General Information of Target

Target ID LDTP16959
Target Name Mas-related G-protein coupled receptor MRG (MAS1L)
Gene Name MAS1L
Gene ID 116511
Synonyms
MRG; Mas-related G-protein coupled receptor MRG; MAS-R; MAS1-like
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MGEHNLLNPGFVGPLVNIHTGDTFYFPNFRASGAQLPGLPSLSYPRRDNVCSLSWPSAEP
CNGYPQPYLGSPVSLNPPFGRTCELARVEDGKGYYREPCAEGGGGGLKREERGRDPGAGP
GAALLPLEPSGPPALGFKYDYAAGGGGGDGGGGAGPPHDPPSCQSLESDSSSSLLNEGNK
GAGAGDPGSLVSPLNPGGGLSASGAPWYPINSRSRKKRKPYSKLQLAELEGEFLVNEFIT
RQRRRELSDRLNLSDQQVKIWFQNRRMKKKRLLLREQALSFF
Target Bioclass
GPCR
Family
G-protein coupled receptor 1 family, Mas subfamily
Subcellular location
Cell membrane
Uniprot ID
P35410
Ensemble ID
ENST00000377127.4
HGNC ID
HGNC:13961
ChEMBL ID
CHEMBL4523857

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 1 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
IA-alkyne
 Probe Info 
C1238(0.00); C797(0.00); C576(0.00); C500(0.00)  LDD0161  [1]

References

1 SP3-FAIMS Chemoproteomics for High-Coverage Profiling of the Human Cysteinome*. Chembiochem. 2021 May 14;22(10):1841-1851. doi: 10.1002/cbic.202000870. Epub 2021 Feb 18.
Mass spectrometry data entry: PXD023056 , PXD023059 , PXD023058 , PXD023057 , PXD023060