General Information of Target

Target ID LDTP18329
Target Name Ferritin heavy polypeptide-like 17 (FTHL17)
Gene Name FTHL17
Gene ID 53940
Synonyms
Ferritin heavy polypeptide-like 17; Cancer/testis antigen 38; CT38
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MALRPEDPSSGFRHSNVVAFINEKMARHTKGPEFYLENISLSWEKVEDKLRAILEDSEVP
SEVKEACTWGSLALGVRFAHRQAQLQRHRVRWLHGFAKLHKSAAQALASDLKKLREQQET
ERKEAASRLRMAQTSLVEVQKERDKELVSPHEWEQGAGWPGLATAGGVCTEGAAEEEEEA
AVAAAGAAGGKGAEEEQRDVEVVAAPVEAMAPPVEAGAAPMETQFPHVEARAASMETTEK
LERILLQLLGDADQEKYTYWGQKEGDLRSVETATSYFSGTTNPWSRASSEPLPVQLPASY
SYSYSSPFSSFSDIPTISPPQATVTAPVPPQLPSDWEAFDTSLWSDGGPHRIDHQEHPRD
RRYSEPHQQRPPVYRRPGDWDCPWCNAVNFSRRDTCFDCGKGIWLQKPH
Target Bioclass
Other
Family
Ferritin family
Uniprot ID
Q9BXU8
Ensemble ID
ENST00000359202.5
HGNC ID
HGNC:3987

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 1 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
DBIA
 Probe Info 
C82(1.62)  LDD2356  [1]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0022  KB02 HGC-27 C82(1.62)  LDD2356  [1]
 LDCM0023  KB03 HGC-27 C82(1.23)  LDD2773  [1]
 LDCM0024  KB05 AGS C82(1.33)  LDD3097  [1]

References

1 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840