General Information of Target

Target ID LDTP13051
Target Name Centrosomal protein of 126 kDa (CEP126)
Gene Name CEP126
Gene ID 57562
Synonyms
KIAA1377; Centrosomal protein of 126 kDa
3D Structure
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2D Sequence (FASTA)
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3D Structure (PDB)
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Sequence
MASDSMSSKQARNHITKGKRQQQHQQIKNRSSISDGDGEDSFIFEANEAWKDFHGSLLRF
YENGELCDVTLKVGSKLISCHKLVLACVIPYFRAMFLSEMAEAKQTLIEIRDFDGDAIED
LVKFVYSSRLTLTVDNVQPLLYAACILQVELVARACCEYMKLHFHPSNCLAVRAFAESHN
RIDLMDMADQYACDHFTEVVECEDFVSVSPQHLHKLLSSSDLNIENEKQVYNAAIKWLLA
NPQHHSKWLDETLAQVRLPLLPVDFLMGVVAKEQIVKQNLKCRDLLDEARNYHLHLSSRA
VPDFEYSIRTTPRKHTAGVLFCVGGRGGSGDPFRSIECYSINKNSWFFGPEMNSRRRHVG
VISVEGKVYAVGGHDGNEHLGSMEMFDPLTNKWMMKASMNTKRRGIALASLGGPIYAIGG
LDDNTCFNDVERYDIESDQWSTVAPMNTPRGGVGSVALVNHVYAVGGNDGMASLSSVERY
DPHLDKWIEVKEMGQRRAGNGVSKLHGCLYVVGGFDDNSPLSSVERYDPRSNKWDYVAAL
TTPRGGVGIATVMGKIFAVGGHNGNAYLNTVEAFDPVLNRWELVGSVSHCRAGAGVAVCS
CLTSQIRDVGHGSNNVVDCM
Target Bioclass
Other
Subcellular location
Midbody
Function Participates in cytokinesis. Necessary for microtubules and mitotic spindle organization. Involved in primary cilium formation.
Uniprot ID
Q9P2H0
Ensemble ID
ENST00000263468.13
HGNC ID
HGNC:29264

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 1 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
DBIA
 Probe Info 
C490(2.88)  LDD3439  [1]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0022  KB02 ECC2 C490(2.36)  LDD2320  [1]
 LDCM0023  KB03 ECC2 C490(3.41)  LDD2737  [1]
 LDCM0024  KB05 SNU-1196 C490(2.88)  LDD3439  [1]

References

1 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840