Details of the Target
General Information of Target
| Target ID | LDTP08175 | |||||
|---|---|---|---|---|---|---|
| Target Name | Adhesion G protein-coupled receptor A1 (ADGRA1) | |||||
| Gene Name | ADGRA1 | |||||
| Gene ID | 84435 | |||||
| Synonyms |
GPR123; KIAA1828; Adhesion G protein-coupled receptor A1; G-protein coupled receptor 123 |
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| 3D Structure | ||||||
| Sequence |
MDLKTVLSLPRYPGEFLHPVVYACTAVMLLCLLASFVTYIVHQSAIRISRKGRHTLLNFC
FHAALTFTVFAGGINRTKYPILCQAVGIVLHYSTLSTMLWIGVTARNIYKQVTKKAPLCL DTDQPPYPRQPLLRFYLVSGGVPFIICGVTAATNIRNYGTEDEDTAYCWMAWEPSLGAFY GPAAIITLVTCVYFLGTYVQLRRHPGRRYELRTQPEEQRRLATPEGGRGIRPGTPPAHDA PGASVLQNEHSFQAQLRAAAFTLFLFTATWAFGALAVSQGHFLDMVFSCLYGAFCVTLGL FVLIHHCAKREDVWQCWWACCPPRKDAHPALDANGAALGRAACLHSPGLGQPRGFAHPPG PCKMTNLQAAQGHASCLSPATPCCAKMHCEPLTADEAHVHLQEEGAFGHDPHLHGCLQGR TKPPYFSRHPAEEPEYAYHIPSSLDGSPRSSRTDSPPSSLDGPAGTHTLACCTQGDPFPM VTQPEGSDGSPALYSCPTQPGREAALGPGHLEMLRRTQSLPFGGPSQNGLPKGKLLEGLP FGTDGTGNIRTGPWKNETTV |
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| Target Bioclass |
GPCR
|
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| Family |
G-protein coupled receptor 2 family, Adhesion G-protein coupled receptor (ADGR) subfamily
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| Subcellular location |
Membrane
|
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| Function | Orphan receptor. | |||||
| Uniprot ID | ||||||
| Ensemble ID | ||||||
| HGNC ID | ||||||
| ChEMBL ID | ||||||
Probe(s) Labeling This Target
ABPP Probe
| Probe name | Structure | Binding Site(Ratio) | Interaction ID | Ref | |
|---|---|---|---|---|---|
|
TFBX Probe Info |
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N.A. | LDD0148 | [1] | |

