General Information of Target

Target ID LDTP19134
Target Name Cancer/testis antigen family 45 member A10 (CT45A10)
Gene Name CT45A10
Gene ID 102723631
Synonyms
Cancer/testis antigen family 45 member A10; Cancer/testis antigen 45A10
3D Structure
Download
2D Sequence (FASTA)
Download
3D Structure (PDB)
Download
Sequence
MTDKTEKVAVDPETVFKRPRECDSPSYQKRQRMALLARKQGAGDSLIAGSAMSKEKKLMT
GHAIPPSQLDSQIDDFTGFSKDGMMQKPGSNAPVGGNVTSSFSGDDLECRETASSPKSQR
EINADIKRKLVKELRCVGQKYEKIFEMLEGVQGPTAVRKRFFESIIKEAARCMRRDFVKH
LKKKLKRMI
Target Bioclass
Other
Family
CT45 family
Uniprot ID
P0DMU9
Ensemble ID
ENST00000611668.4
HGNC ID
HGNC:51263

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 1 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
DBIA
 Probe Info 
C22(1.05)  LDD3311  [1]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0022  KB02 A101D C22(1.92)  LDD2250  [1]
 LDCM0023  KB03 A101D C22(2.81)  LDD2667  [1]
 LDCM0024  KB05 G361 C22(1.05)  LDD3311  [1]

References

1 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840