General Information of Target

Target ID LDTP18428
Target Name EF-hand and coiled-coil domain-containing protein 1 (EFCC1)
Gene Name EFCC1
Gene ID 79825
Synonyms
C3orf73; CCDC48; EF-hand and coiled-coil domain-containing protein 1; Coiled-coil domain-containing protein 48
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MAALIAENFRFLSLFFKSKDVMIFNGLVALGTVGSQELFSVVAFHCPCSPARNYLYGLAA
IGVPALVLFIIGIILNNHTWNLVAECQHRRTKNCSAAPTFLLLSSILGRAAVAPVTWSVI
SLLRGEAYVCALSEFVDPSSLTAREEHFPSAHATEILARFPCKENPDNLSDFREEVSRRL
RYESQLFGWLLIGVVAILVFLTKCLKHYCSPLSYRQEAYWAQYRANEDQLFQRTAEVHSR
VLAANNVRRFFGFVALNKDDEELIANFPVEGTQPRPQWNAITGVYLYRENQGLPLYSRLH
KWAQGLAGNGAAPDNVEMALLPS
Target Bioclass
Other
Uniprot ID
Q9HA90
Ensemble ID
ENST00000436022.2
HGNC ID
HGNC:25692

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 1 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
DBIA
 Probe Info 
C83(1.73); C472(1.31)  LDD2470  [1]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0022  KB02 MGG23 C83(1.73); C472(1.31)  LDD2470  [1]
 LDCM0023  KB03 MGG75 C83(4.56)  LDD2888  [1]
 LDCM0024  KB05 MGG75 C83(5.56)  LDD3305  [1]

References

1 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840