General Information of Target

Target ID LDTP17342
Target Name Putative protein FRMPD2-like (FRMPD2B)
Gene Name FRMPD2B
Synonyms
FRMPD2L1; FRMPD2L2; FRMPD2P1; FRMPD2P2; PDZD5A; PDZD5B; PDZK5A; PDZK5B; Putative protein FRMPD2-like; FERM and PDZ domain-containing protein 2 pseudogene 1; FERM and PDZ domain-containing protein 2B pseudogene; PDZ domain-containing protein 5A
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MSYFPILFFFFLKRCPSYTEPQNLTGVSEFLLLGLSEDPELQPVLAGLFLSMYLVTVLGN
LLIILAVSSDSHLHTPMYFFLSNLSLADIGFTSTTVPKMIVDMQTHSRVISYEGCLTQMS
FFVLFACMDDMLLSVMAYDRFVAICHPLHYRIIMNPRLCGFLILLSFFISLLDSQLHNLI
MLQLTCFKDVDISNFFCDPSQLLHLRCSDTFINEMVIYFMGAIFGCLPISGILFSYYKIV
SPILRVPTSDGKYKAFSTCGSHLAVVCLFYGTGLVGYLSSAVLPSPRKSMVASVMYTVVT
PMLNPFIYSLRNKDIQSALCRLHGRIIKSHHLHPFCYMG
Target Bioclass
Other
Uniprot ID
Q6IN97
HGNC ID
HGNC:16843

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 1 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
BTD
 Probe Info 
C30(0.79)  LDD2097  [1]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0504  Nucleophilic fragment 15a MDA-MB-231 C30(0.79)  LDD2097  [1]
 LDCM0508  Nucleophilic fragment 17a MDA-MB-231 C30(0.59)  LDD2101  [1]

References

1 Nucleophilic covalent ligand discovery for the cysteine redoxome. Nat Chem Biol. 2023 Nov;19(11):1309-1319. doi: 10.1038/s41589-023-01330-5. Epub 2023 May 29.
Mass spectrometry data entry: PXD039908 , PXD029761