General Information of Target

Target ID LDTP15604
Target Name Solute carrier family 2, facilitated glucose transporter member 12 (SLC2A12)
Gene Name SLC2A12
Gene ID 154091
Synonyms
GLUT12; Solute carrier family 2, facilitated glucose transporter member 12; Glucose transporter type 12; GLUT-12
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
METTMGFMDDNATNTSTSFLSVLNPHGAHATSFPFNFSYSDYDMPLDEDEDVTNSRTFFA
AKIVIGMALVGIMLVCGIGNFIFIAALVRYKKLRNLTNLLIANLAISDFLVAIVCCPFEM
DYYVVRQLSWEHGHVLCTSVNYLRTVSLYVSTNALLAIAIDRYLAIVHPLRPRMKCQTAT
GLIALVWTVSILIAIPSAYFTTETVLVIVKSQEKIFCGQIWPVDQQLYYKSYFLFIFGIE
FVGPVVTMTLCYARISRELWFKAVPGFQTEQIRKRLRCRRKTVLVLMCILTAYVLCWAPF
YGFTIVRDFFPTVFVKEKHYLTAFYIVECIAMSNSMINTLCFVTVKNDTVKYFKKIMLLH
WKASYNGGKSSADLDLKTIGMPATEEVDCIRLK
Target Type
Literature-reported
Target Bioclass
Transporter and channel
Family
Major facilitator superfamily, Sugar transporter (TC 2.A.1.1) family, Glucose transporter subfamily
Subcellular location
Cell membrane
Function Insulin-independent facilitative glucose transporter.
TTD ID
T60156
Uniprot ID
Q8TD20
DrugMap ID
TTZO36H
Ensemble ID
ENST00000275230.6
HGNC ID
HGNC:18067

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 1 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
DBIA
 Probe Info 
C601(0.98)  LDD3323  [1]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0022  KB02 769-P C601(1.24)  LDD2246  [1]
 LDCM0023  KB03 769-P C601(1.47)  LDD2663  [1]
 LDCM0024  KB05 SKMEL24 C601(0.98)  LDD3323  [1]

References

1 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840