General Information of Target

Target ID LDTP08914
Target Name Translocating chain-associated membrane protein 1-like 1 (TRAM1L1)
Gene Name TRAM1L1
Gene ID 133022
Synonyms
Translocating chain-associated membrane protein 1-like 1
3D Structure
Download
2D Sequence (FASTA)
Download
3D Structure (PDB)
Download
Sequence
MGLRKKSTKNPPVLSQEFILQNHADIVSCVGMFFLLGLVFEGTAEASIVFLTLQHSVAVP
AAEEQATGSKSLYYYGVKDLATVFFYMLVAIIIHATIQEYVLDKINKRMQFTKAKQNKFN
ESGQFSVFYFFSCIWGTFILISENCLSDPTLIWKARPHSMMTFQMKFFYISQLAYWFHAF
PELYFQKTKKQDIPRQLVYIGLHLFHITGAYLLYLNHLGLLLLVLHYFVELLSHMCGLFY
FSDEKYQKGISLWAIVFILGRLVTLIVSVLTVGFHLAGSQNRNPDALTGNVNVLAAKIAV
LSSSCTIQAYVTWNLITLWLQRWVEDSNIQASCMKKKRSRSSKKRTENGVGVETSNRVDC
PPKRKEKSS
Target Bioclass
Transporter and channel
Family
TRAM family
Subcellular location
Endoplasmic reticulum membrane
Function Stimulatory or required for the translocation of secretory proteins across the ER membrane.
Uniprot ID
Q8N609
Ensemble ID
ENST00000310754.5
HGNC ID
HGNC:28371

Probe(s) Labeling This Target

ABPP Probe
Click To Hide/Show 1 Probe Related to This Target
Probe name Structure Binding Site(Ratio) Interaction ID Ref
DBIA
 Probe Info 
C360(1.34)  LDD3365  [1]

Competitor(s) Related to This Target

Competitor ID Name Cell line Binding Site(Ratio) Interaction ID Ref
 LDCM0022  KB02 OVCAR-3 C360(1.42)  LDD2531  [1]
 LDCM0023  KB03 EFO-27 C360(2.13)  LDD2739  [1]
 LDCM0024  KB05 OVCAR-3 C360(1.34)  LDD3365  [1]

References

1 DrugMap: A quantitative pan-cancer analysis of cysteine ligandability. Cell. 2024 May 9;187(10):2536-2556.e30. doi: 10.1016/j.cell.2024.03.027. Epub 2024 Apr 22.
Mass spectrometry data entry: PXD047840