General Information of Experiment

Probe Name photo_BS  Probe Info 
Probe concentration 10 uM
Criteria Quantification: Probe vs (Probe+Competitor)
Quantitative Method
SILAC
Competitor Name Bromosprine  Competitor Info 
Competitor Concentration 10 mM
In Vivo Experiment Model Model Type Living cell
Derived Tissue Peripheral blood
Disease Model Normal
Model Name Human normal cells (HEK-293T)

Interaction Altas of This Experiment [1]

Enzyme
Click to Show/Hide to Show 1 Protein Related to This Bioclass
Target ID Target Name Binding Ratio
 LDTP16070  Epimerase family protein SDR39U1 (SDR39U1) 2.3
Other
Click to Show/Hide to Show 5 Protein Related to This Bioclass
Target ID Target Name Binding Ratio
 LDTP12369  Bromodomain-containing protein 7 (BRD7) 2.7
 LDTP06304  Bromodomain-containing protein 3 (BRD3) 2.4
 LDTP01074  Bromodomain-containing protein 4 (BRD4) 2.3
 LDTP12059  Bromodomain-containing protein 9 (BRD9) 2.1
 LDTP03322  Bromodomain-containing protein 2 (BRD2) 2.0

References

1 Chemical Proteomic Profiling of Bromodomains Enables the Wide-Spectrum Evaluation of Bromodomain Inhibitors in Living Cells. J Am Chem Soc. 2019 Jul 24;141(29):11497-11505. doi: 10.1021/jacs.9b02738. Epub 2019 Jul 9.