0418  CL3 HEK-293T C708(0.93)  LDD1622  [4]
 LDCM0419  CL30 HEK-293T C708(1.00)  LDD1623  [4]
 LDCM0420  CL31 HEK-293T C708(1.22); C720(0.96)  LDD1624  [4]
 LDCM0421  CL32 HEK-293T C708(1.25); C720(1.03)  LDD1625  [4]
 LDCM0422  CL33 HEK-293T C708(1.14)  LDD1626  [4]
 LDCM0423  CL34 HEK-293T C708(1.37); C720(0.97)  LDD1627  [4]
 LDCM0424  CL35 HEK-293T C708(1.53); C345(0.85); C720(1.11)  LDD1628  [4]
 LDCM0425  CL36 HEK-293T C708(1.48); C720(0.96)  LDD1629  [4]
 LDCM0426  CL37 HEK-293T C708(0.88); C345(0.87)  LDD1630  [4]
 LDCM0428  CL39 HEK-293T C708(0.99)  LDD1632  [4]
 LDCM0429  CL4 HEK-293T C708(0.94)  LDD1633  [4]
 LDCM0430  CL40 HEK-293T C708(1.07)  LDD1634  [4]
 LDCM0431  CL41 HEK-293T C708(1.11)  LDD1635  [4]
 LDCM0432  CL42 HEK-293T C708(0.98)  LDD1636  [4]
 LDCM0433  CL43 HEK-293T C708(1.06); C720(0.95)  LDD1637  [4]
 LDCM0434  CL44 HEK-293T C708(1.13); C720(1.14)  LDD1638  [4]
 LDCM0435  CL45 HEK-293T C708(1.42)  LDD1639  [4]
 LDCM0436  CL46 HEK-293T C708(1.45); C720(1.01)  LDD1640  [4]
 LDCM0437  CL47 HEK-293T C708(1.57); C345(1.09); C720(1.60)  LDD1641  [4]
 LDCM0438  CL48 HEK-293T C708(1.24); C720(1.04)  LDD1642  [4]
 LDCM0439  CL49 HEK-293T C708(0.86); C345(0.90)  LDD1643  [4]
 LDCM0440  CL5 HEK-293T C708(1.02)  LDD1644  [4]
 LDCM0441  CL50 HEK-293T C708(1.02)  LDD1645  [4]
 LDCM0443  CL52 HEK-293T C708(1.16)  LDD1646  [4]
 LDCM0444  CL53 HEK-293T C708(1.09)  LDD1647  [4]
 LDCM0445  CL54 HEK-293T C708(1.04)  LDD1648  [4]
 LDCM0446  CL55 HEK-293T C708(1.17); C720(0.99)  LDD1649  [4]
 LDCM0447  CL56 HEK-293T C708(1.12); C720(1.07)  LDD1650  [4]
 LDCM0448  CL57 HEK-293T C708(1.29)  LDD1651  [4]
 LDCM0449  CL58 HEK-293T C708(1.30); C720(1.06)  LDD1652  [4]
 LDCM0450  CL59 HEK-293T C708(1.41); C345(1.22); C720(1.32)  LDD1653  [4]
 LDCM0451  CL6 HEK-293T C708(1.09)  LDD1654  [4]
 LDCM0452  CL60 HEK-293T C708(1.20); C720(1.08)  LDD1655  [4]
 LDCM0453  CL61 HEK-293T C708(0.87); C345(0.88)  LDD1656  [4]
 LDCM0454  CL62 HEK-293T C708(0.99)  LDD1657  [4]
 LDCM0455  CL63 HEK-293T C708(0.98)  LDD1658  [4]
 LDCM0456  CL64 HEK-293T C708(1.04)  LDD1659  [4]
 LDCM0457  CL65 HEK-293T C708(1.21)  LDD1660  [4]
 LDCM0458  CL66 HEK-293T C708(1.04)  LDD1661  [4]
 LDCM0459  CL67 HEK-293T C708(1.21); C720(0.97)  LDD1662  [4]
 LDCM0460  CL68 HEK-293T C708(1.24); C720(0.99)  LDD1663  [4]
 LDCM0461  CL69 HEK-293T C708(1.00)  LDD1664  [4]
 LDCM0462  CL7 HEK-293T C708(1.05); C720(0.95)  LDD1665  [4]
 LDCM0463  CL70 HEK-293T C708(1.41); C720(0.98)  LDD1666  [4]
 LDCM0464  CL71 HEK-293T C708(1.13); C345(1.01); C720(1.24)  LDD1667  [4]
 LDCM0465  CL72 HEK-293T C708(1.32); C720(1.05)  LDD1668  [4]
 LDCM0466  CL73 HEK-293T C708(1.00); C345(1.54)  LDD1669  [4]
 LDCM0467  CL74 HEK-293T C708(0.94)  LDD1670  [4]
 LDCM0469  CL76 HEK-293T C708(1.02)  LDD1672  [4]
 LDCM0470  CL77 HEK-293T C708(1.08)  LDD1673  [4]
 LDCM0471  CL78 HEK-293T C708(0.95)  LDD1674  [4]
 LDCM0472  CL79 HEK-293T C708(1.05); C720(0.96)  LDD1675  [4]
 LDCM0473  CL8 HEK-293T C708(1.06); C720(0.99)  LDD1676  [4]
 LDCM0474  CL80 HEK-293T C708(1.03); C720(1.08)  LDD1677  [4]
 LDCM0475  CL81 HEK-293T C708(1.13)  LDD1678  [4]
 LDCM0476  CL82 HEK-293T C708(1.23); C720(0.98)  LDD1679  [4]
 LDCM0477  CL83 HEK-293T C708(1.49); C345(0.81); C720(1.15)  LDD1680  [4]
 LDCM0478  CL84 HEK-293T C708(1.27); C720(1.07)  LDD1681  [4]
 LDCM0479  CL85 HEK-293T C708(0.90); C345(1.19)  LDD1682  [4]
 LDCM0480  CL86 HEK-293T C708(0.88)  LDD1683  [4]
 LDCM0481  CL87 HEK-293T C708(0.86)  LDD1684  [4]
 LDCM0482  CL88 HEK-293T C708(0.94)  LDD1685  [4]
 LDCM0483  CL89 HEK-293T C708(1.01)  LDD1686  [4]
 LDCM0484  CL9 HEK-293T C708(1.01)  LDD1687  [4]
 LDCM0485  CL90 HEK-293T C708(1.10)  LDD1688  [4]
 LDCM0486  CL91 HEK-293T C708(0.98); C720(1.09)  LDD1689  [4]
 LDCM0487  CL92 HEK-293T C708(1.08); C720(0.98)  LDD1690  [4]
 LDCM0488  CL93 HEK-293T C708(1.12)  LDD1691  [4]
 LDCM0489  CL94 HEK-293T C708(1.30); C720(0.91)  LDD1692  [4]
 LDCM0490  CL95 HEK-293T C708(1.26); C345(1.06); C720(1.19)  LDD1693  [4]
 LDCM0491  CL96 HEK-293T C708(0.96); C720(1.13)  LDD1694  [4]
 LDCM0492  CL97 HEK-293T C708(0.95); C345(0.89)  LDD1695  [4]
 LDCM0493  CL98 HEK-293T C708(1.03)  LDD1696  [4]
 LDCM0494  CL99 HEK-293T C708(0.90)  LDD1697  [4]
 LDCM0495  E2913 HEK-293T C708(1.06)  LDD1698  [4]
 LDCM0468  Fragment33 HEK-293T C708(0.99)  LDD1671  [4]
 LDCM0427  Fragment51 HEK-293T C708(1.03)  LDD1631  [4]
 LDCM0022  KB02 HEK-293T C708(1.02)  LDD1492  [4]
 LDCM0023  KB03 HEK-293T C708(1.06)  LDD1497  [4]
 LDCM0024  KB05 HEK-293T C708(1.07)  LDD1502  [4]

The Interaction Atlas With This Target

The Protein(s) Related To This Target

Enzyme
Click To Hide/Show 16 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
NADH dehydrogenase flavoprotein 2, mitochondrial (NDUFV2) Complex I 24 kDa subunit family P19404
Dopamine beta-hydroxylase (DBH) Copper type II ascorbate-dependent monooxygenase family P09172
Superoxide dismutase [Cu-Zn] (SOD1) Cu-Zn superoxide dismutase family P00441
Caspase-6 (CASP6) Peptidase C14A family P55212
Parkinson disease protein 7 (PARK7) Peptidase C56 family Q99497
Ubiquitin thioesterase otulin (OTULIN) Peptidase C65 family Q96BN8
Serine protease HTRA2, mitochondrial (HTRA2) Peptidase S1C family O43464
Proteasome subunit beta type-1 (PSMB1) Peptidase T1B family P20618
Phytanoyl-CoA dioxygenase, peroxisomal (PHYH) PhyH family O14832
Mitogen-activated protein kinase 3 (MAPK3) CMGC Ser/Thr protein kinase family P27361
Fibroblast growth factor receptor 3 (FGFR3) Tyr protein kinase family P22607
Ribose-phosphate pyrophosphokinase 1 (PRPS1) Ribose-phosphate pyrophosphokinase family P60891
GTP-binding nuclear protein Ran (RAN) Ran family P62826
Eukaryotic translation initiation factor 2 subunit 3 (EIF2S3) Classic translation factor GTPase family P41091
Transthyretin (TTR) Transthyretin family P02766
E3 ubiquitin-protein ligase NEDD4 (NEDD4) . P46934
Transporter and channel
Click To Hide/Show 5 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Glutamate receptor ionotropic, NMDA 2C (GRIN2C) Glutamate-gated ion channel family Q14957
Junctophilin-3 (JPH3) Junctophilin family Q8WXH2
Nucleoporin p58/p45 (NUP58) NUP58 family Q9BVL2
Alpha-synuclein (SNCA) Synuclein family P37840
Wolframin (WFS1) . O76024
Transcription factor
Click To Hide/Show 2 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Heat shock transcription factor, Y-linked (HSFY1; HSFY2) HSF family Q96LI6
Krueppel-like factor 11 (KLF11) Sp1 C2H2-type zinc-finger protein family O14901
Other
Click To Hide/Show 19 Protein(s) Interacting with This Target
Protein name Family Uniprot ID
Ataxin-1 (ATXN1) ATXN1 family P54253
Cell death-inducing p53-target protein 1 (CDIP1) CDIP1/LITAF family Q9H305
Heat shock-related 70 kDa protein 2 (HSPA2) Heat shock protein 70 family P54652
Axonemal dynein light intermediate polypeptide 1 (DNALI1) Inner dynein arm light chain family O14645
Glial fibrillary acidic protein (GFAP) Intermediate filament family P14136
Phosphatidylinositol 3-kinase regulatory subunit gamma (PIK3R3) PI3K p85 subunit family Q92569
Alpha-2-macroglobulin (A2M) Protease inhibitor I39 (alpha-2-macroglobulin) family P01023
Heat shock protein beta-1 (HSPB1) Small heat shock protein (HSP20) family P04792
Polyubiquitin-B (UBB) Ubiquitin family P0CG47
Gelsolin (GSN) Villin/gelsolin family P06396
Coiled-coil domain-containing protein 50 (CCDC50) . Q8IVM0
DAZ-associated protein 2 (DAZAP2) . Q15038
EPM2A-interacting protein 1 (EPM2AIP1) . Q7L775
Methyl-CpG-binding protein 2 (MECP2) . P51608
RING finger protein 11 (RNF11) . Q9Y3C5
Spartin (SPART) . Q8N0X7
Sprouty-related, EVH1 domain-containing protein 1 (SPRED1) . Q7Z699
TAR DNA-binding protein 43 (TARDBP) . Q13148
Ubiquilin-1 (UBQLN1) . Q9UMX0

References

1 Quantitative and Site-Specific Chemoproteomic Profiling of Targets of Acrolein. Chem Res Toxicol. 2019 Mar 18;32(3):467-473. doi: 10.1021/acs.chemrestox.8b00343. Epub 2019 Jan 15.
2 An Azo Coupling-Based Chemoproteomic Approach to Systematically Profile the Tyrosine Reactivity in the Human Proteome. Anal Chem. 2021 Jul 27;93(29):10334-10342. doi: 10.1021/acs.analchem.1c01935. Epub 2021 Jul 12.
3 N-Acryloylindole-alkyne (NAIA) enables imaging and profiling new ligandable cysteines and oxidized thiols by chemoproteomics. Nat Commun. 2023 Jun 15;14(1):3564. doi: 10.1038/s41467-023-39268-w.
Mass spectrometry data entry: PXD041264
4 Accelerating multiplexed profiling of protein-ligand interactions: High-throughput plate-based reactive cysteine profiling with minimal input. Cell Chem Biol. 2024 Mar 21;31(3):565-576.e4. doi: 10.1016/j.chembiol.2023.11.015. Epub 2023 Dec 19.
Mass spectrometry data entry: PXD044402
5 SP3-FAIMS Chemoproteomics for High-Coverage Profiling of the Human Cysteinome*. Chembiochem. 2021 May 14;22(10):1841-1851. doi: 10.1002/cbic.202000870. Epub 2021 Feb 18.
Mass spectrometry data entry: PXD023056 , PXD023059 , PXD023058 , PXD023057 , PXD023060
6 Enhancing Cysteine Chemoproteomic Coverage through Systematic Assessment of Click Chemistry Product Fragmentation. Anal Chem. 2022 Mar 8;94(9):3800-3810. doi: 10.1021/acs.analchem.1c04402. Epub 2022 Feb 23.
Mass spectrometry data entry: PXD028853
7 Chemoproteomic Profiling by Cysteine Fluoroalkylation Reveals Myrocin G as an Inhibitor of the Nonhomologous End Joining DNA Repair Pathway. J Am Chem Soc. 2021 Dec 8;143(48):20332-20342. doi: 10.1021/jacs.1c09724. Epub 2021 Nov 24.
Mass spectrometry data entry: PXD029255
8 DFT-Guided Discovery of Ethynyl-Triazolyl-Phosphinates as Modular Electrophiles for Chemoselective Cysteine Bioconjugation and Profiling. Angew Chem Int Ed Engl. 2022 Oct 10;61(41):e202205348. doi: 10.1002/anie.202205348. Epub 2022 Aug 22.
Mass spectrometry data entry: PXD033004