General Information of Target

Target ID LDTP16332
Target Name Calcium-activated chloride channel regulator family member 3 (CLCA3P)
Gene Name CLCA3P
Synonyms
CLCA3; Calcium-activated chloride channel regulator family member 3; Calcium-activated chloride channel family member 3; hCLCA3
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MAAPPQLRALLVVVNALLRKRRYHAALAVLKGFRNGAVYGAKIRAPHALVMTFLFRNGSL
QEKLWAILQATYIHSWNLARFVFTYKGLRALQSYIQGKTYPAHAFLAAFLGGILVFGENN
NINSQINMYLLSRVLFALSRLAVEKGYIPEPRWDPFPLLTAVVWGLVLWLFEYHRSTLQP
SLQSSMTYLYEDSNVWHDISDFLVYNKSRPSN
Target Bioclass
Transporter and channel
Family
CLCR family
Subcellular location
Secreted
Uniprot ID
Q9Y6N3
HGNC ID
HGNC:2017
ChEMBL ID
CHEMBL2364708

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 1 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
BTD
 Probe Info 
C205(1.38)  LDD2127  [1]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0534  Nucleophilic fragment 30a MDA-MB-231 C205(1.38)  LDD2127  [1]

References

1 Nucleophilic covalent ligand discovery for the cysteine redoxome. Nat Chem Biol. 2023 Nov;19(11):1309-1319. doi: 10.1038/s41589-023-01330-5. Epub 2023 May 29.
Mass spectrometry data entry: PXD039908 , PXD029761